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JMV6944 作为一种PXR激动剂,以680nM的IC50竞争性抑制hPXR配体结合域(LBD)与PXR的结合,并在新鲜分离的人类原代肝细胞培养物中诱导CYP3A4 mRNA的表达.
JMV6944 作为一种PXR激动剂,以680nM的IC50竞争性抑制hPXR配体结合域(LBD)与PXR的结合,并在新鲜分离的人类原代肝细胞培养物中诱导CYP3A4 mRNA的表达.
规格 | 价格 | 库存 | 数量 |
---|---|---|---|
10 mg | 询价 | 10-14周 | |
50 mg | 询价 | 10-14周 |
产品描述 | JMV6944 is a PXR agonist that competitively inhibits the binding of ligands to the ligand-binding domain (LBD) of human PXR, with an IC50 value of 680 nM. Additionally, JMV6944 induces the expression of CYP3A4 mRNA in cultures of freshly isolated primary human hepatocytes. |
分子量 | 518.71 |
分子式 | C30H38N4O2S |
CAS No. | 2871774-93-3 |
存储 | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
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