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规格 | 价格 | 库存 | 数量 |
---|---|---|---|
1 mg | ¥ 413 | 现货 | |
5 mg | ¥ 1,090 | 现货 | |
10 mg | ¥ 1,720 | 现货 | |
25 mg | ¥ 2,950 | 现货 | |
50 mg | ¥ 4,090 | 现货 | |
100 mg | ¥ 5,510 | 现货 | |
200 mg | ¥ 7,430 | 现货 |
产品描述 | Fz7-21 ((Ac)-LPSDDLEFWCHVMY-NH2) is a peptide antagonist of FZD7 . It antagonises WNT3A-induced Wnt-β-catenin signalling in HEK293 expressing FZD7. Fz7-21 impairs Wnt/β-catenin signaling in HEK293 cells stimulated with exogenous WNT3A (IC50=100 nM) or transfected with a construct expressing WNT3A or WNT1. Fz7-21 also blocks WNT3A-mediated stabilization of β-catenin in mouse L cells (IC50=50 nM). |
靶点活性 | FZD7 CRD (human):58 nM (EC50), FZD7 CRD (mouse):34 nM (EC50) |
别名 | (Ac)-LPSDDLEFWCHVMY-NH2 |
分子量 | 1796.03 |
分子式 | C83H114N18O23S2 |
CAS No. | 2247635-23-8 |
存储 | keep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | ||||||||||||||||||||
溶解度信息 | DMSO: 10 mM | ||||||||||||||||||||
溶液配制表 | |||||||||||||||||||||
DMSO
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