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TargetMol | Compound Library

抗癌化合物库现货

Anti-Cancer Compound Library

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产品编号 L2100

在过去的几十年中癌症的研究和治疗取得了巨大的成功,但癌症仍然是人类面临的巨大挑战,给患者身心健康带来巨大的痛苦。癌细胞具有许多显著不同的生物学特征,表现出无限的增殖潜能,维持自身生长信号的持续稳定,逃避应激信号(例如治疗药物)诱导的细胞凋亡,刺激血管生长,为肿瘤提供营养,同时逃避免疫系统防御和诱导局部慢性炎症,发挥其侵袭和转移能力,表现出异常的代谢活动,并通过突变和表观遗传机制显著改变全基因组的稳定性。 我们根据上述癌细胞显著不同的特征和异常的代谢活动,精心筛选了 9019 个肿瘤相关的小分子化合物,这些化合物都是调节肿瘤细胞代谢、增殖、侵袭、转移通路上的小分子,可用于肿瘤相关的研究以及抗肿瘤药物的筛选,可用于高通量、高内涵筛选。

TargetMol 的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。

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产品编号 L2100

抗癌化合物库

规格

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品描述 产品描述

  • 9019种肿瘤相关的生物活性小分子化合物的特有集合,用于高通量、高内涵筛选;
  • 产品经过临床验证和临床实验,具有生物安全保障和一定的生物活性;
  • 是肿瘤发生机理研究、抗肿瘤药物筛选的有效工具;?
  • 靶点含PI3K、HDAC、mTOR、CDK、Aurora Kinase、JAK等;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS检测技术保证产品高纯度和高质量,减少假阳性发生概率。

Packaging And Storage | TargetMol 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。

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Library Customization | TargetMol 化合物库定制

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Library Customization | TargetMol 化合物库组成

Apoptosis
Autophagy
5-HT Receptor
Endogenous Metabolite
Antibacterial
NF-κB
COX
DNA/RNA Synthesis
Adrenergic Receptor
CDK
Dopamine Receptor
PI3K
EGFR
Potassium Channel
Reactive Oxygen Species
Histamine Receptor
Calcium Channel
VEGFR
Antibiotic
Cytochromes P450
Sodium Channel
HDAC
GABA Receptor
PPAR
Parasite
TRP/TRPV Channel
mTOR
Akt
GPR
ERK
AChR
JAK
Wnt/beta-catenin
Antifungal
Src
Prostaglandin Receptor
HIV Protease
STAT
FLT
Adenosine Receptor
Estrogen Receptor/ERR
PARP
Opioid Receptor
p38 MAPK
PDGFR
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Dehydrogenase
Nucleoside Antimetabolite/Analog
AMPK
GSK-3
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Epigenetic Reader Domain
TNF
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Bcl-2 Family
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c-Met/HGFR
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Androgen Receptor
Ferroptosis
c-Kit
HSP
Cannabinoid Receptor
Bcr-Abl
PKC
MMP
ALK
ATPase
Sirtuin
TGF-beta/Smad
Phosphatase
Kras
IL Receptor
Ras
Aurora Kinase
PDE
HER
JNK
MAPK
Tyrosine Kinases
MEK
DUB
IκB/IKK
NO Synthase
ROCK
P-gp
ADC Cytotoxin
Mitophagy
p53
ROS
Lipoxygenase
SARS-CoV
Serine/threonin kinase
Virus Protease
NMDAR
CXCR
HIF/HIF Prolyl-Hydroxylase
S1P Receptor
DNA-PK
Hedgehog/Smoothened
HSV
IGF-1R
Neurokinin receptor
PKA
RIP kinase
P2X Receptor
Nrf2
NOD
LPL Receptor
BTK
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S6 Kinase
FAK
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Interleukin
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NOS
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MAO
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transporter
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LPA Receptor
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cholecystokinin
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CaMK
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STING
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PTEN
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MLK
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Ligands for Target Protein for PROTAC
Liver X Receptor
PYK2
Glucokinase
NAMPT
PAFR
MT Receptor
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PSMA
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OAT
CRFR
MELK
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ribosome
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Xanthine Oxidase
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ASK
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PKM
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MALT
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IDO
Adiponectin Receptor
DNA gyrase
Hexokinase
PAD
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ATP Citrate Lyase
LRRK2
Aminopeptidase
Decarboxylase
TSH Receptor
PAI-1
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Adenosine Deaminase
p97
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GlyT
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PROTAC Linker
Thioredoxin
Stearoyl-CoA Desaturase (SCD)
Angiotensin-converting Enzyme (ACE)
Thrombopoietin Receptor
cGAS
hCE
Neprilysin

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