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Iptacopan (LNP023) 是一种与factor B 亲和力较高的抑制剂。
Iptacopan (LNP023) 是一种与factor B 亲和力较高的抑制剂。
规格 | 价格 | 库存 | 数量 |
---|---|---|---|
1 mg | ¥ 1,180 | 现货 | |
5 mg | ¥ 2,660 | 现货 | |
10 mg | ¥ 4,320 | 现货 | |
25 mg | ¥ 6,730 | 现货 | |
50 mg | ¥ 8,900 | 现货 | |
100 mg | ¥ 12,200 | 现货 | |
500 mg | ¥ 24,500 | 现货 | |
1 mL x 10 mM (in DMSO) | ¥ 2,920 | 现货 |
产品描述 | Iptacopan (LNP023) is an inhibitor with high affinity for factor B. |
靶点活性 | DPP4:> 100 μM, Cathepsin S:> 30 μM, Cathepsin B:> 100 μM, Cathepsin H:> 100 μM, Cathepsin K:> 100 μM, Caspase-1:> 100 μM, FB:7.9 nM (KD), FB:10 nM, CFB:0.01 μM, 5-LOX:> 30 μM, Apopain:> 100 μM, COX-2 receptor:> 30 μM, Chymase:> 100 μM, Cathepsin G:> 100 μM, CFB:0.012 μM, DPP2:> 100 μM, Blood-coagulation factor Xa:> 100 μM, COX-1 receptor:> 30 μM, Caspase-8:> 100 μM, Cathepsin L:48 μM, Chymotrypsin:> 100 μM |
别名 | LNP023 |
分子量 | 422.52 |
分子式 | C25H30N2O4 |
CAS No. | 1644670-37-0 |
存储 | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
溶解度信息 | DMSO: 55 mg/mL (130.17 mM), Sonication is recommended. | |||||||||||||||||||||||||||||||||||
溶液配制表 | ||||||||||||||||||||||||||||||||||||
DMSO
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