Ac-RYYRWK-NH2 TFA

Name: Ac-RYYRWK-NH2 TFA
Brand: TargetMol
SKU: T40510
Rating: 4.5 (1 reviews)

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产品编号 T40510Cas号 408305-09-9

别名 Ac-RYYRWK-NH2 TFA

Ac-RYYRWK-NH2 is a highly effective and specific partial agonist for the nociceptin receptor (NOP). It demonstrates a remarkable affinity for rat cortical membranes ORL1, with [3H]Ac-RYYRWK-NH2 exhibiting a Kd value of 0.071 nM. However, it shows negligible affinity towards μ-, κ-, or δ-opioid receptors.

Ac-RYYRWK-NH2 TFA

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产品编号 T40510 别名 Ac-RYYRWK-NH2 TFACas号 408305-09-9

规格	价格	库存	数量
100 mg	询价	期货
500 mg	询价	期货

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产品描述	Ac-RYYRWK-NH2 is a highly effective and specific partial agonist for the nociceptin receptor (NOP). It demonstrates a remarkable affinity for rat cortical membranes ORL1, with [3H]Ac-RYYRWK-NH2 exhibiting a Kd value of 0.071 nM. However, it shows negligible affinity towards μ-, κ-, or δ-opioid receptors.
体外活性	[3H]ac-RYYRWK-NH2 binding to rat cortical membranes revealed a single high affinity site for [3H]ac-RYYRWK-NH2 (K d =0.071 nM)[1]. Naloxone benzoylhydrazone displaced [3H]acRYYRWK-NH2 binding to rat cortical membranes (K i =104 nM) and human ORL1 (K i =136 nM) as well as [125I]Tyr14-NC-OH to ORL1 (K i =37 nM) has no affinity for μ-, κ- or δ-opioid receptors[1].
别名	Ac-RYYRWK-NH2 TFA