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AR-M 1000390 hydrochloride (ARM-390 HCl) 是选择性 δ 阿片受体激动剂,EC50为 7.2±0.9 nM。
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AR-M 1000390 hydrochloride (ARM-390 HCl) 是选择性 δ 阿片受体激动剂,EC50为 7.2±0.9 nM。
规格 | 价格 | 库存 | 数量 |
---|---|---|---|
1 mg | ¥ 343 | 现货 | |
5 mg | ¥ 822 | 现货 | |
10 mg | ¥ 1,390 | 现货 | |
25 mg | ¥ 2,750 | 现货 | |
50 mg | ¥ 3,970 | 现货 | |
100 mg | ¥ 5,830 | 现货 | |
1 mL x 10 mM (in DMSO) | ¥ 885 | 现货 |
产品描述 | AR-M 1000390 hydrochloride (ARM-390 HCl) , also known as ARM-390, is a low-internalizing nonpeptidic δ-selective opioid receptor agonist; derivative of SNC 80. Does not trigger acute desensitization of the analgesic response; reduces CFA-induced hyperalgesia. Brain penetrant following systemic administration. |
靶点活性 | δ opioid receptor: |
体外活性 | AR-M 1000390 hydrochloride 不会引发镇痛反应的急性脱敏。 |
体内活性 | AR-M 1000390 hydrochloride 降低了CFA诱导的痛觉过敏。系统给药后能穿透血脑屏障。 |
别名 | ARM390 Hydrochloride, ARM-390 HCl |
分子量 | 384.94 |
分子式 | C23H29ClN2O |
CAS No. | 209808-47-9 |
Smiles | Cl.CCN(CC)C(=O)c1ccc(cc1)C(=C1CCNCC1)c1ccccc1 |
密度 | no data available |
存储 | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
溶解度信息 | H2O: 38.49 mg/mL (100 mM) DMSO: 38.49 mg/mL (100 mM) | |||||||||||||||||||||||||||||||||||
溶液配制表 | ||||||||||||||||||||||||||||||||||||
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