Arzoxifene

Name: Arzoxifene
Brand: TargetMol
SKU: T39259
Price: 655 USD
Availability: InStock
Rating: 4.5 (1 reviews)

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产品编号 T39259Cas号 182133-25-1

别名 SERMIII, LY353381, Arzoxifene

Arzoxifene (LY353381) is an orally active selective estrogen receptor modulator (SERM) exhibiting a fixed ring structure analogous to raloxifene. This compound demonstrates potent antiestrogenic effects on breast cancer and endometrium while displaying minimal side effects. Additionally, Arzoxifene elicits favorable estrogenic effects on bone health and lipid profile.

Arzoxifene

还可以

产品编号 T39259 别名 SERMIII, LY353381, ArzoxifeneCas号 182133-25-1

规格	价格	库存	数量
25 mg	¥ 10,600	6-8周

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产品介绍

生物活性

产品描述	Arzoxifene (LY353381) is an orally active selective estrogen receptor modulator (SERM) exhibiting a fixed ring structure analogous to raloxifene. This compound demonstrates potent antiestrogenic effects on breast cancer and endometrium while displaying minimal side effects. Additionally, Arzoxifene elicits favorable estrogenic effects on bone health and lipid profile.
体外活性	Arzoxifene reduces estrogen receptor expression in endometrial cancer cell lines (ECC-1)[1].
体内活性	Arzoxifene inhibits MCF-7 breast cancer xenograft growth in oophorectomized athymic mice. Arzoxifene is reported to prevent body weight increase in oophorectomized rats[1].
别名	SERMIII, LY353381, Arzoxifene