LUF5771

Name: LUF5771
Brand: TargetMol
SKU: T61307
Price: 186 USD
Availability: InStock
Rating: 4.5 (1 reviews)

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产品编号 T61307Cas号 1141802-49-4

LUF5771 is a highly potent allosteric inhibitor of recombinant luteinizing hormone (recLH) and Org 43553. It exhibits partial activation of the LH receptor with low efficacy [1].

LUF5771

还可以

产品编号 T61307Cas号 1141802-49-4

LUF5771 is a highly potent allosteric inhibitor of recombinant luteinizing hormone (recLH) and Org 43553. It exhibits partial activation of the LH receptor with low efficacy [1].

规格	价格	库存
2 mg	¥ 497	5日内发货
5 mg	¥ 869	5日内发货
1 mL x 10 mM (in DMSO)	¥ 913	5日内发货

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产品介绍

生物活性

产品描述	LUF5771 is a highly potent allosteric inhibitor of recombinant luteinizing hormone (recLH) and Org 43553. It exhibits partial activation of the LH receptor with low efficacy [1].
体外活性	LUF5771 (1 μM or 10 μM) allosteric inhibition is concentration-dependent. LUF5771 significantly increases radioligand dissociation. LUF5771 probably binds to the seven transmembrane domain like Org 43553 does. LUF5771 (10 μM) alone is able to partially activate the LH receptor by 31±4% [1].