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规格 | 价格 | 库存 | 数量 |
---|---|---|---|
1 mg | ¥ 1,130 | 现货 | |
5 mg | ¥ 2,810 | 现货 | |
10 mg | ¥ 4,000 | 现货 | |
25 mg | ¥ 5,880 | 现货 | |
50 mg | ¥ 7,980 | 现货 | |
100 mg | ¥ 10,700 | 现货 | |
200 mg | ¥ 14,300 | 现货 |
产品描述 | M40 acetate is a potent, non-selective galanin receptor antagonist (Ki values are 1.82 and 5.1 nM at GAL1 and GAL2 respectively) that inhibits galanin (1-29) binding in rat brain in vitro (IC50 = 3 - 15 nM). Attenuates the antidepressant effects of fluoxetine and blocks galanin-induced food intake in vivo. Also exhibits weak partial agonist activity at peripheral GAL2 receptors at doses > 100 nM. |
分子量 | 2041.38 |
分子式 | C96H149N23O26 |
CAS No. |
存储 | keep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | ||||||||||||||||||||
溶解度信息 | DMSO: 10 mM | ||||||||||||||||||||
溶液配制表 | |||||||||||||||||||||
DMSO
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