Cimetidine sulfoxide

Name: Cimetidine sulfoxide
Brand: TargetMol
SKU: T38058
Price: 125 USD
Availability: InStock
Rating: 4.5 (1 reviews)

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产品编号 T38058Cas号 54237-72-8

别名 西咪替丁亚砜

Cimetidine sulfoxide (Cimetidine sulphoxide) is a metabolite of Cimetidine, functioning as a histamine H2-receptor antagonist with potential applications in treating peptic ulcer disease and upper gastrointestinal hemorrhage[1].

Cimetidine sulfoxide

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产品编号 T38058 别名 西咪替丁亚砜Cas号 54237-72-8

规格	价格	库存	数量
2 mg	¥ 720	5日内发货

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产品介绍

生物活性

产品描述	Cimetidine sulfoxide (Cimetidine sulphoxide) is a metabolite of Cimetidine, functioning as a histamine H2-receptor antagonist with potential applications in treating peptic ulcer disease and upper gastrointestinal hemorrhage[1].
体外活性	Active transport of Cimetidine across the rat small intestine is observable at lower substrate concentrations (40 and 200 μM), but is masked by passive transfer at higher concentrations (400 μM). Cimetidine sulfoxide is detected after some incubations[2].
体内活性	The enantiomeric composition of Cimetidine sulfoxide is also determined in rat urine (24 h) following the administration of Cimetidine (30 mg/kg; po) to male Wistar rats. The enantiomeric ratio in this case is found to be (+/-) 57:43[3].
别名	西咪替丁亚砜

化学信息

分子量	268.34
分子式	C₁₀H₁₆N₆OS
CAS No.	54237-72-8

储存&溶解度

存储

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.

溶解度信息

DMSO: 83.33 mg/mL (310.54 mM), Sonication and heating to 60℃ are recommended.

溶液配制表

DMSO

	1mg	5mg	10mg	50mg
1 mM	3.7266 mL	18.6331 mL	37.2662 mL	186.3308 mL
5 mM	0.7453 mL	3.7266 mL	7.4532 mL	37.2662 mL
10 mM	0.3727 mL	1.8633 mL	3.7266 mL	18.6331 mL
20 mM	0.1863 mL	0.9317 mL	1.8633 mL	9.3165 mL
50 mM	0.0745 mL	0.3727 mL	0.7453 mL	3.7266 mL
100 mM	0.0373 mL	0.1863 mL	0.3727 mL	1.8633 mL