ZK824859

Name: ZK824859
Brand: TargetMol
SKU: T13409
Price: 185 USD
Availability: InStock
Rating: 4.5 (1 reviews)

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产品编号 T13409Cas号 2271122-53-1

ZK824859 is an oral available and selective inhibitor of urokinase plasminogen activator (uPA)(IC50s of 79 nM, 1580 nM and 1330 nM for human uPA, tPA, and plasmin, respectively).

ZK824859

还可以

产品编号 T13409Cas号 2271122-53-1

ZK824859 is an oral available and selective inhibitor of urokinase plasminogen activator (uPA)(IC50s of 79 nM, 1580 nM and 1330 nM for human uPA, tPA, and plasmin, respectively).

规格	价格	库存
25 mg	¥ 12,800	8-10周
50 mg	¥ 16,800	8-10周
100 mg	¥ 21,500	8-10周

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产品介绍

生物活性

产品描述	ZK824859 is an oral available and selective inhibitor of urokinase plasminogen activator (uPA)(IC50s of 79 nM, 1580 nM and 1330 nM for human uPA, tPA, and plasmin, respectively).
靶点活性	TPA (human):1580 nM , Plasmin (human):1330 nM , uPA (human):79 nM
体外活性	ZK824859 is 5 fold less potent and has lost selectivity in mouse: uPA with IC50 of 410?nM; tPA with IC50 of 910?nM; plasmin with IC50 of 1600?nM compared to human IC50 of 79?nM, 1580?nM and 1330?nM respectively.