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生物碱类天然产物库

生物碱类天然产物库

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产品编号 L6110 Alkaloid Natural Product Library
  库化合物信息   Excel SDF

生物碱是一类活性较强的含氮有机化合物,在中药材中广泛存在,其药用功能逐渐被推广。众多研究发现生物碱的药理活性众多,包括抗肿瘤、抗炎镇痛、抗菌抗病毒、心血管作用、杀虫等。随着对生物碱的深入研究,其将为疾病的治疗提供新的药物来源。

TargetMol 生物碱类天然产物库精选 500 种生物碱类的天然产物,来源包括乌头、长春花、喜树、莨菪、黄连等多种中药材,具有抗肿瘤、抗炎、抗氧化、神经保护等多种功能,例如:从长春花中分离出的生物碱对多种肿瘤细胞有较好的抑制作用,石蒜碱被认为具有很强的抗病毒活性及抗菌作用,延胡乙素等多种异喹啉生物碱具有镇痛活性等。该库可以为从事药物开发和药理研究的客户提供有力工具。

TargetMol的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
TargetMol Compound Library
规格
1 mg
30 μL * 10 mM (in DMSO)
50 μL * 10 mM (in DMSO)
100 μL * 10 mM (in DMSO)
250 μL * 10 mM (in DMSO)
如果上述化合物库无法满足您的需求,您可发送邮件至tech@targetmol.com咨询我们的技术专员,为您量身定制专属化合物库!
咨询化合物库
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产品描述

  • 500种生物碱类天然产物的独特集合,可用于高通量筛选和高内涵筛选;
  • 大部分化合物生物活性明确,具有抗肿瘤、抗炎、抗氧化、神经保护等多种功能;
  • 详细的说明书,化合物结构、靶点信息、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

化合物库定制

TargetMol的化合物可以高度定制! 了解更多

包装和存储

  • 干粉或者DMSO溶液置于带二维码的储存管中,或排列于96孔板/384孔板;
  • 蓝冰运输
获取筛选库化合物信息 (L6110)
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TargetMol Library Books客户使用化合物库发表的文献

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化合物库组成

Apoptosis (55)
Autophagy (50)
Endogenous Metabolite (45)
Antibacterial (35)
AChR (33)
Parasite (28)
NF-κB (25)
AChE (25)
Antifungal (22)
Topoisomerase (15)
Antibiotic (15)
Antioxidant (15)
Influenza Virus (13)
Sodium Channel (13)
5-HT Receptor (12)
Microtubule Associated (12)
Adrenergic Receptor (12)
Potassium Channel (12)
Dopamine Receptor (11)
P450 (11)
Calcium Channel (11)
p38 MAPK (10)
PDE (8)
ADC Cytotoxin (8)
BCL (7)
DNA/RNA Synthesis (7)
ERK (7)
Reactive Oxygen Species (7)
Adenosine Receptor (7)
Virus Protease (6)
P-gp (6)
HIV Protease (6)
Indoleamine 2,3-Dioxygenase (IDO) (6)
Caspase (6)
TNF (6)
STAT (5)
Akt (5)
TRP/TRPV Channel (5)
Anti-infection (5)
COX (5)
TLR (4)
Opioid Receptor (4)
JNK (4)
TGF-beta/Smad (4)
Platelet aggregation (4)
GABA Receptor (4)
IL Receptor (4)
Antifection (3)
ROS (3)
Monoamine Oxidase (3)
AMPK (3)
HDAC (3)
FAK (3)
Antiviral (3)
Drug Metabolite (3)
HER (3)
PARP (3)
Mitophagy (3)
PKC (3)
Ferroptosis (3)
MAO (3)
NOS (3)
Nucleoside Antimetabolite/Analog (3)
Imidazoline Receptor (2)
PKA (2)
HIF (2)
BACE (2)
EGFR (2)
ATPase (2)
PI3K (2)
P2X Receptor (2)
NO Synthase (2)
Serotonin Transporter (2)
Lipoxygenase (2)
cAMP (2)
Aurora Kinase (2)
Dehydrogenase (2)
MMP (2)
RAAS (2)
Beta-Secretase (2)
FAAH (2)
Hedgehog/Smoothened (2)
Prostaglandin Receptor (2)
SARS-CoV (2)
Glucosidase (2)
Smo (2)
iGluR (2)
Histamine Receptor (2)
NADPH (1)
GPR (1)
DYRK (1)
GSK-3 (1)
Arginase (1)
MEK (1)
LPL Receptor (1)
Cannabinoid Receptor (1)
Reverse Transcriptase (1)
FLT (1)
Src (1)
HCV Protease (1)
Hydrogenase (1)
CAT (1)
HIF/HIF Prolyl-Hydroxylase (1)
p53 (1)
S1P Receptor (1)
OCT (1)
CDK (1)
Beta Amyloid (1)
IGF-1R (1)
Bcr-Abl (1)
DNA gyrase (1)
Adiponectin receptor (1)
Monoamine Transporter (1)
E1/E2/E3 Enzyme (1)
Immunology/Inflammation related (1)
Chloride channel (1)
Fatty Acid Synthase (1)
PAK (1)
PDGFR (1)
HSV (1)
Aryl Hydrocarbon Receptor (1)
PAD (1)
DNA (1)
GST (1)
RANKL/RANK (1)
mTOR (1)
VEGFR (1)
BCRP (1)
Cysteine Protease (1)
PGE Synthase (1)
MAPK (1)
cell cycle arrest (1)
Raf (1)
Tyrosine Kinases (1)
MRP (1)
Nrf2 (1)
IκB/IKK (1)
Proteasome (1)

化合物库信息示例

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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