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TargetMol | Compound Library

FDA 上市药物库现货

FDA-Approved Drug Library

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产品编号 L4200

FDA 上市药物库中的所有化合物都具有良好的生物活性、明确的靶点信息,较好的安全性和生物利用度,这些特性可显著加速药物开发和优化,是进行小分子细胞诱导分化和药物重定位理想的工具。详尽的数据资料可以帮助科学家快速完成药物筛选或细胞诱导机制的判断,并为深入揭示其机制机理创造条件。

TargetMol 的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。

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产品编号 L4200

FDA 上市药物库

规格

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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产品描述 产品描述

  • 1840个FDA批准药物的独特集合,可用于高通量筛选和高内涵筛选;
  • 全部得到FDA批准,提供FDA批准编号,用于药物重定位、新的药物靶点筛选的有效工具;
  • 经过了严格的临床前研究和临床试验,生物活性和安全性得到保障;
  • 涵盖多个研究领域:肿瘤、心血管药物、抗炎、免疫、神经系统药物、呼吸系统药物等;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

Packaging And Storage | TargetMol 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。

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Library Customization | TargetMol 化合物库组成

Antibacterial
Antibiotic
Autophagy
Apoptosis
Endogenous Metabolite
Adrenergic Receptor
5-HT Receptor
AChR
Histamine Receptor
Dopamine Receptor
HIV Protease
Sodium Channel
COX
Antifungal
Parasite
Potassium Channel
DNA/RNA Synthesis
Glucocorticoid Receptor
Estrogen/progestogen Receptor
Calcium Channel
Topoisomerase
Cytochromes P450
Ferroptosis
RAAS
SARS-CoV
Serotonin Transporter
VEGFR
PDE
ribosome
Dehydrogenase
Estrogen Receptor/ERR
Microtubule Associated
Mitophagy
Norepinephrine
c-Kit
Nucleoside Antimetabolite/Analog
Reverse Transcriptase
GABA Receptor
HCV Protease
Antifection
Progesterone Receptor
HSV
EGFR
PPAR
PDGFR
Proton pump
Reactive Oxygen Species
ADC Cytotoxin
Androgen Receptor
Influenza Virus
ATPase
Carbonic Anhydrase
HBV
JAK
Cholinesterase (ChE)
Prostaglandin Receptor
Src
Phosphatase
MAO
FGFR
FLT
Thrombin
Proteasome
DNA Alkylator/Crosslinker
Adenosine Receptor
Bcr-Abl
Thyroid hormone receptor(THR)
c-Met/HGFR
MRP
Tyrosine Kinases
ROS
NF-κB
HMG-CoA Reductase
Transferase
DHFR
Virus Protease
PARP
Antifolate
ALK
HDAC
c-RET
Monoamine Oxidase
GNRH Receptor
TRP/TRPV Channel
iGluR
Raf
Drug Metabolite
Opioid Receptor
MMP
SGLT
NO Synthase
PI3K
ABC Transporter
GluR
P-gp
Retinoid Receptor
P2Y Receptor
Factor Xa
PKC
CDK
NMDAR
DNA gyrase
Guanylate cyclase
DPP-4
Endothelin Receptor
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STAT
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LPL Receptor
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IL Receptor
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Trk receptor
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TNF
HER
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Histone Methyltransferase
Integrin
Cell wall
NADPH
Monoamine Transporter
Hedgehog/Smoothened
Vasopressin Receptor
Lipoxygenase
Antiviral
Nrf2
Neurokinin receptor
TAM Receptor
ROS Kinase
CFTR
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Reductase
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FXR
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Molecular Glues
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HIF
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NOS
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ERK
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MT Receptor
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cholecystokinin
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Arginase
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CETP
GSK-3
Melatonin Receptor
Rho
Leukotriene Receptor
Caspase
IRE1
UGT
Gamma-secretase
P2X Receptor
Na-K-Cl cotransporter
Integrase
CCR
CXCR
Xanthine Oxidase
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Akt
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GluCls
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Hydrogenase
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YAP
IFNAR
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gp120/CD4
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Adiponectin Receptor
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GRK
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Glucosidase
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ACK1
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DUB
Telomerase
TGF-beta/Smad
ATP Citrate Lyase
Lipid
MAPK
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STING
Pyroptosis
IκB/IKK
CRISPR/Cas9
PDK
Oxytocin Receptor
Aquaporin
PLK
Platelet aggregation
Anti-infection
NADPH-oxidase
Tyrosinase
NOD-like Receptor (NLR)

Keywords