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TargetMol | Compound Library

FDA 上市药物库现货

FDA-Approved Drug Library

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产品编号 L4200

FDA 上市药物库中的所有化合物都具有良好的生物活性、明确的靶点信息,较好的安全性和生物利用度,这些特性可显著加速药物开发和优化,是进行小分子细胞诱导分化和药物重定位理想的工具。详尽的数据资料可以帮助科学家快速完成药物筛选或细胞诱导机制的判断,并为深入揭示其机制机理创造条件。

TargetMol 的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
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产品编号 L4200

FDA 上市药物库

规格

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品描述 产品描述

  • 1840个FDA批准药物的独特集合,可用于高通量筛选和高内涵筛选;
  • 全部得到FDA批准,提供FDA批准编号,用于药物重定位、新的药物靶点筛选的有效工具;
  • 经过了严格的临床前研究和临床试验,生物活性和安全性得到保障;
  • 涵盖多个研究领域:肿瘤、心血管药物、抗炎、免疫、神经系统药物、呼吸系统药物等;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

Packaging And Storage | TargetMol 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。

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Library Customization | TargetMol 化合物库组成

Antibacterial
Antibiotic
Autophagy
Apoptosis
Endogenous Metabolite
Adrenergic Receptor
5-HT Receptor
AChR
Histamine Receptor
HIV Protease
Dopamine Receptor
Sodium Channel
Parasite
COX
Antifungal
Potassium Channel
Glucocorticoid Receptor
DNA/RNA Synthesis
Estrogen/progestogen Receptor
Calcium Channel
Cytochromes P450
Topoisomerase
SARS-CoV
Ferroptosis
RAAS
VEGFR
Estrogen Receptor/ERR
Serotonin Transporter
PDE
Mitophagy
ribosome
Microtubule Associated
Dehydrogenase
c-Kit
Norepinephrine
Nucleoside Antimetabolite/Analog
Reverse Transcriptase
GABA Receptor
HCV Protease
EGFR
Progesterone Receptor
Antifection
PDGFR
PPAR
HSV
Proton pump
Reactive Oxygen Species
Influenza Virus
ATPase
Carbonic Anhydrase
HBV
JAK
Androgen Receptor
DNA Alkylator/Crosslinker
Cholinesterase (ChE)
Prostaglandin Receptor
FLT
Src
MAO
FGFR
Proteasome
Adenosine Receptor
Phosphatase
Bcr-Abl
NF-κB
HMG-CoA Reductase
Thrombin
Thyroid hormone receptor(THR)
c-Met/HGFR
MRP
Tyrosine Kinases
Raf
ROS
HDAC
Transferase
DHFR
Virus Protease
PARP
Antifolate
iGluR
ALK
c-RET
Monoamine Oxidase
PI3K
GNRH Receptor
TRP/TRPV Channel
Drug Metabolite
MMP
SGLT
NMDAR
ABC Transporter
Opioid Receptor
mTOR
P-gp
Retinoid Receptor
STAT
HIF/HIF Prolyl-Hydroxylase
NO Synthase
P2Y Receptor
Factor Xa
PKC
CDK
DNA gyrase
Guanylate cyclase
DPP-4
Endothelin Receptor
GluR
CaMK
Phospholipase
DNA Methyltransferase
LPL Receptor
DNA Alkylation
IL Receptor
Lipoxygenase
TLR
Trk receptor
MEK
TNF
HER
S1P Receptor
ADC Cytotoxin
Histone Methyltransferase
Integrin
NADPH
Monoamine Transporter
Hedgehog/Smoothened
Vasopressin Receptor
Interleukin
Antiviral
HSP
Nrf2
AMPK
HIF
Neurokinin receptor
TAM Receptor
ROS Kinase
CFTR
Reductase
Cell wall
Glutathione Peroxidase
FXR
ROCK
ERK
Annexin A
Molecular Glues
Isocitrate Dehydrogenase (IDH)
DNA
Ligand for E3 Ligase
Aromatase
GPR
Hydroxylase
AhR
NOS
Histone Demethylase
CaSR
Cholecystokinin Receptor
Cysteine Protease
Aryl Hydrocarbon Receptor
LDL
Gamma-secretase
MT Receptor
Mitochondrial Metabolism
Smo
Fatty Acid Synthase
PAK
IGF-1R
Akt
GPCR19
Bcl-2 Family
Decarboxylase
Neprilysin
GST
Melanocortin Receptor
Complement System
Sigma receptor
Chloride channel
MicroRNA
CRM1
Amino Acids and Derivatives
Ligands for Target Protein for PROTAC
Arginase
Antioxidant
CETP
GSK-3
Melatonin Receptor
Rho
Leukotriene Receptor
Caspase
IRE1
UGT
Na-K-Cl cotransporter
Integrase
CCR
CXCR
Somatostatin
Xanthine Oxidase
Thrombopoietin Receptor
Beta-Secretase
PGE Synthase
Glutathione reductase
Free radical scavengers
Ephrin Receptor
GluCls
RSV
Beta Amyloid
Kras
c-Fms
Oxytocin Receptor
Adenosine Deaminase
CGRP Receptor
Gap Junction Protein
Syk
Ras
Protease-activated Receptor
BTK
NPC1L1
Hydrogenase
RAR/RXR
ROR
DNA-PK
p38 MAPK
YAP
IFNAR
JNK
gp120/CD4
TOPK
VDA
PKA
Wnt/beta-catenin
Serine Protease
CSF-1R
IAP
Myosin
Adiponectin Receptor
MTH1
GRK
Glucagon Receptor
P2X Receptor
GlyT
Glucosidase
Hexokinase
PROTAC Linker
HCN Channel
FAAH
ACK1
Bradykinin Receptor
Angiotensin-converting Enzyme (ACE)
Chk
Epigenetic Reader Domain
DUB
Telomerase
TGF-beta/Smad
ATP Citrate Lyase
Lipid
MAPK
OAT
STING
Pyroptosis
IκB/IKK
CRISPR/Cas9
PDK
Aquaporin
PLK
Platelet aggregation
Anti-infection
NADPH-oxidase
Tyrosinase
NOD-like Receptor (NLR)
PKM
Vitamin

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