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TargetMol | Compound Library

人代谢物化合物库现货

Human Metabolite Library

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产品编号 L2570

人代谢物包括内源性代谢物和外源性代谢物;内源性代谢物,顾名思义,就是人体内产生和发现的一些代谢产物,如柠檬酸循环的任何中间代谢物,这些代谢物参与机体重要的生理过程,可作为潜在的药物先导物。外源性代谢物不在机体内产生与发现,来源于外界,包括药物、毒素和食品添加剂等,研究外源性代谢物在人体内如何发生代谢,有助于加快药物发现和毒理学的研究。在药物发现中,了解药物的代谢物有助于对药物作用机理的研究。 TargetMol 人代谢物化合物库收集了5100 种内源性和外源性代谢物,包括羧酸、氨基酸、生物胺、核苷酸、维生素、单糖、双糖、脂类、碳水化合物等不同种类代谢物。

TargetMol 的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
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产品编号 L2570

人代谢物化合物库

规格

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品描述 产品描述

  • 5100种人代谢物的独特集合,用于高通量、高内涵筛选;
  • 研究人体代谢疾病、探索癌症发病机制和寻找新药的有效工具;
  • 部分化合物已上市或进入临床,具有生物安全保障和良好的生物活性;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

Packaging And Storage | TargetMol 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。

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Library Customization | TargetMol 化合物库定制

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Library Customization | TargetMol 化合物库组成

Endogenous Metabolite
Apoptosis
Antibacterial
Autophagy
Antibiotic
COX
Antifungal
NF-κB
Parasite
5-HT Receptor
HIV Protease
Antioxidant
DNA/RNA Synthesis
Reactive Oxygen Species
Cytochromes P450
Adrenergic Receptor
AChR
Calcium Channel
Histamine Receptor
Dopamine Receptor
GABA Receptor
Influenza Virus
PPAR
Potassium Channel
PDE
Sodium Channel
Estrogen/progestogen Receptor
TNF
Glucocorticoid Receptor
Ferroptosis
Topoisomerase
Prostaglandin Receptor
Estrogen Receptor/ERR
EGFR
PI3K
Dehydrogenase
Virus Protease
Caspase
Microtubule Associated
RAAS
HSV
Cholinesterase (ChE)
p38 MAPK
ERK
SARS-CoV
NO Synthase
HCV Protease
Nucleoside Antimetabolite/Analog
Akt
Mitophagy
MMP
Adenosine Receptor
TRP/TRPV Channel
VEGFR
IL Receptor
Reverse Transcriptase
AMPK
Drug Metabolite
NMDAR
Lipoxygenase
STAT
Nrf2
PKC
Antiviral
HDAC
Tyrosinase
ATPase
PDGFR
Progesterone Receptor
ROS
Anti-infection
iGluR
Antifection
Androgen Receptor
P-gp
PARP
MAO
Bcl-2 Family
c-Kit
JNK
Phosphatase
HBV
Proteasome
JAK
Beta Amyloid
Phospholipase
FGFR
Carbonic Anhydrase
Amino Acids and Derivatives
Reductase
Mitochondrial Metabolism
mTOR
GPR
Opioid Receptor
GluR
FLT
Transferase
CDK
TLR
Wnt/beta-catenin
ribosome
Chloride channel
DNA Alkylator/Crosslinker
Serotonin Transporter
Glucosidase
Norepinephrine
Monoamine Oxidase
MRP
Tyrosine Kinases
Immunology/Inflammation related
Interleukin
HSP
HIF/HIF Prolyl-Hydroxylase
NOS
Src
TGF-beta/Smad
HMG-CoA Reductase
Retinoid Receptor
Aromatase
Neurokinin receptor
Thrombin
Proton pump
DHFR
PKA
Bcr-Abl
Raf
DPP-4
DNA Alkylation
HIF
Cannabinoid Receptor
Gamma-secretase
Epigenetic Reader Domain
CaMK
Sirtuin
MEK
p53
Integrin
Factor Xa
Melatonin Receptor
Antifolate
Cysteine Protease
E1/E2/E3 Enzyme
Hedgehog/Smoothened
CCR
Xanthine Oxidase
IGF-1R
DNA
Trk receptor
IκB/IKK
Platelet aggregation
AhR
Thyroid hormone receptor(THR)
c-Met/HGFR
NADPH
FXR
Aryl Hydrocarbon Receptor
ABC Transporter
Fatty Acid Synthase
SGLT
Acyltransferase
Free radical scavengers
transporter
c-RET
DNA Methyltransferase
NOD
HER
ADC Cytotoxin
Histone Methyltransferase
GSK-3
Monoamine Transporter
CXCR
Endothelin Receptor
PGE Synthase
ALK
P2Y Receptor
BACE
CETP
Glutathione Peroxidase
Serine Protease
Leukotriene Receptor
UGT
MT Receptor
Guanylate cyclase
Lipid
GST
CFTR
Arginase
LTR
Cholecystokinin Receptor
Cell Cycle Arrest
LDL
P2X Receptor
Smo
MAPK
Ligand for E3 Ligase
Hydroxylase
Adenosine Deaminase
Syk
NOD-like Receptor (NLR)
S1P Receptor
LPL Receptor
PERK
CaSR
GNRH Receptor
Serine/threonin kinase
Glucokinase
ROCK
IAP
Annexin A
Adiponectin Receptor
Phosphorylase
DNA gyrase
PROTAC Linker
FAAH
PTEN
Epoxide Hydrolase
Aurora Kinase
Telomerase
ATP Citrate Lyase
OAT
Aminopeptidase
RSV
Neprilysin
PLK
Complement System
TAM Receptor
FAK
ROS Kinase
Imidazoline Receptor
Vitamin
MicroRNA
DNA-PK
IFNAR
Lipase
gp120/CD4
Amylase
CSF-1R
PAFR
GlyT
Molecular Glues
Isocitrate Dehydrogenase (IDH)
Bradykinin Receptor
Angiotensin-converting Enzyme (ACE)
cAMP
Indoleamine 2,3-Dioxygenase (IDO)
Beta-Secretase
GPCR19
Histone Acetyltransferase
Casein Kinase
ATM/ATR
c-Fms
Sigma receptor
Advanced Glycation End Products
Mdm2
Adenylyl Cyclase
NPC1L1
Monocarboxylate transporter
ROR
CRM1
Ligands for Target Protein for PROTAC
YAP
Na+/Ca2+ Exchanger
Cell wall
Histone Demethylase
Tie-2
VDA
c-Myc
Rho
Liver X Receptor
Neurotensin Receptor
IRE1
Glucagon Receptor
Na-K-Cl cotransporter
Hexokinase
Bombesin Receptor
PAK
Vasopressin Receptor
OX Receptor
Thrombopoietin Receptor
DUB
BCRP
Glutathione reductase
STING
Ephrin Receptor
Decarboxylase
ADC Linker
GluCls
Pyroptosis
Carboxypeptidase
CRISPR/Cas9
PDK
GHSR
CGRP Receptor
NADPH-oxidase
S6 Kinase
Ras
Protease-activated Receptor
BTK
Apelin receptor
Taste receptor
Transaminase
stilbene oxidase
Hydrogenase
RAR/RXR
CD38
CYP19A1
Dynamin
NEDD8
Aconitase
DYRK
TOPK
N-Acetylglucosaminyltransferase
Hck
NAMPT
Glutaminase
RANKL/RANK
IDO
Myosin
FLAP
RIP kinase
MTH1
Fas/FasL
Anion Exchanger
HCN Channel
Stearoyl-CoA Desaturase (SCD)
ACK1
Somatostatin
Chk
PAD
KSP
Mucin
Wee1
PSMA
Survivin
LRRK2
CPT
hCE
PAI-1
Acetyl-CoA Carboxylase
GPX
Protease
Oxytocin Receptor
IRAK
p97
PD-1/PD-L1
Kinesin
Drug-Linker Conjugates for ADC
Kras

Keywords