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TargetMol | Compound Library

ReFRAME 相关化合物库现货

ReFRAME Related Library

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产品编号 L9230

2018年Jeff Janes 等人通过数据挖掘和文献查询,构建了ReFRAME 化合物库,在美国国家科学院院刊(PNAS)发表了关于ReFRAME 化合物库的应用和实用性;其中大部分已通过I 期临床研究具有临床安全性,ReFRAME 化合物库临床安全的独特性质将显著缩短候选药物进入临床的时间,降低失败风险,可高效应用于早期药物研发阶段的筛选以及先导化合物的发现。作者分享了ReFRAME 化合物库,旨在促进数据共享和药物发现机会。盖茨基金会和清华大学等创办的全球健康药物研发中心(GHDDI)也将ReFRAME 化合物库应用于抗COVID-19药物研发。
TargetMol 整理了ReFRAME 化合物库包含5084 种化合物,是药物再利用和抗COVID-19药物研发的有效工具。

TargetMol 的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
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产品编号 L9230

ReFRAME 相关化合物库

规格

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品描述 产品描述

  • 5084化合物的独特集合,可用于高通量筛选和高内涵筛选,是药物再利用和抗COVID-19药物研发的有效工具
  • 部分化合物已上市得到FDA、EMA、NMPA等权威部门审批,大部分已通过I期临床研究;
  • 通过结构多样性聚类分析,具有优良的结构多样性,包含2698个聚类簇(相似程度大于70%的为一簇),平均1.2个化合物一个簇;
  • 涵盖多个研究领域:肿瘤、心血管药物、抗炎/免疫、神经系统药物、呼吸系统药物等;
  • 靶点多样,包括5-HT Receptor、Sodium Channel、p38 MAPK、PI3K、MEK等;
  • 详细的说明书,化合物结构、靶点信息、适应症信息、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

包装和储存 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
  • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。

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Apoptosis
Antibacterial
Autophagy
Endogenous Metabolite
Antibiotic
5-HT Receptor
Parasite
Adrenergic Receptor
DNA/RNA Synthesis
COX
Dopamine Receptor
AChR
Antifungal
HIV Protease
Potassium Channel
Calcium Channel
ROS
Histamine Receptor
Sodium Channel
PDE
Cytochromes P450
NF-κB
PI3K
VEGFR
GABA Receptor
Nucleoside Antimetabolite/Analog
Virus Protease
Reactive Oxygen Species
Prostaglandin Receptor
SARS-CoV
PPAR
EGFR
Dehydrogenase
Influenza Virus
p38 MAPK
HCV Protease
Estrogen/progestogen Receptor
Glucocorticoid Receptor
Topoisomerase
iGluR
Estrogen Receptor/ERR
CDK
Akt
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FLT
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TNF
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HDAC
mTOR
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Mitophagy
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Src
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Reverse Transcriptase
TRP/TRPV Channel
Proteasome
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ERK
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STAT
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Monoamine Oxidase
MMP
ATPase
Wnt/beta-catenin
Cholinesterase (ChE)
GluR
MAO
Beta Amyloid
NO Synthase
PKC
MEK
TLR
Antioxidant
Progesterone Receptor
Transferase
Bcr-Abl
Leukotriene Receptor
AMPK
NMDAR
Anti-infection
Aurora Kinase
P-gp
MDM-2/p53
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Raf
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Tyrosine Kinases
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Angiotensin-converting Enzyme (ACE)
DNA Alkylator/Crosslinker
ALK
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Thyroid hormone receptor(THR)
TGF-beta/Smad
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ribosome
LPL Receptor
Retinoid Receptor
Endothelin Receptor
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c-RET
Amino Acids and Derivatives
Gamma-secretase
IGF-1R
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JNK
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Sigma receptor
Factor Xa
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FAK
Cholecystokinin Receptor
TAM Receptor
RSV
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Aromatase
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Guanylate cyclase
DHFR
ATM/ATR
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PAFR
Syk
HER
GNRH Receptor
Vasopressin Receptor
ROCK
MRP
P2X Receptor
Xanthine Oxidase
p53
IκB/IKK
IDO
Indoleamine 2,3-Dioxygenase (IDO)
HMG-CoA Reductase
Chloride channel
Casein Kinase
Platelet aggregation
ROS Kinase
NADPH
CaMK
DNA gyrase
CSF-1R
Smo
Immunology/Inflammation related
Chk
IAP
Monoamine Transporter
CRFR
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DNA Methyltransferase
OX Receptor
PGE Synthase
OXPHOS
LDLR
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PLK
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glycosidase
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PAI-1
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Telomerase
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NOS
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IRE1
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Myosin
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P2Y Receptor
MAPK
GPCR19
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PERK
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LDL
STING
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Ligands for Target Protein for PROTAC
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ATP Citrate Lyase
IKZF
GSNOR
gp120/CD4
HCN Channel
cAMP
Histone Acetyltransferase
CPT
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Advanced Glycation End Products
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ASK
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PI4K
KLF
Hydrogenase
NEDD8
N-Acetylglucosaminyltransferase
VDAC
NR4A
Adiponectin Receptor
Anion Exchanger
CD73
cGAS
TSH Receptor
p62
Ferroportin

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