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TargetMol | Compound Library

神经退行性疾病化合物库现货

Anti-Neurodegenerative Disease Compound Library

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产品编号 L2620

神经退行性疾病是机体神经元结构或功能逐渐丧失而引发的一类疾病,包括肌萎缩侧索硬化症(Amyotrophiclateral sclerosis,ALS)、帕金森病(Parkinson’s disease,PD)、阿尔茨海默病(Alzheimer disease,AD)、亨廷顿氏病(Huntington’s disease,HD)以及脊髓性肌萎缩症(spinal muscular atrophy,SMA)等,目前这类疾病病因尚不明确并无有效治愈手段,且严重威胁着患者的生活质量。 TargetMol 基于目前的研究现状,收集了2154 种与神经退行性疾病相关的化合物,这些化合物或者对神经退行性疾病有一定的疗效,或者作用于神经退行性疾病相关的靶点,可以用于神经退行性疾病相关的药物研发和机制研究。

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产品编号 L2620

神经退行性疾病化合物库

规格

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品描述 产品描述

  • 2154种与神经退行性疾病相关的化合物,可用于高通量和高内涵筛选;
  • 靶点包括AchE, NMDA, CGRP, β-secretase, γ-secretase, Dopamine Receptor, Adenosine Receptor, 5-HT receptor等;
  • 部分化合物已经得到FDA批准上市;
  • 详细的说明书,化合物结构、靶点信息、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

包装和储存 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
  • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。

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Library Customization | TargetMol 化合物库组成

5-HT Receptor
AChR
Dopamine Receptor
Adrenergic Receptor
Apoptosis
Autophagy
GABA Receptor
Endogenous Metabolite
GluR
iGluR
Cholinesterase (ChE)
Histamine Receptor
Opioid Receptor
NMDAR
PDE
Beta Amyloid
Monoamine Oxidase
COX
MAO
Antibacterial
Reactive Oxygen Species
JNK
Serotonin Transporter
NF-κB
Potassium Channel
Gamma-secretase
Parasite
GSK-3
Calcium Channel
Norepinephrine
PPAR
Sodium Channel
Adenosine Receptor
Caspase
Cytochromes P450
TNF
ERK
Nrf2
Influenza Virus
HIV Protease
CDK
CaMK
Akt
LRRK2
Ferroptosis
BACE
Mitophagy
Beta-Secretase
Transferase
Antifungal
Sigma receptor
NO Synthase
PI3K
Phosphatase
Virus Protease
Interleukin
Cannabinoid Receptor
Antibiotic
Dehydrogenase
Mitochondrial Metabolism
Src
p38 MAPK
VEGFR
TRP/TRPV Channel
IL Receptor
MMP
Estrogen/progestogen Receptor
Bcr-Abl
Drug Metabolite
DNA/RNA Synthesis
P-gp
Bcl-2 Family
IκB/IKK
mTOR
SARS-CoV
Phospholipase
Imidazoline Receptor
Antioxidant
Melatonin Receptor
Wnt/beta-catenin
PARP
GlyT
Glucosidase
ROS
Lipoxygenase
Sirtuin
HDAC
AMPK
Anti-infection
Microtubule Associated
Adenylyl Cyclase
MRP
PKC
P2X Receptor
OX Receptor
EGFR
MEK
FLT
c-Kit
Amino Acids and Derivatives
LPL Receptor
P2Y Receptor
PKA
Estrogen Receptor/ERR
AAK1
MT Receptor
FAAH
Aurora Kinase
Epigenetic Reader Domain
MAPK
Prostaglandin Receptor
Trk receptor
Tyrosinase
HIF/HIF Prolyl-Hydroxylase
S1P Receptor
GPCR
NOS
Carbonic Anhydrase
ROR
Histone Methyltransferase
RAAS
AAK1 (AP2 associated kinase 1)
ABC Transporter
HSV
CCR
IGF-1R
Retinoid Receptor
FGFR
Neurokinin receptor
NOD
Ras
HMG-CoA Reductase
NOD-like Receptor (NLR)
Chloride channel
c-Met/HGFR
NADPH
Histone Demethylase
Rho
FXR
Glucocorticoid Receptor
Monoamine Transporter
JAK
PTEN
Epoxide Hydrolase
TGF-beta/Smad
PGE Synthase
Antiviral
Histone Acetyltransferase
transporter
Casein Kinase
c-Fms
MDM-2/p53
S6 Kinase
p53
Advanced Glycation End Products
Transaminase
Monocarboxylate transporter
Integrin
IFNAR
DYRK
MIF
Progesterone Receptor
OCT
HBV
Nucleoside Antimetabolite/Analog
Cysteine Protease
Aryl Hydrocarbon Receptor
CSF-1R
Topoisomerase
UGT
PAFR
Raf
Antifection
Guanylate cyclase
PDGFR
Stearoyl-CoA Desaturase (SCD)
Angiotensin-converting Enzyme (ACE)
DUB
OXPHOS
Acyltransferase
STING
Free radical scavengers
Decarboxylase
RSV
ATM/ATR
Reverse Transcriptase
CRISPR/Cas9
Hydroxylase
CGRP Receptor
Gap Junction Protein
FAK
FOXO3
Thyroid hormone receptor(THR)
Proteasome
ATPase
CAT
NPC1L1
RAR/RXR
HCV Protease
Glutaminyl Cyclase
Na+/Ca2+ Exchanger
Reductase
Arrestin
PERK
Necroptosis
Glutathione Peroxidase
GTPase
c-Myc
CaSR
Serine Protease
Hck
Serine/threonin kinase
Liver X Receptor
Neurotensin Receptor
Glutaminase
ROCK
NR4A
RANKL/RANK
IDO
IAP
Immunology/Inflammation related
Prolyl Endopeptidase (PREP)
Annexin A
E1/E2/E3 Enzyme
Adiponectin Receptor
LDL
GRK
Hexokinase
HCN Channel
Neuropeptide Y Receptor
DNA Alkylation
Bombesin Receptor
PAK
Somatostatin
Chk
PAD
Indoleamine 2,3-Dioxygenase (IDO)
Androgen Receptor
Telomerase
SGLT
ATP Citrate Lyase
OAT
MNK
HSP
TLR
GluCls
PAI-1
Pyroptosis
ALK
Neprilysin
GST
STAT
Aromatase
PDK
HIF
Adenosine Deaminase
Cuproptosis
SGK
REV-ERB
Syk
DNA Methyltransferase
IRAK
Thrombin
Liposome
ROS Kinase
CFTR
MLK
Vitamin
BTK
NMU2R
NMUR

Keywords