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TargetMol | Compound Library

抗糖尿病库现货

Anti-Diabetic Compound Library

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产品编号 L1900

糖尿病是一种以高血糖为特征的代谢性疾病,长期的高血糖会导致全身各种组织功能障碍,如果出现并发症,糖尿病会对生活质量产生重大影响,并可能降低预期寿命,目前仍然无法治愈糖尿病,只能通过饮食调节和药物辅助治疗进行病情控制。 TargetMol 抗糖尿病库包含了 800 个糖尿病相关活性化合物,是研究糖尿病的优良工具和药物筛选的极佳载体。

TargetMol 的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
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产品编号 L1900

抗糖尿病库

规格

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品描述 产品描述

  • 800种生物活性小分子化合物;
  • 靶点包括SGLT、PPAR、DPP-4、OC receptor、AMPK等;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

包装和储存 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
  • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。

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Library Customization | TargetMol 化合物库组成

PPAR
Autophagy
Apoptosis
AMPK
mTOR
NF-κB
Endogenous Metabolite
IGF-1R
JNK
PI3K
Glucagon Receptor
Antibacterial
COX
GSK-3
DPP-4
Akt
SGLT
Potassium Channel
Glucosidase
Antibiotic
Proteasome
CDK
GPCR
STAT
Antioxidant
Ferroptosis
p38 MAPK
Phosphatase
TNF
Influenza Virus
Parasite
Reductase
Sirtuin
Cytochromes P450
DNA-PK
Mitophagy
Dehydrogenase
ERK
Glucokinase
PDE
Reactive Oxygen Species
Src
transporter
Antifungal
IL Receptor
S6 Kinase
MMP
PKC
Prostaglandin Receptor
Adrenergic Receptor
ALK
EGFR
FLT
Lipoxygenase
NO Synthase
AChR
Adenosine Receptor
ATM/ATR
Calcium Channel
FGFR
IκB/IKK
TRP/TRPV Channel
VEGFR
Virus Protease
ATPase
Bcl-2 Family
Beta Amyloid
Cannabinoid Receptor
Caspase
Cholinesterase (ChE)
DNA/RNA Synthesis
HDAC
HIF/HIF Prolyl-Hydroxylase
HIV Protease
Interleukin
Mitochondrial Metabolism
Nrf2
p53
ROS
SARS-CoV
Tyrosinase
Wnt/beta-catenin
Aurora Kinase
FAK
Glucocorticoid Receptor
HSV
JAK
MEK
NADPH
PDGFR
Sodium Channel
5-HT Receptor
ABC Transporter
Antifection
BACE
Casein Kinase
CCR
CETP
c-Met/HGFR
Drug Metabolite
Fatty Acid Synthase
GABA Receptor
HIF
Histamine Receptor
MAPK
NADPH-oxidase
NOD
PDK
Phosphorylase
PKA
ROCK
Serine Protease
SIK
Thrombin
Transferase
Tyrosine Kinases
Androgen Receptor
Bcr-Abl
Bombesin Receptor
Carbonic Anhydrase
CFTR
Chk
c-RET
DNA
E1/E2/E3 Enzyme
Epigenetic Reader Domain
FXR
Glutathione Peroxidase
HBV
Leukotriene Receptor
Liver X Receptor
MAO
MLK
Norepinephrine
NOS
Opioid Receptor
PARP
PERK
P-gp
Phospholipase
PYK2
Raf
Retinoid Receptor
Stearoyl-CoA Desaturase (SCD)
Syk
Topoisomerase
Trk receptor
ACK1
Acyltransferase
Advanced Glycation End Products
Amylase
Annexin A
Anti-infection
Antiviral
Aromatase
Arrestin
Aryl Hydrocarbon Receptor
ATP Citrate Lyase
Beta-Secretase
Bradykinin Receptor
CaMK
CaSR
Cell Cycle Arrest
c-Fms
Chloride channel
c-Kit
CXCR
Cysteine Protease
DNA Alkylation
Dopamine Receptor
DYRK
Epoxide Hydrolase
Estrogen Receptor/ERR
Estrogen/progestogen Receptor
FAAH
FLAP
FOXO1
Free radical scavengers
GluR
GPCR19
GRK
GTPase
Hexokinase
Hippo pathway
Histone Methyltransferase
HMG-CoA Reductase
Immunology/Inflammation related
Integrin
IRAK
LDL
LPL Receptor
LRRK2
LTR
MNK
Monoamine Oxidase
Neurotensin Receptor
NOD-like Receptor (NLR)
NPC1L1
PAI-1
PAK
PI4K
PKM
PROTAC Linker
Proton pump
Pyroptosis
RAAS
Reverse Transcriptase
Rho
S1P Receptor
Serotonin Transporter
SGK
Sigma receptor
Telomerase
TGF-beta/Smad
Tie-2
TLR
YAP
ADC Cytotoxin
IGF-2R
BTK
PGC-1α

Keywords