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规格 | 价格 | 库存 | 数量 |
---|---|---|---|
1 mg | ¥ 346 | 现货 | |
2 mg | ¥ 513 | 现货 | |
5 mg | ¥ 823 | 现货 | |
10 mg | ¥ 1,360 | 现货 | |
25 mg | ¥ 2,450 | 现货 | |
50 mg | ¥ 3,680 | 现货 | |
100 mg | ¥ 5,280 | 现货 | |
1 mL x 10 mM (in DMSO) | ¥ 981 | 现货 |
产品描述 | Regorafénib N-oxyde M2 is an active metabolite of Regorafenib. Regorafenib is a multi-target inhibitor for VEGFR1/2/3, PDGFRβ, RET, Kit, and Raf-1 (IC50s: 13/4.2/46, 1.5, 22, 7, and 2.5 nM). |
靶点活性 | VEGFR1:13nM , RET:22nM , VEGFR2:4.2nM , c-Kit:7nM , Raf-1:2.5 nM , PDGFRβ:1.5nM , VEGFR3:46nM |
别名 | 瑞戈非尼杂质 13 |
分子量 | 498.81 |
分子式 | C21H15ClF4N4O4 |
CAS No. | 835621-11-9 |
存储 | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
溶解度信息 | DMSO: Slightly soluble |
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