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Search Results for " human "

Targets Recommended: cholecystokinin

4386

抑制剂 & 化合物

792

天然产物

33

化合物库

2

TargetMol 试剂盒

6839

重组蛋白

64

同位素标记化合物

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Cat. No.	Product Name
L2500	人内源代谢化合物库		499 compounds
	499 种内源性生物活性化合物的独特集合，用于高通量、高内涵筛选；
L2570	人代谢物化合物库		4454 compounds
	4454 种人代谢物的独特集合，用于高通量、高内涵筛选；
L2501	人内源代谢化合物库 Plus		1283 compounds
	1283种内源性生物活性化合物的独特集合，用于高通量、高内涵筛选。
L9410	共价抑制剂库		1920 compounds
	1920 种小分子的独特集合，包含已发现的共价抑制剂以及包含某些共价反应基团常见弹头的分子，如氯乙酰基，2-氯丙酰基，丙烯酰基，1-丙-2-炔基，1-丁-2-炔基，酮羰基，二硫键等，可以用于共价抑制剂药物研发；
L2540	肠道微生物代谢化合物库		614 compounds
	614 种肠道微生物代谢物的集合，可以用于高通量和高内涵筛选；
L1380	转录因子库		695 compounds
	695 种转录因子靶向、结构新颖的化合物；
L4660	神经疾病库Plus		1246 compounds
	1246 种神经系统相关、结构新颖的化合物；
L9400	PPI抑制剂库		485 compounds
	485 种已知活性的 PPI 相关的抑制剂，可用于高通量、高内涵筛选；
L2150	抗癌药物库		3080 compounds
	3080 个具有抗癌活性小分子的独特集合，生物活性已经临床前实验证实，可用于高通量、高内涵筛选；
L2160	抗癌活性化合物库		3188 compounds
	3188 种具有抗肿瘤活性的化合物的特有集合，用于高通量、高内涵筛选；
L2300	离子通道库		931 compounds
	931 种与离子通道相关的生物活性小分子化合物的特有集合，用于离子通道相关的疾病和药物研究，可用于高通量筛选和高内涵筛选；
L1580	GPCR库Plus		338 compounds
	338 种GPCR 靶向、结构新颖的化合物；
L2100	抗癌化合物库		7234 compounds
	7234 种肿瘤相关的生物活性小分子化合物的特有集合，用于高通量、高内涵筛选；
L2120	抗癌临床化合物库		2545 compounds
	2545 个具有抗癌活性小分子的独特集合，可用于高通量高内涵筛选。
L7000	活性脂质化合物库		385 compounds
	385 种生物活性小分子化合物，用于高通量、高内涵筛选；
L1500	GPCR靶点分子库		1940 compounds
	1940 种与 G 蛋白及其耦联受体相关的生物活性小分子化合物，所有小分子都具有良好的生物和药理活性，部分是 FDA 批准的上市药物；
L8700	铁死亡化合物库		779 compounds
	779 种与铁死亡通路相关的化合物，可用于高通量和高内涵筛选；
L8200	抗衰老化合物库		3279 compounds
	3279 个抗衰老化合物的独特集合，可用于高通量筛选和高内涵筛选；
L8300	染色质修饰分子库		250 compounds
	250 种染色质化学修饰相关的生物活性小分子化合物的特有集合，用于高通量、高内涵筛选；
L2110	抗癌上市药物库		1779 compounds
	1779 个具有抗癌活性小分子的独特集合，所有化合物都经过了严格的临床前研究和临床试验，由FDA、EMA 或NMPA 批准上市，可用于高通量、高内涵筛选。
L2180	抗肿瘤库Plus		1468 compounds
	1468 种抗肿瘤相关、结构新颖的化合物；
L9000	细胞凋亡化合物库		1760 compounds
	1760 种与凋亡相关的生物活性小分子化合物的特有集合，多用于研究肿瘤发生发展机制和抗癌药物筛选等。可用于高通量筛选和高内涵筛选；
L7200	钙通道分子库		140 compounds
	140 种钙通道相关化合物的独特集合，可用于高通量筛选和高内涵筛选；
L2191	抗乳腺癌化合物库		1939 compounds
	1939 种与乳腺癌相关的化合物，可以用于抗乳腺癌药物研发和药理研究；
L1800	抗感染化合物库		2938 compounds
	2938 种具有抗感染活性的化合物的特有集合，包括抗细菌、抗真菌、抗巨细胞病毒、抗HIV、抗SARS、抗流感等活性；
L9600	多肽分子库		791 compounds
	791 种多肽类分子，可用于多肽药物开发及信号转导通路和作用机制研究；
L6820	烟草单体化合物库		747 compounds
	747种烟草单体化合物的独特集合，可用于高通量筛选和高内涵筛选
L4300	Wnt/Hedgehog/Notch 通路化合物库		237 compounds
	237 个Wnt & Hedgehog & Notch 靶点相关的生物活性小分子化合物的特有集合，用于相关通路的研究及药物的筛选，可用于高通量、高内涵筛选。
L6120	黄酮类天然产物库		514 compounds
	514 种黄酮类天然产物的独特集合，可用于高通量筛选和高内涵筛选；
L2194	抗结直肠癌化合物库		1545 compounds
	1545 种与结直肠癌相关的化合物，可以用于高通量和高内涵筛选；
L1710	抗COVID-19化合物库		1133 compounds
	1133 种对SARS-CoV-2有抑制作用或潜在抑制作用的化合物集合，可用于高通量和高内涵筛选；
L6500	微生物天然产物库		550 compounds
	550 种微生物来源的生物活性小分子化合物的特有集合，用于高通量、高内涵筛选；
DO1200	药物靶点库		53200 compounds
	数量多，含53200种小分子化合物，是高通量筛选的有力工具；

化合物库

人内源代谢化合物库

Cat.No: L2500

Compounds: 499

人代谢物化合物库

Cat.No: L2570

Compounds: 4454

人内源代谢化合物库 Plus

Cat.No: L2501

Compounds: 1283

共价抑制剂库

Cat.No: L9410

Compounds: 1920

肠道微生物代谢化合物库

Cat.No: L2540

Compounds: 614

转录因子库

Cat.No: L1380

Compounds: 695

神经疾病库Plus

Cat.No: L4660

Compounds: 1246

PPI抑制剂库

Cat.No: L9400

Compounds: 485

抗癌药物库

Cat.No: L2150

Compounds: 3080

抗癌活性化合物库

Cat.No: L2160

Compounds: 3188

离子通道库

Cat.No: L2300

Compounds: 931

Cat.No: L1580

Compounds: 338

抗癌化合物库

Cat.No: L2100

Compounds: 7234

抗癌临床化合物库

Cat.No: L2120

Compounds: 2545

活性脂质化合物库

Cat.No: L7000

Compounds: 385

GPCR靶点分子库

Cat.No: L1500

Compounds: 1940

铁死亡化合物库

Cat.No: L8700

Compounds: 779

抗衰老化合物库

Cat.No: L8200

Compounds: 3279

染色质修饰分子库

Cat.No: L8300

Compounds: 250

抗癌上市药物库

Cat.No: L2110

Compounds: 1779

抗肿瘤库Plus

Cat.No: L2180

Compounds: 1468

细胞凋亡化合物库

Cat.No: L9000

Compounds: 1760

钙通道分子库

Cat.No: L7200

Compounds: 140

抗乳腺癌化合物库

Cat.No: L2191

Compounds: 1939

抗感染化合物库

Cat.No: L1800

Compounds: 2938

多肽分子库

Cat.No: L9600

Compounds: 791

烟草单体化合物库

Cat.No: L6820

Compounds: 747

Wnt/Hedgehog/Notch 通路化合物库

Cat.No: L4300

Compounds: 237

黄酮类天然产物库

Cat.No: L6120

Compounds: 514

抗结直肠癌化合物库

Cat.No: L2194

Compounds: 1545

抗COVID-19化合物库

Cat.No: L1710

Compounds: 1133

微生物天然产物库

Cat.No: L6500

Compounds: 550

药物靶点库

Cat.No: DO1200

Compounds: 53200

Cat. No.	Product Name	Form	Specificity Of Inhibition
C0066	Human CD34+ Cell Enrichment Kit (positive selection) 人 CD34+ 细胞富集试剂盒 (阴选)	Suspension in bottle	适用于从人脐带血单个核细胞（CBMC）或外周血单个核细胞（PBMC）中富集 CD34+ 细胞。
C0065	Human CD3+ T Cell Isolation Kit (negative selection) 人 CD3+ T 细胞分选试剂盒 (阴选)	Suspension in bottle	适用于从人 PBMC 中分选出 CD3+ T 细胞。

TargetMol 试剂盒

人 CD34+ 细胞富集试剂盒 (阴选)

Cat.No: C0066

人 CD3+ T 细胞分选试剂盒 (阴选)

Cat.No: C0065

Cat. No.	Product Name	Target	Signaling Pathways
TP2030	Gastrin I, human Gastrin I (human)	cholecystokinin	GPCR/G Protein
	Gastrin I, human (Gastrin I (human)) 是胃中产生的内源性肽，通过 CCK2 受体增加大鼠的胃蛋白酶原和酸分泌。
TP1143L	Fibrinopeptide A, human acetate Fibrinopeptide A, human acetate(25422-31-5 free base),Human fibrinopeptide A acetate	Others	Others
	Fibrinopeptide A, human acetate (Human fibrinopeptide A acetate)(25422-31-5 free base) 是一种 16 个残基的短多肽，由凝血酶从纤维蛋白原上切割下来。纤维蛋白肽 A (FPA) 由纤维蛋白原蛋白的 N 末端 Aα 区域在被凝血酶切割后产生。
TP1174	Endothelin-2 (49-69), human Human endothelin-2,Endothelin-2, human,Endothelin-2 (human, canine),人内皮素2	Others	Others
	Endothelin-2 (49-69), human (Human endothelin-2) 是一种由 21 个氨基酸组成的血管活性肽。它可与 G 蛋白连接的跨膜受体，ET-RA 和ET-RB 结合。
TP1240	ACTH (18-39) TFA (human) CLIP (human) (TFA)	Others	Others
	Adrenocorticotropic Hormone (ACTH) (18-39), human TFA (CLIP human TFA) 是一种似皮质促素中叶肽，由垂体中叶的促黑素细胞产生。
T7489	MART-1 (26-35) (human) MART-1 (26-35) human	Others	Others
	MART-1 (26-35) (human) (MART-1 (26-35) human) 是一种 MART-1 蛋白 26 到 35 氨基酸片段。
T8231	ACTH (1-39) human Adrenocorticotropic Hormone (ACTH) (1-39), human,ACTH (1-39), human,丝拉克肽	Others	Others
	Adrenocorticotropic Hormone (ACTH) (1-39), human (ACTH (1-39), human) 是黑皮质素受体激动剂。
TP1187	C-Type Natriuretic Peptide (CNP) (1-22), human CNP (1-22), human	RAAS	Endocrinology/Hormones
	C-Type Natriuretic Peptide (CNP) (1-22), human 是一种利钠肽受体 B (NPR-B) 激动剂，是一种 CNP 的 1-22 片段。它对生理激动剂组胺和 5-HT 刺激或直接由 Forskolin 刺激的 cAMP 合成具有抑制作用。其中CNP 是一种有效的、内皮衍生的松弛剂和生长抑制因子。
TP2018L	GIP (human) acetate GIP (human) acetate(100040-31-1 Free base)	IGF-1R	Tyrosine Kinase/Adaptors
	GIP (human) acetate 是葡萄糖依赖性胰岛素分泌的刺激剂和胃酸分泌的弱抑制剂。 GIP (human) acetate 在脂质代谢和肥胖的发展中起着至关重要的作用。
T8221	Insulin (human) INSULIN,甘精胰岛素,胰岛素,Insulin(human)	IGF-1R	Tyrosine Kinase/Adaptors
	Insulin (human) 是一种多肽激素，可以促进糖原的合成，调节血液中的葡萄糖水平。Insulin (human) 具有降血糖活性，临床上用于治疗糖尿病患者的高血糖。
TP1082L	Neuropeptide AF (human) acetate Neuropeptide AF (93-110), human Acetate,Neuropeptide AF (human) acetate (192387-38-5 Free base)	Opioid Receptor	Endocrinology/Hormones; GPCR/G Protein; Neuroscience
	Neuropeptide AF (human) acetate (Neuropeptide AF (human) acetate (192387-38-5 Free base)) 属于抗阿片类神经肽，是 Neuropeptide AF (human) 衍生物，可调节脂肪细胞代谢。
TP1923L1	ELA-14(human) acetate ELA-14(human) acetate (1886973-05-2 free base)	Apelin receptor; Arrestin	GPCR/G Protein
	ELA-14(human) acetate 是 ELA 的一个片段，它与 APJ 结合，激活 Gαi1 和 β-arrestin-2 信号通路，并类似于其亲本内源性肽诱导受体内化。
T7577	Angiotensin III, human, mouse 血管紧张素III,Angiotensin III, human, mouse(3TFA)	RAAS	Endocrinology/Hormones
	Angiotensin III, human, mouse (Angiotensin III, human, mouse(3TFA)) 是一种七肽，是血管紧张素 2 型受体 (AT2R) 激动剂，能够作用于 AT2R (IC50:0.648 nM)及 AT1R (IC50:21.1nM)。
T19584L	TNF-α (31-45), human acetate TNF-α (31-45), human acetate(144796-71-4 free base)	Others	Others
	TNF-α (31-45), human acetate(144796-71-4 free base) 是一种肿瘤坏死因子-α 的肽。
TP1900L1	Hemopressin (human, mouse) acetate Hemopressin (human, mouse) acetate(1314035-51-2 free base)	Cannabinoid Receptor	GPCR/G Protein
	Hemopressin (human, mouse) acetate(1314035-51-2 free base) 是一种衍生自血红蛋白 α1 链的九肽，是从大鼠脑匀浆中分离出来的。 Hemopressin 是 CB1 大麻素受体的口服活性、选择性和反向激动剂。 Hemopressin 在炎性疼痛模型中发挥镇痛作用。
T40412L	BAD (103-127) (human) acetate BAD (103-127) (human) acetate (331762-68-6 Free base)	Others	Others
	BAD (103-127) (human) acetate 是一种来自于 BAD 的 BH3结构域的25-mer Bad 多肽，可拮抗 Bcl-xl 的作用。
TP1295	Angiotensin I (human, mouse, rat) Angiotensin 1 Human,血管紧张素 1 (人)	Others	Others
	Angiotensin I (human, mouse, rat) 是血管紧张素Ⅱ的前体物质，在血管紧张素转化酶 (ACE) 的参与下裂解成血管紧张素Ⅱ。
TP1219	Atrial Natriuretic Peptide (ANP) (1-28), human, porcine Acetate ANP (1-28), human, porcineANP(1-28)
	Atrial Natriuretic Peptide (ANP) (1-28), human, porcine Acetate 是颗粒鸟苷酸环化酶的刺激剂，已被发现通过增加环鸟苷单磷酸的合成来保护分离的心肌细胞免受复氧诱导的高收缩。Atrial Natriuretic Peptide (ANP) (1-28), human, porcine Acetate 也有助于在反复运动期间刺激脂解，并在运动期间控制脂解。
TP1257L	Adrenomedullin (AM) (22-52), human acetate Adrenomedullin (AM) (22-52), human acetate（159899-65-7 Free base）	CGRP Receptor	GPCR/G Protein; Neuroscience
	Adrenomedullin (AM) (22-52), human acetate 是猫后肢血管床中 CGRP 受体和肾上腺髓质素受体的拮抗剂。
T19309L1	Endothelin 1 (swine, human) acetate Endothelin 1 (swine, human) acetate(117399-94-7 free base)	Endothelin Receptor	GPCR/G Protein
	Endothelin 1 (swine, human) acetate(117399-94-7 free base) 是一种合成肽，其序列为人和猪内皮素 1。它是一种有效的内源性血管收缩剂，通过两种类型的受体 ETA 和 ETB 起作用。
TP2092L	Apelin-17 (human, bovine) acetate Apelin-17 (human, bovine) acetate(217082-57-0 free base)	HIV Protease	Microbiology/Virology; Proteases/Proteasome
	Apelin-17 (human, bovine) acetate(217082-57-0 free base) 是一种内源性 apelin 受体激动剂。有效抑制毛喉素刺激的 cAMP 积累 (pIC50 = 9.94)。
TP1737L	Urotensin II (114-124), human acetate Urotensin II (114-124), human acetate(251293-28-4 free base)	GPR	Endocrinology/Hormones; GPCR/G Protein
	Urotensin II (114-124), human acetate(251293-28-4 free base) 是一种 11 个氨基酸残基肽，是一种有效的血管收缩剂和孤儿受体 GPR14 的激动剂。
TP1880L1	PAMP-12 (human, porcine) acetate PAMP-12 (human, porcine) acetate(196305-05-2 free base)	Others	Others
	PAMP-12 (human, porcine) acetate (PAMP-12 (human, porcine) acetate (196305-05-2 free base)) 是 ir-PAMP 的主要成分，由 AM 前体加工而成，PAMP-20 也是如此，并且可能参与心血管控制。
TP1144L	Corticotropin-releasing factor (human) acetate Corticotropin-releasing factor (human) acetate (86784-80-7 Free base)	CRFR	GPCR/G Protein
	Corticotropin-releasing factor (human) acetate 刺激垂体前叶合成和分泌促肾上腺皮质激素。
TP1627L	Prepro VIP (111-122), human acetate Prepro VIP (111-122), human acetate(123025-94-5 free base)	Others	Others
	Prepro VIP (111-122), human acetate(123025-94-5 free base) 是一种前血管活性肠多肽 (VIP) 衍生肽，对应于残基 111-122。
TP1244L1	ACTH (1-10) Acetate (human) Adrenocorticotropic Hormone (ACTH) (1-10), human acetate(2791-05-1 Free base)	Others	Others
	Adrenocorticotropic Hormone (ACTH) (1-10), human acetate 是促肾上腺皮质激素的一个片段。 Adrenocorticotropic Hormone (ACTH) (1-10), human acetate 仅在 100 和 1000 nM 时具有较弱的 α-MSH 效力。
T21608L	β-Interleukin I (163-171), human Acetate β-Interleukin I (163-171), human Acetate(106021-96-9 Free base)	Others	Others
	β-Interleukin I (163-171), human Acetate 是一种参与调节免疫反应、炎症反应和造血的肽。
TP1007L	β-Amyloid (1-42), acetate (human) β-Amyloid (1-42), human acetate (107761-42-2 Free base)
	β-Amyloid (1-42), acetate (human) 是由 42 个氨基酸组成的肽，是 β-Amyloid 的一部分，常用于阿尔茨海默病造模。
TP1732L	Galanin (1-30), human acetate 醋酸甘丙肽,Galanin (1-30), human acetate(119418-04-1 Free base)	Others	Others
	Galanin (1-30), human acetate (Galanin ) 是一种 30 个氨基酸的神经肽。它是 GalR1 和 GalR2 受体的激动剂，Kis 均为 1 nM。
TP2056L	Acetyl-Calpastatin (184-210)(human) acetate Acetyl-Calpastatin (184-210) (human) acetate(123714-50-1 Free base )	Cysteine Protease	Proteases/Proteasome
	Acetyl-Calpastatin (184-210)(human) acetate 是一种有效，选择性和可逆的钙蛋白酶 (calpain) 抑制剂，对 μ-钙蛋白酶和组织蛋白酶 L 的 Ki 值分别为 0.2 nM 和 6 μM。
TP1618L	PACAP-38 (31-38), human, mouse, rat acetate PACAP-38 (31-38), human, mouse, rat acetate(138764-85-9 Free base)	PACAP	GPCR/G Protein
	PACAP-38 (31-38), human, mouse, rat acetate 是 PAC1 受体的激活剂。PACAP-38 (31-38), human, mouse, rat acetate 对交感神经元 NPY 和儿茶酚胺的产生具有强效、有效和持续的刺激作用，可用于神经营养和神经保护研究。
TP1628L	Activated Protein C (390-404), human acetate Activated Protein C (390-404), human acetate(146340-20-7 Free base)	APC	Cell Cycle/Checkpoint
	Activated Protein C (390-404), human acetate (Activated Protein C ) 抑制 APC 抗凝活性。
TP2499	Human IgE Pentapeptide HEPP acetate Human IgE Pentapeptide HEPP acetate (62087-72-3 Free base）
	Human IgE Pentapeptide HEPP acetate 是一种五肽，在几种不同体系中均不能产生 IgE 抑制作用，可用于治疗结膜炎。
T21649L	GnRH Associated Peptide (1-13) Acetate（human） GnRH Associated Peptide (GAP) (1-13), human Acetate (100111-07-7 Free base),GnRH Associated Peptide (1-13), Acetate（human） (100111-07-7 Free base)	Others	Others
	GnRH Associated Peptide (GAP) (1-13), human Acetate 被发现是催乳素分泌的有效抑制剂并刺激促性腺激素的释放。用对应于 GAP 序列的肽进行主动免疫导致催乳素分泌大大增加。
T38193L	β-Endorphin (1-27) (human) acetate β-Endorphin (1-27) (human) acetate(76622-84-9 Free base)	Opioid Receptor	Endocrinology/Hormones; GPCR/G Protein; Neuroscience
	β-Endorphin (1-27) (human) acetate 存在于大脑垂体和下丘脑中，具有镇痛活性。 β-Endorphin (1-27) (human) acetate 是一种阿片受体激动剂，对 μ-阿片受体和 δ-阿片受体具有较好的亲和力。
TP1996	MCH(human, mouse, rat) MCH (human, mouse, rat),黑色素聚集激酶素(MCH)( 大鼠)	GPR; Melanin-concentrating Hormone Receptor (MCHR)	Endocrinology/Hormones; GPCR/G Protein
	MCH(human, mouse, rat) 是MCH-R 肽激动剂，对 CHO 细胞系中 MCH-2R 高度敏感，激活 MCH-1R 和 MCH-2R 的IC50 值分别为 0.3 和 1.5 nM，EC50值对分别为 3.9 和 0.1 nM。
T39392L	C-Type Natriuretic Peptide (1-22) acetate（human） C-Type Natriuretic Peptide (CNP) (1-22), human acetate(1966153-17-2 Free base)	Others	Others
	C-Type Natriuretic Peptide (CNP) (1-22), human acetate 是一种利钠肽受体 B (NPR-B) 的激动剂，一种内皮衍生的松弛剂和生长抑制因子。 C-Type Natriuretic Peptide (CNP) (1-22), human acetate 抑制由组胺和 5-HT 或直接由毛喉素刺激的 cAMP 合成。
TP2044L	α-CGRP (human) acetate 人类降钙素基因相关肽 1,α-CGRP (human) acetate (90954-53-3 free base)	Others	Others
	α-CGRP (human) acetate 是一种由 37 个氨基酸组成的调节性神经肽。它是一种有效的血管扩张剂，具有正性肌力作用和变时性作用。
T38470	Obestatin (human)
	Obestatin (human) 是一种由 preproghrelin 经过剪切形成的G蛋白欧联实体39的内源性配体，可以剂量依赖的方式抑制进食，可用于研究肥胖。
TP1651L	Proinsulin C-peptide human acetate 醋酸胰岛素原C-肽(55-89),人,Proinsulin C-peptide human acetate (33017-11-7 Free base)	Others	Others
	Proinsulin C-peptide human acetate (Proinsulin C-peptide human acetate (33017-11-7 Free base)) 是一种由31个氨基酸残基组成的多肽，它连接胰岛素原的 A 链和 B 链以确保正确折叠，具有生物活性并调节细胞功能。
TP1070L	PACAP (1-27), human, ovine, rat acetate PACAP 1-27 acetate,PACAP (1-27), human, ovine, rat acetate(127317-03-7 free base)	PACAP	GPCR/G Protein
	PACAP (1-27), human, ovine, rat acetate (PACAP 1-27 acetate)(127317-03-7 free base) 是一种新的神经肽，最初从牛下丘脑中分离出来，也存在于人和大鼠中。
TP1359L	Amyloid β Peptide (42-1)(human) acetate Amyloid β Peptide (42-1)(human) acetate(317366-82-8 free base)	Beta Amyloid	Neuroscience
	Amyloid β Peptide (42-1)(human) acetate 是淀粉样蛋白 β 肽 (1-42) 的无活性形式。Amyloid β Peptide (42-1)(human) acetate 是由 42 个氨基酸组成的肽，其在阿尔茨海默病的发病机制中起关键作用。
T21484	BNP (1-32), human	Others	Others
	BNP (1-32), human 是一种脑利钠肽。
T76840	Vunakizumab Anti-Human IL17A Recombinant Antibody	IL Receptor	Immunology/Inflammation
	Vunakizumab 是一种靶向 IL-17A 的人源化 IgGκ 单克隆抗体，常与白细胞介素 22 链接形成 Vunakizumab-IL22 来研究流感病毒引起的肺免疫损伤。Vunakizumab 可用于研究银屑病关节炎，通过与IL-17A结合发挥作用。
TP1705	Gastrin I (1-14), human	Others	Others
	Gastrin I (1-14), human 是人胃泌素 I 肽的 1-14 片段。其中Gastrin I 是内源性胃肠肽激素。Gastrin 是胃酸分泌的主要激素调节剂。
TP1004L	Beta-MSH (1-22) (human) acetate Beta-MSH (1-22) (human) acetate (17908-57-5 Free base),醋酸Β-促黑激素(人)	Melanocortin Receptor	GPCR/G Protein; Neuroscience
	Beta-MSH (1-22) (human) acetate (Beta-MSH (1-22) (human) acetate (17908-57-5 Free base)) 是一种 22 肽，是一种内源性黑皮质素 4 受体 (MC4-R) 激动剂。
TP1116L	Kinetensin acetate(103131-69-7 free base) Kinetensin (human) acetate	Neurotensin Receptor	GPCR/G Protein
	Kinetensin acetate(103131-69-7 free base) 是从经胃蛋白酶处理的人血浆中分离出来的。它是一种神经降压素样肽。
TP1949L	PEN (human) aceate	GPCR19	GPCR/G Protein
	PEN (human) aceate 是丰富的下丘脑神经肽之一，源自 ProSAAS 前蛋白，是 GPR83 的内源性配体。
TP1842L	Angiotensinogen (1-14), human acetate	Endogenous Metabolite	Metabolism
	Angiotensinogen (1-14), human acetate 是血管紧张素原的片段，它是肾素-血管紧张素系统的被动底物。
TP1863L	Glucagon (19-29), human acetate	Glucagon Receptor	GPCR/G Protein
	Glucagon (19-29), human acetate 是一种从胰高血糖素加工而来的 COOH 末端片段，是一种有效的胰岛素分泌抑制剂。
TP2030L1	Gastrin I (human) acetate Gastrin I (human) acetate(10047-33-3 free base),Gastrin-17 acetate,Little gastrin I acetate,胃膜素醋酸盐	cholecystokinin	GPCR/G Protein
	Gastrin I (human) acetate (Gastrin-17 acetate) 是在胃中产生的内源性肽，通过胆囊收缩素 2 (CCK2) 受体增加胃酸分泌。

化合物

Gastrin I, human

Cat.No: TP2030

Synonym: Gastrin I (human)

Target: cholecystokinin

Fibrinopeptide A, human acetate

Cat.No: TP1143L

Synonym: Fibrinopeptide A, human acetate(25422-31-5 free base),Human fibrinopeptide A acetate

Target: Others

Endothelin-2 (49-69), human

Cat.No: TP1174

Synonym: Human endothelin-2,Endothelin-2, human,Endothelin-2 (human, canine),人内皮素2

Target: Others

ACTH (18-39) TFA (human)

Cat.No: TP1240

Synonym: CLIP (human) (TFA)

Target: Others

MART-1 (26-35) (human)

Cat.No: T7489

Synonym: MART-1 (26-35) human

Target: Others

ACTH (1-39) human

Cat.No: T8231

Synonym: Adrenocorticotropic Hormone (ACTH) (1-39), human,ACTH (1-39), human,丝拉克肽

Target: Others

C-Type Natriuretic Peptide (CNP) (1-22), human

Cat.No: TP1187

Synonym: CNP (1-22), human

Target: RAAS

GIP (human) acetate

Cat.No: TP2018L

Synonym: GIP (human) acetate(100040-31-1 Free base)

Target: IGF-1R

Insulin (human)

Cat.No: T8221

Synonym: INSULIN,甘精胰岛素,胰岛素,Insulin(human)

Target: IGF-1R

Neuropeptide AF (human) acetate

Cat.No: TP1082L

Synonym: Neuropeptide AF (93-110), human Acetate,Neuropeptide AF (human) acetate (192387-38-5 Free base)

Target: Opioid Receptor

ELA-14(human) acetate

Cat.No: TP1923L1

Synonym: ELA-14(human) acetate (1886973-05-2 free base)

Target: Apelin receptor, Arrestin

Angiotensin III, human, mouse

Cat.No: T7577

Synonym: 血管紧张素III,Angiotensin III, human, mouse(3TFA)

Target: RAAS

TNF-α (31-45), human acetate

Cat.No: T19584L

Synonym: TNF-α (31-45), human acetate(144796-71-4 free base)

Target: Others

Hemopressin (human, mouse) acetate

Cat.No: TP1900L1

Synonym: Hemopressin (human, mouse) acetate(1314035-51-2 free base)

Target: Cannabinoid Receptor

BAD (103-127) (human) acetate

Cat.No: T40412L

Synonym: BAD (103-127) (human) acetate (331762-68-6 Free base)

Target: Others

Angiotensin I (human, mouse, rat)

Cat.No: TP1295

Synonym: Angiotensin 1 Human,血管紧张素 1 (人)

Target: Others

Atrial Natriuretic Peptide (ANP) (1-28), human, porcine Acetate

Cat.No: TP1219

Synonym: ANP (1-28), human, porcineANP(1-28)

Adrenomedullin (AM) (22-52), human acetate

Cat.No: TP1257L

Synonym: Adrenomedullin (AM) (22-52), human acetate（159899-65-7 Free base）

Target: CGRP Receptor

Endothelin 1 (swine, human) acetate

Cat.No: T19309L1

Synonym: Endothelin 1 (swine, human) acetate(117399-94-7 free base)

Target: Endothelin Receptor

Apelin-17 (human, bovine) acetate

Cat.No: TP2092L

Synonym: Apelin-17 (human, bovine) acetate(217082-57-0 free base)

Target: HIV Protease

Urotensin II (114-124), human acetate

Cat.No: TP1737L

Synonym: Urotensin II (114-124), human acetate(251293-28-4 free base)

Target: GPR

PAMP-12 (human, porcine) acetate

Cat.No: TP1880L1

Synonym: PAMP-12 (human, porcine) acetate(196305-05-2 free base)

Target: Others

Corticotropin-releasing factor (human) acetate

Cat.No: TP1144L

Synonym: Corticotropin-releasing factor (human) acetate (86784-80-7 Free base)

Target: CRFR

Prepro VIP (111-122), human acetate

Cat.No: TP1627L

Synonym: Prepro VIP (111-122), human acetate(123025-94-5 free base)

Target: Others

ACTH (1-10) Acetate (human)

Cat.No: TP1244L1

Synonym: Adrenocorticotropic Hormone (ACTH) (1-10), human acetate(2791-05-1 Free base)

Target: Others

β-Interleukin I (163-171), human Acetate

Cat.No: T21608L

Synonym: β-Interleukin I (163-171), human Acetate(106021-96-9 Free base)

Target: Others

β-Amyloid (1-42), acetate (human)

Cat.No: TP1007L

Synonym: β-Amyloid (1-42), human acetate (107761-42-2 Free base)

Galanin (1-30), human acetate

Cat.No: TP1732L

Synonym: 醋酸甘丙肽,Galanin (1-30), human acetate(119418-04-1 Free base)

Target: Others

Acetyl-Calpastatin (184-210)(human) acetate

Cat.No: TP2056L

Synonym: Acetyl-Calpastatin (184-210) (human) acetate(123714-50-1 Free base )

Target: Cysteine Protease

PACAP-38 (31-38), human, mouse, rat acetate

Cat.No: TP1618L

Synonym: PACAP-38 (31-38), human, mouse, rat acetate(138764-85-9 Free base)

Target: PACAP

Activated Protein C (390-404), human acetate

Cat.No: TP1628L

Synonym: Activated Protein C (390-404), human acetate(146340-20-7 Free base)

Target: APC

Human IgE Pentapeptide HEPP acetate

Cat.No: TP2499

Synonym: Human IgE Pentapeptide HEPP acetate (62087-72-3 Free base）

GnRH Associated Peptide (1-13) Acetate（human）

Cat.No: T21649L

Synonym: GnRH Associated Peptide (GAP) (1-13), human Acetate (100111-07-7 Free base),GnRH Associated Peptide (1-13), Acetate（human） (100111-07-7 Free base)

Target: Others

β-Endorphin (1-27) (human) acetate

Cat.No: T38193L

Synonym: β-Endorphin (1-27) (human) acetate(76622-84-9 Free base)

Target: Opioid Receptor

MCH(human, mouse, rat)

Cat.No: TP1996

Synonym: MCH (human, mouse, rat),黑色素聚集激酶素(MCH)( 大鼠)

Target: GPR, Melanin-concentrating Hormone Receptor (MCHR)

C-Type Natriuretic Peptide (1-22) acetate（human）

Cat.No: T39392L

Synonym: C-Type Natriuretic Peptide (CNP) (1-22), human acetate(1966153-17-2 Free base)

Target: Others

α-CGRP (human) acetate

Cat.No: TP2044L

Synonym: 人类降钙素基因相关肽 1,α-CGRP (human) acetate (90954-53-3 free base)

Target: Others

Obestatin (human)

Cat.No: T38470

Proinsulin C-peptide human acetate

Cat.No: TP1651L

Synonym: 醋酸胰岛素原C-肽(55-89),人,Proinsulin C-peptide human acetate (33017-11-7 Free base)

Target: Others

PACAP (1-27), human, ovine, rat acetate

Cat.No: TP1070L

Synonym: PACAP 1-27 acetate,PACAP (1-27), human, ovine, rat acetate(127317-03-7 free base)

Target: PACAP

Amyloid β Peptide (42-1)(human) acetate

Cat.No: TP1359L

Synonym: Amyloid β Peptide (42-1)(human) acetate(317366-82-8 free base)

Target: Beta Amyloid

BNP (1-32), human

Cat.No: T21484

Target: Others

Cat.No: T76840

Synonym: Anti-Human IL17A Recombinant Antibody

Target: IL Receptor

Gastrin I (1-14), human

Cat.No: TP1705

Target: Others

Beta-MSH (1-22) (human) acetate

Cat.No: TP1004L

Synonym: Beta-MSH (1-22) (human) acetate (17908-57-5 Free base),醋酸Β-促黑激素(人)

Target: Melanocortin Receptor

Kinetensin acetate(103131-69-7 free base)

Cat.No: TP1116L

Synonym: Kinetensin (human) acetate

Target: Neurotensin Receptor

PEN (human) aceate

Cat.No: TP1949L

Target: GPCR19

Angiotensinogen (1-14), human acetate

Cat.No: TP1842L

Target: Endogenous Metabolite

Glucagon (19-29), human acetate

Cat.No: TP1863L

Target: Glucagon Receptor

Gastrin I (human) acetate

Cat.No: TP2030L1

Synonym: Gastrin I (human) acetate(10047-33-3 free base),Gastrin-17 acetate,Little gastrin I acetate,胃膜素醋酸盐

Target: cholecystokinin

Cat. No.	Product Name	Target	Signaling Pathways
TP2167	β-CGRP, human acetate β-CGRP, human acetate (101462-82-2 free),CGRP-II (Human) (acetate),Human β-CGRP acetate	CGRP Receptor	GPCR/G Protein; Neuroscience
	β-CGRP, human acetate 是降钙素肽之一，通过受体活性修饰蛋白 (RAMP) 和降钙素受体样受体 (CRLR) 的复合物发挥作用（对于 CRLR/RAMP1 和 CRLR，IC50：1 nM 和 300 nM /RAMP2 在单元格中）。
T7040	Angiotensin II human DRVYIHPF,Angiotensin II,Hypertensin II,血管紧张素Ⅱ,Ang II,血管紧张素II	Apoptosis; RAAS	Apoptosis; Endocrinology/Hormones
	Angiotensin II human (Ang II) 是一种生物活性肽，一种血管收缩剂。Angiotensin II 可以与 AT1R 和 AT2R 相互作用，调节人类血压，刺激交感神经，增加醛固酮生物合成和肾脏活动。
T41030	γ-Globulins from human blood	Others	Others
	γ-Globulins, a protein fraction found in human blood, comprise a class of proteins with potent antibody activity that safeguards against bacterial and viral infections. These γ-globulins are specifically utilized in the treatment of common variable immunodeficiency.
T13433	β-Endorphin, human	Others	Others
	β-Endorphin, human, a prominent endogenous peptide, existing in the hypophysis cerebri and hypothalamus,and is an agonist of opioid receptor.
T6377	Aloperine	Apoptosis; Virus Protease; HIV Protease; Antibiotic; Autophagy	Apoptosis; Autophagy; Microbiology/Virology; Proteases/Proteasome
	Aloperine 是一种在苦参类植物中的生物碱，其具有抗癌，抗炎、抗肿瘤和抗病毒特性，可用于研究过敏性接触性皮炎湿疹和其他皮肤炎症。
TN2283	Tripterifordin	HIV Protease	Microbiology/Virology; Proteases/Proteasome
	Tripterifordin 在 H9 淋巴细胞中显示出抗 HIV 复制活性，EC50值为 3100 nM。
T2S1040	Jolkinolide B	ERK; IL Receptor; BCL; p38 MAPK; TNF; NF-κB; Akt; Caspase; PI3K; JAK; JNK; STAT; mTOR	Angiogenesis; Apoptosis; Chromatin/Epigenetic; Cytoskeletal Signaling; Immunology/Inflammation; JAK/STAT signaling; MAPK; NF-κB; PI3K/Akt/mTOR signaling; Proteases/Proteasome; Stem Cells
	Jolkinolide B 是一种从 Euphorbia fischeriana Steud 的根中分离出来的具有生物活性的二萜。 Jolkinolide B 诱导癌细胞凋亡。 Jolkinolide B 可用于预防和治疗骨溶解的研究。
T3020	Sclareol	Apoptosis; Others	Apoptosis; Others
	Sclareol 是一种从快乐鼠尾草中分离出来的拉丹型二萜，对多种人类 Y 细胞系具有生长抑制和细胞毒活性，诱导细胞凋亡。
T9503	PHYTOSPHINGOSINE	Apoptosis	Apoptosis
	Phytosphingosine 是具有抗癌作用的一种磷脂。在癌细胞中，它通过 caspase 8 的激活和 Bax 转位诱导细胞凋亡。
T10021	1-Methylxanthine	Endogenous Metabolite	Metabolism
	1-Methylxanthine 是咖啡因衍生物，是咖啡因和茶碱 (1,3-二甲基黄嘌呤，TP) 在人体尿代谢产物，能够提高肿瘤细胞的放射敏感性。
TQ0217	Gomisin G 戈米辛G,戈米辛 G	P450; HIV Protease	Metabolism; Microbiology/Virology; Proteases/Proteasome
	Gomisin G 是一种有抗HIV 活性的天然产物。
TN4417	Larixyl acetate	Others	Others
	Larixyl acetate 是一种生物活性化学物质。
T11363	Ganoderic acid F	Others	Others
	Ganoderic acid F 是一种灵芝酸。它具有抗肿瘤和抗转移的活性，与抑制血管生成和涉及细胞增殖和细胞死亡，致癌作用，氧化应激，钙信号传导和内质网应激的蛋白质改变等机制相关。
T0474	Erythromycin ethylsuccinate EES,琥乙红霉素	ribosome; HIV Protease; Antibacterial; Antibiotic; Autophagy	Autophagy; Microbiology/Virology; Proteases/Proteasome
	Erythromycin ethylsuccinate (EES) 是一种由红链霉菌产生的大环内酯类抗生素，有潜力用于多种细菌感染。它具有抗 HIV-1病毒活性。
Fr16741	Oxindole 2-吲哚酮,板蓝根,Indolin-2-one	Others; HIV Protease	Microbiology/Virology; Others; Proteases/Proteasome
	Oxindole (Indolin-2-one) 是一种芳族杂环砌块，其衍生物是激酶抑制剂研究中的主要成分。
T2942	Psoralen Ficusin,Furocoumarin,补骨脂素,psoralene	Apoptosis; Influenza Virus; HIV Protease; DNA/RNA Synthesis	Apoptosis; Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology; Proteases/Proteasome
	Psoralen (Ficusin) 是从补骨脂种子中提取的一种香豆素。它具有如抗癌、抗氧化、抗抑郁、抗癌、抗菌、抗病毒等多种生物学特性。
TN2069	Picrocrocin 藏红花,苦番紅花素	Apoptosis	Apoptosis
	Picrocrocin 是一种从椰菜花中发现的类胡萝卜素，对 SKMEL-2 人恶性黑色素瘤细胞具有生长抑制作用，具有抗癌作用。
T10005L	1,2-Dipalmitoyl-sn-glycerol 3-phosphate sodium	Endogenous Metabolite	Metabolism
	1,2-Dipalmitoyl-sn-glycerol 3-phosphate sodium 是一种人内源性代谢物，是一种磷酸酯。
T5061	Lumichrome 7,8-Dimethylalloxazine,光色素	Apoptosis; Endogenous Metabolite	Apoptosis; Metabolism
	Lumichrome 是人类体内的内源性化合物，由核黄素光降解产生。它利用p53 依赖机制抑制人肺癌细胞生长并诱导凋亡。
T2865	Oleanolic Acid Oleanic acid,Caryophyllin,齐墩果酸	HIV Protease; Endogenous Metabolite; Antibiotic; Autophagy	Autophagy; Metabolism; Microbiology/Virology; Proteases/Proteasome
	Oleanolic Acid (Caryophyllin) 是具有抗癌活性的一种天然产物。
T3822	Bellidifolin Bellidifoline,龙胆山酮酚,Bellidifolium,雏菊叶龙胆酮	Others; HIV Protease	Microbiology/Virology; Others; Proteases/Proteasome
	Bellidifolin (Bellidifoline) 是从獐牙菜的茎中提取的一种呫吨酮，它能作为病毒蛋白 R 的抑制剂，具有保肝、降血糖、抗炎、抗氧化、抗肿瘤作用。
T0966	Sennoside A 番泻苷A,NSC 112929,番泻苷 A	MAO; HIV Protease	Metabolism; Microbiology/Virology; Neuroscience; Proteases/Proteasome
	Sennoside A (NSC-112929) 是在番泻叶的叶子和豆荚中大量发现的蒽醌苷，抑制 HIV-1 复制。
TN1103	Diphyllin 山荷叶素,二叶草素	ATPase; Proton pump; Influenza Virus; HIV Protease	Membrane transporter/Ion channel; Microbiology/Virology; Proteases/Proteasome
	Diphyllin 是一种从Justicia procumbens 中分离的芳基萘木脂素，是HIV-1的有效抑制剂，IC50 为 0.38 μM。它是V-ATPase 抑制剂，IC50值为 17 nM，可抑制人破骨细胞中的溶酶体酸化。它抑制NO 产生，IC50值为 50 μM ，具有抗癌和抗炎活性。
T6841	Fumagillin NSC9168,烟曲霉素,Amebacilin	Others; HIV Protease; Antibiotic; Parasite	Microbiology/Virology; Others; Proteases/Proteasome
	Fumagillin (Amebacilin) 由烟曲霉菌中提取的一种抗菌药，有抗阿米巴活性。它通过抑制 HIV-1 viral protein R 活性来抑制 HIV‐1感染。
T8689	Chloroquine CQ,氯喹	SARS-CoV; TLR; HIV Protease; Antibiotic; Parasite; Autophagy	Autophagy; Immunology/Inflammation; Microbiology/Virology; Proteases/Proteasome
	Chloroquine 是一种 Toll 样受体抑制剂，可以抑制自噬。Chloroquine 具有抗疟疾和抗炎活性，广泛用于治疗疟疾和类风湿性关节炎。Chloroquine 还具有抗 SARS-CoV-2 (COVID-19) 活性、抗 HIV-1 活性。
T8116	Azulene 甘菊蓝,奥苷菊环,Bicyclo[5.3.0]Decapentaene	Others; HIV Protease	Microbiology/Virology; Others; Proteases/Proteasome
	Azulene (Bicyclo[5.3.0]Decapentaene) 是萘的异构体，具有高抗HIV 活性。它是从洋甘菊精油中分离出来的一种化学支架。
T5S1133	Ganoderic acid D 灵芝酸D,灵芝酸 D	Apoptosis; Sirtuin	Apoptosis; Chromatin/Epigenetic; DNA Damage/DNA Repair
	Ganoderic acid D 是高度氧化的四环三萜，是灵芝的主要活性成分，可诱导 HeLa 人宫颈癌细胞凋亡。它上调 SIRT3的蛋白质表达并通过 SIRT3 诱导脱乙酰化的亲环蛋白 D 。它抑制结肠癌细胞的能量重编程，包括结肠癌细胞中的葡萄糖摄取，乳酸、丙酮酸和乙酰辅酶的产生。
T2177	Kaempferol Kempferol,山柰酚,山奈酚,Robigenin	Apoptosis; Estrogen Receptor/ERR; Mitophagy; Estrogen/progestogen Receptor; HIV Protease; Endogenous Metabolite; Parasite; Autophagy	Apoptosis; Autophagy; Endocrinology/Hormones; Metabolism; Microbiology/Virology; Proteases/Proteasome
	Kaempferol (Robigenin) 属于天然类黄酮，是一种 ERRα 和 ERRγ 的反向激动剂。Kaempferol 具有抗肿瘤、抗炎、抗氧化、抗菌和抗病毒等多种活性。
T0492	Dimethyl fumarate 富马酸二甲酯,DMF	Reactive Oxygen Species; HIV Protease; Nrf2; Endogenous Metabolite; Autophagy	Autophagy; Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB; Proteases/Proteasome
	Dimethyl fumarate (DMF) 是具有口服活性且可透过血脑屏障的Nrf2激活剂，可诱导抗氧化剂基因表达上调。它是一种富马酸盐衍生物，可作抗炎和免疫调节剂，可研究多发性硬化症。
TN2004	Obtusin 1,7-二羟基-2,3,8-三甲氧基-6-甲基蒽-9,10-二酮,决明素	MAO; Monoamine Oxidase	Metabolism; Neuroscience
	Obtusin 是来自决明子种子，是一种高度选择性和竞争性的人单胺氧化酶-A 抑制剂，IC50=11.12 μM，Ki=6.15 μM。它在神经退行性疾病，尤其是焦虑和抑郁中起预防作用。
T0437	Inosine INO 495,NSC 20262,肌苷	ROS; Endogenous Metabolite; Adenosine Receptor	GPCR/G Protein; Immunology/Inflammation; Metabolism; Neuroscience
	Inosine (NSC-20262) 是由腺苷分解代谢产生的一种内源性嘌呤核苷，是腺苷受体A1R 和A2AR 的激动剂，具有抗炎免疫调节，抗伤害和神经保护作用。
T2S0731	Trilobatin 三叶苷,三叶甙,P-Phlorizin	Amylase	Metabolism
	Trilobatin (P-Phlorizin) 是源自Lithocarpus polystachyusRehd 的甜味剂，是一种HIV-1抑制剂，靶向 Gp41 包膜蛋白，具有神经保护作用。它还是SGLT1/2抑制剂，可选择性诱导人肝母细胞瘤细胞增殖。
T2789	Scutellarin 黄岑素,野黄芩苷,Breviscapin,Breviscapinun,Breviscapine,Scutellarein-7-glucuronide	Akt; HIV Protease; STAT	Cytoskeletal Signaling; JAK/STAT signaling; Microbiology/Virology; PI3K/Akt/mTOR signaling; Proteases/Proteasome; Stem Cells
	Scutellarin (Scutellarein-7-glucuronide) 是从黄芩中分离的黄酮，可抑制破骨细胞中 RANKL 介导的 MAPK 和 NF-κB 信号通路，并下调 HCC 细胞中的 STAT3/Girdin/Akt 信号通路。
T4962	Zingibroside R1 Ginsenoside Z-R1,姜状三七皂苷R1,姜状三七苷R1	HIV Protease	Microbiology/Virology; Proteases/Proteasome
	Zingibroside R1 (Ginsenoside Z-R1) 是分离自Panax japonicasC. A. Meyer 根部的一种三萜皂苷，有HIV-1、抗肿瘤和抗血管生成活性。它对 EAT 细胞的 2-脱氧-D-葡萄糖的摄取具有抑制作用，IC50值为91.3 μM。
T1284	Megestrol acetate SC10363,醋酸甲地孕酮,BDH1298	Glucocorticoid Receptor; Estrogen/progestogen Receptor; Progesterone Receptor; HIV Protease; Autophagy	Autophagy; Endocrinology/Hormones; Microbiology/Virology; Others; Proteases/Proteasome
	Megestrol acetate (BDH1298) 是具有口服活性的合成孕激素。它还具有抗雄激素特性，可用于治疗厌食症和恶病质。
T1131	Ivermectin MK-933,伊维菌素	Mitophagy; GluCls; P2X Receptor; SARS-CoV; HIV Protease; Antibiotic; Parasite; Autophagy; HSV	Autophagy; Membrane transporter/Ion channel; Microbiology/Virology; Neuroscience; Proteases/Proteasome
	Ivermectin (MK-933) 是谷氨酸门控氯离子通道激活剂，具有抗寄生虫活性。它特异性抑制Impα/β1 介导的核导入，还抑制牛疱疹病毒 1 复制并抑制BoHV-1DNA 聚合酶的核输入。它具有很强的抗病毒活性。它也是P2X4和 α7nAChRs 的正异构效应物。
T7991	2-Hydroxycinnamic acid 邻羟基肉桂酸(邻香豆酸),(E)-3-(2-羟基苯基)丙烯酸	Others; SARS-CoV; HIV Protease	Microbiology/Virology; Others; Proteases/Proteasome
	2-Hydroxycinnamic acid 是从肉桂的甲醇提取物中分离出的一种天然产物，具有光氧化活性。它对HIV/SARS-CoV S 假病毒的感染具有抑制作用，IC50为 0.3 mM。
T2728	Limonin Dictamnolactone,Limonoic acid 3,19:16,17 dilactone,柠檬苦素,Obaculactone,Citrolimonin	Apoptosis; HIV Protease; Endogenous Metabolite	Apoptosis; Metabolism; Microbiology/Virology; Proteases/Proteasome
	Limonin (Citrolimonin) 是柑橘类水果中富含的一种三萜类天然产物，具有抗病毒和抗肿瘤活性。
TN2883	3',4'-Dimethoxyflavone	Others; PARP	Chromatin/Epigenetic; DNA Damage/DNA Repair; Others
	3',4'-Dimethoxyflavone 是类黄酮化合物的参考标准，类黄酮化合物具有多种药用活性。
T3122	Fangchinoline Tetrandrine B,防己诺林碱,(+)-Limacine,Hanfangichin B,防己醇灵,(+)-Fangchinoline	Apoptosis; FAK; HIV Protease; Autophagy	Angiogenesis; Apoptosis; Autophagy; Cytoskeletal Signaling; Microbiology/Virology; Proteases/Proteasome; Tyrosine Kinase/Adaptors
	Fangchinoline (Tetrandrine B) 是从Stephaniatetrandra 中分离出来的，一种具有广泛生物学活性的天然产物。它是新型HIV-1抑制剂，通过损害 gp160 蛋白水解过程来抑制 HIV-1 复制。它靶向Focal adhesion kinase (FAK)并抑制肿瘤细胞中 FAK 介导的的信号传导途径。
T16791	Rottlerin Mallotoxin,NSC 56346,粗糠柴苦素,NSC 94525	CaMK; Apoptosis; Others; HIV Protease; PKA; PKC; Autophagy	Apoptosis; Autophagy; Chromatin/Epigenetic; Cytoskeletal Signaling; Microbiology/Virology; Neuroscience; Others; Proteases/Proteasome; Tyrosine Kinase/Adaptors
	Rottlerin (NSC-56346) 是一种从Mallotus Philippinensis 中得到的天然产物，是 PKC 的特异性抑制剂，抑制HIV-1整合和狂犬病病毒感染。它通过活化 caspase 3 诱导细胞凋亡.
T3730	Methyl gallate NSC 363001,Gallicin,Gallic acid methyl ester,Gallincin,没食子酸甲酯	Reactive Oxygen Species; HIV Protease; Reverse Transcriptase; Antibacterial	Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB; Proteases/Proteasome
	Methyl gallate (Gallincin) 是具有抗氧化，抗癌和抗炎活性的植物酚类。它也可抑制细菌活性。它还具有抗HIV-1和HIV-1酶的抑制活性。
TN6796	2'-FUCOSYLLACTOSE 2'-Fucosyl-D-lactose,2'-岩藻糖基乳糖	Others	Others
	2'-FUCOSYLLACTOSE (2'-Fucosyl-D-lactose) 是一种含岩藻糖的寡糖。
T4P2931	Linoleic acid 9,12-octadecadienoic acid,亚油酸,α-亚油酸,acidelinoleique,9,12-Linoleic acid	Others; Endogenous Metabolite	Metabolism; Others
	Linoleic acid (9,12-octadecadienoic acid) 是一种多不饱和脂肪酸，存在于坚果、种子和植物性油中。它是膜磷脂的一部分，作为膜流动性的结构成分来维持表皮透皮水屏障。它通过氧化作用引起血红蛋白和红细胞损伤。
T5782	Bevirimat YK FH312,MPC-4326,PA-457,贝韦立马	HIV Protease	Microbiology/Virology; Proteases/Proteasome
	Bevirimat (PA-457) 是一种 HIV-1 成熟抑制剂，可在病毒体成熟过程中阻断 Gag 衣壳 (CA) 前体 CA-SPI 裂解为成熟的 CA 蛋白。
T2830	Betulinic acid 白桦脂酸,桦木酸,ALS-357,Lupatic acid,Betulic acid	Apoptosis; Mitophagy; NF-κB; HIV Protease; Topoisomerase; Endogenous Metabolite; Aminopeptidase; Autophagy	Apoptosis; Autophagy; DNA Damage/DNA Repair; Metabolism; Microbiology/Virology; NF-κB; Proteases/Proteasome
	Betulinic acid (ALS-357) 是从白桦树皮中分离出来的一种五环三萜类天然产物，是真核细胞拓扑异构酶 I 的抑制剂，IC50值为 5 μM，具有抗逆转录病毒、抗疟疾、抗癌和抗炎特性。
T7203	Oglufanide 奥谷法奈,L-Glutamyl-L-tryptophan,H-Glu-Trp-OH	VEGFR; HCV Protease; Endogenous Metabolite	Angiogenesis; Metabolism; Microbiology/Virology; Proteases/Proteasome; Tyrosine Kinase/Adaptors
	Oglufanide (H-Glu-Trp-OH) 是一种从小牛胸腺中分离出来的二肽免疫调节剂，可抑制血管内皮生长因子，可刺激细胞内细菌感染和对丙型肝炎病毒的免疫反应。
T2775	Baicalin 黄芩苷,黄岑苷,Baicalein 7-O-β-D-glucuronide	NF-κB; HIV Protease; GABA Receptor; Autophagy	Autophagy; Membrane transporter/Ion channel; Microbiology/Virology; Neuroscience; NF-κB; Proteases/Proteasome
	Baicalin (Baicalein 7-O-β-D-glucuronide) 是一种从黄芩中分离出来的脯氨酰内肽酶抑制剂，具有抗氧化、抗肿瘤、抗 HIV 的特性。
T6S2391	L-Chicoric Acid (-)-Chicoric acid,trans-Caffeoyltartaric acid,Chicoric acid,L-菊苣酸,dicaffeoyltartaric acid,菊苣酸	Others; HIV Protease	Microbiology/Virology; Others; Proteases/Proteasome
	L-Chicoric Acid (trans-Caffeoyltartaric acid) 是一种二咖啡酰酒石酸，是一种选择性可逆的 HIV-1 整合酶抑制剂，IC50约为 100 nM。它还可抑制 HIV-1 复制。
T0070	Pentoxifylline Oxpentifylline,PTX,己酮可可碱,BL-191	HIV Protease; PDE; Adenosine Receptor; Autophagy	Autophagy; GPCR/G Protein; Metabolism; Microbiology/Virology; Neuroscience; Proteases/Proteasome
	Pentoxifylline (PTX) 是一种具有口服活性的磷酸二酯酶非选择性抑制剂，具有免疫调节、抗炎、抗纤溶、抗增殖和血液流变学改善作用。它可研究周围血管疾病、脑血管疾病和其他一些涉及局部微循环缺陷的疾病。
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天然产物

β-CGRP, human acetate

Cat.No: TP2167

Synonym: β-CGRP, human acetate (101462-82-2 free),CGRP-II (Human) (acetate),Human β-CGRP acetate

Target: CGRP Receptor

Angiotensin II human

Cat.No: T7040

Synonym: DRVYIHPF,Angiotensin II,Hypertensin II,血管紧张素Ⅱ,Ang II,血管紧张素II

Target: Apoptosis, RAAS

γ-Globulins from human blood

Cat.No: T41030

Target: Others

β-Endorphin, human

Cat.No: T13433

Target: Others

Cat.No: T6377

Target: Apoptosis, Virus Protease, HIV Protease, Antibiotic, Autophagy

Cat.No: TN2283

Target: HIV Protease

Cat.No: T2S1040

Target: ERK, IL Receptor, BCL, p38 MAPK, TNF, NF-κB, Akt, Caspase, PI3K, JAK, JNK, STAT, mTOR

Cat.No: T3020

Target: Apoptosis, Others

PHYTOSPHINGOSINE

Cat.No: T9503

Target: Apoptosis

1-Methylxanthine

Cat.No: T10021

Target: Endogenous Metabolite

Cat.No: TQ0217

Synonym: 戈米辛G,戈米辛 G

Target: P450, HIV Protease

Larixyl acetate

Cat.No: TN4417

Target: Others

Ganoderic acid F

Cat.No: T11363

Target: Others

Erythromycin ethylsuccinate

Cat.No: T0474

Synonym: EES,琥乙红霉素

Target: ribosome, HIV Protease, Antibacterial, Antibiotic, Autophagy

Cat.No: Fr16741

Synonym: 2-吲哚酮,板蓝根,Indolin-2-one

Target: Others, HIV Protease

Cat.No: T2942

Synonym: Ficusin,Furocoumarin,补骨脂素,psoralene

Target: Apoptosis, Influenza Virus, HIV Protease, DNA/RNA Synthesis

Cat.No: TN2069

Synonym: 藏红花,苦番紅花素

Target: Apoptosis

1,2-Dipalmitoyl-sn-glycerol 3-phosphate sodium

Cat.No: T10005L

Target: Endogenous Metabolite

Cat.No: T5061

Synonym: 7,8-Dimethylalloxazine,光色素

Target: Apoptosis, Endogenous Metabolite

Cat.No: T2865

Synonym: Oleanic acid,Caryophyllin,齐墩果酸

Target: HIV Protease, Endogenous Metabolite, Antibiotic, Autophagy

Cat.No: T3822

Synonym: Bellidifoline,龙胆山酮酚,Bellidifolium,雏菊叶龙胆酮

Target: Others, HIV Protease

Cat.No: T0966

Synonym: 番泻苷A,NSC 112929,番泻苷 A

Target: MAO, HIV Protease

Cat.No: TN1103

Synonym: 山荷叶素,二叶草素

Target: ATPase, Proton pump, Influenza Virus, HIV Protease

Cat.No: T6841

Synonym: NSC9168,烟曲霉素,Amebacilin

Target: Others, HIV Protease, Antibiotic, Parasite

Cat.No: T8689

Synonym: CQ,氯喹

Target: SARS-CoV, TLR, HIV Protease, Antibiotic, Parasite, Autophagy

Cat.No: T8116

Synonym: 甘菊蓝,奥苷菊环,Bicyclo[5.3.0]Decapentaene

Target: Others, HIV Protease

Ganoderic acid D

Cat.No: T5S1133

Synonym: 灵芝酸D,灵芝酸 D

Target: Apoptosis, Sirtuin

Cat.No: T2177

Synonym: Kempferol,山柰酚,山奈酚,Robigenin

Target: Apoptosis, Estrogen Receptor/ERR, Mitophagy, Estrogen/progestogen Receptor, HIV Protease, Endogenous Metabolite, Parasite, Autophagy

Dimethyl fumarate

Cat.No: T0492

Synonym: 富马酸二甲酯,DMF

Target: Reactive Oxygen Species, HIV Protease, Nrf2, Endogenous Metabolite, Autophagy

Cat.No: TN2004

Synonym: 1,7-二羟基-2,3,8-三甲氧基-6-甲基蒽-9,10-二酮,决明素

Target: MAO, Monoamine Oxidase

Cat.No: T0437

Synonym: INO 495,NSC 20262,肌苷

Target: ROS, Endogenous Metabolite, Adenosine Receptor

Cat.No: T2S0731

Synonym: 三叶苷,三叶甙,P-Phlorizin

Target: Amylase

Cat.No: T2789

Synonym: 黄岑素,野黄芩苷,Breviscapin,Breviscapinun,Breviscapine,Scutellarein-7-glucuronide

Target: Akt, HIV Protease, STAT

Zingibroside R1

Cat.No: T4962

Synonym: Ginsenoside Z-R1,姜状三七皂苷R1,姜状三七苷R1

Target: HIV Protease

Megestrol acetate

Cat.No: T1284

Synonym: SC10363,醋酸甲地孕酮,BDH1298

Target: Glucocorticoid Receptor, Estrogen/progestogen Receptor, Progesterone Receptor, HIV Protease, Autophagy

Cat.No: T1131

Synonym: MK-933,伊维菌素

Target: Mitophagy, GluCls, P2X Receptor, SARS-CoV, HIV Protease, Antibiotic, Parasite, Autophagy, HSV

2-Hydroxycinnamic acid

Cat.No: T7991

Synonym: 邻羟基肉桂酸(邻香豆酸),(E)-3-(2-羟基苯基)丙烯酸

Target: Others, SARS-CoV, HIV Protease

Cat.No: T2728

Synonym: Dictamnolactone,Limonoic acid 3,19:16,17 dilactone,柠檬苦素,Obaculactone,Citrolimonin

Target: Apoptosis, HIV Protease, Endogenous Metabolite

3',4'-Dimethoxyflavone

Cat.No: TN2883

Target: Others, PARP

Cat.No: T3122

Synonym: Tetrandrine B,防己诺林碱,(+)-Limacine,Hanfangichin B,防己醇灵,(+)-Fangchinoline

Target: Apoptosis, FAK, HIV Protease, Autophagy

Cat.No: T16791

Synonym: Mallotoxin,NSC 56346,粗糠柴苦素,NSC 94525

Target: CaMK, Apoptosis, Others, HIV Protease, PKA, PKC, Autophagy

Cat.No: T3730

Synonym: NSC 363001,Gallicin,Gallic acid methyl ester,Gallincin,没食子酸甲酯

Target: Reactive Oxygen Species, HIV Protease, Reverse Transcriptase, Antibacterial

2'-FUCOSYLLACTOSE

Cat.No: TN6796

Synonym: 2'-Fucosyl-D-lactose,2'-岩藻糖基乳糖

Target: Others

Cat.No: T4P2931

Synonym: 9,12-octadecadienoic acid,亚油酸,α-亚油酸,acidelinoleique,9,12-Linoleic acid

Target: Others, Endogenous Metabolite

Cat.No: T5782

Synonym: YK FH312,MPC-4326,PA-457,贝韦立马

Target: HIV Protease

Cat.No: T2830

Synonym: 白桦脂酸,桦木酸,ALS-357,Lupatic acid,Betulic acid

Target: Apoptosis, Mitophagy, NF-κB, HIV Protease, Topoisomerase, Endogenous Metabolite, Aminopeptidase, Autophagy

Cat.No: T7203

Synonym: 奥谷法奈,L-Glutamyl-L-tryptophan,H-Glu-Trp-OH

Target: VEGFR, HCV Protease, Endogenous Metabolite

Cat.No: T2775

Synonym: 黄芩苷,黄岑苷,Baicalein 7-O-β-D-glucuronide

Target: NF-κB, HIV Protease, GABA Receptor, Autophagy

L-Chicoric Acid

Cat.No: T6S2391

Synonym: (-)-Chicoric acid,trans-Caffeoyltartaric acid,Chicoric acid,L-菊苣酸,dicaffeoyltartaric acid,菊苣酸

Target: Others, HIV Protease

Cat.No: T0070

Synonym: Oxpentifylline,PTX,己酮可可碱,BL-191

Target: HIV Protease, PDE, Adenosine Receptor, Autophagy

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Species：

Expression System：

Tag：

Cat. No.	Product Name	Species	Expression System
TMPY-00811	Human cytomegalovirus (HCMV) Glycoprotein B/gB Protein Human cytωlovirus (HCMV) Glycoprotein B/gB	CMV	HEK293 Cells
	Human cytomegalovirus (HCMV) Glycoprotein B/gB Protein is expressed in HEK293 mammalian cells. The predicted molecular weight is 92 kDa and the accession number is P13201.
TMPY-01201	Human cytomegalovirus (HCMV) Glycoprotein B/gB Protein (His) Human cytωlovirus (HCMV) Glycoprotein B/gB	CMV	HEK293 Cells
	Human cytomegalovirus (HCMV) Glycoprotein B/gB Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 93.2 kDa and the accession number is P13201.
TMPH-03764	YAP1 Protein, Human, Recombinant (His) YAP1-2gamma,YAP2L,YAP65	Human	P. pastoris (Yeast)
	Transcriptional regulator which can act both as a coactivator and a corepressor and is the critical downstream regulatory target in the Hippo signaling pathway that plays a pivotal role in organ size control and tumor suppression by restricting proliferation and promoting apoptosis. The core of this pathway is composed of a kinase cascade wherein STK3/MST2 and STK4/MST1, in complex with its regulatory protein SAV1, phosphorylates and activates LATS1/2 in complex with its regulatory protein MOB1,...
TMPH-00007	HMGCR Protein, Human, Recombinant (His) HMGCR,3-hydroxy-3-methylglutaryl-coenzyme A reductase	Human	E. coli
	Catalyzes the conversion of (3S)-hydroxy-3-methylglutaryl-CoA (HMG-CoA) to mevalonic acid, the rate-limiting step in the synthesis of cholesterol and other isoprenoids, thus plays a critical role in cellular cholesterol homeostasis. HMGCR is the main target of statins, a class of cholesterol-lowering drugs.
TMPH-00009	OGT Protein, Human, Recombinant (His & SUMO) OGT,O-GlcNAc transferase subunit p110,O-linked N-acetylgluco...	Human	E. coli
	OGT Protein, Human, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 62.5 kDa and the accession number is O15294.
TMPH-00010	MMP-14 Protein, Human, Recombinant (His & SUMO) Membrane-type-1 matrix metalloproteinase,MMP14,Membrane-type...	Human	E. coli
	Endopeptidase that degrades various components of the extracellular matrix such as collagen. Activates progelatinase A. Essential for pericellular collagenolysis and modeling of skeletal and extraskeletal connective tissues during development. May be involved in actin cytoskeleton reorganization by cleaving PTK7. Acts as a positive regulator of cell growth and migration via activation of MMP15. Involved in the formation of the fibrovascular tissues in association with pro-MMP2. Cleaves ADGRB1 to...
TMPY-00810	Human cytomegalovirus (HCMV) Glycoprotein B/gB Protein (hFc) Human cytωlovirus (HCMV) Glycoprotein B/gB	CMV	HEK293 Cells
	Human cytomegalovirus (HCMV) Glycoprotein B/gB Protein (hFc) is expressed in HEK293 mammalian cells with Fc tag. The predicted molecular weight is 118 kDa and the accession number is P13201.
TMPJ-01470	SCF Protein, Human, Recombinant Mast Cell Growth Factor,c-Kit ligand,KITLG,MGF,Stem Cell Fac...	Human	E. coli
	Stem Cell Factor (SCF) is a hematopoietic growth factor that exerts its activity at the early stages of hematopoiesis. SCF stimulates the proliferation of myeloid, erythroid, and lymphoid progenitors in bone marrow cultures and has been shown to act synergistically with colony stimulating factors.
TMPY-00812	Human cytomegalovirus (HCMV) Glycoprotein B/gB Protein (aa 1-700, hFc) Human cytωlovirus (HCMV) Glycoprotein B/gB	CMV	HEK293 Cells
	Human cytomegalovirus (HCMV) Glycoprotein B/gB Protein (aa 1-700, hFc) is expressed in HEK293 mammalian cells with Fc tag. The predicted molecular weight is 104 kDa and the accession number is P13201.
TMPK-01466	HLA-A02:01&B2M&HPV 16 E6 (KLPQLCTEL) Tetramer Protein, Human, MHC (His & Avi) Human* papillomavirus type 16,E6,HPV16	Human	HEK293 Cells
	Human papillomavirus (HPV) 16 infection is a necessary condition for the pathogenesis and development of cervical cancer. The E6 protein is expressed by the HPV16 E6 gene and promotes malignant phenotype transformation, which is an important mechanism for the occurrence and development of cervical cancer.
TMPK-01467	HLA-A02:01&B2M&HPV 16 E6 (KLPQLCTEL) Monomer Protein, Human, MHC (His & Avi) HPV16,E6,Human* papillomavirus type 16	Human	HEK293 Cells
	Human papillomavirus (HPV) 16 infection is a necessary condition for the pathogenesis and development of cervical cancer. The E6 protein is expressed by the HPV16 E6 gene and promotes malignant phenotype transformation, which is an important mechanism for the occurrence and development of cervical cancer.
TMPJ-01471	Activin A Protein, Human, Mouse, Rat, Cynomolgus, Rhesus, Recombinant Activin A,INHBA,Inhibin beta A chain,Inhibin β A chain	Human/Mouse/Rat	HEK293 Cells
	Activin and inhibin are two closely related protein complexes that have almost directly opposite biological effects. Activins, members of the TGF-beta superfamily, are disulfide-linked dimeric proteins originally purified from gonadal fluids as proteins that stimulated pituitary follicle stimulating hormone (FSH) release. Inhibins/activins are involved in regulating a number of diverse functions such as hypothalamic and pituitary hormone secretion, gonadal hormone secretion, germ cell developm...
TMPH-01773	ELANE Protein, Human, Recombinant (GST) Neutrophil elastase,ELA2,Medullasin,Elastase-2,ELANE,Bone ma...	Human	E. coli
	Modifies the functions of natural killer cells, monocytes and granulocytes. Inhibits C5a-dependent neutrophil enzyme release and chemotaxis. Capable of killing E.coli but not S.aureus in vitro; digests outer membrane protein A (ompA) in E.coli and K.pneumoniae. ELANE Protein, Human, Recombinant (GST) is expressed in E. coli expression system with N-GST tag. The predicted molecular weight is 52.6 kDa and the accession number is P08246.
TMPH-01488	HLA-B Protein, Human, Recombinant (E. coli, His) HLA-B,Human leukocyte antigen B,HLA class I histoco...	Human	E. coli
	HLA-B Protein, Human, Recombinant (E. coli, His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 38.9 kDa and the accession number is P01889.
TMPJ-00541	CD177 Protein, Human, Recombinant (His) PRV-1,HNA-2a,Human Neutrophil Alloantigen 2a,CD177,...	Human	HEK293 Cells
	CD177 is polymorphic and has at least two alleles: PRV1 and NB1. Human PRV1 is a Glycosyl-Phosphatidylinositol (GPI)-linked cell surface glycoprotein that belongs to the uPAR/CD59/Ly6 family of receptors. PRV1 is expressed by neutrophils and neutrophil precursors,and changes in expression serve as diagnostic markers for myeloproliferative disorders such as polycythemia vera and essential thrombocythemia. PRV1 may also be expressed by Erythroblasts, B cells, and Monocytes. NB1, a Glycosyl-Phospha...
TMPJ-01099	IL-15RA Protein, Human, Recombinant (hFc, Human Cells) interleukin-15 receptor subunit α,IL15RA,interleukin-15 rece...	Human	HEK293 Cells
	Interleukin 15 Receptor alpha (IL-15Rα) is a transmembrane glycoprotein that plays a pleiotropic role in immune development and function, including the positive maintenance of lymphocyte homeostasis. IL-15Rα chain can bind soluble IL-15 and “transpresent” cytokine to the cells, allowing them to respond to IL-15. Soluble IL-15Rα can function as a specific high-affinity IL-15 antagonist. The soluble IL-15/IL-15Rα complexes exhibit a strong agonistic activity which is mediated through membrane-boun...
TMPH-01070	CD177 Protein, Human, Recombinant (GST & His) Human neutrophil alloantigen 2a,CD177,PRV1,Polycyth...	Human	E. coli
	CD177 Protein, Human, Recombinant (GST & His) is expressed in E. coli expression system with N-6xHis-GST tag. The predicted molecular weight is 63.6 kDa and the accession number is Q8N6Q3.
TMPH-02019	REG3A Protein, Human, Recombinant (GST) Regenerating islet-derived protein 3-alpha,REG3A,Regeneratin...	Human	E. coli
	Bactericidal C-type lectin which acts exclusively against Gram-positive bacteria and mediates bacterial killing by binding to surface-exposed carbohydrate moieties of peptidoglycan. Regulates keratinocyte proliferation and differentiation after skin injury via activation of EXTL3-PI3K-AKT signaling pathway. REG3A Protein, Human, Recombinant (GST) is expressed in E. coli expression system with N-GST tag. The predicted molecular weight is 43.6 kDa and the accession number is Q06141.
TMPU-00003	STAT2 Protein, Human, Recombinant (His)	Human	E. coli
	Signal transducer and activator of transcription that mediates signaling by type I IFNs (IFN-alpha and IFN-beta). Following type I IFN binding to cell surface receptors, Jak kinases (TYK2 and JAK1) are activated, leading to tyrosine phosphorylation of STAT1 and STAT2. The phosphorylated STATs dimerize, associate with ISGF3G/IRF-9 to form a complex termed ISGF3 transcription factor, that enters the nucleus. ISGF3 binds to the IFN stimulated response element (ISRE) to activate the transcription of...
TMPZ-00006	SPINK9 Protein, Human, Recombinant (His) LEKTI2	Human	HEK298 Cells
	SPINK9 specifically inhibits KLK5, which may contribute to the regulation of the desquamation process in skin by inhibiting KLK5. SPINK9 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 7.37 kDa and the accession number is Q5DT21.
TMPY-02881	RAGE Protein, Human, Recombinant RAGE,advanced glycosylation end product-specific receptor	Human	HEK293 Cells
	RAGE Protein, Human, Recombinant is expressed in HEK293 mammalian cells. The predicted molecular weight is 35 kDa and the accession number is A0A1U9X785.
TMPY-04330	Mer Protein, Human, Recombinant MER proto-oncogene, tyrosine kinase,RP38,MER,c-mer,Tyro12,c-...	Human	HEK293 Cells
	Mer Protein, Human, Recombinant is expressed in HEK293 mammalian cells. The predicted molecular weight is 54 kDa and the accession number is Q12866.
TMPY-01010	NGF Protein, Human, Recombinant Beta-NGF,神经生长因子,β-NGF,NGFB,nerve growth factor (β polypeptid...	Human	CHO Cells
	NGF Protein, Human, Recombinant is expressed in CHO mammalian cells. The predicted molecular weight is 13.2 kDa and the accession number is P01138.
TMPY-00132	Mesothelin Protein, Human, Recombinant MPF,SMRP,Mesothelin	Human	HEK293 Cells
	Mesothelin Protein, Human, Recombinant is expressed in HEK293 mammalian cells. The predicted molecular weight is 32.4 kDa and the accession number is Q13421-3.
TMPY-04104	LIF Protein, Human, Recombinant CDF,DIA,白血病抑制因子,MLPLI,Leukemia Inhibitory Factor,HILDA	Human	HEK293 Cells
	LIF Protein, Human, Recombinant is expressed in HEK293 mammalian cells. The predicted molecular weight is 19.7 kDa and the accession number is P15018-1.
TMPY-02327	HGF Protein, Human, Recombinant SF,hepatocyte growth factor (hepapoietin A,HGFB,F-TCF,F-TCFB...	Human	CHO Cells
	HGF Protein, Human, Recombinant is expressed in CHO mammalian cells. The predicted molecular weight is 79.7 kDa and the accession number is P14210-1.
TMPY-01560	EGF Protein, Human, Recombinant URG,epidermal growth factor,表皮生长因子,HOMG4	Human	E. coli
	EGF Protein, Human, Recombinant is expressed in E. coli expression system. The predicted molecular weight is 6.35 kDa and the accession number is P01133-1.
TMPJ-01430	NovoNectin Protein, Human, Recombinant NovoNectin,Cold-insoluble globulin,FN,CIG,Fibronectin,Fibron...	Human	E. coli
	Fibronectin1(FN1) is a secreted protein and contains 12 fibronectin type-I domains,fibronectin type-II domains and 16 fibronectin type-III domains.Recombinant human fibronectin fragment, is a protein of ~63 kDa containing a central cell-binding domain, a high affinity heparin-binding domain II,and CS1 site within the alternatively spliced III CS region of human fibronectin. Cells bind to a VLA-4 ligand, a CS-I site, and a VLA-5 ligand, a cell attachment domain, and virus vectors binds to a hepar...
TMPY-03484	TCPTP Protein, Human, Recombinant TCPTP,protein tyrosine phosphatase, non-receptor type 2,PTPT...	Human	Baculovirus Insect Cells
	TCPTP Protein, Human, Recombinant is expressed in Baculovirus insect cells. The predicted molecular weight is 36.8 kDa and the accession number is P17706-1.
TMPJ-00042	TSLP Protein, Human, Recombinant TSLP,Thymic stromal lymphopoietin	Human	E. coli
	Thymic stromal lymphopoietin (TSLP) is a novel member of the hemopoietic cytokine family that promotes the development of B cells and shares overlapping activity with IL-7. The human TSLP protein comprises a 28 amino acids (aa) signal sequence and 131 aa mature region. Human TSLP has two isoforms lfTSLP and sfTSLP produced by alternative splicing . lfTSLP is expressed in a number of tissues including heart, liver and prostate, and sfTSLP (63aa) is predominantly expressed in keratinocytes of oral...
TMPY-03782	Albumin Protein, Human, Recombinant PRO0883,albumin,FDAH,PRO0903,PRO1341,ANALBA	Human	P. pastoris (Yeast)
	Albumin Protein, Human, Recombinant is expressed in yeast. The predicted molecular weight is 66.4 kDa and the accession number is P02768-1.
TMPY-00875	Leptin Protein, Human, Recombinant OBS,leptin,OB,LEPD	Human	E. coli
	Leptin Protein, Human, Recombinant is expressed in E. coli expression system. The predicted molecular weight is 16 kDa and the accession number is A4D0Y8.
TMPY-00395	Insulin Protein, Human, Recombinant IDDM1,MODY10,ILPR,IDDM2,IRDN,IDDM,insulin,INS	Human	P. pastoris (Yeast)
	INS (Insulin) is a Protein Coding gene. This gene encodes insulin, a peptide hormone that plays a vital role in the regulation of carbohydrate and lipid metabolism. After removal of the precursor signal peptide, proinsulin is post-translationally cleaved into three peptides: the B chain and A chain peptides, which are covalently linked via two disulfide bonds to form insulin, and C-peptide. The binding of insulin to the insulin receptor (INSR) stimulates glucose uptake. Diseases associated with ...
TMPZ-00004	DNAJC16 Protein, Human, Recombinant (His) ERDJ8,KIAA0962	Human	HEK296 Cells
	DNAJC16 plays an important role in regulating the size of autophagosomes during the formation process. DNAJC16 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 24.86 kDa and the accession number is Q9Y2G8.
TMPZ-00001	Endothelin-3 Protein, Human, Recombinant (His) Preproendothelin-3,PPET3	Human	HEK293 Cells
	Endothelins are endothelium-derived vasoconstrictor peptides. Endothelin-3 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 24.42 kDa and the accession number is P14138.
TMPZ-00005	Carboxypeptidase Q Protein, Human, Recombinant (His) PGCP,LCH1	Human	HEK297 Cells
	CPQ may play an important role in the hydrolysis of circulating peptides. Catalyzes the hydrolysis of dipeptides with unsubstituted terminals into amino acids. May play a role in the liberation of thyroxine hormone from its thyroglobulin (Tg) precursor. Carboxypeptidase Q Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 49.72 kDa and the accession number is Q9Y646.
TMPH-01632	MRC1 Protein, Human, Recombinant (His) Human mannose receptor,C-type lectin domain family ...	Human	E. coli
	Mediates the endocytosis of glycoproteins by macrophages. Binds both sulfated and non-sulfated polysaccharide chains.; (Microbial infection) Acts as phagocytic receptor for bacteria, fungi and other pathogens.; (Microbial infection) Acts as a receptor for Dengue virus envelope protein E.; (Microbial infection) Interacts with Hepatitis B virus envelope protein. MRC1 Protein, Human, Recombinant (His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 69.9...
TMPK-00419	PDGF R alpha/PDGFRA Protein, Human, Recombinant (His & Avi) RHEPDGFRA,PDGFR-2,CD140A,PDGFR2,MGC74795,PDGF R α/PDGFRA Pro...	Human	HEK293 Cells
	Platelet-derived growth factor is commonly known as a mitogen. Many research data suggest a role for PDGF-beta R in the mitogenic response of mesangial cells. There are four members of PDGF family known as PDGF-A chain, PDGF-B chain, PDGF-C chain and PDGF-D chain, which in active forms are dimers. As far as two receptors PDGF-alpha R and PDGF-beta R are known to bind PDGF. PDGF R alpha/PDGFRA Protein, Human, Recombinant (His & Avi) is expressed in HEK293 mammalian cells with C-His-Avi tag. The p...
TMPY-00749	FGF-2 Protein, Human, Recombinant fibroblast growth factor 2 (basic),FGF-2,FGFB,HBGF-2,BFGF	Human	E. coli
	FGF-2 Protein, Human, Recombinant is expressed in E. coli expression system. The predicted molecular weight is 16.5 kDa and the accession number is P09038-4.
TMPY-04803	DLL4 Protein, Human, Recombinant δ-like 4 (Drosophila),delta-like 4 (Drosophila),Delta-like 4...	Human	HEK293 Cells
	DLL4 Protein, Human, Recombinant is expressed in HEK293 mammalian cells. The predicted molecular weight is 55 kDa and the accession number is Q9NR61.
TMPY-03441	SAE1 Protein, Human, Recombinant SUA1,SUMO1 activating enzyme subunit 1,HSPC140,UBLE1A,AOS1	Human	Baculovirus Insect Cells
	SAE1 Protein, Human, Recombinant is expressed in Baculovirus insect cells. The predicted molecular weight is 38.6 kDa and the accession number is Q9UBE0.
TMPY-04751	VRK1 Protein, Human, Recombinant PCH1,vaccinia related kinase 1,PCH1A	Human	Baculovirus Insect Cells
	VRK1 Protein, Human, Recombinant is expressed in Baculovirus insect cells. The predicted molecular weight is 45.6 kDa and the accession number is Q99986.
TMPY-03274	CXCL11 Protein, Human, Recombinant SCYB9B,I-TAC,chemokine (C-X-C motif) ligand 11,H174,SCYB11,I...	Human	E. coli
	I-TAC, also known as CXCL11, is a small cytokine belonging to the CXC chemokine family. It is highly expressed in peripheral blood leukocytes, pancreas and liver, with moderate levels in thymus, spleen and lung and low expression levels were in small intestine, placenta and prostate. The I-TAC chemokine elicits its effects on its target cells by interacting with the cell surface chemokine receptor CXCR3, with a higher affinity than do the other ligands for this receptor, CXCL9 and CXCL10. I-TAC ...
TMPJ-00915	HSP40 Protein, Human, Recombinant (His) HDJ1,HSPF1,DNAJ1,Heat Shock 40 kDa Protein 1,HSP40,hDj-1,DNA...	Human	E. coli
	DnaJ Homolog Subfamily B Member 1 (DNAJB1) is a member of the heat shock protein family. Heat shock proteins (HSPs) are a highly conserved family of stress response proteins. HSPs function primarily as molecular chaperones, facilitating the folding of other cellular proteins, preventing protein aggregation, or targeting improperly folded proteins to specific degradative pathways. DNAJB1 regulates cellular processes by aiding in the folding, transport and assembly. DNAJB1 contains a J-domain whic...
TMPK-00420	PDGF R alpha/PDGFRA Protein, Human, Recombinant (His & Avi), Biotinylated RHEPDGFRA,PDGFRA,PDGF R α/PDGFRA Protein, Human, Re...	Human	HEK293 Cells
	Platelet-derived growth factor is commonly known as a mitogen. Many research data suggest a role for PDGF-beta R in the mitogenic response of mesangial cells. There are four members of PDGF family known as PDGF-A chain, PDGF-B chain, PDGF-C chain and PDGF-D chain, which in active forms are dimers. As far as two receptors PDGF-alpha R and PDGF-beta R are known to bind PDGF. PDGF R alpha/PDGFRA Protein, Human, Recombinant (His & Avi), Biotinylated is expressed in HEK293 mammalian cells with C-His-...
TMPY-03432	KEAP1 Protein, Human, Recombinant kelch like ECH associated protein 1,INRF2,KLHL19,KEAP-1	Human	Baculovirus Insect Cells
	KEAP1 Protein, Human, Recombinant is expressed in Baculovirus insect cells. The predicted molecular weight is 69.7 kDa and the accession number is Q14145.
TMPY-03050	CXCL5 Protein, Human, Recombinant ENA-78,SCYB5,chemokine (C-X-C motif) ligand 5	Human	E. coli
	CXCL5 Protein, Human, Recombinant is expressed in E. coli expression system. The predicted molecular weight is 7.8 kDa and the accession number is P42830.
TMPY-03890	CD81 Protein, Human, Recombinant S5.7,CVID6,TSPAN28,TAPA1,CD81 molecule	Human	HEK293 Cells
	CD81 Protein, Human, Recombinant is expressed in HEK293 mammalian cells. The predicted molecular weight is 9.9 kDa and the accession number is A0A024RCB7.
TMPY-04018	LRG1 Protein, Human, Recombinant HMFT1766,leucine-rich α-2-glycoprotein 1,LRG,leucine-rich al...	Human	HEK293 Cells
	LRG1 Protein, Human, Recombinant is expressed in HEK293 mammalian cells. The predicted molecular weight is 35.1 kDa and the accession number is AAH34389.1.
TMPY-04683	CD47 Protein, Human, Recombinant MER6,CD47 molecule,OA3,IAP	Human	HEK293 Cells
	CD47 Protein, Human, Recombinant is expressed in HEK293 mammalian cells. The predicted molecular weight is 14.5 kDa and the accession number is Q08722-3.
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重组蛋白

Human cytomegalovirus (HCMV) Glycoprotein B/gB Protein

Cat.No: TMPY-00811

Species: CMV

Expression System: HEK293 Cells

Human cytomegalovirus (HCMV) Glycoprotein B/gB Protein (His)

Cat.No: TMPY-01201

Species: CMV

Expression System: HEK293 Cells

YAP1 Protein, Human, Recombinant (His)

Cat.No: TMPH-03764

Species: Human

Expression System: P. pastoris (Yeast)

HMGCR Protein, Human, Recombinant (His)

Cat.No: TMPH-00007

Species: Human

Expression System: E. coli

OGT Protein, Human, Recombinant (His & SUMO)

Cat.No: TMPH-00009

Species: Human

Expression System: E. coli

MMP-14 Protein, Human, Recombinant (His & SUMO)

Cat.No: TMPH-00010

Species: Human

Expression System: E. coli

Human cytomegalovirus (HCMV) Glycoprotein B/gB Protein (hFc)

Cat.No: TMPY-00810

Species: CMV

Expression System: HEK293 Cells

SCF Protein, Human, Recombinant

Cat.No: TMPJ-01470

Species: Human

Expression System: E. coli

Human cytomegalovirus (HCMV) Glycoprotein B/gB Protein (aa 1-700, hFc)

Cat.No: TMPY-00812

Species: CMV

Expression System: HEK293 Cells

HLA-A*02:01&B2M&HPV 16 E6 (KLPQLCTEL) Tetramer Protein, Human, MHC (His & Avi)

Cat.No: TMPK-01466

Species: Human

Expression System: HEK293 Cells

HLA-A*02:01&B2M&HPV 16 E6 (KLPQLCTEL) Monomer Protein, Human, MHC (His & Avi)

Cat.No: TMPK-01467

Species: Human

Expression System: HEK293 Cells

Activin A Protein, Human, Mouse, Rat, Cynomolgus, Rhesus, Recombinant

Cat.No: TMPJ-01471

Species: Human/Mouse/Rat

Expression System: HEK293 Cells

ELANE Protein, Human, Recombinant (GST)

Cat.No: TMPH-01773

Species: Human

Expression System: E. coli

HLA-B Protein, Human, Recombinant (E. coli, His)

Cat.No: TMPH-01488

Species: Human

Expression System: E. coli

CD177 Protein, Human, Recombinant (His)

Cat.No: TMPJ-00541

Species: Human

Expression System: HEK293 Cells

IL-15RA Protein, Human, Recombinant (hFc, Human Cells)

Cat.No: TMPJ-01099

Species: Human

Expression System: HEK293 Cells

CD177 Protein, Human, Recombinant (GST & His)

Cat.No: TMPH-01070

Species: Human

Expression System: E. coli

REG3A Protein, Human, Recombinant (GST)

Cat.No: TMPH-02019

Species: Human

Expression System: E. coli

STAT2 Protein, Human, Recombinant (His)

Cat.No: TMPU-00003

Species: Human

Expression System: E. coli

SPINK9 Protein, Human, Recombinant (His)

Cat.No: TMPZ-00006

Species: Human

Expression System: HEK298 Cells

RAGE Protein, Human, Recombinant

Cat.No: TMPY-02881

Species: Human

Expression System: HEK293 Cells

Mer Protein, Human, Recombinant

Cat.No: TMPY-04330

Species: Human

Expression System: HEK293 Cells

NGF Protein, Human, Recombinant

Cat.No: TMPY-01010

Species: Human

Expression System: CHO Cells

Mesothelin Protein, Human, Recombinant

Cat.No: TMPY-00132

Species: Human

Expression System: HEK293 Cells

LIF Protein, Human, Recombinant

Cat.No: TMPY-04104

Species: Human

Expression System: HEK293 Cells

HGF Protein, Human, Recombinant

Cat.No: TMPY-02327

Species: Human

Expression System: CHO Cells

EGF Protein, Human, Recombinant

Cat.No: TMPY-01560

Species: Human

Expression System: E. coli

NovoNectin Protein, Human, Recombinant

Cat.No: TMPJ-01430

Species: Human

Expression System: E. coli

TCPTP Protein, Human, Recombinant

Cat.No: TMPY-03484

Species: Human

Expression System: Baculovirus Insect Cells

TSLP Protein, Human, Recombinant

Cat.No: TMPJ-00042

Species: Human

Expression System: E. coli

Albumin Protein, Human, Recombinant

Cat.No: TMPY-03782

Species: Human

Expression System: P. pastoris (Yeast)

Leptin Protein, Human, Recombinant

Cat.No: TMPY-00875

Species: Human

Expression System: E. coli

Insulin Protein, Human, Recombinant

Cat.No: TMPY-00395

Species: Human

Expression System: P. pastoris (Yeast)

DNAJC16 Protein, Human, Recombinant (His)

Cat.No: TMPZ-00004

Species: Human

Expression System: HEK296 Cells

Endothelin-3 Protein, Human, Recombinant (His)

Cat.No: TMPZ-00001

Species: Human

Expression System: HEK293 Cells

Carboxypeptidase Q Protein, Human, Recombinant (His)

Cat.No: TMPZ-00005

Species: Human

Expression System: HEK297 Cells

MRC1 Protein, Human, Recombinant (His)

Cat.No: TMPH-01632

Species: Human

Expression System: E. coli

PDGF R alpha/PDGFRA Protein, Human, Recombinant (His & Avi)

Cat.No: TMPK-00419

Species: Human

Expression System: HEK293 Cells

FGF-2 Protein, Human, Recombinant

Cat.No: TMPY-00749

Species: Human

Expression System: E. coli

DLL4 Protein, Human, Recombinant

Cat.No: TMPY-04803

Species: Human

Expression System: HEK293 Cells

SAE1 Protein, Human, Recombinant

Cat.No: TMPY-03441

Species: Human

Expression System: Baculovirus Insect Cells

VRK1 Protein, Human, Recombinant

Cat.No: TMPY-04751

Species: Human

Expression System: Baculovirus Insect Cells

CXCL11 Protein, Human, Recombinant

Cat.No: TMPY-03274

Species: Human

Expression System: E. coli

HSP40 Protein, Human, Recombinant (His)

Cat.No: TMPJ-00915

Species: Human

Expression System: E. coli

PDGF R alpha/PDGFRA Protein, Human, Recombinant (His & Avi), Biotinylated

Cat.No: TMPK-00420

Species: Human

Expression System: HEK293 Cells

KEAP1 Protein, Human, Recombinant

Cat.No: TMPY-03432

Species: Human

Expression System: Baculovirus Insect Cells

CXCL5 Protein, Human, Recombinant

Cat.No: TMPY-03050

Species: Human

Expression System: E. coli

CD81 Protein, Human, Recombinant

Cat.No: TMPY-03890

Species: Human

Expression System: HEK293 Cells

LRG1 Protein, Human, Recombinant

Cat.No: TMPY-04018

Species: Human

Expression System: HEK293 Cells

CD47 Protein, Human, Recombinant

Cat.No: TMPY-04683

Species: Human

Expression System: HEK293 Cells

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Cat. No.	Product Name	Target	Signaling Pathways
T11655	Indomethacin-D4 Indometacin-D4,吲哚美辛-D4	CDK	Cell Cycle/Checkpoint
	Indomethacin-D4 is a deuterium labeled Indomethacin. Indomethacin is a potent and nonselective inhibitor of COX1 and COX2, with IC50s of 18 nM and 26 nM for human COX-1 and COX-2, respectively, in CHO cells.
TMIH-0521	Silibinin-d3
	Silibinin-d3 是 Silibinin 的氘代化合物。Silibinin 的 CAS 号为 22888-70-6。Silibinin 是水飞蓟的主要活性成分，具有抗癌和化疗预防作用，能抑制细胞增殖和迁移。
T12638	(R)-Praziquantel-d11 (R)-吡喹酮 D11,(R)-Praziquantel D11	5-HT Receptor	GPCR/G Protein; Neuroscience
	(R)-Praziquantel D11 is the deuterium labeled (R)-Praziquantel. (R)-Praziquantel is the active enantiomer of Praziquantel, is a partial the human 5-HT2B receptor agonist
T13291	VD3-D6 Vitamin D3-26,26,26,27,27,27-d6	Others	Others
	VD3-D6 is the deuterated form of Vitamin D3; tools for determination of Vitamin D3 metabolites in human serum.
T19489	O-Desmethyl gefitinib D8	EGFR	Angiogenesis; JAK/STAT signaling; Tyrosine Kinase/Adaptors
	O-Desmethyl gefitinib D8 is a deuterium labeled O-Desmethyl gefitinib that is an active metabolite of Gefitinib in human plasma.
T10368	Aripiprazole (D8) OPC-14597 D8	Others	Others
	Aripiprazole D8 (OPC-14597 D8) is the deuterium-labeled Aripiprazole. Aripiprazole is a human 5-HT1A receptor partial agonist (Ki: 4.2 nM).
T12487	Piroxicam D3 吡罗昔康 D3,CP-16171 D3	Others	Others
	Piroxicam D3 is deuterium labeled Piroxicam. Piroxicam is a COX inhibitor(human monocyte COX-1 and COX-2 with IC50s of 47, 25 μM , respectively) .
T11229	Erlotinib-d6 OSI-774 D6,NSC 718781 D6,CP-358774 D6	Others	Others
	Erlotinib is a directly acting inhibitor EGFR tyrosine kinase inhibitor with an IC50 of 2 nM for human EGFR. Erlotinib D6 is a deuterium labeled Erlotinib .
T70615	TAS-303
	TAS-303 is a selective norepinephrine reuptake inhibitor which displays significant norepinephrine transporter (NET) inhibitory activity toward serotonin or dopamine transporters. Radioligand-binding studies showed that TAS-303 selectively and potently inhibited [3H]norepinephrine binding to the human NET.
T71300	Pentoxifylline-d6
	Pentoxifylline-d6 is intended for use as an internal standard for the quantification of pentoxifylline by GC- or LC-MS. Pentoxifylline is a hemorrheologic agent. It increases the deformability of washed isolated human erythrocytes when used at a concentration of 100 µM. Pentoxifylline (1, 2, and 3 mM) inhibits ADP-induced platelet aggregation in isolated human whole blood. It inhibits thrombus formation induced by ADP in a hamster cheek pouch model when administered at doses of 5, 10, and 20 mg/...
T10349	Apixaban 13C,d3 Apixaban 13CD3,BMS-562247-01 13CD3	Others	Others
	Apixaban 13CD3 (BMS-562247-01 13CD3) is a deuterium-labeled Apixaban. Apixaban is a reversible inhibitor of Factor Xa (Ki: 0.08 nM and 0.17 nM in human and rabbit).
T10610	Brexpiprazole-d8 OPC-34712 D8	Others	Others
	Brexpiprazole D8 (OPC-34712 D8) is a deuterium-labeled Brexpiprazole. Brexpiprazole is a partial agonist of human 5-HT1A and dopamine receptors (Ki: 0.12 nM and 0.3 nM).
T11995	Melatonin-d4 N-Acetyl-5-methoxytryptamine D5,Melatonin D5,褪黑素 D5	Others	Others
	Melatonin D5, a deuterium-labeled version of melatonin, is a hormone produced by the pineal gland, known for its role as a selective ATF-6 inhibitor that promotes apoptosis in human hepatoma cells via COX-2 downregulation. Additionally, it activates melatonin receptors and exhibits antioxidative and anti-inflammatory properties.
T11276	Fexofenadine-d6 MDL-16455-d6,Terfenadine carboxylate-d6	Histamine Receptor	GPCR/G Protein; Immunology/Inflammation; Neuroscience
	Fexofenadine-d6 (MDL-16455-d6) 是 Fexofenadine 的氘代物，可用做检测人血浆中非索非那定浓度的内标。
T10611	Brexpiprazole S-oxide D8 DM-3411 D8	Dopamine Receptor; 5-HT Receptor	GPCR/G Protein; Neuroscience
	Brexpiprazole S-oxide D8 (DM-3411 D8) is a deuterium labeled Brexpiprazole S-oxide. Brexpiprazole S-oxide is a main metabolite of Brexpiprazole. Brexpiprazole is a partial agonist of human 5-HT1A and dopamine receptors (Kis: 0.12 nM and 0.3 nM).
T11246	Etoricoxib-d4 MK-0663 D4,依托考昔 D4,L-791456 D4,Etoricoxib D4	Others	Others
	Etoricoxib D4 is a non steroidal anti-inflammatory agent, acting as a selective and orally active COX-2 inhibitor, with IC50s of 1.1 μM and 116 μM for COX-2 and COX-1 in human whole blood.Etoricoxib D4 is a deuterium labeled Etoricoxib.
T35695	Oleic Acid-13C
	Oleic acid-13C is intended for use as an internal standard for the quantification of oleic acid by GC- or LC-MS. Oleic acid is a monounsaturated fatty acid and a major component of membrane phospholipids that has been found in human plasma, cell membranes, and adipose tissue.1,2 It contributes approximately 17% of the total fatty acids esterified to phosphatidylcholine, the major phospholipid class in porcine platelets.1 Oleic acid inhibits collagen-stimulated platelet aggregation by approximate...
T71303	Flufenamic Acid-d4
	Flufenamic acid-d4 is intended for use as an internal standard for the quantification of flufenamic acid by GC- or LC-MS. Flufenamic acid is a non-steroidal anti-inflammatory drug (NSAID) and COX inhibitor (IC50s = 3 and 9.3 µM for human COX-1 and COX-2, respectively). Flufenamic acid inhibits TNF-α-induced increases in COX-2 levels and NF-κB activation in HT-29 colon cancer cells in a concentration-dependent manner. It inhibits calcium influx induced by fMLP or A23187 in human polymorphonuclear...
T35915	Erlotinib-13C6 Erlotinib-13C6
	Erlotinib-13C6 (CP-358774-13C6) is a 13C-labeled Erlotinib. Erlotinib is a directly acting EGFR tyrosine kinase inhibitor, with an IC50 of 2 nM for human EGFR[1]. Erlotinib reduces EGFR autophosphorylation in intact tumor cells with an IC50 of 20 nM. Erlotinib is used for the treatment of non-small cell lung cancer[1].Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process[2]...
TMIH-0359	Mycophenolic Acid-d3 Phenyl Glucuronide
	Mycophenolic Acid-d3 Phenyl Glucuronide 是 Mycophenolic Acid Phenyl Glucuronide 的氘代化合物。Mycophenolic Acid Phenyl Glucuronide 的 CAS 号为 31528-44-6。Mycophenolic acid glucuronide是人血浆中mycophenolic acid的葡糖甙代谢产物。
TMIJ-0434	p-Benzoquinone-d4
	p-Benzoquinone-d4 是 p-Benzoquinone 的氘代化合物。p-Benzoquinone 的 CAS 号为 106-51-4。p-Benzoquinone 是一种超氧化物清除剂。它是一种在人体血液中发现的有毒代谢物。
TMIJ-0456	Malathion-d7
	Malathion-d7 是 Malathion 的氘代化合物。Malathion 的 CAS 号为 121-75-5。Malathion 是一种杀虫剂，是一种有机磷酸酯的副交感神经药物，不可逆地与胆碱酯酶结合，具有相对较低的人体毒性。
TMIJ-0451	Malathion-d10
	Malathion-d10 是 Malathion 的氘代化合物。Malathion 的 CAS 号为 121-75-5。Malathion 是一种杀虫剂，是一种有机磷酸酯的副交感神经药物，不可逆地与胆碱酯酶结合，具有相对较低的人体毒性。
T73711	Atomoxetine-d3 hydrochloride
	Atomoxetine-d3 hydrochloride 是氘代标记的Atomoxetine hydrochloride。Atomoxetine hydrochloride 是去甲肾上腺素重吸收抑制剂，与人NET，SERT 和DAT 的放射性配体结合的 Ki 分别为5，77和1451 nM。
TMID-0010	Mavacamten-d6
	Mavacamten-d6 是 Mavacamten 的氘代化合物。Mavacamten 的 CAS 号为 1642288-47-8。MYK-461 是一种可口服的心肌肌球蛋白 ATP 酶抑制剂，在牛心脏和人心脏中的IC50值分别为 490和711 nM。
TMIH-0198	DM-3411-d8 Brexpiprazole Metabolite
	DM-3411-d8 是 DM-3411 的氘代化合物。DM-3411 的 CAS 号为 913611-97-9。Brexpiprazole是人5-HT1A和多巴胺受体的部分激动剂，Ki分别为0.12 和 0.3 nM。它也是5-HT2A受体的拮抗剂，Ki为 0.47 nM，可作为非典型抗精神病药。
T71326	1,3,7-Trimethyluric Acid-d9
	1,3,7-Trimethyluric acid-d9 is intended for use as an internal standard for the quantification of 1,3,7-trimethyluric acid by GC- or LC-MS. 1,3,7-Trimethyluric acid is a derivative of uric acid and a metabolite of caffeine. It is formed from caffeine by the cytochrome P450 isoform CYP3A4. 1,3,7-Trimethyluric acid scavenges hydroxyl radicals in a cell-free assay and inhibits t-butyl hydroperoxide-induced lipid peroxidation by 56.5% in isolated human erythrocyte membranes.
T73820	Bosentan-d4
	Bosentan-d4 是 Bosentan 的氘代物。Bosentan 是一种有效的endothelin-1 (ET)拮抗剂，在人的 SMC 细胞中，作用于ETA 和ETB 受体，Ki 值分别为 4.7 nM 和 95 nM。
TMIJ-0108	rac-Hesperetin-13C-d3 rac-Diosmin EP Impurity G-13C-d3
	rac-Hesperetin-13C-d3 是 rac-Hesperetin 的 13C 和氘代化合物。rac-Hesperetin 的 CAS 号为 69097-99-0。
T71893	Clobetasol Propionate-d5
	Clobetasol propionate-d5 is intended for use as an internal standard for the quantification of clobetasol propionate by GC- or LC-MS. Clobetasol propionate is a corticosteroid. It binds to glucocorticoid receptors in a cell-free assay and inhibits proliferation of primary human skin fibroblasts when used at a concentration of 5 µg/ml. Topical administration of clobetasol propionate reduces croton oil-induced ear edema in mice. Formulations containing clobetasol propionate have been used in the t...
T71302	Norfluoxetine-d5 HCl
	Norfluoxetine-d5 is intended for use as an internal standard for the quantification of norfluoxetine by GC- or LC-MS. Norfluoxetine is an active metabolite of the antidepressant fluoxetine. It is formed from fluoxetine by the cytochrome P450 (CYP) isoforms CYP2C9, CYP2C19, and CYP3A. Norfluoxetine inhibits serotonin (5-HT) uptake in rat brain synaptosomal membrane preparations (Ki = 44.7 nM) and isolated human platelets (IC50 = ~15 nM). It has been found in the tissues of fish exposed to wastewa...
TMIJ-0332	Taurolithocholic Acid-d5 Sodium Salt (Major)
	Taurolithocholic Acid-d5 Sodium Salt (Major) 是 Taurolithocholic Acid Sodium Salt 的氘代化合物。Taurolithocholic Acid Sodium Salt 的 CAS 号为 6042-32-6。Taurolithocholic acid sodium salt 是抑胆剂和Ca2+激动剂，可抑制放射性配体与毒蕈碱 M1 结合。
T35790	Palmitic acid-1,2,3,4-13C4 Palmitic Acid-13C (C1, C2, C3, and C4 labeled)
	Palmitic acid-13C (C1, C2, C3, and C4 labeled) is intended for use as an internal standard for the quantification of palmitic acid by GC- or LC-MS. Palmitic acid is a common 16-carbon saturated fat that represents 10-20% of human dietary fat intake and comprises approximately 25 and 65% of human total plasma lipids and saturated fatty acids, respectively.1,2Acylation of palmitic acid to proteins facilitates anchoring of membrane-bound proteins to the lipid bilayer and trafficking of intracellula...
TMIH-0209	Elobixibat-d5
	Elobixibat-d5 是 Elobixibat 的氘代化合物。Elobixibat 的 CAS 号为 439087-18-0。Elobixibat 是回肠胆汁酸转运蛋白的抑制剂（小鼠、人和犬 IBAT 的 IC50：0.13 nM、0.53 nM 和 5.8 nM）。 Elobixibat 可用于慢性特发性便秘的研究。
TMIH-0368	Naringenin-d4
	Naringenin-d4 是 Naringenin 的氘代化合物。Naringenin 的 CAS 号为 480-41-1。Naringenin是葡萄柚中主要的黄烷酮，可作为抗氧化剂、自由基清除剂、抗炎剂、碳水化合物代谢促进剂、免疫系统调节剂。
TMIJ-0215	Doxofylline-d4
	Doxofylline-d4 是 Doxofylline 的氘代化合物。Doxofylline 的 CAS 号为 69975-86-6。Doxofylline 是腺苷 A1 受体拮抗剂，且能抑制磷酸二酯酶 IV，用于治疗哮喘。
TMID-0118	Doxofylline-d6
	Doxofylline-d6 是 Doxofylline 的氘代化合物。Doxofylline 的 CAS 号为 69975-86-6。Doxofylline 是腺苷 A1 受体拮抗剂，且能抑制磷酸二酯酶 IV，用于治疗哮喘。
T71286	Guaifenesin-d3
	Guaifenesin-d3 is intended for use as an internal standard for the quantification of guaifenesin by GC- or LC-MS. Guaifenesin is an expectorant. It inhibits production of mucin 5AC (MUC5AC), reduces mucus viscosity and elasticity, and increases the mucociliary transport rate of endogenous particles in primary human tracheobronchial epithelial cells in a concentration-dependent manner. Guaifenesin increases phenol red secretion, a marker of expectorant activity, in rats.3 Formulations containing ...
TMIJ-0470	Folpet-d4
	Folpet-d4 是 Folpet 的氘代化合物。Folpet 的 CAS 号为 133-07-3。Folpet 是一种广泛使用的二甲酰亚胺类杀菌剂，可诱发小鼠胃肠道肿瘤，主要发生在十二指肠，对人支气管上皮细胞也有细胞毒作用。
T69758	Flutamide-d7
	Flutamide-d7 is intended for use as an internal standard for the quantification of flutamide by GC- or LC-MS. Flutamide is an androgen receptor antagonist and prodrug form of 2-hydroxy flutamide. Flutamide is converted to 2-hydroxy flutamide by the cytochrome P450 (CYP) isoform CYP1A2 in human liver microsomes. It is cytotoxic to PC3 and LNCaP prostate cancer cells with IC50 values of 98.8 and 81.8 µM, respectively. Flutamide (50 mg/kg per day) reduces tumor growth in a PC-82 mouse xenograft mo...
T71145	Racecadotril-d5
	Racecadotril-d5 is intended for use as an internal standard for the quantification of racecadotril by GC- or LC-MS. Racecadotril is a prodrug form of the neprilysin (NEP) inhibitor thiorphan. In vivo, racecadotril reduces or prevents castor oil-induced diarrhea without delaying intestinal transit in rats when administered at doses of 80 or 100 mg/kg, respectively. It also decreases the duration of diarrhea and increases body weight gain in a neonatal gnotobiotic pig model of human rotavirus-indu...
T71211	Rizatriptan-d6 benzoate salt
	Rizatriptan-d6 is intended for use as an internal standard for the quantification of rizatriptan by GC- or LC-MS. Rizatriptan is an agonist of the serotonin receptor subtypes 5-HT1B and 5-HT1D. It is selective for 5-HT1B and 5-HT1D receptors over 5-HT1A receptors. Rizatriptan induces vasoconstriction in isolated human middle meningeal arteries. In vivo, rizatriptan reduces head grooming, the number of oculotemporal strokes, eye blinking, and one-eye closures in a Cacna1a mutant transgenic mou...
T38356	1,2-Dipalmitoyl-13C-sn-glycero-3-PC
	1,2-Dipalmitoyl-13C-sn-glycero-3-PC is intended for use as an internal standard for the quantification of 1,2-dipalmitoyl-sn-glycero-3-PC by GC- or LC-MS. 1,2-Dipalmitoyl-sn-glycero-3-PC (DPPC) is a zwitterionic glycerophospholipid commonly used in the formation of lipid monolayers, bilayers, and liposomes for use in a variety of applications.1,2,3,4 It has been used in the formation of proteoliposomes for implantation of γ-glutamyl transpeptidase into human erythrocyte membranes.3 Incorporation...
T35789	Palmitic acid-1-13C
	Palmitic acid-13C is intended for use as an internal standard for the quantification of palmitic acid by GC- or LC-MS. Palmitic acid is a 16-carbon saturated fatty acid. It comprises approximately 25% of human total plasma lipids.1 It increases protein levels of COX-2 in RAW 264.7 cells when used at a concentration of 75 μM.2 Palmitic acid is involved in the acylation of proteins to anchor membrane-bound proteins to the lipid bilayer.2,3,4,5,6 \|1. Santos, M.J., López-Jurado, M., Llopis, J., et a...
T35783	Zearalenone-13C18 Zearalenone-13C18
	Zearalenone-13C18is intended for use as an internal standard for the quantification of zearalenone by GC- or LC-MS. Zearalenone is a mycotoxin that has been found inFusariumand has estrogenic activities.1It binds to human estrogen receptor α (ERα) and ERβ (IC50s = 9 and 5.8 nM, respectively).2Zearalenone induces precocious development of mammary tissues in young female pigs and prepucial enlargement in young male pigs.3Zearalenone (1.5-5 mg/kg of diet) induces hyperestrogenism in pigs. It also i...
T36059	Dichlorphenamide-13C6 Dichlorphenamide-13C6
	Dichlorphenamide-13C6is intended for use as an internal standard for the quantification of dichlorphenamide by GC- or LC-MS. Dichlorphenamide is a sulfonamide and an orally bioavailable carbonic anhydrase (CA) inhibitor (Kis = 1.20, 38, 50, and 50 nM for the human CA isoforms CAI, CAII, CAIX, and CAXII, respectively).1It lowers intraocular pressure in rabbits when 50 μl of a 10% solution is applied topically to the eye.2Dichlorphenamide rescues the potassium deficiency and prevents insulin-induc...
T71143	Ambroxol-d5
	Ambroxol-d5 is intended for use as an internal standard for the quantification of ambroxol by GC- or LC-MS. Ambroxol is an expectorant and active metabolite of bromhexine. It decreases short-circuit currents in electrically stimulated isolated canine tracheal epithelial cells when applied submucosally. Ambroxol decreases IL-13-induced production of mucin 5AC (MUC5AC) in primary human airway epithelial cells and inhibits IL-13-induced decreases in the mucociliary transport rate of endogenous part...
TMIJ-0519	Fosaprepitant-d4 Dimeglumine
	Fosaprepitant-d4 Dimeglumine 是 Fosaprepitant Dimeglumine 的氘代化合物。Fosaprepitant Dimeglumine 的 CAS 号为 265121-04-8。Fosaprepitant dimeglumine 是 Aprepitant 的前药。它是一种神经激肽 1 受体拮抗剂，可用于预防化疗引起的恶心呕吐。
TMID-0175	DL-α-Hydroxyglutaric acid disodium salt-d4
	DL-α-Hydroxyglutaric acid disodium salt-d4 是 DL-α-Hydroxyglutaric acid disodium salt 的氘代化合物。DL-α-Hydroxyglutaric acid disodium salt 的 CAS 号为 40951-21-1。DL-α-Hydroxyglutaric acid disodium salt 是一种 α-羟基酸，由 (R) -5-oxy-2-tetrahydrofuran 羧酸水解形成，在人类神经代谢疾病 D-α-羟基戊二酸尿症中过量产生。DL-α-Hydroxyglutaric acid disodium salt 是α-酮戊二酸 (α-KG)的拮抗剂，可抑制多种α-KG 依赖性双加氧酶。
T35775	HT-2 Toxin-13C22 HT-2 Toxin-13C22
	HT-2 toxin-13C22is intended for use as an internal standard for the quantification of HT-2 toxin by GC- or LC-MS. HT-2 toxin is a type A trichothecene mycotoxin and an active, deacetylated metabolite of the trichothecene mycotoxin T-2 toxin .1,2Like T-2 toxin, HT-2 toxin inhibits protein synthesis and cell proliferation in plants.2HT-2 toxin also reduces viability of HepG2, A549, HEp-2, Caco-2, A-204, U937, Jurkat, and RPMI-8226 cancer cells with IC50values ranging from 3.1 to 23 ng/ml and human...
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同位素标记化合物

Indomethacin-D4

Cat.No: T11655

Synonym: Indometacin-D4,吲哚美辛-D4

Target: CDK

Cat.No: TMIH-0521

(R)-Praziquantel-d11

Cat.No: T12638

Synonym: (R)-吡喹酮 D11,(R)-Praziquantel D11

Target: 5-HT Receptor

Cat.No: T13291

Synonym: Vitamin D3-26,26,26,27,27,27-d6

Target: Others

O-Desmethyl gefitinib D8

Cat.No: T19489

Target: EGFR

Aripiprazole (D8)

Cat.No: T10368

Synonym: OPC-14597 D8

Target: Others

Cat.No: T12487

Synonym: 吡罗昔康 D3,CP-16171 D3

Target: Others

Cat.No: T11229

Synonym: OSI-774 D6,NSC 718781 D6,CP-358774 D6

Target: Others

Cat.No: T70615

Pentoxifylline-d6

Cat.No: T71300

Apixaban 13C,d3

Cat.No: T10349

Synonym: Apixaban 13CD3,BMS-562247-01 13CD3

Target: Others

Brexpiprazole-d8

Cat.No: T10610

Synonym: OPC-34712 D8

Target: Others

Cat.No: T11995

Synonym: N-Acetyl-5-methoxytryptamine D5,Melatonin D5,褪黑素 D5

Target: Others

Fexofenadine-d6

Cat.No: T11276

Synonym: MDL-16455-d6,Terfenadine carboxylate-d6

Target: Histamine Receptor

Brexpiprazole S-oxide D8

Cat.No: T10611

Synonym: DM-3411 D8

Target: Dopamine Receptor, 5-HT Receptor

Cat.No: T11246

Synonym: MK-0663 D4,依托考昔 D4,L-791456 D4,Etoricoxib D4

Target: Others

Cat.No: T35695

Flufenamic Acid-d4

Cat.No: T71303

Cat.No: T35915

Synonym: Erlotinib-13C6

Mycophenolic Acid-d3 Phenyl Glucuronide

Cat.No: TMIH-0359

p-Benzoquinone-d4

Cat.No: TMIJ-0434

Cat.No: TMIJ-0456

Cat.No: TMIJ-0451

Atomoxetine-d3 hydrochloride

Cat.No: T73711

Cat.No: TMID-0010

Cat.No: TMIH-0198

Synonym: Brexpiprazole Metabolite

1,3,7-Trimethyluric Acid-d9

Cat.No: T71326

Cat.No: T73820

rac-Hesperetin-13C-d3

Cat.No: TMIJ-0108

Synonym: rac-Diosmin EP Impurity G-13C-d3

Clobetasol Propionate-d5

Cat.No: T71893

Norfluoxetine-d5 HCl

Cat.No: T71302

Taurolithocholic Acid-d5 Sodium Salt (Major)

Cat.No: TMIJ-0332

Palmitic acid-1,2,3,4-13C4

Cat.No: T35790

Synonym: Palmitic Acid-13C (C1, C2, C3, and C4 labeled)

Cat.No: TMIH-0209

Cat.No: TMIH-0368

Cat.No: TMIJ-0215

Cat.No: TMID-0118

Cat.No: T71286

Cat.No: TMIJ-0470

Cat.No: T69758

Racecadotril-d5

Cat.No: T71145

Rizatriptan-d6 benzoate salt

Cat.No: T71211

1,2-Dipalmitoyl-13C-sn-glycero-3-PC

Cat.No: T38356

Palmitic acid-1-13C

Cat.No: T35789

Zearalenone-13C18

Cat.No: T35783

Synonym: Zearalenone-13C18

Dichlorphenamide-13C6

Cat.No: T36059

Synonym: Dichlorphenamide-13C6

Cat.No: T71143

Fosaprepitant-d4 Dimeglumine

Cat.No: TMIJ-0519

DL-α-Hydroxyglutaric acid disodium salt-d4

Cat.No: TMID-0175

HT-2 Toxin-13C22

Cat.No: T35775

Synonym: HT-2 Toxin-13C22

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