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TargetMol | Compound Library

抗感染化合物库现货

Anti-Infection Compound Library

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产品编号 L1800

当外来生物进入人体并造成伤害时就会发生感染,这些引起感染的外来生物称为病原体,例如细菌、病毒、真菌和寄生虫等。有些感染是轻微的几乎不可察觉,但有些感染严重甚至危及生命,且对治疗有抵抗力。

针对上述情况,TargetMol 精选了3260 种具有抗菌、抗病毒以及抗寄生虫等抗感染活性的化合物的组成抗感染化合物库,以用于抗感染研究中的药物高通量筛选、确认药物靶点以及其他医药研发和科研领域。

TargetMol 的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
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产品编号 L1800

抗感染化合物库

规格

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品描述 产品描述

  • 3260种具有抗感染活性的化合物的特有集合,包括抗细菌、抗真菌、抗巨细胞病毒、抗HIV、抗SARS、抗流感等活性;
  • 含有磺胺类,氨基糖苷类,四环素类和大环内酯类等化合物,是筛选新型抗感染药的有效工具;可用于高通量筛选和高内涵筛选;
  • 通过前期临床研究和临床实验,生物活性和安全性已经得到验证;其中一些抗感染化合物已得到FDA批准上市;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

包装和储存 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
  • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。

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Library Customization | TargetMol 化合物库组成

Antibacterial
Antibiotic
Antifungal
Parasite
HIV Protease
Autophagy
Apoptosis
Endogenous Metabolite
Influenza Virus
Antiviral
DNA/RNA Synthesis
SARS-CoV
HCV Protease
Virus Protease
HBV
NF-κB
HSV
Anti-infection
Nucleoside Antimetabolite/Analog
Topoisomerase
Antifection
Antioxidant
COX
Cytochromes P450
Reactive Oxygen Species
Reverse Transcriptase
Dehydrogenase
Histamine Receptor
ribosome
Mitophagy
AChR
Cholinesterase (ChE)
Potassium Channel
STAT
TLR
Dopamine Receptor
Ferroptosis
GABA Receptor
Adenosine Receptor
Calcium Channel
IL Receptor
PKC
Phosphatase
TNF
5-HT Receptor
p38 MAPK
ROS
Sodium Channel
TRP/TRPV Channel
ATPase
Caspase
Microtubule Associated
MMP
PI3K
Akt
Proton pump
RSV
Adrenergic Receptor
AMPK
CDK
HDAC
PPAR
Tyrosinase
PDE
Drug Metabolite
EGFR
Estrogen/progestogen Receptor
HSP
Phospholipase
Bcl-2 Family
NO Synthase
NOS
PARP
Src
DNA gyrase
ERK
Glucocorticoid Receptor
JAK
Nrf2
VEGFR
CCR
CXCR
Estrogen Receptor/ERR
Mitochondrial Metabolism
Wnt/beta-catenin
Bcr-Abl
DHFR
HIF/HIF Prolyl-Hydroxylase
JNK
Lipoxygenase
P-gp
PKA
Cysteine Protease
Fatty Acid Synthase
Glucosidase
Interleukin
MAO
mTOR
PDGFR
Serine Protease
Transferase
Beta Amyloid
CaMK
Carbonic Anhydrase
DNA Methyltransferase
Epigenetic Reader Domain
Immunology/Inflammation related
Proteasome
Antifolate
ATM/ATR
c-Kit
Histone Methyltransferase
Retinoid Receptor
S1P Receptor
TGF-beta/Smad
DUB
FLT
Gamma-secretase
Histone Demethylase
IκB/IKK
Monoamine Oxidase
NADPH
NMDAR
PI4K
Sirtuin
STING
Thrombin
Tyrosine Kinases
ABC Transporter
Chloride channel
DNA
DprE1
Glucokinase
GSK-3
Hedgehog/Smoothened
HIF
HMG-CoA Reductase
IFNAR
MEK
NADPH-oxidase
Opioid Receptor
P2Y Receptor
p97
PERK
Reductase
Serine/threonin kinase
Xanthine Oxidase
ADC Cytotoxin
Acetyl-CoA Carboxylase
Acyltransferase
Adenosine Deaminase
Aminopeptidase
Amylase
Aurora Kinase
Cannabinoid Receptor
Casein Kinase
Cell wall
c-Met/HGFR
DNA-PK
Free radical scavengers
GPCR
Lipid
Liver X Receptor
MAPK
MicroRNA
Monoamine Transporter
P2X Receptor
p53
Prostaglandin Receptor
Raf
RIP kinase
S6 Kinase
Syk
Telomerase
transporter
AhR
Androgen Receptor
Arginase
BCRP
cAMP
Chk
CRISPR/Cas9
FAAH
FAK
FGFR
gp120/CD4
IGF-1R
iGluR
Indoleamine 2,3-Dioxygenase (IDO)
LPL Receptor
MRP
Norepinephrine
Platelet aggregation
Pyroptosis
Ras
Serotonin Transporter
Amino Acids and Derivatives
Annexin A
Aromatase
BACE
Complement System
CRM1
DNA Alkylation
DNA Alkylator/Crosslinker
Dynamin
Factor Xa
GluCls
Glutathione Peroxidase
Guanylate cyclase
Histone Acetyltransferase
IAP
Integrase
Integrin
Leukotriene Receptor
LTR
MNK
NOD
NOD-like Receptor (NLR)
PAK
PD-1/PD-L1
PGE Synthase
PKM
Progesterone Receptor
Stearoyl-CoA Desaturase (SCD)
Thyroid hormone receptor(THR)
UGT
BTK
ACK1
Adiponectin Receptor
Advanced Glycation End Products
ALK
Aryl Hydrocarbon Receptor
ATP Citrate Lyase
ATTECs
Beta-Secretase
BMI-1
Bombesin Receptor
CFTR
CGRP Receptor
c-Myc
CSF-1R
Decarboxylase
E1/E2/E3 Enzyme
EBI2/GPR183
Endothelin Receptor
Ephrin Receptor
Epoxide Hydrolase
FKBP
FXR
Gap Junction Protein
GluR
Glutaminase
Glutathione reductase
GlyT
GNRH Receptor
GPX
GST
Hck
Hexokinase
Hydrogenase
Hydroxylase
IRAK
IRE1
LDL
Ligands for Target Protein for PROTAC
LIM Kinase
Lipase
MAGL
Mdm2
Molecular Glues
Monocarboxylate transporter
MTH1
Myosin
Na-K-Cl cotransporter
Neurokinin receptor
OCT
PDK
PLK
Porcupine
Protease-activated Receptor
PTEN
RAAS
Rho
ROCK
SGK
SGLT
Sigma receptor
Somatostatin
TAM Receptor
Thrombopoietin Receptor
TOPK
Transketolase
Trk receptor
VDA
YAP

Keywords