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TargetMol | Compound Library

FDA 上市药物库现货

FDA-Approved Drug Library

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产品编号 L4200

FDA 上市药物库中的所有化合物都具有良好的生物活性、明确的靶点信息,较好的安全性和生物利用度,这些特性可显著加速药物开发和优化,是进行小分子细胞诱导分化和药物重定位理想的工具。详尽的数据资料可以帮助科学家快速完成药物筛选或细胞诱导机制的判断,并为深入揭示其机制机理创造条件。

TargetMol 的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。

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产品编号 L4200

FDA 上市药物库

规格

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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产品描述 产品描述

  • 1840个FDA批准药物的独特集合,可用于高通量筛选和高内涵筛选;
  • 全部得到FDA批准,提供FDA批准编号,用于药物重定位、新的药物靶点筛选的有效工具;
  • 经过了严格的临床前研究和临床试验,生物活性和安全性得到保障;
  • 涵盖多个研究领域:肿瘤、心血管药物、抗炎、免疫、神经系统药物、呼吸系统药物等;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

Packaging And Storage | TargetMol 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。

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Library Customization | TargetMol 化合物库组成

Antibacterial
Antibiotic
Autophagy
Apoptosis
Endogenous Metabolite
Adrenergic Receptor
5-HT Receptor
AChR
Histamine Receptor
Dopamine Receptor
HIV Protease
Sodium Channel
COX
Antifungal
Parasite
Potassium Channel
DNA/RNA Synthesis
Glucocorticoid Receptor
Estrogen/progestogen Receptor
Calcium Channel
Topoisomerase
Cytochromes P450
Ferroptosis
RAAS
SARS-CoV
Serotonin Transporter
VEGFR
Mitophagy
PDE
ribosome
Microtubule Associated
Dehydrogenase
Estrogen Receptor/ERR
c-Kit
Norepinephrine
HCV Protease
Nucleoside Antimetabolite/Analog
Reverse Transcriptase
GABA Receptor
Antifection
EGFR
Progesterone Receptor
PDGFR
HSV
PPAR
Proton pump
ADC Cytotoxin
Reactive Oxygen Species
Influenza Virus
ATPase
Carbonic Anhydrase
HBV
JAK
Androgen Receptor
DNA Alkylator/Crosslinker
Cholinesterase (ChE)
Prostaglandin Receptor
FLT
Src
Phosphatase
MAO
FGFR
Thrombin
Proteasome
Adenosine Receptor
Bcr-Abl
NF-κB
Thyroid hormone receptor(THR)
c-Met/HGFR
MRP
Tyrosine Kinases
Raf
ROS
HDAC
HMG-CoA Reductase
Transferase
DHFR
Virus Protease
PARP
Antifolate
ALK
c-RET
Monoamine Oxidase
PI3K
GNRH Receptor
TRP/TRPV Channel
iGluR
Drug Metabolite
Opioid Receptor
MMP
SGLT
ABC Transporter
mTOR
P-gp
Retinoid Receptor
NO Synthase
P2Y Receptor
Factor Xa
PKC
CDK
NMDAR
DNA gyrase
Guanylate cyclase
DPP-4
Endothelin Receptor
GluR
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STAT
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LPL Receptor
DNA Alkylation
IL Receptor
TLR
Trk receptor
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TNF
S1P Receptor
HER
Histone Methyltransferase
Integrin
NADPH
Monoamine Transporter
Hedgehog/Smoothened
Vasopressin Receptor
Lipoxygenase
Antiviral
Nrf2
AMPK
Neurokinin receptor
TAM Receptor
ROS Kinase
CFTR
Reductase
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ERK
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Molecular Glues
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Interleukin
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HIF
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NOS
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CaSR
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Cysteine Protease
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MT Receptor
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IGF-1R
DNA
Akt
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GST
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CRM1
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Ligands for Target Protein for PROTAC
Arginase
Antioxidant
CETP
GSK-3
Melatonin Receptor
Rho
Leukotriene Receptor
Vitamin
Caspase
IRE1
UGT
Na-K-Cl cotransporter
Integrase
CCR
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Somatostatin
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Beta-Secretase
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NPC1L1
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DNA-PK
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YAP
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Adiponectin Receptor
MTH1
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GlyT
Glucosidase
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FAAH
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ACK1
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Chk
Epigenetic Reader Domain
DUB
TGF-beta/Smad
Telomerase
Lipid
ATP Citrate Lyase
MAPK
OAT
STING
Pyroptosis
IκB/IKK
CRISPR/Cas9
PDK
Aquaporin
PLK
Platelet aggregation
Anti-infection
NADPH-oxidase
Tyrosinase
NOD-like Receptor (NLR)

Keywords