购物车
  • 全部删除
  • TargetMol
    您的购物车当前为空
TargetMol | Compound Library

抗纤维化化合物库现货

Anti-Fibrosis Compound Library

Rating icon 很棒
产品编号 L9810

纤维化(fibrosis)是一种病理改变,主要表现为器官组织内纤维结缔组织增多,实质细胞减少,持续进展可致器官结构破坏和功能减退,乃至衰竭,严重威胁人类健康和生命。纤维化可发生于多种器官,常见的包括肺脏、肝脏、肾脏、骨髓等。纤维化通常由各种刺激导致的慢性炎症性反应引起,包括:持续性感染,自身免疫反应,过敏性反应,化学刺激,射线和组织损伤等。

TargetMol 抗纤维化化合物库收集了1800 种抗纤维化分子和潜在的抗纤维化分子,包括相关靶点如TGFβ、TNFα、MMP 的抑制剂、抗氧化剂及抗炎分子等,是研究纤维化机制和开发抗纤维化药物的良好工具。

TargetMol 的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
资源下载
化合物库相关信息
Excel
SDF
联系我们获取更多批次信息

产品编号 L9810

抗纤维化化合物库

规格

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品特性 产品特性

  • 1800种潜在的抗纤维化分子,是研究纤维化的有效工具,可以用于高通量筛选和高内涵筛选;
  • 靶点包括TGFβ、TNFα、MMP、EGFR、NADPH-oxidase等;
  • 部分化合物已经得到FDA批准上市;?
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

Packaging And Storage | TargetMol 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。

使用TargetMol产品
发表顶级期刊文献

引用更多关于TargetMol产品的科学文献吧!

查看更多

SCI 文献

Library Customization | TargetMol 化合物库定制

Compound Library | TargetMol
您可以通过点击按钮
定制您专属的化合物!
联系专属定制

Library Customization | TargetMol 化合物库组成

Apoptosis
Autophagy
NF-κB
PI3K
Reactive Oxygen Species
COX
VEGFR
Endogenous Metabolite
PDGFR
MMP
mTOR
p38 MAPK
Antioxidant
Akt
ERK
Wnt/beta-catenin
Antibacterial
TNF
AMPK
Raf
TGF-beta/Smad
GSK-3
c-Kit
CDK
JNK
FGFR
Ras
FLT
MEK
IκB/IKK
Src
IL Receptor
DNA-PK
MAPK
Parasite
EGFR
CFTR
Antibiotic
S6 Kinase
ALK
STAT
Ferroptosis
Caspase
JAK
ATM/ATR
NO Synthase
Mitophagy
HIV Protease
Antifungal
Calcium Channel
Hedgehog/Smoothened
Influenza Virus
RIP kinase
Bcr-Abl
NOD
Aurora Kinase
PPAR
PKC
Cytochromes P450
PDK
c-Met/HGFR
DNA/RNA Synthesis
ROS
Lipoxygenase
c-RET
Interleukin
Bcl-2 Family
IRAK
Mitochondrial Metabolism
Nrf2
PKA
Rho
PDE
NOD-like Receptor (NLR)
Potassium Channel
NOS
Dehydrogenase
Virus Protease
Tyrosine Kinases
IGF-1R
Casein Kinase
c-Fms
Tyrosinase
ROCK
Topoisomerase
MLK
Cholinesterase (ChE)
P-gp
Prostaglandin Receptor
Trk receptor
Beta Amyloid
PI4K
AChR
HIF/HIF Prolyl-Hydroxylase
FAK
HSV
PGE Synthase
TLR
HDAC
Syk
p53
Kras
ATPase
NADPH
Glutathione Peroxidase
TRP/TRPV Channel
Adrenergic Receptor
E1/E2/E3 Enzyme
Smo
Chk
Antiviral
GABA Receptor
Sodium Channel
Chloride channel
HCV Protease
Integrin
Adenosine Receptor
BACE
RAAS
Phosphatase
Serine Protease
Drug Metabolite
Glucosidase
PTEN
Epigenetic Reader Domain
MNK
SARS-CoV
HER
Proteasome
Carbonic Anhydrase
Transferase
Estrogen/progestogen Receptor
Tie-2
TOPK
Estrogen Receptor/ERR
PARP
CSF-1R
SIK
HSP
Porcupine
Free radical scavengers
Ephrin Receptor
transporter
ASK
Ligand for E3 Ligase
ribosome
LPA Receptor
GPR
Phospholipase
5-HT Receptor
Anti-infection
TAM Receptor
Monoamine Oxidase
S1P Receptor
LPL Receptor
Reductase
c-Myc
MRP
HBV
Serine/threonin kinase
Aryl Hydrocarbon Receptor
IAP
Immunology/Inflammation related
LDL
Molecular Glues
Opioid Receptor
CCR
LRRK2
Retinoid Receptor
KLF
HIF
PLK
SGK
NADPH-oxidase
Mdm2
Proton pump
Histone Methyltransferase
LTR
Histamine Receptor
GTPase
Cysteine Protease
FXR
Leukotriene Receptor
RANKL/RANK
MAO
Glucocorticoid Receptor
IRE1
UGT
Gamma-secretase
DNA gyrase
Antifection
DNA Alkylation
ACK1
CaMK
Lipid
Beta-Secretase
Acyltransferase
Aminopeptidase
Sirtuin
PAI-1
MELK
GST
Cannabinoid Receptor
Gap Junction Protein
Microtubule Associated
AhR
BTK
PROTACs
Adenylyl Cyclase
GSNOR
Monocarboxylate transporter
NPC1L1
RAR/RXR
DHFR
ROR
Dynamin
MyD88
YAP
Arginase
IFNAR
DYRK
Histone Demethylase
PERK
gp120/CD4
Galectin
N-Acetylglucosaminyltransferase
Cholecystokinin Receptor
AAK1
Hck
Cell Cycle Arrest
Liver X Receptor
PYK2
Amylase
iGluR
Myosin
Haspin Kinase
P2X Receptor
ABC Transporter
Anion Exchanger
Guanylate cyclase
Fatty Acid Synthase
PAK
FAAH
Somatostatin
PAD
cAMP
GluR
DNA
DUB
Indoleamine 2,3-Dioxygenase (IDO)
SGLT
ATP Citrate Lyase
BCRP
OXPHOS
Glutathione reductase
STING
Histone Acetyltransferase
cGAS
Pyroptosis
RSV
Methionine Adenosyltransferase (MAT)
Hippo pathway
GPX
Reverse Transcriptase
Aromatase
CRISPR/Cas9
Hydroxylase
Adenosine Deaminase
Discoidin Domain Receptor (DDR)
Platelet aggregation
BMI-1
Thrombin
PD-1/PD-L1
PKM
ADC Cytotoxin

Keywords