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SR-12062作为神经肽受体1 (NTSR1) 的全激动剂,表现出显著的高效能和增强的药效。在NTSR1上,该化合物的EC50值为2 μM,并完全激活受体(Emax=100%)。相较于母化合物1(EC50=178 μM;Emax=17%),SR-12062的效力提高了约90倍。
SR-12062作为神经肽受体1 (NTSR1) 的全激动剂,表现出显著的高效能和增强的药效。在NTSR1上,该化合物的EC50值为2 μM,并完全激活受体(Emax=100%)。相较于母化合物1(EC50=178 μM;Emax=17%),SR-12062的效力提高了约90倍。
规格 | 价格 | 库存 | 数量 |
---|---|---|---|
10 mg | 询价 | 10-14周 | |
50 mg | 询价 | 10-14周 |
产品描述 | SR-12062 functions as a full agonist at neurotensin receptor 1 (NTSR1), demonstrating notable efficacy and increased potency. Its EC50 value on NTSR1 is 2 μM, with complete receptor activation (Emax=100%). Compared to the parent compound 1 (EC50=178 μM; Emax=17%), SR-12062 shows approximately 90-fold greater potency. |
别名 | SR12062, SR 12062 |
分子量 | 415.48 |
分子式 | C25H25N3O3 |
CAS No. | 1623019-77-1 |
存储 | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
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