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PDE2/PDE10-IN-1
还可以产品编号 T12393Cas号 1426833-08-0
PDE2/PDE10-IN-1 is a inhibitor of phosphodiesterase 2 (PDE2) and PDE10(IC50s of 29 and 480 nM, respectively).
PDE2/PDE10-IN-1
还可以产品编号 T12393Cas号 1426833-08-0
PDE2/PDE10-IN-1 is a inhibitor of phosphodiesterase 2 (PDE2) and PDE10(IC50s of 29 and 480 nM, respectively).
| 规格 | 价格 | 库存 | 数量 |
|---|---|---|---|
| 25 mg | ¥ 10,600 | 6-8周 | |
| 50 mg | ¥ 13,800 | 6-8周 | |
| 100 mg | ¥ 17,500 | 6-8周 | |
| 1 mL x 10 mM (in DMSO) | ¥ 4,400 | 6-8周 |
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化学信息
| 产品描述 | PDE2/PDE10-IN-1 is a inhibitor of phosphodiesterase 2 (PDE2) and PDE10(IC50s of 29 and 480 nM, respectively). |
| 靶点活性 | PDE4D (human):5890 nM, PDE11A (human):6920 nM, PDE10A (rat):480 nM, PDE2A (human):29 nM |
| 体外活性 | PDE2/PDE10-IN-1 inhibits PDE2 and PDE10(IC50 of 29 and 480 nM, respectively). PDE2/PDE10-IN-1 is also inactive up to a concentration of 125 μg/mL in a bacterial mutagenicity assay. PDE2/PDE10-IN-1 also inhibits PDE11A and PDE4D with IC50s of 6920 nM and 5890 nM, respectively. In addition PDE2/PDE10-IN-1 does not show significant inhibition of a panel of CYP450 enzymes (CYP1A2, 2C9, 2D6, 2C19, and 3A4). |
| 体内活性 | PDE2/PDE10-IN-1, which is orally bioavailable, occupies PDE2 with an ED50 of 21 mg/kg. |
| 分子量 | 295.73 |
| 分子式 | C15H10ClN5 |
| CAS No. | 1426833-08-0 |
| 密度 | 1.49 g/cm3 (Predicted) |
储存&溶解度
| 存储 | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
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