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High affinity and potent ghrelin receptor inverse agonist (Ki values are 4.9 and 31 nM in COS7 and HEK293T cells, respectively). Blocks ghrelin receptor-mediated Gq- and G13-dependent signaling pathways.
High affinity and potent ghrelin receptor inverse agonist (Ki values are 4.9 and 31 nM in COS7 and HEK293T cells, respectively). Blocks ghrelin receptor-mediated Gq- and G13-dependent signaling pathways.
规格 | 价格 | 库存 | 数量 |
---|---|---|---|
1 mg | 询价 | 期货 |
产品描述 | High affinity and potent ghrelin receptor inverse agonist (Ki values are 4.9 and 31 nM in COS7 and HEK293T cells, respectively). Blocks ghrelin receptor-mediated Gq- and G13-dependent signaling pathways. |
分子量 | 902.13 |
分子式 | C51H67N9O6 |
CAS No. | 1394288-22-2 |
密度 | 1.212 g/cm3 (Predicted) |
存储 | keep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | ||||||||||
溶解度信息 | H2O: 2 mg/mL (2.22 mM), Sonication is recommended. | ||||||||||
溶液配制表 | |||||||||||
H2O
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