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Cat. No.	Product Name
L1510	核受体化合物库	531 compounds
	531 个核受体作用化合物的独特集合，可用于高通量筛选和高内涵筛选；
L2610	神经递质受体化合物库	1513 compounds
	1513 种与神经递质受体相关的化合物，用于高通量、高内涵筛选；
L2700	肾上腺素能受体化合物库	193 compounds
	193 种特异靶向肾上腺素受体的生物活性小分子化合物的集合，是相关疾病药物筛选的有效工具；
L2800	5-羟色胺分子库	268 compounds
	268 种生物活性小分子化合物，用于高通量、高内涵筛选；
L3300	组胺&褪黑色素化合物库	153 compounds
	153 种生物活性小分子化合物，用于高通量、高内涵筛选；
L7600	趋化因子抑制剂库	59 compounds
	59 种趋化因子或其受体抑制剂的独特集合，可用于高通量筛选和高内涵筛选；
L2195	抗前列腺癌化合物库	2070 compounds
	2070 种与前列腺癌相关的化合物，可以用于高通量和高内涵筛选
L2191	抗乳腺癌化合物库	1939 compounds
	1939 种与乳腺癌相关的化合物，可以用于抗乳腺癌药物研发和药理研究；
L2193	抗肝癌化合物库	1787 compounds
	1787 种与肝癌相关的化合物，可以用于抗肝癌药物研发和药理研究；
L9830	抗帕金森病化合物库	857 compounds
	857 种帕金森病相关的化合物集合，可用于高通量和高内涵筛选；
L1400	MAPK 抑制剂库	365 compounds
	365 种与MAPK 信号通路相关的生物活性小分子化合物的特有集合，可用于高通量筛选和高内涵筛选；
L7110	抗高血压化合物库	678 compounds
	678 种高血压相关的小分子，用于高通量和高内涵筛选；
L4100	TGF-β/Smad靶点化合物库	184 compounds
	184 个 TGF-β/Smad 靶点相关的小分子化合物的特有集合，用于高通量、高内涵筛选；
L9000	细胞凋亡化合物库	1760 compounds
	1760 种与凋亡相关的生物活性小分子化合物的特有集合，多用于研究肿瘤发生发展机制和抗癌药物筛选等。可用于高通量筛选和高内涵筛选；
L9840	抗阿尔茨海默症化合物库	986 compounds
	986 种阿尔茨海默症相关的化合物集合，可用于高通量和高内涵筛选；

Cat. No.	Product Name	Target	Signaling Pathways
T21723L	EGF Receptor Peptide Acetate EGF Receptor Peptide Acetate (96249-43-3 Free base),Epidermal Growth Factor Receptor Peptide Acetate(96249-43-3 Free base)	Others	Others
	Epidermal Growth Factor Receptor Peptide Acetate (Epidermal Growth Factor Receptor Peptide Acetate (96249-43-3 Free base)) 存在于细胞表面，通过与其特异性配体的结合而被激活。EGFR 属于受体酪氨酸激酶(RTK) 的 ErbB 家族。
T37793	A2B receptor antagonist 2 A2B receptor antagonist 2	Adenosine Receptor	GPCR/G Protein; Neuroscience
	A2B receptor antagonist 2 是腺苷受体 A2B 的拮抗剂（rA1 的 Ki = 2.30 μM，rA2A 的 Ki = 6.8 μM，hA2B 的 3.44 μM）。
T4031	S1p receptor agonist 1 S1p-receptor-agonist-1	S1P Receptor; LPL Receptor	GPCR/G Protein
	S1p receptor agonist 1 (S1p-receptor-agonist-1) 是有口服活性的S1P 受体激动剂，具有诱导 S1P1 内化的活性，EC50为9.83 nM。它有潜力用于关节炎和实验性自身免疫性脑炎)的相关研究。
T38287	C3a Receptor Agonist C3a receptor agonist 1,C3a受体激动剂,Complement 3a Receptor Agonist	Complement System	Immunology/Inflammation
	C3a Receptor Agonist (C3a receptor agonist 1) 结合免疫系统补体途径中的G 蛋白偶联C3a 受体(C3aRs)。在肠缺血再灌注损伤模型中，C3aR 的激活可防止中性粒细胞动员。C3aRs 在成年小鼠的神经祖细胞和未成熟神经元上表达。C3a 在体外刺激神经祖细胞的分化。
T37792	A2A receptor antagonist 1 CPI-444 analog,A2A receptor antagonist 1	Adenosine Receptor	GPCR/G Protein; Neuroscience
	A2A receptor antagonist 1 (CPI-444 analog)是腺苷 A2A 和 A1受体的拮抗剂，Ki 值分别为4和264 nM。
T10250	ADRA1D receptor antagonist 1 HCl ADRA1D receptor antagonist 1 HCl（1191908-24-3 free base）	Adrenergic Receptor	GPCR/G Protein; Neuroscience
	ADRA1D receptor antagonist 1 HCl 是一种具有口服活性、高效性和选择性的 α1D 肾上腺素受体拮抗剂（Ki：1.6 nM），具有潜在的抗增殖活性。
T60075	Dopamine D2 receptor agonist-2 Dopamine D2 Receptor	Dopamine Receptor	GPCR/G Protein; Neuroscience
	Dopamine D2 receptor agonist-2 (Dopamine D2 Receptor) 是靶向多巴胺D2受体的配体。
T3177	Orexin 2 Receptor Agonist OX2R	OX Receptor	GPCR/G Protein; Neuroscience
	Orexin 2 Receptor Agonist (OX2R) 是一种选择性有效的OX2R 激动剂， EC50为23 nM。
T9579L	GLP-1 receptor agonist 9 citrate GLP-1 receptor agonist 9 citrate (2401892-71-3 Free base)	Glucagon Receptor	GPCR/G Protein
	GLP-1 receptor agonist 9 citrate 是 GLP-1 的激动剂。
T11349	GABAA receptor agent 1	GABA Receptor	Membrane transporter/Ion channel; Neuroscience
	GABAA receptor agent 1 是GABAA 受体的高亲和力配体，有抗惊厥活性。
T9244	σ1 Receptor antagonist-1	Sigma receptor	GPCR/G Protein
	σ1 Receptor antagonist-1 是高选择性的 sigma 1受体拮抗剂，pKi 为10.28。它抑制细胞生长，在 G0/G1 期阻滞细胞周期并诱导 MCF-7/ADR 细胞凋亡。
TP1422	Interleukin (IL)-6 Receptor	Others	Others
	Interleukin (IL)-6 Receptor 是一种肽，来源于白细胞介素6受体。
T10058	A2B receptor antagonist 1	Adenosine Receptor	GPCR/G Protein; Neuroscience
	A2B receptor antagonist 1 是一个有效的 A2B 腺苷受体 (A2B adenosine receptor) 拮抗剂。
T13736	Interferon receptor inducer-1	IFNAR	Immunology/Inflammation
	Interferon receptor inducer-1 是一种干扰素(IFN)受体诱导剂，可用于干扰素诱导参与的紊乱性疾病的研究。
T5586	cFMS Receptor Inhibitor II	c-Fms	Tyrosine Kinase/Adaptors
	cFMS Receptor Inhibitor II 是 CSF-1R 激酶抑制剂。其中 CSF-1 是细胞因子。
T5829	H4 Receptor antagonist 1	Histamine Receptor	GPCR/G Protein; Immunology/Inflammation; Neuroscience
	H4 Receptor antagonist 1 是选择性组胺 H4受体反向激动剂，其IC50值为19 nM。
T37734	AMPA receptor modulator-2	GluR	Neuroscience
	AMPA receptor modulator-2 是 AMPA 受体的有效调节剂，在 TARPγ2 依赖性 AMPA 受体上的pIC50为 10.1。
T9247	Vanilloid receptor antagonist 1 4-(7-Hydroxy-2-isopropyl-4-oxoquinazolin-3(4H)-yl)benzonitrile	TRP/TRPV Channel	Membrane transporter/Ion channel
	Vanilloid receptor antagonist 1 (4-(7-Hydroxy-2-isopropyl-4-oxoquinazolin-3(4H)-yl)benzonitrile) 是香草酸受体的有效拮抗剂。
T11211	EP4 receptor antagonist 1	Prostaglandin Receptor	GPCR/G Protein; Immunology/Inflammation
	EP4 receptor antagonist 1 是一种有效的特异性前列腺素 EP4受体拮抗剂，对人和小鼠 EP4受体的 IC50分别为6.1 nM 和16.2 nM。 EP4 receptor antagonist 1 可用于癌症免疫治疗的研究。
T8848	GPR34 receptor antagonist 2 Tyrosine, N-[(2E)-3-(4'-chloro[1,1'-biphenyl]-4-yl)-1-oxo-2-propen-1-yl]-O-(phenylmethyl)-,gpr34-receptor-antagonist-2	Others	Others
	GPR34 receptor antagonist 2 (Tyrosine, N-[(2E)-3-(4'-chloro[1,1'-biphenyl]-4-yl)-1-oxo-2-propen-1-yl]-O-(phenylmethyl)-) 是一种GPR34受体拮抗剂，可用于研究免疫疾病、炎性疾病。
T12912	Sigma-1 receptor antagonist 3	Sigma receptor; HER	Angiogenesis; GPCR/G Protein; JAK/STAT signaling; Tyrosine Kinase/Adaptors
	Sigma-1 receptor antagonist 3 是 Sigma-1受体选择性拮抗剂，Ki 为 1.14 nM。它抑制 hERG，IC50为 1.54μM。它在神经性疼痛方面有研究的价值。
T7740	Protease-Activated Receptor-4 diTFA Protease-Activated Receptor-4 diTFA(245443-52-1(free base))	Protease-activated Receptor	GPCR/G Protein
	Protease-Activated Receptor-4 diTFA 是蛋白酶激活受体 4 (PAR4) 激动剂。
T1824	TGR5 Receptor Agonist	GPCR19	GPCR/G Protein
	TGR5 Receptor Agonist 是一种TGR5(GPCR19)激动剂。
T12910	Sigma-1 receptor antagonist 1	Sigma receptor	GPCR/G Protein
	Sigma-1 receptor antagonist 1 是一种有效、特异性的 sigma-1 受体拮抗剂。 Sigma-1 receptor antagonist 1 具有抗神经性疼痛活性，可用于治疗神经性疼痛研究。
T12911	Sigma-1 receptor antagonist 2	Sigma receptor	GPCR/G Protein
	Sigma-1 receptor antagonist 2 是有效的sigma 1受体选择性拮抗剂，与 σ1 和 σ2 受体结合的Ki 分别为 3.88 和 1288 nM。
T21620	Adenosine receptor antagonist 4	Adenosine Receptor	GPCR/G Protein; Neuroscience
	Adenosine receptor antagonist 4 是一种腺苷受体拮抗剂。
TP1704	Galanin Receptor Ligand M35 TFA	Neuropeptide Y Receptor	GPCR/G Protein; Neuroscience
	Galanin Receptor Ligand M35 TFA(142846-71-7 free base) 是一种高亲和力配体和甘丙肽受体拮抗剂 (Kd=0.1 nM)。
T10307	AMPA receptor modulator-1	iGluR	Membrane transporter/Ion channel; Neuroscience
	AMPA receptor modulator-1可被谷氨酸激活，从而调节离子通道。
T4521	Edg-2 receptor inhibitor 1 SAR-100842	LPA Receptor	GPCR/G Protein
	Edg-2 receptor inhibitor 1 (SAR-100842) 是一种提取的 Edg-2 受体抑制剂 (IC50: <0.1 μM)。
T14127	Adenosine A1 receptor activator T62	Adenosine Receptor	GPCR/G Protein; Neuroscience
	Adenosine A1 receptor activator T62 是腺苷 A1 受体的变构增强剂，有镇痛作用。
T37908	Glucocorticoid receptor agonist-1	Glucocorticoid Receptor; ADC Cytotoxin	Antibody-drug Conjugate/ADC Related; Endocrinology/Hormones
	Glucocorticoid receptor agonist-1是一种强效糖皮质激素受体激动剂，其 IC50 值为 2.8 nM。
T15785	LPA1 receptor antagonist 1 LPA1 R antagonist 1	LPA Receptor	GPCR/G Protein
	LPA1 receptor antagonist 1(LPA1 R antagonist 1) 是一种具有选择性和高效性的溶血磷脂酸 (LPA1) 受体拮抗剂( IC50 : 25 nM)，可用于研究特发性肺纤维化。
T15249	Estrogen receptor modulator 1	Estrogen Receptor/ERR	Endocrinology/Hormones
	Estrogen receptor modulator 1 是一种有效的、具有口服活性的、选择性雌激素受体(estrogen receptor)调节剂 (SERM)，其 pIC50为 0.46。它能够诱导 Tamoxifen 耐药、激素非依赖性异种移植瘤的消退。
T9157	GP130 receptor agonist-1 N-(4-Fluorophenyl)-4-phenyl-2-thiazolami	Interleukin	Immunology/Inflammation
	GP130 receptor agonist-1 (N-(4-Fluorophenyl)-4-phenyl-2-thiazolami) 是一种有效的、口服有活性的、可透过血脑屏障的 GP130受体激动剂。它对 NMDA 诱导的神经毒性具有神经保护作用。
T22466	Adenosine receptor A1 antagonist 5	cAMP	GPCR/G Protein
	Adenosine receptor A1 antagonist 5 可作为一种腺苷拮抗剂，是一种氧嘌呤，可作为杀虫剂和虫害防治剂，对血压升高有抑制作用。
T11137	(E)-GABAB receptor antagonist 1	GABA Receptor	Membrane transporter/Ion channel; Neuroscience
	(E)-GABAB receptor antagonist 1 是 GABAB receptor antagonist 1 的反式结构。(E)-GABAB receptor antagonist 1 降低 GABA 诱导的 IP3 (三磷酸肌醇) 产生，IC50 为 37.9 μM。GABAB receptor antagonist 1是选择性的 GABAB (γ-氨基丁酸) 受体的负变构调节剂。
T12247	NOT Receptor Modulator 1 2-(3-(2-(4-chlorophenyl)imidazo[1,2-a]pyridin-6-yl)phenyl)propan-2-ol	Others	Others
	NOT Receptor Modulator 1 (2-(3-(2-(4-chlorophenyl)imidazo[1,2-a]pyridin-6-yl)phenyl)propan-2-ol) 是核受体 NOT 调节剂。
T11077	Dopamine D2 receptor antagonist-1	Others	Others
	Dopamine D2 receptor antagonist-1，一种对多巴胺D2受体（D2R）表现出亚毫摩尔级别亲和力的负变构调节剂（NAM）。
T7674	Thrombin Receptor Activator for Peptide	Protease-activated Receptor	GPCR/G Protein
	Thrombin Receptor Activator for Peptide 也称为凝血因子 II 受体 (1-5) 或蛋白酶激活受体 1 (1-5)，用于研究冠心病 (CHD)。
T60087	cFMS Receptor Inhibitor IV 5-cyano-N-(2,5-di(piperidin-1-yl)phenyl)furan-2-carboxamide	c-Fms	Tyrosine Kinase/Adaptors
	cFMS Receptor Inhibitor IV 是 c-Fms 酪氨酸激酶的抑制剂。
T77508	A2B receptor antagonist 2 hydrochloride	Others	Others
	A2B receptor antagonist 2 hydrochloride 是腺苷受体 A2B 的拮抗剂（rA1 的 Ki = 2.30 μM，rA2A 的 Ki = 6.8 μM，hA2B 的 3.44 μM）
T78646	Estrogen receptor antagonist 8	Estrogen/progestogen Receptor	Endocrinology/Hormones
	Estrogen receptor antagonist 8 作为一种雌激素受体(ER)拮抗剂，具有抗子宫活性和潜在的抗肿瘤活性，可用于研究卵巢功能障碍。
T4312	GPR120 Agonist 2 GPR120 receptor agonist	GPR	Endocrinology/Hormones; GPCR/G Protein
	GPR120 Agonist 2 是一种选择性 GPR120激动剂。
T67915	Succinate/succinate receptor antagonist 1	Others	Others
	Succinate/succinate receptor antagonist 1 是一种有效的琥珀酸受体拮抗剂。Succinate/succinate receptor antagonist 1 中断牙龈组织中的琥珀酸信号，抑制琥珀酸受体 1 (SucnRl Antagonist 1) 的激活，对琥珀酸受体 1的 IC50 值为 20 μΜ。Succinate/succinate receptor antagonist 1 可用于治疗牙周病。
T7513	Protease-Activated Receptor-2, amide 蛋白酶活化的受体-2，酰胺,SLIGKV-NH2,H-丝氨酰亮氨酰异亮氨酰甘氨酰赖氨酰缬氨酰NH2	Protease-activated Receptor	GPCR/G Protein
	Protease-Activated Receptor-2, amide (SLIGKV-NH2) 是 PAR2 的激动剂，IC50为 10.4 M。
T38836L	Protease-Activated Receptor-1, PAR-1 Agonist acetate	Protease-activated Receptor	GPCR/G Protein
	Protease-Activated Receptor-1, PAR-1 Agonist acetate 是一种选择性蛋白酶激活受体 1 (PAR-1) 激动剂肽。它对应于 PAR1 栓系配体，可以选择性地模拟凝血酶通过该受体的作用。
T22009	CB2 receptor agonist 2 ZINC72105556,4-Quinolone-3-Carboxamide Furan CB2 Agonist,CB2受体拮抗剂2	Cannabinoid Receptor	GPCR/G Protein
	CB2 receptor agonist 2 (ZINC72105556) 是有效和选择性的 CB2 受体激动剂。对 CB2 的 Ki 为 8.5 nM。CB2 receptor agonist 2 对 CB2 具有高亲和力和选择性。
T61813	AMPA receptor antagonist-3	iGluR	Membrane transporter/Ion channel; Neuroscience
	AMPA receptor antagonist-3 是一种AMPA 受体拮抗剂。
T61068	AMPA receptor antagonist-2	iGluR	Membrane transporter/Ion channel; Neuroscience
	AMPA receptor antagonist-2是一种AMPA 受体拮抗剂。
T67946	EP2 receptor antagonist-2	Prostaglandin Receptor	GPCR/G Protein; Immunology/Inflammation
	EP2 receptor antagonist-2 (CID891729)为EP2受体拮抗剂，能够抑制PGE2诱导的EP2受体激活，并阻断由N-甲基-D-天冬氨酸(NMDA)引起的乳酸脱氢酶(LDH)释放。

Cat. No.	Product Name	Target	Signaling Pathways
TN1217	2'-O-Methylisoliquiritigenin	Dopamine Receptor; 5-HT Receptor; GABA Receptor	GPCR/G Protein; Membrane transporter/Ion channel; Neuroscience
	2'-O-Methylisoliquiritigenin 是从洋甘草中分离出来的一种天然产物，是由 NR 中特异性诱导的酶合成的。它上调 5-HT、NE、DA 和 GABA 途径，对 NE 通路有显著影响。
TN1465	Cannabigerol	NOS; 5-HT Receptor; ROS	GPCR/G Protein; Immunology/Inflammation; Neuroscience
	Cannabigerol 是一种植物大麻素，是一种高亲和力 α2-肾上腺素能受体激动剂、中度亲和力 5-HT1A 受体拮抗剂和低亲和力 CB1/CB2受体拮抗剂。它可降低眼压，有潜力治疗青光眼。
TQ0119	Cirsimaritin	GABA Receptor	Membrane transporter/Ion channel; Neuroscience
	Cirsimaritin 具有抗菌、抗炎、抗肿瘤、抗氧化特性和肾脏保护作用。 Cirsimaritin 与 GABAA 受体上的苯二氮卓位点结合较弱。
T5754	Kavain	NF-κB; GABA Receptor	Membrane transporter/Ion channel; Neuroscience; NF-κB
	Kavain 是从卡瓦胡椒中分离出来的卡瓦酸内酯，可以正向调控GABAA 受体，具有抗焦虑作用。
TN2247	Swertisin	Adenosine Receptor	GPCR/G Protein; Neuroscience
	Swertisin 是从日本紫菜中分离出的 C-葡萄糖基黄酮，是腺苷 A1 受体拮抗剂，具有抗糖尿病、抗炎和抗氧化作用。
TN1015	Meranzin	Adrenergic Receptor; Immunology/Inflammation related	GPCR/G Protein; Immunology/Inflammation; Neuroscience
	Meranzin 是从传统中药 Chaihu-Shugan-San (CSS) 中的生物活性化合物，是从紫茉莉叶中分离出的，能够调节共有的 α2-肾上腺素受体，并参与 AMPA-ERK1/2-BDNF 信号传导。它有潜在的预防动脉粥样硬化和抑郁症合并症。
T3782	Jujuboside A	transporter; GABA Receptor	Membrane transporter/Ion channel; Metabolism; Neuroscience
	Jujuboside A 是从中药酸枣仁中提取的一种糖苷，可用于失眠和焦虑的相关研究。
T7557	Guvacine hydrochloride	GABA Receptor	Membrane transporter/Ion channel; Neuroscience
	Guvacine hydrochloride 是从槟榔中得到的一种生物碱，是 GABA 摄取抑制剂，IC50为 10 μM。它对几种克隆的 GABA 转运体具有适度的选择性。
T0076	Paliperidone 9-羟基利培酮,帕潘立酮,9-hydroxyrisperidone	Dopamine Receptor; 5-HT Receptor; Adrenergic Receptor; Histamine Receptor	GPCR/G Protein; Immunology/Inflammation; Neuroscience
	Paliperidone (9-hydroxyrisperidone) 是 Risperidone 的主要活性代谢产物，是多巴胺 D2 拮抗剂和5-HT2A 拮抗剂。它用作非典型抗精神病药，用于精神分裂症的急性及维持治疗。它对α1和α2肾上腺素能受体和 H1组胺能受体也有拮抗作用。
T2815	Puerarin 葛根素,Kakonein	5-HT Receptor	GPCR/G Protein; Neuroscience
	Puerarin (Kakonein) 是从葛根中提取的一种异黄酮，是一种5-HT2C 受体拮抗剂。
T9113	Myristicin Myristicine,肉豆蔻醚	IL Receptor; Anti-infection; BCL; P450; PARP; 5-HT Receptor; Caspase; GABA Receptor; NO Synthase	Apoptosis; Chromatin/Epigenetic; DNA Damage/DNA Repair; GPCR/G Protein; Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; Microbiology/Virology; Neuroscience; Proteases/Proteasome
	Myristicin (Myristicine) 是一种在香料和伞形植物中发现的天然产物。肉豆蔻素具有抗胆碱能、抗菌和肝保护作用，还具有抗炎作用，其通过钙途径抑制dsrna 刺激的巨噬细胞中的NO、细胞因子、趋化因子和生长因子。Myristicin 可以诱导细胞凋亡，其特征是改变线粒体膜电位、细胞色素c 释放、Caspase-3激活、parp 切割和DNA 断裂。
T8036	6-Methylflavone	GABA Receptor	Membrane transporter/Ion channel; Neuroscience
	6-Methylflavone 是α1β2γ2L 和α1β2GABAA 受体激活剂。
T6S2099	Geraniin	Antioxidant; TNF	Apoptosis; oxidation-reduction
	Geraniin 是一种肿瘤坏死因子α释放抑制剂，其IC50值为 43 μM，具有抗肿瘤、抗炎和抗高血糖活性。
TN1023	Miltirone	P450; GABA Receptor	Membrane transporter/Ion channel; Metabolism; Neuroscience
	Miltirone 是存在于丹参中的一种天然产物，可作为中枢苯二氮受体部分激动剂，IC50值为 0.3 μM。
T0525	Flopropione 夫洛丙酮,Phloropropiophenone	5-HT Receptor; Transferase	GPCR/G Protein; Metabolism; Neuroscience
	Flopropione (Phloropropiophenone) 是一种解痉剂，用作 5-HT1A 受体拮抗剂，也是儿茶酚-O-甲基转移酶抑制剂。
T6S0630	Hypaconitine	P450; TNF	Apoptosis; Metabolism
	Hypaconitine 是从乌头属种分离的一种高毒性成分，可研究风湿病。
T3S2100	(-)-Securinine 一叶秋碱,Securinine	GABA Receptor	Membrane transporter/Ion channel; Neuroscience
	(-)-Securinine (Securinine) 是来自叶底珠的一种生物碱，也是 GABAA 受体拮抗剂。
T2720	Ginsenoside Rc Panaxoside Rc,人参皂苷Rc,人参皂苷 Rc	Others; TNF; GABA Receptor; Interleukin	Apoptosis; Immunology/Inflammation; Membrane transporter/Ion channel; Neuroscience; Others
	Ginsenoside Rc (Panaxoside Rc) 是人参中的一种人参皂苷，可抑制 TNF-α 和 IL-1β 的表达。它增强 GABA 受体 A 介导的离子通道电流。
T6648	Rotundine Gindarine,L-Tetrahydropalmatine,Caseanine,罗通定,(-)-Tetrahydropalmatine	Dopamine Receptor; 5-HT Receptor	GPCR/G Protein; Neuroscience
	Rotundine (Gindarine) 是多巴胺D1、D2和D3受体的拮抗剂，IC50值分别为 166、1.4 和 3.3 μM。它也是5-HT1A 的拮抗剂，IC50值为 370 nM。
T6S0654	Isocorynoxeine 7-Isocorynoxeine,异去氢钩藤碱	5-HT Receptor	GPCR/G Protein; Neuroscience
	Isocorynoxeine (7-Isocorynoxeine) 是钩藤中的一种生物碱，剂量依赖性抑制5-HT2A 受体介导的电流反应，IC50为 72.4 μM。
T3369	Nuciferine (-)-Nuciferine,VLT 049,荷叶碱,Sanjoinine E	Dopamine Receptor; 5-HT Receptor	GPCR/G Protein; Neuroscience
	Nuciferine ((-)-Nuciferine) 是一种在埃及蓝睡莲和水芙蓉中发现的生物碱，是5-HT2A、5-HT2B 和5-HT2C 拮抗剂，IC50分别为 478 nM、1 μM 和 131 nM。它也是5-HT7的反向激动剂，IC50为 150 nM。
T5799	Arecaidine hydrochloride	Others	Others
	Arecaidine hydrochloride 是一种具有高效 GABA 吸收抑制功能的吡啶生物碱。它是 H+偶联的氨基酸转运蛋白 1 (PAT1，SLC36A1) 的底物，能够竞争性抑制 L-脯氨酸的摄取。
TN1032	Geissoschizine methyl ether 缝籽木嗪甲醚,缝籽嗪甲醚	5-HT Receptor	GPCR/G Protein; Neuroscience
	Geissoschizine methyl ether 是从钩藤中发现的一种生物碱，是 Yokukansan 的主要活性成分，具有精神药物作用。它是一种有效的 5-羟色胺 A 受体激动剂，是 Yokukansan 改善攻击性和社交性的候选药物。
T1681	Aminophylline 氨茶碱,Phyllocontin	PDE; Adenosine Receptor	GPCR/G Protein; Metabolism; Neuroscience
	Aminophylline (Phyllocontin) 是一种竞争性非选择性磷酸二酯酶抑制剂，具有支气管扩张作用。它是竞争性的腺苷受体拮抗剂，有用于哮喘研究的潜力。
T4S1637	gamma-Mangostin Normangostin,γ-倒捻子素	Others; 5-HT Receptor	GPCR/G Protein; Neuroscience; Others
	gamma-Mangostin (Normangostin) 是从药用植物山竹的果壳中提纯的一种天然产物，是一种竞争性5-HT2A 受体拮抗剂。它是运甲状腺素蛋白原纤维化抑制剂，与甲状腺素结合位点结合并稳定了 TTR 四聚体，具有抗高血压、预防结肠癌等作用。
TN2268	Tetrahydromagnolol	Cannabinoid Receptor; GPR; GABA Receptor	Endocrinology/Hormones; GPCR/G Protein; Membrane transporter/Ion channel; Neuroscience
	Tetrahydromagnolol 是 Magnolol 的主要代谢产物，是一种弱的GPR55受体拮抗剂。它是选择性大麻素CB2受体激动剂，EC50为 170 nM，Ki 为 416 nM，对CB2受体的选择性比 CB1 受体高 20 倍。
T6519	Gramine NSC 16892,芦竹碱,Donaxine	Adiponectin receptor; Reverse Transcriptase; Adrenergic Receptor	GPCR/G Protein; Microbiology/Virology; Neuroscience
	Gramine (Donaxine) 是从芦竹中得到的一种生物碱，是脂联素受体激动剂，对 AdipoR2 和 AdipoR1 的 IC50值分别为 3.2 和 4.2 µM。它也是小鼠和人β2-肾上腺素受体激动剂，具有抗肿瘤、抗炎和抗病毒作用。
T6662	Scopine 东莨菪醇,6,7-Epoxytropine	Adrenergic Receptor	GPCR/G Protein; Neuroscience
	Scopine (6,7-Epoxytropine) 是一种山莨菪碱的代谢物，是一种 α1-肾上腺素受体激动剂，用于治疗急性循环性休克。
T5S1882	Songorine 准葛尔乌头碱,Napellonine,Zongorine,Bullatine G	Others; GABA Receptor	Membrane transporter/Ion channel; Neuroscience; Others
	Songorine (Napellonine) 是从乌头属中分离出的一种二萜生物碱，具有抗癌、抗心律不齐和抗炎活性。它是大鼠脑中的GABAA 受体拮抗剂，有用于上皮性卵巢癌的研究潜力。
T4S0217	HOMOPLANTAGININ	TNF; NF-κB	Apoptosis; NF-κB
	Homoplantaginin 是来自中药荔枝草的一种类黄酮，具有抗炎和抗氧化活性。
T8268	6,2'-Dihydroxyflavone 6,2-二羟基黄酮,6,2'-二羟基黄酮	GABA Receptor	Membrane transporter/Ion channel; Neuroscience
	6,2'-Dihydroxyflavone 是一种新型GABAA 受体拮抗剂。
T1711	Harmine Telepathine,去氢骆驼蓬碱	MAO; 5-HT Receptor; DYRK	Cell Cycle/Checkpoint; GPCR/G Protein; Metabolism; Neuroscience; Tyrosine Kinase/Adaptors
	Harmine (Telepathine) 是一种从山茱萸种子中分离出来的生物碱，具有抗癌和抗炎活性。它是双特异性酪氨酸磷酸化调节激酶抑制剂，对5-HT2A 血清素受体具有高亲和力，Ki 值为 397 nM。
T2979	DL-Menthol DL-薄荷醇,Hexahydrothymol,(±)-Menthol,薄荷醇	GABA Receptor; AChE	Membrane transporter/Ion channel; Neuroscience
	DL-Menthol ((±)-Menthol) 是单萜醇 (–)-薄荷醇和 (+)-薄荷醇的外消旋混合物，已在大麻中发现。它与 GABAA 受体的激活有关。
TN1052	Lindleyin	Estrogen Receptor/ERR; Estrogen/progestogen Receptor	Endocrinology/Hormones
	Lindleyin 是从 Rhei rhizoma 中分离得到，通过雌激素受体介导激素作用。它能够与 ERα结合，有类似雌激素的作用。
T2850	Bicuculline 荷包牡丹碱,(+)-Bicuculline,d-Bicuculline	GABA Receptor	Membrane transporter/Ion channel; Neuroscience
	Bicuculline ((+)-Bicuculline) 是从东北延胡索中提取的一种生物碱，能阻断 Ca2+激活钾 (SK) 通道。它是一种竞争性的神经递质 GABAA 受体拮抗剂，IC50为 2 μM。
T19931	Gentisein NSC 329491,NSC329491,NSC-329491	Serotonin Transporter	Neuroscience
	Gentisein (NSC-329491) 是 Mangiferin 的主要代谢物，有效抑制 5-HT 的摄取，IC50为 4.7 µM。
T0892	Diphylline 二羟丙茶碱,Dyphylline,Diprophylline	PDE; Adenosine Receptor	GPCR/G Protein; Metabolism; Neuroscience
	Diphylline (Diprophylline) 是一种A1/A2腺苷受体拮抗剂，也是环状核苷酸磷酸二酯酶抑制剂。它是一种黄嘌呤衍生物，具有支气管扩张和血管扩张作用，有用于治疗慢性支气管炎和肺气肿的潜力。
T1396	Bemegride 贝美格,Bemegrid,3-Ethyl-3-methylglutarimide,Agipnon	GABA Receptor	Membrane transporter/Ion channel; Neuroscience
	Bemegride (3-Ethyl-3-methylglutarimide) 是一种中枢神经系统兴奋剂和巴比妥类中毒的解毒剂。
T2749	Ginkgolide A 银杏内酯A,BN-52020	GABA Receptor; Endogenous Metabolite	Membrane transporter/Ion channel; Metabolism; Neuroscience
	Ginkgolide A (BN-52020) 是从银杏叶提取出来的一种天然产物，是 GABA 拮抗剂，有用于多种炎症和免疫疾病的研究潜力。
TN1849	Kuwanon H	GPR; Bombesin Receptor	Endocrinology/Hormones; GPCR/G Protein
	Kuwanon H 是分离自桑白皮的黄酮类化合物，具有拮抗非肽类蛙皮素受体的活性。Kuwanon H 特异性抑制细胞内胃泌激素释放肽 CRP 与GRP-preferring 受体的结合，Ki 为 290 nM。
T6S0627	Mesaconitine 新乌碱,新乌头碱；中乌头碱	TNF	Apoptosis
	Mesaconitine 是乌头属植物的一种主要活性成分，通过循环 AMP 和刺激中枢 β-肾上腺素能系统具有镇痛活性，还有抗炎活性。
T5S0543	Isocurcumenol	Apoptosis; Estrogen Receptor/ERR; Reductase	Apoptosis; Endocrinology/Hormones; Metabolism
	Isocurcumenol 是从莪术中分离得到的一种天然产物，是一种ERα抑制剂，对 DLA 和 KB 癌细胞的IC50分别为 99.1 µg/mL 和 178.2 µg/mL，具有抗肿瘤活性。
TN2865	(E)-3,4,5-Trimethoxycinnamic acid O-Methylsinapic acid,3,4,5-三甲氧基肉桂酸,3,4,5-Trimethoxy-trans-cinnamic acid,3,4,5-Trimethoxyphenylacrylic acid	Others	Others
	(E)-3,4,5-Trimethoxycinnamic acid (O-Methylsinapic acid) 是一种来自羌活根和根茎的天然产物。
T6S1256	Ruscogenin	NOS; NF-κB; NOD-like Receptor (NLR)	Immunology/Inflammation; NF-κB
	Ruscogenin 是一种重要甾体皂苷元，提取自麦冬。它能够抑制 TXNIP/NLRP3炎症体激活和 MAPK 途径，改善脑缺血诱导的血脑屏障功能障碍，具有显著抗血栓、抗炎作用。
T2879	Fisetin 漆黄素,非瑟酮	TNF; Sirtuin; PPAR	Apoptosis; Chromatin/Epigenetic; DNA Damage/DNA Repair; Metabolism
	Fisetin 是在许多水果和蔬菜中发现的一种天然黄酮醇，有抗氧化、抗癌和神经保护作用。
T3698	alpha-Asarone α-Asarone,trans-Asarone,α-细辛脑	P450; GABA Receptor; HMG-CoA Reductase	Membrane transporter/Ion channel; Metabolism; Neuroscience
	alpha-Asarone (trans-Asarone) 是来自胡萝卜的一种天然产物，具有抗抑郁等功效。
T13768	(+)-Medicarpin	Estrogen/progestogen Receptor	Endocrinology/Hormones
	(+)-Medicarpin, a pterocarpan, is an isoflavonoid compound derived from multiple medicinal plant species such as Sophora japonica, Zollernia paraensis, Platymiscium yucatamun, Machaerium aristulatum, and Platymiscium floribundum. It exhibits potent inhibition of osteoclastogenesis and facilitates bone healing and increased bone mass through osteoblast differentiation, which is mediated by the estrogen receptor (ER) β.
T6S1597	Mulberroside A 桑皮苷 A,桑皮苷A	TNF; Tyrosinase; Interleukin	Apoptosis; Immunology/Inflammation; Proteases/Proteasome
	Mulberroside A 是桑中的一种主要活性成分，可降低TNF-α、IL-1β和IL-6的表达，抑制 NALP3、caspase-1 和 NF-κB 的激活以及 ERK、JNK 和 p38 的磷酸化。它抑制蘑菇酪氨酸酶，具有抗炎和抗细胞凋亡作用。
T5940	Proxyphylline 羟丙茶碱,7-(2-Hydroxypropyl)theophylline	PDE; Adenosine Receptor	GPCR/G Protein; Metabolism; Neuroscience
	Proxyphylline (7-(2-Hydroxypropyl)theophylline) 是甲基黄嘌呤衍生物，可用作心脏活化剂、血管扩张剂和支气管扩张剂。
TN2437	Serotonin 5-羟基色胺,5-hydroxytryptamine,血清素,五羟色胺,5-HT	Others; 5-HT Receptor; Endogenous Metabolite; Transferase	GPCR/G Protein; Metabolism; Neuroscience; Others
	Serotonin (5-hydroxytryptamine) 是 CNS 中的单胺神经递质和内源性5-HT 受体激动剂。它也是儿茶酚 O-甲基转移酶(COMT) 的抑制剂，Ki 值为 44 μM。
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Cat. No.	Product Name	Species	Expression System
TMPY-03739	Transferrin Receptor/TFRC Protein, Cynomolgus, Rhesus, Recombinant (His) transferrin receptor	Cynomolgus,Rhesus	HEK293 Cells
	Transferrin Receptor/TFRC Protein, Cynomolgus, Rhesus, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 77.5 kDa and the accession number is XP_005545315.1&NP_001244232.1.
TMPY-01053	Prolactin Receptor Protein, Human, Recombinant (His) hPRLrI,PRLR,MFAB,HPRL,prolactin receptor	Human	HEK293 Cells
	Prolactin Receptor Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 26 kDa and the accession number is P16471-1.
TMPY-01146	Insulin Receptor Protein, Human, Recombinant (long isoform, His) HHF5,CD220,insulin receptor	Human	HEK293 Cells
	Insulin Receptor Protein, Human, Recombinant (long isoform, His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 107 kDa and the accession number is P06213-1.
TMPY-01725	Leptin Receptor Protein, Human, Recombinant (His) LEPRD,OB-R,OBR,LEP-R,CD295,leptin receptor	Human	HEK293 Cells
	Leptin Receptor Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 95 kDa and the accession number is P48357-1.
TMPY-01873	Transferrin Receptor/TFRC Protein, Human, Recombinant (His) TFR1,p90,CD71,TFR,transferrin receptor,T9,TRFR,TR	Human	HEK293 Cells
	Transferrin Receptor/TFRC Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 77.4 kDa and the accession number is AAA61153.1.
TMPY-05096	Transferrin Receptor/TFRC Protein, Human, Recombinant (N-hFc) CD71,T9,transferrin receptor,TFR1,p90,TRFR,TFR,TR	Human	HEK293 Cells
	Transferrin Receptor/TFRC Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 103.6 kDa and the accession number is CAA25527.1.
TMPY-02294	Transferrin Receptor/TFRC Protein, Mouse, Recombinant (His) 2610028K12Rik,p90,E430033M20Rik,AI426448,TFR,AU015758,Mtvr1,...	Mouse	HEK293 Cells
	Transferrin Receptor/TFRC Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 78.3 kDa and the accession number is Q62351.
TMPY-06661	Transferrin Receptor/TFRC Protein, Rat, Recombinant (His) transferrin receptor	Rat	HEK293 Cells
	Transferrin Receptor/TFRC Protein, Rat, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 78.59 kDa and the accession number is Q99376.
TMPY-02434	Prolactin Receptor Protein, Rat, Recombinant (His) prolactin receptor,RATPRLR,MGC105486	Rat	HEK293 Cells
	Prolactin Receptor Protein, Rat, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 26 kDa and the accession number is P05710-1.
TMPY-04395	Insulin Receptor Protein, Human, Recombinant (His & GST) HHF5,insulin receptor,CD220	Human	Baculovirus Insect Cells
	Insulin Receptor Protein, Human, Recombinant (His & GST) is expressed in Baculovirus insect cells with His and GST tag. The predicted molecular weight is 72.3 kDa and the accession number is P06213-1.
TMPK-01200	Nogo Receptor/RTN4R Protein, Cynomolgus, Recombinant (His) NGR,NOGOR,RTN4R,NgR1,Nogo receptor,Nogo-66 rece...	Cynomolgus	HEK293 Cells
	NOGO Receptor 1 (RTN4R) regulates axonal growth, as well as axon regeneration after injury. The gene maps to the 22q11.2 schizophrenia susceptibility locus and is thus a strong functional and positional candidate gene.RTN4R may modulate the genetic risk or clinical expression of schizophrenia in a subset of patients and identify additional studies that will be necessary to clarify the role of RTN4R in psychiatric phenotypes.
TMPY-01612	CD155/PVR Protein, Rhesus, Recombinant (His) poliovirus receptor	Rhesus	HEK293 Cells
	CD155/PVR Protein, Rhesus, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 35.8 kDa and the accession number is Q0MSE6.
TMPY-01149	Insulin Receptor Protein, Human, Recombinant (short isoform, His) Insulin Receptor,HHF5,CD220	Human	HEK293 Cells
	Insulin Receptor Protein, Human, Recombinant (short isoform, His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 106 kDa and the accession number is P06213-2.
TMPY-03144	Nogo Receptor/RTN4R Protein, Human, Recombinant (His) NGR,reticulon 4 receptor,NOGOR	Human	HEK293 Cells
	Nogo Receptor/RTN4R Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 46.8 kDa and the accession number is Q9BZR6.
TMPH-03388	Transferrin Receptor/TFRC Protein, Rat, Recombinant (His & SUMO) Tfrc,Transferrin receptor protein 1	Rat	E. coli
	Transferrin Receptor/TFRC Protein, Rat, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 35.9 kDa and the accession number is Q99376.
TMPY-05283	Insulin Receptor Protein, Human, Recombinant (long isoform, His), Biotinylated CD220,Insulin Receptor,HHF5	Human	HEK293 Cells
	Insulin Receptor Protein, Human, Recombinant (long isoform, His), Biotinylated is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 107 kDa and the accession number is P06213-1.
TMPY-02984	Prolactin Receptor Protein, Mouse, Recombinant (His) Pr-1,Pr-3,AI987712,prolactin receptor,Prlr,Prlr-rs1	Mouse	HEK293 Cells
	Prolactin Receptor Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 26 kDa and the accession number is P07321.
TMPH-00932	Androgen receptor Protein, Human, Recombinant (His & Myc & SUMO) Nuclear receptor subfamily 3 group C member 4,AR,NR...	Human	E. coli
	Androgen receptor Protein, Human, Recombinant (His & Myc & SUMO) is expressed in E. coli.
TMPY-05025	Thrombin Receptor Protein, Human, Recombinant (His) TR,PAR1,HTR,coagulation factor II (thrombin) receptor	Human	HEK293 Cells
	Thrombin Receptor Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 10.2 kDa and the accession number is A0A024RAP7.
TMPY-01566	Prolactin Receptor Protein, Mouse, Recombinant (His & hFc) prolactin receptor,Prlr,Pr-3,Pr-1,Prlr-rs1,AI987712	Mouse	HEK293 Cells
	Prolactin Receptor Protein, Mouse, Recombinant (His & hFc) is expressed in HEK293 mammalian cells with His and hFc tag. The predicted molecular weight is 52.5 kDa and the accession number is Q08501-1.
TMPY-01056	Nogo Receptor/RTN4R Protein, Human, Recombinant (His & hFc) NOGOR,reticulon 4 receptor,NGR	Human	HEK293 Cells
	Nogo Receptor/RTN4R Protein, Human, Recombinant (His & hFc) is expressed in HEK293 mammalian cells with His and hFc tag. The predicted molecular weight is 73 kDa and the accession number is Q9BZR6.
TMPY-02934	IL-2RG Protein, Rat, Recombinant (His) interleukin 2 receptor, γ,interleukin 2 recepto...	Rat	HEK293 Cells
	IL-2RG Protein, Rat, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 29.5 kDa and the accession number is Q68FU6.
TMPY-04717	CD122/IL2RB Protein, Rhesus, Recombinant (His) interleukin 2 receptor, β,interleukin 2 recepto...	Rhesus	HEK293 Cells
	CD122/IL2RB Protein, Rhesus, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 26.1 kDa and the accession number is H9Z8K1.
TMPY-00874	Leptin Receptor Protein, Human, Recombinant (His & hFc) LEP-R,OBR,CD295,OB-R,LEPRD,leptin receptor	Human	HEK293 Cells
	Leptin Receptor Protein, Human, Recombinant (His & hFc) is expressed in HEK293 mammalian cells with His and hFc tag. The predicted molecular weight is 121.4 kDa and the accession number is P48357-1.
TMPY-05274	IL-23R Protein, Human, Recombinant (His) interleukin 23 receptor	Human	HEK293 Cells
	IL-23R Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 39.3 kDa and the accession number is AAM44229.1.
TMPY-02987	Vitamin D Receptor/VDR Protein, Mouse, Recombinant (His) vitamin D (1,25- dihydroxyvitamin D3) receptor,Nr1i...	Mouse	Baculovirus Insect Cells
	Vitamin D Receptor/VDR Protein, Mouse, Recombinant (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 49.28 kDa and the accession number is P48281.
TMPY-01163	Nogo Receptor/RTN4R Protein, Mouse, Recombinant (His) Rtn4r,NgR,NgR1,reticulon 4 receptor,NOGOR	Mouse	HEK293 Cells
	Nogo Receptor/RTN4R Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 47 kDa and the accession number is Q99PI8.
TMPY-02706	Vitamin D Receptor/VDR Protein, Human, Recombinant (His) PPP1R163,vitamin D (1,25- dihydroxyvitamin D3) receptor<...	Human	Baculovirus Insect Cells
	Vitamin D Receptor/VDR Protein, Human, Recombinant (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 50 kDa and the accession number is P11473.
TMPY-05102	CD122/IL2RB Protein, Rat, Recombinant (His) interleukin 2 receptor, β,interleukin 2 recepto...	Rat	HEK293 Cells
	CD122/IL2RB Protein, Rat, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 26.4 kDa and the accession number is P26896.
TMPJ-00154	IL-15RA Protein, Mouse, Recombinant (hFc, Human Cells) sIL-15 receptor subunit α,Il15ra,Interleukin-15	Mouse	HEK293 Cells
	Mouse interleukin-15 receptor subunit alpha, also known as Il15ra, is a high-affinity receptor for interleukin-15. Il15ra associates as a heterotrimer with the IL-2 receptor beta and gamma subunits (Common gamma chain, or gamma c) to initiate signal transduction. It can signal both in cis and trans where IL15R from one subset of cells presents IL15 to neighboring IL2RG-expressing cells. Il15ra is expressed in special cells including a wide variety of Tand B cells and non-lymphoid cells. Human Il...
TMPY-04649	ROR1 Protein, Human, Recombinant (His) dJ537F10.1,NTRKR1,receptor tyrosine kinase-like orp...	Human	HEK293 Cells
	ROR1 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 43.4 kDa and the accession number is Q01973.
TMPJ-00994	LTBR Protein, Mouse, Recombinant (hFc) Tnfcr,Lymphotoxin-beta receptor,Tumor necrosis fact...	Mouse	HEK293 Cells
	It is a single-pass type I membrane protein and contains 4 TNFR-Cys repeats. The protein is a member of the tumor necrosis factor (TNF) family of receptors. It is expressed on the surface of most cell types, including cells of epithelial and myeloid lineages, but not on T and B lymphocytes. The protein is the receptor for the heterotrimeric lymphotoxin containing LTA and LTB, and for TNFS14/LIGHT. It promotes apoptosis via TRAF3 and TRAF5 and may play a role in the development of lymphoid organs...
TMPY-00085	Calcitonin receptor Protein, Human, Recombinant (aa 1-153, hFc) CTR,CTR1,CT-R,calcitonin receptor,CRT	Human	HEK293 Cells
	Calcitonin receptor Protein, Human, Recombinant (aa 1-153, hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 42.1 kDa and the accession number is P30988-2.
TMPY-06022	FOLR1 Protein, Cynomolgus, Rhesus, Recombinant (His) folate receptor 1 (adult)	Cynomolgus,Rhesus	HEK293 Cells
	FOLR1 Protein, Cynomolgus, Rhesus, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 26.3 kDa and the accession number is A0A2K5UR19&NP_001181576.1.
TMPY-03951	IL-18R alpha Protein, Cynomolgus, Recombinant (hFc) interleukin 18 receptor 1	Cynomolgus	HEK293 Cells
	IL-18R alpha Protein, Cynomolgus, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 61.1 kDa and the accession number is F7H8F9.
TMPY-01883	EPOR Protein, Human, Recombinant (His) erythropoietin receptor,EPO-R	Human	HEK293 Cells
	EPOR Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 26.3 kDa and the accession number is P19235-1.
TMPY-01221	Nogo Receptor/RTN4R Protein, Mouse, Recombinant (His & hFc) NgR1,reticulon 4 receptor,NgR,Rtn4r,NOGOR	Mouse	HEK293 Cells
	Nogo Receptor/RTN4R Protein, Mouse, Recombinant (His & hFc) is expressed in HEK293 mammalian cells with His and hFc tag. The predicted molecular weight is 73.8 kDa and the accession number is Q99PI8.
TMPY-00181	Endothelin B Receptor Protein, Human, Recombinant (His) ETBR,ET-B,ET-BR,ETB,HSCR2,endothelin receptor type ...	Human	HEK293 Cells
	Endothelin B Receptor Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 9.5 kDa and the accession number is P24530-1.
TMPY-03860	Endothelin B Receptor Protein, Human, Recombinant (mFc) ET-B,endothelin receptor type B,ETB,ETBR,ETRB,ET-BR...	Human	HEK293 Cells
	Endothelin B Receptor Protein, Human, Recombinant (mFc) is expressed in HEK293 mammalian cells with mFc tag. The predicted molecular weight is 34.4 kDa and the accession number is P24530-1.
TMPY-00418	IL-21R Protein, Mouse, Recombinant (His) interleukin 21 receptor,NILR	Mouse	HEK293 Cells
	IL-21R Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 26.3 kDa and the accession number is AAL82636.1.
TMPY-04818	EGFR Protein, Cynomolgus, Recombinant (His) epidermal growth factor receptor	Cynomolgus	HEK293 Cells
	EGFR Protein, Cynomolgus, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 70.1 kDa and the accession number is A0A2K5WK39.
TMPY-02335	OSMR Protein, Mouse, Recombinant (His) oncostatin M receptor,OSMRB	Mouse	HEK293 Cells
	OSMR Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 83.7 kDa and the accession number is O70458-1.
TMPY-02824	IL-18R alpha Protein, Rat, Recombinant (hFc) interleukin 18 receptor 1	Rat	HEK293 Cells
	IL-18R alpha Protein, Rat, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 62.5kDa and the accession number is A0A8I6A1C2.
TMPY-05090	CD25/IL2R alpha Protein, Rat, Recombinant (His) interleukin 2 receptor, α,CD25/IL2R α,interleukin 2...	Rat	Baculovirus Insect Cells
	CD25/IL2R alpha Protein, Rat, Recombinant (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 25.9 kDa and the accession number is A6JLS0.
TMPY-00317	Calcitonin receptor Protein, Human, Recombinant (aa 25-154, hFc) CTR,calcitonin receptor,CRT,CTR1,CT-R	Human	HEK293 Cells
	Calcitonin receptor Protein, Human, Recombinant (aa 25-154, hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 43.9 kDa and the accession number is P30988-1.
TMPY-05617	Transferrin Receptor/TFRC Protein, Human, Recombinant (His), Biotinylated TRFR,p90,TR,TFR,CD71,TFR1,T9,transferrin receptor	Human	HEK293 Cells
	Transferrin Receptor/TFRC Protein, Human, Recombinant (His), Biotinylated is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 77.4 kDa and the accession number is P02786.
TMPY-03776	CD25/IL2R alpha Protein, Cynomolgus, Recombinant interleukin 2 receptor, α,interleukin 2 recepto...	Cynomolgus	HEK293 Cells
	CD25/IL2R alpha Protein, Cynomolgus, Recombinant is expressed in HEK293 mammalian cells. The predicted molecular weight is 22.4 kDa and the accession number is H6WS54.
TMPY-03644	CD25/IL2R alpha Protein, Cynomolgus, Recombinant (His) interleukin 2 receptor, alpha,CD25/IL2R α,interleuk...	Cynomolgus	HEK293 Cells
	CD25/IL2R alpha Protein, Cynomolgus, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 38.1 kDa and the accession number is H6WS54.
TMPJ-00335	TGFBR2 Protein, Mouse, Recombinant (His) TGFR-2,TGF-beta type II receptor,Transforming growt...	Mouse	HEK293 Cells
	TGFBR2 Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with C-6xHis tag. The predicted molecular weight is 25-38 KDa and the accession number is Q62312-2.
TMPY-05644	CD25/IL2R alpha Protein, Rhesus, Recombinant (His & Avi), Biotinylated interleukin 2 receptor, α,CD25/IL2R α,interleukin 2...	Rhesus	HEK293 Cells
	CD25/IL2R alpha Protein, Rhesus, Recombinant (His & Avi), Biotinylated is expressed in HEK293 mammalian cells with His and Avi tag. The predicted molecular weight is 24.9 kDa and the accession number is Q5MNY4.
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Cat. No.	Product Name	Target	Signaling Pathways
T14687	Deucravacitinib BMS-986165	Tyrosine Kinases; JAK; IFNAR; Interleukin	Angiogenesis; Chromatin/Epigenetic; Immunology/Inflammation; JAK/STAT signaling; Stem Cells; Tyrosine Kinase/Adaptors
	Deucravacitinib (BMS-986165) 是一种高选择性、口服生物可利用的变构 TYK2 抑制剂，用于治疗自身免疫性疾病。它通过稳定调节 JH2 结构域来阻断受体介导的 Tyk2 激活，可抑制IL-12/23和 I 型IFN 途径。它选择性结合 TYK2 假激酶 (JH2) 结构域，IC50为1.0 nM。
T10113	3-Hydroxy agomelatine D3	5-HT Receptor	GPCR/G Protein; Neuroscience
	3-Hydroxy agomelatine D3 is a deuterium labeled 3-Hydroxy agomelatine. 3-Hydroxy agomelatine is an Agomelatine metabolite and a 5-HT2C receptor antagonist (IC50: 3.2 μM; Ki: 1.8 μM).
T11197	Enclomiphene D4 hydrochloride (E)-Clomiphene D4 hydrochloride,Enclomifene D4 hydrochloride,trans-Clomiphene D4 hydrochloride	Others	Others
	Enclomiphene D4 hydrochloride ((E)-Clomiphene D4 hydrochloride; trans-Clomiphene D4 hydrochloride; Enclomifene D4 hydrochloride) is a potent and orally active oestrogen receptor antagonist, with antioestrogenic property.Enclomiphene D4 hydrochloride ((E)-Clomiphene D4 hydrochloride; trans-Clomiphene D4 hydrochloride; Enclomifene D4 hydrochloride) is a deuterium labeled Enclomiphene.
T70332	JNJ-61393215
	JNJ-61393215 is a novel selective orexin-1 receptor (OX1R) antagonist.
T69673	Deucrictibant
	Deucrictibant is a bradykinin receptor antagonist.
T11867	Loperamide-d6 hydrochloride R-18553 D6 hydrochloride	Others	Others
	Loperamide D6 hydrochloride, a deuterium-labeled variant of Loperamide hydrochloride, acts as an opioid receptor agonist utilized for diarrhea treatment.
T12046	Mirtazapine D3 Org3770 D3,6-Azamianserin D3,米氮平 D3	5-HT Receptor	GPCR/G Protein; Neuroscience
	Mirtazapine D3 is a deuterium labeled Mirtazapine. Mirtazapine is an inhibitor of 5-HT receptor .
T11592	Hydroxyzine D8	Others	Others
	Hydroxyzine D8, a deuterium-labeled version of Hydroxyzine, acts as a histamine H1-receptor antagonist.
T19341	Glycerol phenylbutyrate-D15 HPN-100-D15	Sigma receptor	GPCR/G Protein
	Glycerol phenylbutyrate-D15 is a deuterium-labeled Glycerol phenylbutyrate. Glycerol phenylbutyrate is a sigma-2 (σ2) receptor ligand (pKi: 8.02).
T19342	Glycerol phenylbutyrate-D5 HPN-100-D5	Sigma receptor	GPCR/G Protein
	Glycerol phenylbutyrate-D5 is a deuterium-labeled Glycerol phenylbutyrate. Glycerol phenylbutyrate is a sigma-2 (σ2) receptor ligand (pKi: 8.02).
TMIH-0314	Lurasidone-d8 HCl
	Lurasidone-d8 HCl 是 Lurasidone HCl 的氘代化合物。Lurasidone HCl 的 CAS 号为 367514-88-3。Lurasidone hydrochloride 是多巴胺 D2和5-HT7的拮抗剂，IC50值分别为 1.68 和 0.495 nM，用于治疗精神分裂症和双相情感障碍。它也是5-HT1A受体的部分激动剂，IC50值为 6.75 nM。
TMIH-0235	Finerenone-d5
	Finerenone-d5 是 Finerenone 的氘代化合物。Finerenone 的 CAS 号为 1050477-31-0。Finerenone 是一种选择性、具有口服活性的、非甾体类盐皮质激素受体拮抗剂 (IC50=18 nM)。与糖皮质激素受体、雄激素受体和孕酮受体相比，它表现出良好的选择性 (>500-fold)。它在心肾疾病研究中具有潜在的应用前景，如 2 型糖尿病和慢性肾脏疾病。
T11536	Haloperidol (D4') Haloperidol D4',氟哌啶醇 (D4')	Others	Others
	Haloperidol D4' is deuterium-labeled haloperidol. Haloperidol is a dopamine D2 receptor antagonist.
T11295	Flibanserin-d4 BIMT-17BS D4,BIMT-17 D4,Flibanserin D4	Others	Others
	Flibanserin, a compound identified as BIMT-17, acts as a complete agonist at the serotonin 5-HT1A receptor, with a binding affinity (Ki) of 1 nM, while functioning as an antagonist at the 5-HT2A receptor with a 49 nM affinity. Flibanserin D4 represents a deuterium-labeled version of Flibanserin.
T12638	(R)-Praziquantel-d11 (R)-吡喹酮 D11,(R)-Praziquantel D11	5-HT Receptor	GPCR/G Protein; Neuroscience
	(R)-Praziquantel D11 is the deuterium labeled (R)-Praziquantel. (R)-Praziquantel is the active enantiomer of Praziquantel, is a partial the human 5-HT2B receptor agonist
T12329	Ospemifene D4 FC-1271a D4	Estrogen/progestogen Receptor	Endocrinology/Hormones
	Ospemifene D4 is a deuterium labeled Ospemifene. Ospemifene is a selective and orally active modulator of estrogen receptor.
T11675	Irbesartan-d4 厄贝沙坦 D4,SR-47436 D4,BMS-186295 D4	Others	Others
	Irbesartan D4, a deuterium-labeled variant of Irbesartan, is a highly potent and specific antagonist of the angiotensin II type 1 (AT1) receptor.
TMIH-0461	Prucalopride-13C-d3
	Prucalopride-13C-d3 是 Prucalopride 的 13C 和氘代化合物。Prucalopride 的 CAS 号为 179474-81-8。Prucalopride 是一种选择性、高亲和力的 5-HT4A/4B 受体激动剂，Ki为2.5和 8 nM。它对 5-HT4A/4B 受体的选择性是其他 5-HT 受体亚型的 290 倍以上。
T10818	Ciprofibrate D6	Others	Others
	Ciprofibrate D6 is a deuterium-labeled Ciprofibrate. Ciprofibrate is an agonist of peroxisome proliferator-activated receptor.
T13204	Trimethobenzamide D6	Others	Others
	Trimethobenzamide D6 is deuterium labeled Trimethobenzamide. Trimethobenzamide is a the D2 receptor blocker. Trimethobenzamide is an antiemetic.
T10241	Acrivastine D7 BW825C D7	Others	Others
	Acrivastine D7 is a deuterium labeled Acrivastine. Acrivastine is a short acting antagonist of histamine 1 receptor.
TMIH-0102	Avatrombopag-d8
	Avatrombopag-d8 是 Avatrombopag 的氘代化合物。Avatrombopag 的 CAS 号为 570406-98-3。Avatrombopag 是一种新型口服血小板生成素 (TPO) 受体激动剂，可激活 TPO 受体并增加巨核细胞增殖/分化和血小板生成。
T11869	Losartan (D4 Carboxylic Acid) E-3174 D4,氯沙坦羧酸 D4,EXP-3174 D4	Others	Others
	Losartan D4 Carboxylic Acid is the deuterium labeled Losartan, which is an angiotensin II receptor antagonist.
T11591	Hydroxyzine D4 羟嗪 D4	Others	Others
	Hydroxyzine D4 is a deuterium-labeled variation of Hydroxyzine, a chemical compound known for its anticholinergic, anxiolytic, and analgesic properties. It is classified as a heterocyclic histamine H1-receptor antagonist.
T12176	Naratriptan D3 Hydrochloride GR-85548A D3	Others	Others
	Naratriptan D3 Hydrochloride is the deuterium labeled Naratriptan, is a selective agonist of 5-HT1 receptor subtype.
T12698	Regorafenib-d3 Regorafenib D3,BAY 73-4506 D3	Others	Others
	Regorafenib D3 is a deuterium labeled Regorafenib. Regorafenib is a multi-targeted receptor inhibitor of tyrosine kinase.
TMIH-0486	Ramelteon-d5
	Ramelteon-d5 是 Ramelteon 的氘代化合物。Ramelteon 的 CAS 号为 196597-26-9。Ramelteon 是强效高选择性和可口服的MT1/MT2激动剂，Ki值分别为 14 和 112 pM，有用于失眠症的研究潜力。
TMIH-0485	Ramelteon-d3
	Ramelteon-d3 是 Ramelteon 的氘代化合物。Ramelteon 的 CAS 号为 196597-26-9。Ramelteon 是强效高选择性和可口服的MT1/MT2激动剂，Ki值分别为 14 和 112 pM，有用于失眠症的研究潜力。
T19234	Cetirizine D8 dihydrochloride 盐酸西替利嗪 D8	Histamine Receptor	GPCR/G Protein; Immunology/Inflammation; Neuroscience
	Cetirizine D8 dihydrochloride is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagonist.
T12806	(S)-Mirtazapine D3 (S)-Org3770 D3,(S)-6-Azamianserin D3	5-HT Receptor	GPCR/G Protein; Neuroscience
	(S)-Mirtazapine D3 is a deuterium labeled (S)-Mirtazapine. (S)-Mirtazapine is a stereoselective antagonist of 5-HT2 receptor. (S)-Mirtazapine is metabolized by CYP2D6 and CYP1A2.
T13137	TGFβRI-IN-1	TGF-beta/Smad	Stem Cells
	TGFβRI-IN-1 is an oral active and selective inhibitor of TGFβ receptor type I (TGFβRI) kinase(IC50 values of 2 nM and 7.6 μM for TGFβRI and TGFβRII, respectively ).
T12631	(R)-Mirtazapine D3 (R)-6-Azamianserin D3,(R)-Org3770 D3	5-HT Receptor	GPCR/G Protein; Neuroscience
	(R)-Mirtazapine D3 is a deuterium labeled (R)-Mirtazapine.(R)-Mirtazapine is a antagonist of 5-HT3 receptor.
T10670	Candesartan-d4 坎地沙坦 D4,CV-11974 D4	Others	Others
	Candesartan D4 is the deuterium labeled Candesartan. Candesartan is an antagonist of angiotensin II receptor.
T13076	Tamoxifen-d5 ICI 47699-d5,(Z)-Tamoxifen-d5,trans-Tamoxifen-d5	HSP	Cytoskeletal Signaling; Metabolism
	Tamoxifen-d5 is a deuterium labeled Tamoxifen. Tamoxifen is a selective modulator of estrogen receptor (SERM). Tamoxifen is a potent activator of Hsp90 and enhances the Hsp90 molecular chaperone ATPase activity.
T12760	Rotigotine D7 Hydrochloride N-0923 D7 Hydrochloride	Others	Others
	Rotigotine D7 Hydrochloride is the deuterium labeled Rotigotine(N-0923), which is an agonist of dopamine D2 and D3 receptor.
T19233	Cetirizine D4 dihydrochloride Cetirizine D4 dihydrochloride (1219803-84-5 free base)	Others	Others
	Cetirizine D4 dihydrochloride is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagonist.
T10368	Aripiprazole (D8) OPC-14597 D8	Others	Others
	Aripiprazole D8 (OPC-14597 D8) is the deuterium-labeled Aripiprazole. Aripiprazole is a human 5-HT1A receptor partial agonist (Ki: 4.2 nM).
T38602	(E/Z)-Eltrombopag 13C4 (E/Z)-Eltrombopag 13C4,(E/Z)-SB-497115 13C4
	(E/Z)-Eltrombopag 13C4 ((E/Z)-SB-497115 13C4) is a mixture complex of E-Eltrombopag and Z-Eltrombopag, with 13C labeled. Z-Eltrombopag is a thrombopoietin (TPO) receptor agonist developed for certain conditions that lead to thrombocytopenia.
T19297	Doxazosin D8 UK 33274 D8	Others	Others
	Doxazosin D8 (UK 33274 D8) is a deuterium labeled Doxazosin (UK 33274).Doxazosin, a quinazoline derivative, selectively antagonizes postsynaptic AP1 adrenergic receptor.
T12300	Olmesartan-d4 RNH-6270 D4,奥美沙坦 D4	Others	Others
	Olmesartan D4 is the deuterium labeled Olmesartan. Olmesartan is an antagonist of angiotensin II receptor (AT1R) used to treat high blood pressure.
T19191	Alosetron-d3 Alosetron D3,GR 68755 D3,GR 68755X D3	Others	Others
	Alosetron D3 (GR 68755 D3) is a deuterium-labeled Alosetron. Alosetron is an antagonist of 5HT3-receptor.
T19190	Alosetron D3 Hydrochloride GR-68755C D3	Others	Others
	Alosetron D3 (GR 68755 D3) Hydrochloride is a deuterium-labeled Alosetron. Alosetron is an antagonist of 5HT3-receptor.
TMIJ-0185	Telmisartan-13C-d3
	Telmisartan-13C-d3 是 Telmisartan 的 13C 和氘代化合物。Telmisartan 的 CAS 号为 144701-48-4。Telmisartan 是一种血管紧张素II 1型受体拮抗剂，能够抑制其活性，IC50值为 9.2 nM。
T10559	Blonanserin D8 AD-5423 D8	Others	Others
	Blonanserin D8 is a deuterium-labeled Blonanserin. Blonanserin (AD-5423) is a dopamine D2/5-HT2 receptor antagonist with an atypical antipsychotic effect.
T12210	Netupitant D6 CID-6451149 D6	Others	Others
	Netupitant D6 is the deuterium labeled Netupitant, which is a selective and orally active antagonist of neurokinin-1 receptor.
T11208	Enzalutamide-d3 MDV3100 D3	Others	Others
	Enzalutamide D3 is a deuterium labeled Enzalutamide . Enzalutamide is an androgen receptor (AR) antagonist with an IC50 of 36 nM in LNCaP prostate cells.
T11870	Losartan D4 氯沙坦 D4,DuP-753 D4	Others	Others
	Losartan D4, the deuterium-labeled version of Losartan, functions as an angiotensin II receptor antagonist. It inhibits the interaction between angiotensin II and AT1 receptors by competing for binding, achieving an IC50 value of 20 nM.
TMIJ-0162	Dexamethasone-d4
	Dexamethasone-d4 是 Dexamethasone 的氘代化合物。Dexamethasone 的 CAS 号为 50-02-2。Dexamethasone是一种糖皮质激素受体激动剂和一种 IL 受体调节剂。在脂多糖诱导的巨噬细胞炎症反应中，它抑制含有炎性 microRNA-155 的外泌体的产生。
T12550	Propranolol-d7 hydrochloride Propranolol D7 hydrochloride	Others	Others
	Propranolol D7 hydrochloride is a deuterium labeled Propranolol hydrochloride. Propranolol hydrochloride is a nonselective antagonist of β-adrenergic receptor (βAR).
T10440	Azilsartan-d5 TAK-536 D5	Others	Others
	Azilsartan (TAK-536) D5 is the deuterium-labeled Azilsartan. Azilsartan is a specific antagonist of the angiotensin II type 1 receptor.
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