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TargetMol | Compound Library

非甾体类抗炎化合物库现货

Nonsteroidal Anti-Inflammatory Compound Library

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产品编号 L4710

非甾体抗炎药(Nonsteroidal Antiinflammatory Drugs,NSAIDs)是一类不含皮质激素甾体结构的抗炎药,NSAIDs 自阿司匹林于1898年首次合成后,100多年来已有百余种上千个品牌上市,这类药物包括阿司匹林、对乙酰氨基酚、吲哚美辛、萘普生、萘普酮、双氯芬酸、布洛芬、尼美舒利、罗非昔布、塞来昔布等,该类药物通过抑制环氧化酶、减少前列腺素的合成,从而发挥抗炎、抗风湿、止痛、退热和抗凝血等作用,在临床上广泛用于骨关节炎、类风湿性关节炎、多种发热和各种疼痛症状的缓解。 TargetMol 非甾体类抗炎化合物库收集了609 种非甾体类的抗炎相关化合物,可用于抗炎相关的药理研究和药物开发。

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产品编号 L4710

非甾体类抗炎化合物库

规格

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品描述 产品描述

  • 609种非甾体类的抗炎相关化合物,可用于高通量和高内涵筛选;
  • 包含常见非甾体抗炎药活性成分,如阿司匹林、吲哚美辛、舒林酸、布洛芬、吡罗昔康等;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR和HPLC技术保证产品高纯度。

Packaging And Storage | TargetMol 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。

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Library Customization | TargetMol 化合物库组成

COX
Histamine Receptor
Apoptosis
Autophagy
Antibacterial
NF-κB
IL Receptor
ROS
TNF
Reactive Oxygen Species
Lipoxygenase
NOS
TLR
Endogenous Metabolite
Antioxidant
Interleukin
Antiviral
Parasite
NO Synthase
Prostaglandin Receptor
Antibiotic
PPAR
CXCR
Influenza Virus
Antifungal
CCR
Cytochromes P450
PGE Synthase
5-HT Receptor
HIV Protease
Ferroptosis
Virus Protease
Adrenergic Receptor
MRP
ERK
Nrf2
Potassium Channel
AChR
Dopamine Receptor
p38 MAPK
NOD
AhR
LTR
TRP/TRPV Channel
Aryl Hydrocarbon Receptor
STAT
Phospholipase
Norepinephrine
STING
IRAK
NOD-like Receptor (NLR)
NADPH
Mitophagy
Wnt/beta-catenin
Calcium Channel
PDE
Antifection
JAK
Xanthine Oxidase
SARS-CoV
IκB/IKK
HCV Protease
Estrogen/progestogen Receptor
Glutathione Peroxidase
HBV
Caspase
Akt
DNA/RNA Synthesis
AMPK
Sodium Channel
NADPH-oxidase
Chloride channel
ATPase
Dehydrogenase
IFNAR
Reductase
JNK
Tyrosine Kinases
Leukotriene Receptor
iGluR
Immunology/Inflammation related
Drug Metabolite
MMP
Bcl-2 Family
Retinoid Receptor
HDAC
Carbonic Anhydrase
PI3K
Adenosine Receptor
Cell wall
gp120/CD4
Phosphatase
Progesterone Receptor
Estrogen Receptor/ERR
MAO
UGT
Gamma-secretase
Raf
Opioid Receptor
HSV
CaMK
Acyltransferase
Aminopeptidase
Free radical scavengers
transporter
ALK
ribosome
Gap Junction Protein
S6 Kinase
Tyrosinase
FAK
ROS Kinase
PD-1/PD-L1
Proteasome
Transferase
NPC1L1
Monocarboxylate transporter
MALT
Histone Methyltransferase
Src
Amino Acids and Derivatives
RAAS
Lipase
GSK-3
Galectin
N-Acetylglucosaminyltransferase
PARP
Cell Cycle Arrest
Cysteine Protease
VEGFR
IAP
Glucocorticoid Receptor
Topoisomerase
FLAP
PAFR
CDK
NMDAR
ABC Transporter
Mitochondrial Metabolism
Monoamine Transporter
Anion Exchanger
PAK
FAAH
Cholinesterase (ChE)
PTEN
Chk
Epoxide Hydrolase
Epigenetic Reader Domain
DNA
mTOR
Androgen Receptor
Telomerase
TGF-beta/Smad
MAPK
P-gp
HSP
Trk receptor
Sirtuin
PAI-1
RSV
Beta Amyloid
Aromatase
GABA Receptor
Hydroxylase
HIF
MEK
FGFR
Platelet aggregation
Syk
Anti-infection
Ras
Thrombin
p53
Monoamine Oxidase
HER
BTK

Keywords