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TargetMol | Compound Library

抗心血管疾病化合物库现货

Anti-Cardiovascular Disease Compound Library

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产品编号 L5400

心血管疾病泛指由于动脉粥样硬化、高脂血症、血液黏稠、高血压等所导致的心脏、大脑及全身组织发生的缺血性或出血性疾病,例如心绞痛、心肌梗塞、中风等,是全球死亡的首要原因。不同类型疾病的发病机制不同,各种抗氧化、抗高血脂、抗缺血、抑制血小板聚集和抗炎物质都具有降低心血管疾病风险的作用。某些天然产物具有抑制粘附分子、细胞因子和趋化因子基因表达,抑制血小板功能,增强内皮细胞一氧化氮释放,抑制平滑肌活化的作用,这些化合物都是心血管疾病药物筛选中的重要工具。 TargetMol 抗心血管疾病化合物库是由 1793 个心血管疾病相关的化合物组成的综合筛选库,用于心血管疾病的相关研究和高通量高内涵筛选。

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产品编号 L5400

抗心血管疾病化合物库

规格

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品描述 产品描述

  • 1793种心血管疾病相关的生物活性小分子化合物的特有集合,用于高通量、高内涵筛选;
  • 靶点包括膜转运体、离子通道等心血管疾病相关靶点;
  • 大部分产品是经FDA、EMA或NMPA批准上市的药物,是研究心血管相关疾病的有效工具;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

包装和储存 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
  • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。

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Library Customization | TargetMol 化合物库组成

Adrenergic Receptor
Calcium Channel
Apoptosis
PDE
Autophagy
VEGFR
Endogenous Metabolite
COX
Sodium Channel
Potassium Channel
5-HT Receptor
Antibacterial
AChR
TNF
NF-κB
RAAS
PDGFR
Dopamine Receptor
Parasite
Angiotensin-converting Enzyme (ACE)
IL Receptor
FGFR
c-Kit
Histone Acetyltransferase
PARP
FLT
Histamine Receptor
Reactive Oxygen Species
PPAR
CDK
HMG-CoA Reductase
Drug Metabolite
Cytochromes P450
EGFR
Factor Xa
PKC
p38 MAPK
Adenosine Receptor
BACE
Epigenetic Reader Domain
Antioxidant
JAK
Antibiotic
ATPase
Carbonic Anhydrase
Antifungal
IGF-1R
Interleukin
c-Met/HGFR
Mitophagy
ERK
DNA/RNA Synthesis
Src
Influenza Virus
c-RET
Akt
Beta-Secretase
Ferroptosis
Norepinephrine
Thrombin
NO Synthase
HIV Protease
P2Y Receptor
TRP/TRPV Channel
Glucocorticoid Receptor
Prostaglandin Receptor
SARS-CoV
Phospholipase
PI3K
Caspase
P-gp
Virus Protease
PKA
Beta Amyloid
HDAC
GABA Receptor
Anti-infection
Proteasome
iGluR
Raf
ROS
Guanylate cyclase
Cholinesterase (ChE)
Lipoxygenase
CaMK
Nrf2
STAT
GSK-3
MRP
Bcr-Abl
Mitochondrial Metabolism
c-Fms
Monoamine Oxidase
Proton pump
Integrin
Dehydrogenase
Tyrosine Kinases
Serine Protease
ROCK
NMDAR
Aurora Kinase
AMPK
Hydroxylase
NOD-like Receptor (NLR)
NADPH
Tie-2
Wnt/beta-catenin
Serotonin Transporter
MAO
Topoisomerase
Bcl-2 Family
IκB/IKK
Acetyl-CoA Carboxylase
MEK
NOD
Tyrosinase
Chloride channel
Na+/Ca2+ Exchanger
Serine/threonin kinase
Nucleoside Antimetabolite/Analog
FXR
LDL
P2X Receptor
Opioid Receptor
HSV
MMP
GluR
Acyltransferase
Trk receptor
TAM Receptor
Microtubule Associated
HIF/HIF Prolyl-Hydroxylase
GPCR
NOS
Amino Acids and Derivatives
CETP
JNK
Glutathione Peroxidase
Liver X Receptor
Myosin
DPP-4
Fatty Acid Synthase
Chk
Epoxide Hydrolase
cAMP
mTOR
PGE Synthase
TLR
Ephrin Receptor
RSV
Neprilysin
HIF
Sigma receptor
Protease-activated Receptor
FAK
Imidazoline Receptor
p53
Thyroid hormone receptor(THR)
Arginase
DNA Alkylator/Crosslinker
Reductase
Estrogen Receptor/ERR
Leukotriene Receptor
LDLR
Immunology/Inflammation related
CSF-1R
Na-K-Cl cotransporter
HCN Channel
Endothelin Receptor
Androgen Receptor
TGF-beta/Smad
Lipid
MAPK
HSP
Sirtuin
transporter
ALK
Reverse Transcriptase
PDK
MDM-2/p53
Platelet aggregation
Syk
NADPH-oxidase
Ras
S6 Kinase
Adenylyl Cyclase
Transferase
Monocarboxylate transporter
DHFR
ROR
Histone Methyltransferase
MTP
Estrogen/progestogen Receptor
Factor VIIa
LPL Receptor
LTR
Histone Demethylase
PERK
Rho
Antifolate
PYK2
Amylase
Prolyl Endopeptidase (PREP)
UGT
Gamma-secretase
ABC Transporter
Glucosidase
Antifection
Monoamine Transporter
DNA Alkylation
FAAH
Xanthine Oxidase
Thrombopoietin Receptor
DNA
OXPHOS
Aminopeptidase
PAI-1
Casein Kinase
FKBP
SGK
Gap Junction Protein
DNA Methyltransferase
AhR
CFTR
NPC1L1
DNA-PK
HCV Protease
DprE1
YAP
IFNAR
Lipase
Necroptosis
MIF
TOPK
Phosphatase
Progesterone Receptor
OCT
N-Acetylglucosaminyltransferase
CaSR
HBV
VDAC
Cell Cycle Arrest
Cysteine Protease
Neurotensin Receptor
Glucokinase
Aryl Hydrocarbon Receptor
IDO
IAP
IRE1
Annexin A
Photosystem (PS)
FLAP
RIP kinase
Adiponectin Receptor
PAFR
GRK
Arp2/3 Complex
DNA gyrase
GlyT
Anion Exchanger
Isocitrate Dehydrogenase (IDH)
CCR
ACK1
Vasopressin Receptor
Indoleamine 2,3-Dioxygenase (IDO)
SGLT
ATP Citrate Lyase
BCRP
OAT
Antiviral
LRRK2
GPCR19
AIM2
Decarboxylase
ASK
GST
Retinoid Receptor
KRas
Aromatase
CRISPR/Cas9
RXFP receptor
PLK
Cuproptosis
Cannabinoid Receptor
Discoidin Domain Receptor (DDR)
IRAK
p97
ROS Kinase
MLK
HER
PKM
S1P Receptor
ADC Cytotoxin
Sodium-dependent phosphate transporter
Vitamin
BTK
PGC-1α

Keywords