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5-HT1A/5-HT7受体拮抗剂(5-HT1A Ki=8 nM,Kb=0.04 nM;5-HT7 Ki=451 nM,Kb=460 nM)具有 PDE4B/PDE7A 抑制活性(PDE4BIC50=80.4μM;PDE7AIC50=151.3μM),其抗抑郁样作用强于作为参考活性分子的依西酞普兰。
5-HT1A/5-HT7受体拮抗剂(5-HT1A Ki=8 nM,Kb=0.04 nM;5-HT7 Ki=451 nM,Kb=460 nM)具有 PDE4B/PDE7A 抑制活性(PDE4BIC50=80.4μM;PDE7AIC50=151.3μM),其抗抑郁样作用强于作为参考活性分子的依西酞普兰。
规格 | 价格 | 库存 | 数量 |
---|---|---|---|
25 mg | ¥ 10,600 | 10-14周 | |
50 mg | ¥ 13,800 | 10-14周 | |
100 mg | ¥ 17,500 | 10-14周 |
产品描述 | This compound is a dual 5-HT1A/5-HT7 receptor antagonist (5-HT1A Ki = 8 nM, Kb = 0.04 nM; 5-HT7 Ki = 451 nM, Kb = 460 nM) with additional inhibitory activity against PDE4B/PDE7A (PDE4B IC50 = 80.4 μM; PDE7A IC50 = 151.3 μM). Its antidepressant-like effect surpasses that of the reference agent, escitalopram. |
分子量 | 409.56 |
分子式 | C25H35N3O2 |
CAS No. | 2511632-55-4 |
存储 | Shipping with blue ice. |
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