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SNT-207858
还可以产品编号 T12946Cas号 1104080-42-3
SNT-207858 is a selective, blood brain barrier penetrating, potent and orally active antagonist of melanocortin-4 (MC-4) receptor. SNT207858 has an IC50 of 22 nM (binding) and 11 nM (function) on the MC-4 receptor.
SNT-207858
还可以产品编号 T12946Cas号 1104080-42-3
SNT-207858 is a selective, blood brain barrier penetrating, potent and orally active antagonist of melanocortin-4 (MC-4) receptor. SNT207858 has an IC50 of 22 nM (binding) and 11 nM (function) on the MC-4 receptor.
| 规格 | 价格 | 库存 | 数量 |
|---|---|---|---|
| 25 mg | ¥ 10,600 | 6-8周 | |
| 50 mg | ¥ 13,800 | 6-8周 | |
| 100 mg | ¥ 17,500 | 6-8周 |
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| 产品描述 | SNT-207858 is a selective, blood brain barrier penetrating, potent and orally active antagonist of melanocortin-4 (MC-4) receptor. SNT207858 has an IC50 of 22 nM (binding) and 11 nM (function) on the MC-4 receptor. |
| 靶点活性 | MC-4 receptor (function):11 nM , MC-4 receptor (binding):22 nM |
| 体外活性 | SNT207858 binds to the MC-4 receptor with an affinity of 22 nM, and shows a 170-fold selectivity vs. MC-3 and a 40-fold selectivity vs. MC-5. |
| 体内活性 | In mice,the tumor induced weight loss significantly reduced by SNT207858 (30 mg/kg; oral administration; once daily; 15 days). |
| 分子量 | 689.54 |
| 分子式 | C32H45Cl4N5O3 |
| CAS No. | 1104080-42-3 |
| 密度 | no data available |
储存&溶解度
| 存储 | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
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比如您的给药剂量是 10 mg/kg ，每只动物体重 20 g ，给药体积 100 μL ， 
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