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规格 | 价格 | 库存 | 数量 |
---|---|---|---|
1 mg | ¥ 774 | 现货 | |
5 mg | ¥ 1,790 | 现货 | |
10 mg | ¥ 2,630 | 现货 | |
25 mg | ¥ 4,140 | 现货 | |
50 mg | ¥ 5,680 | 现货 | |
100 mg | ¥ 7,680 | 现货 | |
500 mg | ¥ 15,300 | 现货 | |
1 mL x 10 mM (in DMSO) | ¥ 2,100 | 现货 |
产品描述 | CB1 inverse agonist 1 (MRL-650) is an orally active and selective CB1 agonist. The IC50s for CB1 and CB2 are 7.5 nM and 4100 nM, respectively. CB1 inverse agonist 1 shows anorexigenic effects. |
靶点活性 | CB1:7.5 nM, CB2:4100 nM |
体内活性 | CB1 inverse agonist 1(0.3-3 mg/kg)呈剂量依赖性地抑制摄食行为[1]。 |
别名 | MRL-650 |
分子量 | 514.79 |
分子式 | C25H18Cl3N3O3 |
CAS No. | 852315-00-5 |
存储 | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | ||||||||||||||||||||||||||||||
溶解度信息 | DMSO: 45 mg/mL (87.41 mM) | ||||||||||||||||||||||||||||||
溶液配制表 | |||||||||||||||||||||||||||||||
DMSO
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