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ST3932 is a ST1535 metabolite, is a adenosine A2A receptor antagonist(Kis of 8 nM and 33 nM for A2A and A1 receptors, respectively).
ST3932 is a ST1535 metabolite, is a adenosine A2A receptor antagonist(Kis of 8 nM and 33 nM for A2A and A1 receptors, respectively).
规格 | 价格 | 库存 | 数量 |
---|---|---|---|
25 mg | ¥ 11,700 | 6-8周 | |
50 mg | ¥ 15,300 | 6-8周 | |
100 mg | ¥ 19,500 | 6-8周 |
产品描述 | ST3932 is a ST1535 metabolite, is a adenosine A2A receptor antagonist(Kis of 8 nM and 33 nM for A2A and A1 receptors, respectively). |
靶点活性 | A2A receptor:ki: 8 nM , A1 receptor:33 nM (ki) |
体外活性 | ST3932 is a ST1535 metabolite, acts as an adenosine A2A receptor antagonist(Kis of 8 nM and 33 nM for A2A and A1 receptors, respectively). ST3932 inhibits agonist-induced cAMP accumulation(IC50 : 450 nM). |
体内活性 | In mice, Haloperidol-induced catalepsy antagonized by ST3932 (10, 20, 40 mg/kg, p.o.), and increases motor activity . ST3932 (20, 40 mg/kg, i.p.) significantly increases the number of contralateral turns induced by l-DOPA in rats. |
分子量 | 288.31 |
分子式 | C12H16N8O |
CAS No. | 1246018-21-2 |
密度 | 1.62 g/cm3 (Predicted) |
存储 | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
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