• TargetMol
    您的购物车当前为空
TargetMol | Compound Library

抗心血管疾病化合物库现货

Anti-Cardiovascular Disease Compound Library

Rating icon 很棒
产品编号 L5400

心血管疾病泛指由于动脉粥样硬化、高脂血症、血液黏稠、高血压等所导致的心脏、大脑及全身组织发生的缺血性或出血性疾病,例如心绞痛、心肌梗塞、中风等,是全球死亡的首要原因。不同类型疾病的发病机制不同,各种抗氧化、抗高血脂、抗缺血、抑制血小板聚集和抗炎物质都具有降低心血管疾病风险的作用。某些天然产物具有抑制粘附分子、细胞因子和趋化因子基因表达,抑制血小板功能,增强内皮细胞一氧化氮释放,抑制平滑肌活化的作用,这些化合物都是心血管疾病药物筛选中的重要工具。

TargetMol 抗心血管疾病化合物库是由 1793 个心血管疾病相关的化合物组成的综合筛选库,用于心血管疾病的相关研究和高通量高内涵筛选。

TargetMol 的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
资源下载
化合物库相关信息
Excel
SDF
联系我们获取更多批次信息

产品编号 L5400

抗心血管疾病化合物库

规格

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品描述 产品描述

  • 1793种心血管疾病相关的生物活性小分子化合物的特有集合,用于高通量、高内涵筛选;
  • 靶点包括膜转运体、离子通道等心血管疾病相关靶点;
  • 大部分产品是经FDA、EMA或NMPA批准上市的药物,是研究心血管相关疾病的有效工具;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

包装和储存 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
  • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。

使用TargetMol产品
发表顶级期刊文献

引用更多关于TargetMol产品的科学文献吧!

查看更多

Library Customization | TargetMol 化合物库定制

Compound Library | TargetMol
您可以通过点击按钮
定制您专属的化合物!
联系专属定制

Library Customization | TargetMol 化合物库组成

Adrenergic Receptor
Apoptosis
Calcium Channel
PDE
Autophagy
VEGFR
Endogenous Metabolite
COX
Sodium Channel
Potassium Channel
NF-κB
Antibacterial
5-HT Receptor
TNF
AChR
ROS
RAAS
PDGFR
Dopamine Receptor
Parasite
Angiotensin-converting Enzyme (ACE)
IL Receptor
FGFR
p38 MAPK
c-Kit
Interleukin
PARP
Histone Acetyltransferase
Histamine Receptor
FLT
PPAR
ERK
Reactive Oxygen Species
Akt
Drug Metabolite
CDK
NO Synthase
Cytochromes P450
HMG-CoA Reductase
EGFR
PKC
Adenosine Receptor
Factor Xa
DNA/RNA Synthesis
Antifungal
BACE
JAK
Epigenetic Reader Domain
PI3K
Antioxidant
Prostaglandin Receptor
Antibiotic
Carbonic Anhydrase
Caspase
IGF-1R
Influenza Virus
ATPase
Src
Ferroptosis
c-Met/HGFR
Mitophagy
c-RET
Thrombin
HIV Protease
JNK
Beta-Secretase
PKA
TRP/TRPV Channel
Norepinephrine
SARS-CoV
Nrf2
Phospholipase
P2Y Receptor
Glucocorticoid Receptor
STAT
NOD-like Receptor (NLR)
GSK-3
Wnt/beta-catenin
Cholinesterase (ChE)
CaMK
P-gp
Beta Amyloid
HDAC
GABA Receptor
Proteasome
Integrin
iGluR
Mitochondrial Metabolism
Lipoxygenase
Virus Protease
Raf
Guanylate cyclase
AMPK
Anti-infection
MRP
Bcr-Abl
c-Fms
MEK
Monoamine Oxidase
Proton pump
Dehydrogenase
Tyrosine Kinases
Serine Protease
Serotonin Transporter
ROCK
LDLR
NMDAR
Aurora Kinase
Acetyl-CoA Carboxylase
Hydroxylase
Tyrosinase
NADPH
Tie-2
Glutathione Peroxidase
MAO
Topoisomerase
MMP
Bcl-2 Family
IκB/IKK
NOD
Microtubule Associated
Chloride channel
Amino Acids and Derivatives
Na+/Ca2+ Exchanger
CETP
PERK
Serine/threonin kinase
Nucleoside Antimetabolite/Analog
Liver X Receptor
FXR
LDL
P2X Receptor
Opioid Receptor
Fatty Acid Synthase
HSV
GluR
mTOR
TGF-beta/Smad
Acyltransferase
TLR
Trk receptor
TAM Receptor
FAK
HIF/HIF Prolyl-Hydroxylase
GPCR
NOS
Myosin
DPP-4
Chk
Epoxide Hydrolase
cAMP
PGE Synthase
MAPK
HSP
Sirtuin
Ephrin Receptor
RSV
Neprilysin
HIF
Ras
Sigma receptor
Protease-activated Receptor
Imidazoline Receptor
p53
Thyroid hormone receptor(THR)
Histone Methyltransferase
Arginase
DNA Alkylator/Crosslinker
Reductase
Estrogen Receptor/ERR
Leukotriene Receptor
CSF-1R
Immunology/Inflammation related
RIP kinase
UGT
Na-K-Cl cotransporter
HCN Channel
Endothelin Receptor
Androgen Receptor
Lipid
transporter
PAI-1
ALK
Reverse Transcriptase
PDK
MDM-2/p53
Platelet aggregation
Syk
NADPH-oxidase
S6 Kinase
Vitamin
MTP
Adenylyl Cyclase
Transferase
Monocarboxylate transporter
DHFR
ROR
Estrogen/progestogen Receptor
Factor VIIa
LPL Receptor
LTR
IFNAR
Histone Demethylase
Necroptosis
Phosphatase
Rho
Antifolate
PYK2
Amylase
Prolyl Endopeptidase (PREP)
Annexin A
Gamma-secretase
ABC Transporter
Glucosidase
Antifection
Monoamine Transporter
DNA Alkylation
FAAH
CCR
Xanthine Oxidase
Thrombopoietin Receptor
glycosidase
DNA
OXPHOS
Aminopeptidase
GPCR19
ASK
Casein Kinase
FKBP
SGK
Gap Junction Protein
DNA Methyltransferase
IRAK
AhR
CFTR
MLK
NPC1L1
DNA-PK
HCV Protease
DprE1
YAP
Lipase
MIF
TOPK
Progesterone Receptor
OCT
N-Acetylglucosaminyltransferase
CaSR
HBV
VDAC
Cell Cycle Arrest
Cysteine Protease
Neurotensin Receptor
Glucokinase
Aryl Hydrocarbon Receptor
IDO
IAP
IRE1
Photosystem (PS)
FLAP
Adiponectin Receptor
PAFR
GRK
Arp2/3 Complex
DNA gyrase
GlyT
Anion Exchanger
Isocitrate Dehydrogenase (IDH)
Hedgehog/Smoothened
Vasopressin Receptor
ACK1
CXCR
Indoleamine 2,3-Dioxygenase (IDO)
SGLT
ATP Citrate Lyase
BCRP
OAT
Antiviral
STING
LRRK2
AIM2
Decarboxylase
GST
Retinoid Receptor
Kras
Aromatase
CRISPR/Cas9
RXFP receptor
PLK
Cuproptosis
Cannabinoid Receptor
Discoidin Domain Receptor (DDR)
Tight Junction Protein
p97
ROS Kinase
HER
PKM
S1P Receptor
ADC Cytotoxin
Sodium-dependent phosphate transporter
BTK
PGC-1α

Keywords