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顶部产品描述包装和储存文件下载化合物库定制化合物库组成
TargetMol | Compound Library

抗癌临床化合物库现货

Anti-Cancer Clinical Compound Library

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产品编号 L2120

尽管在过去的几十年中癌症的研究和治疗取得了巨大的成功，但癌症仍然是人类面临的巨大挑战，给患者身心健康带来巨大的痛苦。癌细胞具有许多显著不同的生物学特征，表现出无限的增殖潜能，维持自身生长信号的持续稳定，逃避应激信号(例如治疗药物)诱导的细胞凋亡，刺激血管生长，为肿瘤提供营养，同时逃避免疫系统防御和诱导局部慢性炎症，发挥其侵袭和转移能力，表现出异常的代谢活动，并通过突变和表观遗传机制显著改变全基因组的稳定性。 抗癌活性的药物是临床研究的热点之一，根据文献报道和有关公开资料，我们收集了2680 个具有抗癌活性或潜在抗癌活性的处于临床试验阶段的化合物，组成抗癌临床化合物库，可用于癌症相关研究及高通量高内涵筛选。

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产品编号 L2120

抗癌临床化合物库

规格

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品描述 产品描述

  • 2680个具有抗癌活性小分子的独特集合，可用于高通量高内涵筛选；
  • 生物活性已经临床前实验证实，所有化合物均已进入临床实验阶段的抗癌化合物；
  • 包括肺癌、乳腺癌、白血病、淋巴瘤等15种癌症，是癌症相关研究的有效筛选工具；
  • 作用靶点涉及PI3K,HDAC, mTOR, CDK, JAK 等癌症相关靶点；
  • 结构多样，药效显著，可渗透细胞；
  • 详细的说明书，化合物结构、靶点信息、IC50值、活性描述等；
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确，纯度高，减少假阳性。

Packaging And Storage | TargetMol 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管；
  • 干粉蓝冰运输，DMSO溶液干冰运输；
  • 排布：96孔板：1st & 12th 空白对照，384孔板：1st & 2nd & 23th & 24th空白对照。

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Supporting Files | TargetMol 文件下载

化合物库操作手册 (635 KB) Targetmol化合物库目录 (60.2 MB)

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Library Customization | TargetMol 化合物库组成

Apoptosis
Autophagy
5-HT Receptor
Endogenous Metabolite
Adrenergic Receptor
DNA/RNA Synthesis
Antibacterial
Dopamine Receptor
Antibiotic
Histamine Receptor
COX
VEGFR
EGFR
Sodium Channel
PI3K
Calcium Channel
Potassium Channel
CDK
FLT
Cytochromes P450
Glucocorticoid Receptor
PDGFR
Parasite
Topoisomerase
Reactive Oxygen Species
JAK
HIV Protease
c-Kit
HDAC
FGFR
Microtubule Associated
c-Met/HGFR
PPAR
mTOR
Dehydrogenase
AChR
Src
Ferroptosis
NF-κB
Prostaglandin Receptor
GABA Receptor
Tyrosine Kinases
Antifungal
Mitophagy
Nucleoside Antimetabolite/Analog
SARS-CoV
Estrogen/progestogen Receptor
Androgen Receptor
ADC Cytotoxin
Adenosine Receptor
Estrogen Receptor/ERR
Bcr-Abl
Raf
GPR
HER
Influenza Virus
PARP
Akt
iGluR
PDE
BTK
Aurora Kinase
HSP
Epigenetic Reader Domain
ALK
P-gp
MEK
p38 MAPK
Serotonin Transporter
TRP/TRPV Channel
Opioid Receptor
HSV
Norepinephrine
RAAS
ROS
c-RET
ATPase
ERK
Trk receptor
DNA Alkylator/Crosslinker
Phosphatase
HBV
PKC
NMDAR
Endothelin Receptor
Histone Methyltransferase
HCV Protease
GSK-3
Virus Protease
Bcl-2 Family
c-Fms
TNF
TAM Receptor
HIF/HIF Prolyl-Hydroxylase
Proton pump
CXCR
Chk
DNA-PK
Progesterone Receptor
E1/E2/E3 Enzyme
Guanylate cyclase
SGLT
STAT
Retinoid Receptor
AMPK
HIF
FAK
p53
S1P Receptor
Carbonic Anhydrase
LPL Receptor
Caspase
DNA Alkylation
IL Receptor
Vasopressin Receptor
TLR
Reverse Transcriptase
Kras
Antioxidant
Antifolate
P2X Receptor
Mitochondrial Metabolism
MMP
Interleukin
Nrf2
ROS Kinase
CFTR
Proteasome
Gamma-secretase
Hedgehog/Smoothened
IGF-1R
TGF-beta/Smad
ATM/ATR
PLK
Syk
Mdm2
Transferase
DHFR
P2Y Receptor
GNRH Receptor
PKA
ROCK
CSF-1R
IAP
GluR
Beta Amyloid
S6 Kinase
Kinesin
Integrin
JNK
MRP
Wnt/beta-catenin
MAO
Drug Metabolite
Antifection
Lipoxygenase
Indoleamine 2,3-Dioxygenase (IDO)
Ligand for E3 Ligase
Neurokinin receptor
DNA Methyltransferase
HMG-CoA Reductase
RIP kinase
Smo
OX Receptor
DNA
Antiviral
Sirtuin
Casein Kinase
Cannabinoid Receptor
Sigma receptor
Monoamine Oxidase
Histone Demethylase
Pim
Glucagon Receptor
Molecular Glues
Isocitrate Dehydrogenase (IDH)
PAK
Bradykinin Receptor
IκB/IKK
Phospholipase
Hydroxylase
IRAK
NADPH
Glutathione Peroxidase
Serine Protease
Leukotriene Receptor
DPP-4
CCR
Cholinesterase (ChE)
Xanthine Oxidase
Ephrin Receptor
GHSR
Thrombin
NO Synthase
Chloride channel
PROTACs
CRM1
YAP
IFNAR
Tie-2
Melatonin Receptor
CaSR
Cholecystokinin Receptor
Serine/threonin kinase
FXR
Aryl Hydrocarbon Receptor
IDO
ABC Transporter
Monoamine Transporter
Neuropeptide Y Receptor
Fatty Acid Synthase
KSP
CaMK
Wee1
PGE Synthase
STING
Aminopeptidase
GPCR19
CRFR
RSV
Aromatase
CGRP Receptor
Ras
AhR
NOS
ROR
LTR
PERK
Rho
PYK2
NAMPT
Glutaminase
Annexin A
MT Receptor
Na-K-Cl cotransporter
Somatostatin
DUB
MAPK
OAT
Free radical scavengers
transporter
Decarboxylase
ribosome
Melanocortin Receptor
PDK
Adenosine Deaminase
NOD
Tyrosinase
Protease-activated Receptor
PD-1/PD-L1
NEDD8
Amino Acids and Derivatives
Ligands for Target Protein for PROTAC
Arginase
Reductase
Cell wall
VDA
c-Myc
Kisspeptin
Cysteine Protease
IRE1
LDL
DNA gyrase
Glucosidase
Hexokinase
HCN Channel
Telomerase
ATP Citrate Lyase
BCRP
Beta-Secretase
Acyltransferase
Porcupine
CD73
GST
LPA Receptor
Oxytocin Receptor
Gap Junction Protein
Discoidin Domain Receptor (DDR)
p97
NOD-like Receptor (NLR)
MLK
Advanced Glycation End Products
NPC1L1
Monocarboxylate transporter
Hydrogenase
MALT
DYRK
RAR/RXR 
TOPK
GTPase
Galectin
N-Acetylglucosaminyltransferase
Hck
Liver X Receptor
Neurotensin Receptor
Glucokinase
Stemness kinase
Myosin
UGT
PAFR
MTH1
GRK
GlyT
Anion Exchanger
Thioredoxin
ACK1
MNK
Survivin
Histone Acetyltransferase
ASK
GluCls
PAI-1
Pyroptosis
MELK
Methionine Adenosyltransferase (MAT)
Neprilysin
Hippo pathway
PI4K
KLF
Aquaporin
RXFP receptor
SGK
Complement System
NADPH-oxidase
BMI-1
Imidazoline Receptor

Keywords

Anti Cancer Clinical Compound LibraryAntiCancer Clinical Compound Library
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