JWH 251, a cannabimimetic indole, has a high affinity tothe central cannabinoid (CB1) receptor (Ki = 29 nM) and a comparatively modest affinity for the peripheral cannabinoid (CB2) receptor (Ki = 146 nM). JWH 251 can stimulates GTPγS and bind to CB1 and CB2 receptors with EC50 values of 29 and 8.3 nM, respectively.
JWH-251
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产品编号 T32341Cas号 864445-39-6
JWH 251, a cannabimimetic indole, has a high affinity tothe central cannabinoid (CB1) receptor (Ki = 29 nM) and a comparatively modest affinity for the peripheral cannabinoid (CB2) receptor (Ki = 146 nM). JWH 251 can stimulates GTPγS and bind to CB1 and CB2 receptors with EC50 values of 29 and 8.3 nM, respectively.
JWH 251, a cannabimimetic indole, has a high affinity tothe central cannabinoid (CB1) receptor (Ki = 29 nM) and a comparatively modest affinity for the peripheral cannabinoid (CB2) receptor (Ki = 146 nM). JWH 251 can stimulates GTPγS and bind to CB1 and CB2 receptors with EC50 values of 29 and 8.3 nM, respectively.
化学信息
分子量
319.44
分子式
C22H25NO
CAS No.
864445-39-6
密度
1.03 g/cm3 (Predicted)
储存&溶解度
存储
Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.
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