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TargetMol | Compound Library

抗乳腺癌化合物库现货

Anti-Breast Cancer Compound Library

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产品编号 L2191

乳腺癌是乳腺恶性肿瘤,是全球女性发病率较高的癌症,约占女性癌症患者的20%,也是100多个国家癌症死亡的主要原因。近年来全球乳腺癌发病率一直呈上升趋势。 乳腺癌根据病理分型可分为非浸润性癌,早期浸润性癌,浸润性癌。根据分子分型可分为雌激素受体阳性乳腺癌(ER+PR+HER2-),HER2阳性乳腺癌(ER-PR-HER2+),三阴性乳腺癌(ER-PR-HER2-)。不同类型的乳腺癌,从治疗方法到预后都是非常不同,需要针对已经明确的致癌位点,探索相关靶点来设计相应的药物。 TargetMol 抗乳腺癌库收集了2440 种与乳腺癌相关的化合物,包含了已经报道的有乳腺癌治疗作用的化合物,以及相关的靶点通路(HER-2, VEGF, EGFR, PARP, CDK4/6, HSP, PD-1, SET7/9, BRCA 等),是乳腺癌药物研发的良好工具。

TargetMol 的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
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产品编号 L2191

抗乳腺癌化合物库

规格

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品描述 产品描述

  • 2440种与乳腺癌相关的化合物,可以用于抗乳腺癌药物研发和药理研究;
  • 靶点包含HER-2, VEGF, EGFR, PARP, CDK4/6, HSP, PD-1, SET7/9, BRCA等;
  • 部分化合物已上市或已进入临床期;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

Packaging And Storage | TargetMol 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。

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Library Customization | TargetMol 化合物库组成

Apoptosis
Autophagy
NF-κB
PI3K
CDK
EGFR
Reactive Oxygen Species
VEGFR
COX
PPAR
mTOR
Akt
Endogenous Metabolite
HDAC
PARP
AMPK
GSK-3
FGFR
Antibacterial
HSP
TGF-beta/Smad
PDGFR
ERK
Estrogen/progestogen Receptor
FLT
c-Kit
Src
Estrogen Receptor/ERR
IκB/IKK
DNA-PK
Parasite
TNF
DNA/RNA Synthesis
HER
p38 MAPK
Wnt/beta-catenin
STAT
Progesterone Receptor
S6 Kinase
Antioxidant
ATM/ATR
Antibiotic
Ferroptosis
Caspase
IL Receptor
HIV Protease
ALK
c-Met/HGFR
RIP kinase
Microtubule Associated
JNK
PKC
Influenza Virus
PDK
NOD
Calcium Channel
Gamma-secretase
Aurora Kinase
Cytochromes P450
Antifungal
JAK
PD-1/PD-L1
Topoisomerase
c-RET
Mitophagy
PKA
Bcr-Abl
Bcl-2 Family
IRAK
NO Synthase
Raf
ROS
Lipoxygenase
IGF-1R
PI4K
Dehydrogenase
MAPK
MEK
NOS
Prostaglandin Receptor
Potassium Channel
p53
MMP
Nrf2
Phosphatase
Virus Protease
Tyrosine Kinases
Chk
Casein Kinase
Tyrosinase
FAK
NOD-like Receptor (NLR)
Mitochondrial Metabolism
Epigenetic Reader Domain
Beta Amyloid
TAM Receptor
TRP/TRPV Channel
PDE
Androgen Receptor
c-Fms
GABA Receptor
AChR
HIF/HIF Prolyl-Hydroxylase
HCV Protease
P-gp
Sirtuin
Aromatase
Drug Metabolite
HSV
PTEN
Interleukin
TLR
Trk receptor
Histone Methyltransferase
Nucleoside Antimetabolite/Analog
SIK
transporter
5-HT Receptor
Syk
Sodium Channel
Ras
PROTACs
Carbonic Anhydrase
Serine/threonin kinase
ROCK
PGE Synthase
Antiviral
MELK
GPR
PLK
HIF
Proteasome
DYRK
Histone Demethylase
NADPH
Tie-2
Pim
Serine Protease
Adrenergic Receptor
Glucocorticoid Receptor
E1/E2/E3 Enzyme
Antifection
Opioid Receptor
Fatty Acid Synthase
Cholinesterase (ChE)
CaMK
Cannabinoid Receptor
Anti-infection
ATPase
Chloride channel
Transferase
ADC Cytotoxin
Integrin
RAAS
Histamine Receptor
Rho
PYK2
MAO
Aryl Hydrocarbon Receptor
CSF-1R
IAP
Glucosidase
Hedgehog/Smoothened
SARS-CoV
Free radical scavengers
Ephrin Receptor
Retinoid Receptor
SGK
DHFR
ROR
Adenosine Receptor
BACE
Glutathione Peroxidase
GTPase
MRP
GNRH Receptor
HBV
Leukotriene Receptor
Immunology/Inflammation related
IRE1
LDL
GluR
DUB
Wee1
BCRP
Survivin
Phospholipase
MLK
S1P Receptor
Kinesin
BTK
Mdm2
RAR/RXR
Dopamine Receptor
YAP
DNA Alkylator/Crosslinker
LTR
IFNAR
TOPK
c-Myc
Cholecystokinin Receptor
Hck
Antifolate
Cysteine Protease
Glutaminase
RANKL/RANK
ABC Transporter
DNA Alkylation
FAAH
CCR
CXCR
cAMP
Indoleamine 2,3-Dioxygenase (IDO)
Beta-Secretase
MNK
STING
LRRK2
PAI-1
RSV
GST
GPX
Reverse Transcriptase
Discoidin Domain Receptor (DDR)
AhR
Proton pump
NPC1L1
NUDIX hydrolase
MyD88
LPL Receptor
Reductase
Lipase
PERK
gp120/CD4
Melatonin Receptor
OCT
AAK1
Cell Cycle Arrest
Liver X Receptor
Glucokinase
Myosin
FLAP
UGT
PAFR
Haspin Kinase
GRK
NMDAR
DNA gyrase
Hexokinase
Smo
PROTAC Linker
ACK1
Endothelin Receptor
Somatostatin
Epoxide Hydrolase
KSP
DNA
Telomerase
SGLT
ATP Citrate Lyase
OXPHOS
Glutathione reductase
Acyltransferase
Aminopeptidase
Histone Acetyltransferase
Decarboxylase
cGAS
HuR
Pyroptosis
Ligand for E3 Ligase
CRISPR/Cas9
Adenosine Deaminase
Gap Junction Protein
DAPK
Platelet aggregation
NADPH-oxidase
DNA Methyltransferase
APC/C
Thrombin
Protease-activated Receptor
ROS Kinase
CFTR
Monoamine Oxidase
PKM

Keywords