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TargetMol | Compound Library

抗糖尿病库现货

Anti-Diabetic Compound Library

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产品编号 L1900

糖尿病是一种以高血糖为特征的代谢性疾病,长期的高血糖会导致全身各种组织功能障碍,如果出现并发症,糖尿病会对生活质量产生重大影响,并可能降低预期寿命,目前仍然无法治愈糖尿病,只能通过饮食调节和药物辅助治疗进行病情控制。 TargetMol 抗糖尿病库包含了 800 个糖尿病相关活性化合物,是研究糖尿病的优良工具和药物筛选的极佳载体。

TargetMol 的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
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产品编号 L1900

抗糖尿病库

规格

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品描述 产品描述

  • 800种生物活性小分子化合物;
  • 靶点包括SGLT、PPAR、DPP-4、OC receptor、AMPK等;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

Packaging And Storage | TargetMol 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。

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Library Customization | TargetMol 化合物库定制

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Library Customization | TargetMol 化合物库组成

PPAR
Autophagy
Apoptosis
AMPK
mTOR
NF-κB
Endogenous Metabolite
IGF-1R
JNK
PI3K
Glucagon Receptor
Antibacterial
GSK-3
COX
DPP-4
Akt
SGLT
Potassium Channel
Proteasome
Glucosidase
Antibiotic
STAT
CDK
GPR
Antioxidant
Parasite
Phosphatase
p38 MAPK
Ferroptosis
TNF
Cytochromes P450
Sirtuin
Influenza Virus
DNA-PK
Reductase
Mitophagy
Glucokinase
Src
Dehydrogenase
PDE
ERK
Reactive Oxygen Species
IL Receptor
transporter
Antifungal
S6 Kinase
PKC
MMP
Lipoxygenase
Prostaglandin Receptor
Adrenergic Receptor
EGFR
FLT
NO Synthase
ALK
Adenosine Receptor
Virus Protease
VEGFR
Mitochondrial Metabolism
Interleukin
IκB/IKK
ATM/ATR
FGFR
HDAC
HIV Protease
ATPase
Wnt/beta-catenin
Caspase
Calcium Channel
TRP/TRPV Channel
ROS
DNA/RNA Synthesis
SARS-CoV
Bcl-2 Family
Beta Amyloid
Nrf2
Cannabinoid Receptor
AChR
Tyrosinase
HIF/HIF Prolyl-Hydroxylase
c-Met/HGFR
Glucocorticoid Receptor
HSV
Aurora Kinase
PDGFR
JAK
Cholinesterase (ChE)
MEK
FAK
p53
NADPH
Histamine Receptor
CETP
PKA
Serine Protease
ROCK
Phosphorylase
Tyrosine Kinases
SIK
Drug Metabolite
ABC Transporter
Antifection
Fatty Acid Synthase
CCR
MAPK
Trk receptor
PDK
5-HT Receptor
Casein Kinase
GABA Receptor
HIF
NOD
Thrombin
NOS
Carbonic Anhydrase
BACE
Glutathione Peroxidase
Transferase
PERK
PARP
PYK2
Amylase
MAO
Topoisomerase
Bcr-Abl
Raf
HBV
Liver X Receptor
Leukotriene Receptor
FXR
E1/E2/E3 Enzyme
Opioid Receptor
Stearoyl-CoA Desaturase (SCD)
Chk
Epigenetic Reader Domain
DNA
P-gp
Bombesin Receptor
Epoxide Hydrolase
Norepinephrine
Androgen Receptor
CFTR
MLK
Retinoid Receptor
Phospholipase
c-RET
Syk
NADPH-oxidase
Sodium Channel
Chloride channel
Histone Methyltransferase
Estrogen/progestogen Receptor
LPL Receptor
Arrestin
DYRK
RAAS
Tie-2
GTPase
Advanced Glycation End Products
Proton pump
NPC1L1
Dopamine Receptor
Integrin
YAP
LTR
CaSR
Estrogen Receptor/ERR
Annexin A
LDL
Rho
Serotonin Transporter
Cell Cycle Arrest
Cysteine Protease
Neurotensin Receptor
NAMPT
FOXO1
Aryl Hydrocarbon Receptor
Immunology/Inflammation related
FLAP
GRK
Hexokinase
DNA Alkylation
ACK1
Bradykinin Receptor
CXCR
GluR
CaMK
TGF-beta/Smad
ATP Citrate Lyase
Beta-Secretase
Acyltransferase
TLR
LRRK2
Free radical scavengers
GPCR19
PROTAC Linker
PAK
FAAH
Telomerase
MNK
Antiviral
Pyroptosis
c-Fms
PI4K
SGK
IRAK
HMG-CoA Reductase
PKM
PAI-1
Hippo pathway
Reverse Transcriptase
Aromatase
Anti-infection
c-Kit
Sigma receptor
NOD-like Receptor (NLR)
S1P Receptor
Monoamine Oxidase
ADC Cytotoxin
IGF-2R
BTK
PGC-1α

Keywords