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Targets Recommended: Reactive Oxygen Species

3952

抑制剂 & 化合物

376

天然产物

27

化合物库

233

重组蛋白

103

同位素标记化合物

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Cat. No.	Product Name
L2160	抗癌活性化合物库		3188 compounds
	3188 种具有抗肿瘤活性的化合物的特有集合，用于高通量、高内涵筛选；
L9850	口服活性化合物库		2427 compounds
	2427 种口服活性化合物独特集合，可用于高通量筛选和高内涵筛选
L4010	已知活性化合物库		22555 compounds
	22555 个已知活性化合物的集合，可用于高通量筛选、高内涵筛选、细胞诱导和靶点确认；
L9900	药用辅料化合物库		182 compounds
	182 种 FDA 批准药品中的非活性成分集合
L4150	新颖已知活性精选库		989 compounds
	989 种百里挑一的活性化合物；
L7000	活性脂质化合物库		385 compounds
	385 种生物活性小分子化合物，用于高通量、高内涵筛选；
L4000	经典已知活性库		14439 compounds
	14439 个已知活性化合物的集合，可用于高通量筛选、高内涵筛选、细胞诱导和靶点确认；
D7800	新颖已知活性库		8118 compounds
	提高成功率：新增8118种已知活性化合物，提高实验成功率。
L6900	稀有天然产物库		693 compounds
	693 种稀有天然产物的集合，可以用于高通量和高内涵筛选；
L1500	GPCR靶点分子库		1940 compounds
	1940 种与 G 蛋白及其耦联受体相关的生物活性小分子化合物，所有小分子都具有良好的生物和药理活性，部分是 FDA 批准的上市药物；
L6810	中药单体化合物库		2755 compounds
	2755 种中药来源的单体化合物，是药物开发、药理研究等领域的有力工具；
L6800	中国药典收录天然产物库		2051 compounds
	2051 种中国药典收录的天然产物，是药物开发、药理研究等领域的有力工具；
L1580	GPCR库Plus		338 compounds
	338 种GPCR 靶向、结构新颖的化合物；
L6750	活血化瘀中药单体库		580 compounds
	580种来源于常见活血化瘀中药的单体化合物，是药物开发、药理研究等领域的有效工具。
L2521	糖酵解化合物库		555 compounds
	555 种糖酵解相关的活性化合物，可用于高通量和高内涵筛选
L7800	高溶解性片段库		2728 compounds
	2728 种片段分子合集，数量适中，是 FBDD 方法新药筛选的有力工具。
L6110	生物碱类天然产物库		500 compounds
	500 种生物碱类天然产物的独特集合，可用于高通量筛选和高内涵筛选；
L1720	核苷类化合物库		334 compounds
	334 种核苷类化合物，包括核苷酸、核苷酸类似物及衍生物等，适用于抗病毒、抗肿瘤、抗真菌、抗抑郁等药物的研发；
L2500	人内源代谢化合物库		499 compounds
	499 种内源性生物活性化合物的独特集合，用于高通量、高内涵筛选；
L6120	黄酮类天然产物库		514 compounds
	514 种黄酮类天然产物的独特集合，可用于高通量筛选和高内涵筛选；
L5100	含氟化合物库		574 compounds
	574 个含氟化合物的独特集合，可用于高通量筛选和高内涵筛选；
L6210	藏药化合物库		747 compounds
	747 种藏药来源的天然产物分子集合，可以用于高通量和高内涵筛选；
L6220	蒙药化合物库		950 compounds
	950 种蒙药来源的天然产物分子集合，可以用于高通量和高内涵筛选；
L8720	细胞焦亡化合物库		1066 compounds
	1066 种细胞焦亡相关的化合物，可以用于细胞焦亡相关研究。
L6740	抗结直肠癌中药单体化合物库		382 compounds
	382 种抗结直肠癌相关的中药单体集合，是药物开发、药理研究的有效工具；
L6400	海洋天然产物库		144 compounds
	144 种海洋来源的单体化合物，是药物开发、药理研究等领域的有力工具；
L6820	烟草单体化合物库		747 compounds
	747种烟草单体化合物的独特集合，可用于高通量筛选和高内涵筛选

化合物库

抗癌活性化合物库

Cat.No: L2160

Compounds: 3188

口服活性化合物库

Cat.No: L9850

Compounds: 2427

已知活性化合物库

Cat.No: L4010

Compounds: 22555

药用辅料化合物库

Cat.No: L9900

Compounds: 182

新颖已知活性精选库

Cat.No: L4150

Compounds: 989

活性脂质化合物库

Cat.No: L7000

Compounds: 385

经典已知活性库

Cat.No: L4000

Compounds: 14439

新颖已知活性库

Cat.No: D7800

Compounds: 8118

稀有天然产物库

Cat.No: L6900

Compounds: 693

GPCR靶点分子库

Cat.No: L1500

Compounds: 1940

中药单体化合物库

Cat.No: L6810

Compounds: 2755

中国药典收录天然产物库

Cat.No: L6800

Compounds: 2051

Cat.No: L1580

Compounds: 338

活血化瘀中药单体库

Cat.No: L6750

Compounds: 580

糖酵解化合物库

Cat.No: L2521

Compounds: 555

高溶解性片段库

Cat.No: L7800

Compounds: 2728

生物碱类天然产物库

Cat.No: L6110

Compounds: 500

核苷类化合物库

Cat.No: L1720

Compounds: 334

人内源代谢化合物库

Cat.No: L2500

Compounds: 499

黄酮类天然产物库

Cat.No: L6120

Compounds: 514

含氟化合物库

Cat.No: L5100

Compounds: 574

藏药化合物库

Cat.No: L6210

Compounds: 747

蒙药化合物库

Cat.No: L6220

Compounds: 950

细胞焦亡化合物库

Cat.No: L8720

Compounds: 1066

抗结直肠癌中药单体化合物库

Cat.No: L6740

Compounds: 382

海洋天然产物库

Cat.No: L6400

Compounds: 144

烟草单体化合物库

Cat.No: L6820

Compounds: 747

Cat. No.	Product Name	Target	Signaling Pathways
TP1555L1	Fibronectin Active Fragment Control acetate Fibronectin Active Fragment Control acetate(97461-84-2 Free base)
	Fibronectin Active Fragment Control acetate 是纤连蛋白的活性片段，这是一种糖蛋白。
T5401	GSK2983559 active metabolite GSK2983559,RIPK2 inhibitor 1,RIPK2-IN-1	RIP kinase	Apoptosis; NF-κB
	GSK2983559 active metabolite (RIPK2-IN-1) 是一种受体相互作用蛋白-2 激酶抑制剂。
TP1555	Fibronectin Active Fragment Control
	Fibronectin is a high-molecular weight (~440kDa) extracellular matrix glycoprotein that binds to membrane-spanning receptor proteins called integrins.In addition to integrins, fibronectin also binds extracellular matrix components such as collagen, fibrin
T14122	Active-mono-sulfone-PEG8-acid	Others	Others
	Active-mono-sulfone-PEG8-acid is a polyethylene glycol (PEG) derivative serving as a linker for PROTAC synthesis[1].
T10480	Bay 41-4109 (less active enantiomer)	HBV	Microbiology/Virology
	Bay 41-4109 less active enantiomer shows less activity than Bay 41-4109. BAY 41-4109 is a potent HBV inhibitor (IC50: 53 nM).
T19667	R-138727 Prasugrel active metabolite	Others	Others
	R-138727 is a novel P2Y12 receptor inhibitor.
T29705	AG-2000 Free Base Lansoprazole sulfenamide active metabolite	Others	Others
	AG-2000 Free Base is a bio-active chemical. Detailed information has not been published.
T13646	Desisobutyryl-ciclesonide CIC-AP,Ciclesonide active principle	Others	Others
	Desisobutyryl-ciclesonide has an affinity for glucocorticoid receptors. Desisobutyryl-ciclesonide is the active metabolite of Ciclesonide.
T29704	AG-1812 free base UNII-6RI44GB0V9,HE078804,AC1MIZB6,Lansoprazole disulfide active metabolite	Others	Others
	ABT-1812 is a bio-active chemical.
T9966	GSK-1520489A	Wee1	Cell Cycle/Checkpoint
	GSK-1520489 A 是一种活性 PKMYT1 抑制剂。
T8580	Bupranolol	Adrenergic Receptor	GPCR/G Protein; Neuroscience
	Bupranolol 是竞争性的、口服活性的、非选择性的β-adrenoceptor 拮抗剂，无固有的拟交感神经活性。
T1292	Tiapride hydrochloride	Dopamine Receptor	GPCR/G Protein; Neuroscience
	Tiapride 是一种大脑中 D2/3 多巴胺受体的选择性阻滞剂。它用于治疗各种精神和神经系统疾病，包括运动障碍、酒精戒断综合征、精神病的阴性症状以及老年人的攻击和激动。
T8348	Phentolamine	Adrenergic Receptor	GPCR/G Protein; Neuroscience
	Phentolamine 是一种 alpha-1 和 alpha-2 选择性肾上腺素能受体拮抗剂。
T9732	VY-3-135	Fatty Acid Synthase	Metabolism
	VY-3-135 是口服有效的乙酰辅酶 A 合成酶 2 (ACSS2)选择性抑制剂，IC50为 44 nM，对重组人 ACSS1 或 ACSS3 没有抑制活性。它有效抑制 ACSS2 依赖性脂肪酸代谢，但对肿瘤中的基因表达没有影响。
T8734	Choline	Others	Others
	Choline hydroxide 是一种普遍存在的水溶性营养素，通常与 B 族维生素有关。
T9565	OSBPL7-IN-1	Others	Others
	OSBPL7-IN-1 是口服有效的氧甾醇结合蛋白样 7 (OSBPL7)抑制剂。它促进质膜上ABCA1的增加，但不影响 mRNA 表达。
T34896	Tofisopam Emandaxin,托非索洋,Grandaxin	Others	Others
	Tofisopam (Grandaxin) 是2,3-苯二氮卓类化合物，具有抗焦虑活性，可口服。
T20525	Chloramphenicol palmitate	Antibacterial; Antibiotic	Microbiology/Virology
	Chloramphenicol palmitate 是一种广谱抗生素，对革兰氏阳性和革兰氏阴性细菌具有活性。 Chloramphenicol palmitate 可用于在含有氯霉素抗性基因的转化细胞中作为细菌选择剂的研究。
T9805	BAY 2666605	PDE	Metabolism
	BAY 2666605 是一种具有口服活性的 PDE3A 和 PDE3B 抑制剂，IC50 分别为 87 nM 和 50 nM。 BAY 2666605 具有抗癌作用。
T9590	T-1095	SGLT; transporter	GPCR/G Protein; Metabolism
	T-1095 是一种口服有活性的Na+-葡萄糖协同转运蛋白选择性抑制剂，能够抑制 SGLT1 (IC50:22.8 µm) 及 SGLT2 (IC50:2.3 µm) 。它可用于研究糖尿病。
T11689	ITI-214 ITI214	PDE	Metabolism
	ITI-214 是一种中枢神经系统活性抑制剂，具有口服生物活性的PDE1抑制剂 (Kiof 58 pM)，对其他 PDE 家族成员和一系列酶、受体、转运体和离子通道具有良好的选择性，在各种运动和认知功能的动物模型中显示出有效性。
T40732	TMPD dihydrochloride	Others	Others
	TMPD dihydrochloride 是酶促转化氧化还原的活性底物和用于还原血红素过氧化物酶的电子供体。
T9164	BMS-986242 BMS986242	IDO; Indoleamine 2,3-Dioxygenase (IDO)	Metabolism
	BMS-986242 是具有口服具有活力、强效的、选择性的 indoleamine-2,3-dioxygenase 1 抑制剂，可用于研究癌症。
T2629	UNC2881	TAM Receptor	Tyrosine Kinase/Adaptors
	UNC2881 是一种特异性Mer 激酶抑制剂，可抑制稳态的Mer 激酶磷酸化，其IC50=22 nM。
T2678	LB42708	Transferase	Metabolism
	LB42708 是一种口服有活力的特异性法尼基转移酶抑制剂。它对H-Ras、N-Ras 和K-Ras4B 的法尼基化均有抑制作用，其IC50分别为 0.8 nM、1.2 nM 和 2.0 nM。
T7686	Ramiprilat	RAAS	Endocrinology/Hormones
	Ramiprilat 是 Ramipril 的活性代谢物，是一种口服有活力的血管紧张素转换酶 (ACE) 抑制剂，其 Ki=7 pM。它可用于研究心力衰竭以及高血压。
T17158	trans-AUCB t-AUCB	Epoxide Hydrolase	Metabolism
	trans-AUCB (t-AUCB) 是口服具有活力的、选择性的可溶性环氧水解酶 (sEH) 抑制剂，对人，小鼠和大鼠的 sEH 的IC50分别为 1.3 nM，8 nM，8 nM。它具有抗神经胶质瘤特性。
T9303	MRTX1133	Ras	GPCR/G Protein; MAPK
	MRTX1133 是一种 KRAS G12D 抑制剂 (KD=0.2 pM)，具有强效性、选择性和非共价性。MRTX1133 对 KRAS G12D 突变的肿瘤具有抑制活性，而对 KRAS 野生型肿瘤无抑制活性。
T8581	Flecainide hydrochloride	Others	Others
	Flecainide hydrochloride 是一种用于预防和治疗异常快速心率的药物。这包括室性和室上性心动过速。
T9977	SGK1-IN-4	SGK	Metabolism
	SGK1-IN-4 是 SGK1 的特异性抑制剂，可用于骨关节炎研究。
T7503	Upadacitinib 乌帕替尼,ABT-494	JAK	Angiogenesis; Chromatin/Epigenetic; JAK/STAT signaling; Stem Cells
	Upadacitinib (ABT-494) 是高效选择性的，具有口服活性的 JAK1抑制剂，IC50为43 nM，可用于多种自身免疫性疾病的研究。它对 JAK1 的选择性约为 JAK2 的 74 倍。
T36670	JNJ-67856633	MALT	Immunology/Inflammation
	JNJ-67856633 是口服有效的、选择性的、变构性的 MALT1 protease 抑制剂。在某些情况下，JNJ-67856633可以导致肿瘤停滞。
T21593	AAL-993	VEGFR	Angiogenesis; Tyrosine Kinase/Adaptors
	AAL-993 是口服有效的VEGFR 选择性抑制剂，抑制 VEGFR1、VEGFR2 和 VEGFR3 的IC50分别为 130 nM、23 nM 和 18 nM，对其他酪氨酸激酶的抑制作用较弱。AAL-993 具有抗血管生成和抗肿瘤的活性。
T4628	Seladelpar MBX 8025	PPAR	DNA Damage/DNA Repair; Metabolism
	Seladelpar (MBX 8025) 是一种有效的，具有口服活性的，特异性PPAR-δ激动剂，EC50为 2 nM。
T22304	Desciclovir BW A515U,地昔洛韦,6-Deoxyacyclovir,DCV	Antifection	Microbiology/Virology
	Desciclovir (DCV) 是抗疱疹药物阿昔洛韦的前药，口服有活性，在体内被黄嘌呤氧化酶转化成为阿昔洛韦。
T60024	CFT7455 Cemsidomide	Ligand for E3 Ligase	PROTAC
	CFT7455 (Cemsidomide) 是一种抗癌剂，对 cereblon E3 连接酶具有高亲和力，Kd 为 0.9 nM。 CFT7455 是锌指转录因子 Ikaros (IKZF1) 和 Aiolos (IKZF3) 的口服活性降解剂。
T9786	Lu AF27139	P2X Receptor	Membrane transporter/Ion channel; Neuroscience
	Lu AF27139 是一种有效的选择性 P2X7 受体拮抗剂（人和大鼠的 IC50 分别为 12 和 2.4 nM，小鼠、人和大鼠的 Ki 分别为 22、54 和 13 nM）。 Lu AF27139 可用于中枢神经系统疾病研究。
T28167	NGB 2904 NGB2904 HCl,NGB-2904,NGB2904	Others; Dopamine Receptor; 5-HT Receptor	GPCR/G Protein; Neuroscience; Others
	NGB 2904 是一种具有口服活性的、选择性的多巴胺(DA) D3受体拮抗剂，可用于具可卡因成瘾。
T21976	ONO-8130	Prostaglandin Receptor	GPCR/G Protein; Immunology/Inflammation
	ONO-8130 是前列腺素 EP1 受体选择性拮抗剂，口服有活力，能够阻断 L6 脊髓中ERK 的磷酸化。它可缓解环磷酰胺致膀胱炎小鼠的膀胱疼痛，可用于研究间质性膀胱炎。
T9627	PHD-1-IN-1	HIF/HIF Prolyl-Hydroxylase	Chromatin/Epigenetic; Metabolism
	PHD-1-IN-1 是口服有效的缺氧诱导因子脯氨酰羟化酶结构域 1抑制剂，IC50为 0.034 μM。它与活性位 Fe2+具有独特的单齿结合相互作用，并诱导形成一个 “Arg367-out” 口袋。
T0600	10,11-Dihydrocarbamazepine 双氢卡马西平,10,11-二氢卡马西平,Dihydrocarbamazepine	Others	Others
	10,11-Dihydrocarbamazepine (Dihydrocarbamazepine) 是一种 Oxcarbazepine 的活性代谢物，也是一种有机中间体。Oxcarbazepine 能够几乎完全的、迅速的转化为 10,11-Dihydrocarbamazepine，可能具有抗惊厥效果。
T10826	CK-666	HIV Protease; Microtubule Associated	Cytoskeletal Signaling; Microbiology/Virology; Proteases/Proteasome
	CK-666 是一种肌动蛋白相关蛋白 Arp2/3 复合物的细胞渗透性抑制剂。它与 Arp2/3 复合物结合，稳定复合物的非活性状态，阻止 Arp2 和 Arp3 亚基进入活化的丝状短节距构象。
T2578	Didanosine ddI,去羟肌苷,2',3'-Dideoxyinosine	HIV Protease; Reverse Transcriptase	Microbiology/Virology; Proteases/Proteasome
	Didanosine (ddI) 是一种逆转录酶抑制剂，IC50为490nM。
T21793	CGP 35348	GABA Receptor	Membrane transporter/Ion channel; Neuroscience
	CGP 35348 是 GABAB 受体的选择性拮抗剂 (EC50 = 34 μM)。 CGP 35348 可用于研究白化新生小鼠脑损伤后的神经肌肉协调和空间学习。
T22675	Co 102862 V 102862	Others; Sodium Channel	Membrane transporter/Ion channel; Others
	Co 102862 是一种电压门控钠通道阻滞剂。 Co 102862 可用于抗惊厥的研究。
T1448	Dasatinib BMS-354825,达沙替尼	Apoptosis; Bcr-Abl; Src; c-Kit; Autophagy	Angiogenesis; Apoptosis; Autophagy; Cytoskeletal Signaling; Tyrosine Kinase/Adaptors
	Dasatinib (BMS-354825) 是一种酪氨酸激酶抑制剂，抑制 Src 和 Bcr-Abl (Ki=16/30 pM)，具有口服活性和 ATP 竞争性。Dasatinib 具有抗肿瘤活性，用于治疗白血病和淋巴瘤等。
T22436	Takeda-6d	VEGFR	Angiogenesis; Tyrosine Kinase/Adaptors
	Takeda-6d 是一种新型、有效的 DFG-out RAF/血管内皮生长因子受体 2 (VEGFR2) 抑制剂，IC50 分别为 7.0 nM 和 2.2 nM。
T1072	Loxeen Pridinol methanesulfonate,Α,Α-二苯基-1-哌啶丙醇(普立地诺甲磺酸盐 )	AChR	Neuroscience
	Loxeen (Pridinol methanesulfonate) 用作抗胆碱能药物和抗帕金森病药物。
T2316	Omarigliptin MK-3102,奥格列汀	Proteasome; DPP-4	Proteases/Proteasome; Ubiquitination
	Omarigliptin (MK-3102) 是高效选择性 DPP4抑制剂，IC50=为1.6nM。
T1613	Hydralazine hydrochloride Hydralazine HCl,Apresoline,盐酸肼屈嗪	MAO; HIF/HIF Prolyl-Hydroxylase	Chromatin/Epigenetic; Metabolism; Neuroscience
	Hydralazine hydrochloride (Apresoline) 是一种直接作用的血管舒张剂，可抗高血压。

化合物

Fibronectin Active Fragment Control acetate

Cat.No: TP1555L1

Synonym: Fibronectin Active Fragment Control acetate(97461-84-2 Free base)

GSK2983559 active metabolite

Cat.No: T5401

Synonym: GSK2983559,RIPK2 inhibitor 1,RIPK2-IN-1

Target: RIP kinase

Fibronectin Active Fragment Control

Cat.No: TP1555

Active-mono-sulfone-PEG8-acid

Cat.No: T14122

Target: Others

Bay 41-4109 (less active enantiomer)

Cat.No: T10480

Target: HBV

Cat.No: T19667

Synonym: Prasugrel active metabolite

Target: Others

AG-2000 Free Base

Cat.No: T29705

Synonym: Lansoprazole sulfenamide active metabolite

Target: Others

Desisobutyryl-ciclesonide

Cat.No: T13646

Synonym: CIC-AP,Ciclesonide active principle

Target: Others

AG-1812 free base

Cat.No: T29704

Synonym: UNII-6RI44GB0V9,HE078804,AC1MIZB6,Lansoprazole disulfide active metabolite

Target: Others

Cat.No: T9966

Target: Wee1

Cat.No: T8580

Target: Adrenergic Receptor

Tiapride hydrochloride

Cat.No: T1292

Target: Dopamine Receptor

Cat.No: T8348

Target: Adrenergic Receptor

Cat.No: T9732

Target: Fatty Acid Synthase

Cat.No: T8734

Target: Others

Cat.No: T9565

Target: Others

Cat.No: T34896

Synonym: Emandaxin,托非索洋,Grandaxin

Target: Others

Chloramphenicol palmitate

Cat.No: T20525

Target: Antibacterial, Antibiotic

Cat.No: T9805

Target: PDE

Cat.No: T9590

Target: SGLT, transporter

Cat.No: T11689

Synonym: ITI214

Target: PDE

TMPD dihydrochloride

Cat.No: T40732

Target: Others

Cat.No: T9164

Synonym: BMS986242

Target: IDO, Indoleamine 2,3-Dioxygenase (IDO)

Cat.No: T2629

Target: TAM Receptor

Cat.No: T2678

Target: Transferase

Cat.No: T7686

Target: RAAS

Cat.No: T17158

Synonym: t-AUCB

Target: Epoxide Hydrolase

Cat.No: T9303

Target: Ras

Flecainide hydrochloride

Cat.No: T8581

Target: Others

Cat.No: T9977

Target: SGK

Cat.No: T7503

Synonym: 乌帕替尼,ABT-494

Target: JAK

Cat.No: T36670

Target: MALT

Cat.No: T21593

Target: VEGFR

Cat.No: T4628

Synonym: MBX 8025

Target: PPAR

Cat.No: T22304

Synonym: BW A515U,地昔洛韦,6-Deoxyacyclovir,DCV

Target: Antifection

Cat.No: T60024

Synonym: Cemsidomide

Target: Ligand for E3 Ligase

Cat.No: T9786

Target: P2X Receptor

Cat.No: T28167

Synonym: NGB2904 HCl,NGB-2904,NGB2904

Target: Others, Dopamine Receptor, 5-HT Receptor

Cat.No: T21976

Target: Prostaglandin Receptor

Cat.No: T9627

Target: HIF/HIF Prolyl-Hydroxylase

10,11-Dihydrocarbamazepine

Cat.No: T0600

Synonym: 双氢卡马西平,10,11-二氢卡马西平,Dihydrocarbamazepine

Target: Others

Cat.No: T10826

Target: HIV Protease, Microtubule Associated

Cat.No: T2578

Synonym: ddI,去羟肌苷,2',3'-Dideoxyinosine

Target: HIV Protease, Reverse Transcriptase

Cat.No: T21793

Target: GABA Receptor

Cat.No: T22675

Synonym: V 102862

Target: Others, Sodium Channel

Cat.No: T1448

Synonym: BMS-354825,达沙替尼

Target: Apoptosis, Bcr-Abl, Src, c-Kit, Autophagy

Cat.No: T22436

Target: VEGFR

Cat.No: T1072

Synonym: Pridinol methanesulfonate,Α,Α-二苯基-1-哌啶丙醇(普立地诺甲磺酸盐 )

Target: AChR

Cat.No: T2316

Synonym: MK-3102,奥格列汀

Target: Proteasome, DPP-4

Hydralazine hydrochloride

Cat.No: T1613

Synonym: Hydralazine HCl,Apresoline,盐酸肼屈嗪

Target: MAO, HIF/HIF Prolyl-Hydroxylase

Cat. No.	Product Name	Target	Signaling Pathways
T11351	Galanthamine N-Oxide	AChE	Neuroscience
	Galanthamine N-Oxide 是分离于Zephyranthes concolor 的球茎中的一种生物碱。它抑制电鳗乙酰胆碱酯酶，EC50=26.2 μM。它是TcAChE，hAChE 和 hBChE 酶活性位点中底物调节的显著抑制剂。
T4S1114	Dryocrassin ABBA 东北贯众素,Dryocrassin	Influenza Virus; Antibacterial	Microbiology/Virology
	Dryocrassin ABBA (Dryocrassin) 是一种从苦参中提取的黄酮类天然产物，具有抗病毒和抗菌活性。它抑制树突状细胞的免疫刺激功能，延长同种异体皮肤移植成活率。
T3858	macranthoidin A 灰毡毛忍冬皂苷甲,金银花	Others	Others
	Macranthoidin A 是一种具有口服活性的、提取于金银花中的皂苷。它对四氯化碳，对乙酰氨基酚和镉所致的肝损伤具有保护作用，对耳巴豆油的溶胀具有明显的抑制作用。
T1560	Prednisolone 氢化泼尼松,Predonine,Hydroretrocortine,泼尼松龙,Metacortandralone	Glucocorticoid Receptor; Endogenous Metabolite	Endocrinology/Hormones; Metabolism
	Prednisolone (Hydroretrocortine) 是有口服活性的皮质类固醇和糖皮质激素。它的抗炎特性约为氢化可的松的四倍，同时减少了水和盐的保留。它能够用于眼部抗炎研究。
T5784	Topotecan NSC 609669,拓扑替康,SKF 104864A	Topoisomerase; Autophagy	Autophagy; DNA Damage/DNA Repair
	Topotecan (NSC-609669) 是一种拓扑异构酶 I 抑制剂，通过抑制 DNA 拓扑异构酶起抗肿瘤作用，可用于治疗卵巢癌。
T1611	Isotretinoin 13-cis-Retinoic acid,异维A酸	Retinoid Receptor; Endogenous Metabolite; Autophagy	Autophagy; Metabolism
	Isotretinoin (13-cis-Retinoic acid) 是一种天然存在的维甲酸，具有潜在的抗肿瘤活性。它结合并激活核视黄酸受体 (RAR)，活化的 RARs 作为促进细胞分化和凋亡的转录因子。它是一种类维生素A 和维生素A 衍生物，用于治疗严重的痤疮和某些形式的皮肤、头颈癌。
T1326	Gentamicin sulfate SCH9724,Gentamycin sulfate,NSC-82261,硫酸庆大霉素	ribosome; DHFR; Antibacterial; Antibiotic	Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism; Microbiology/Virology
	Gentamicin sulfate (SCH9724) 是一种广谱的氨基糖苷类抗生素，具有口服活性。Gentamicin sulfate 可以用于抑制敏感生物体中的蛋白质合成。
T0974	Novobiocin Sodium Albamycinsodium,新生霉素钠,Cathomycin,Albamycin	Potassium Channel; DNA gyrase; Topoisomerase; Antibacterial; Antibiotic; ABC; Autophagy	Autophagy; DNA Damage/DNA Repair; Membrane transporter/Ion channel; Microbiology/Virology
	Novobiocin Sodium (Albamycinsodium) 是源自 Streptomyces niveus 的抗生素。它的化学结构类似于香豆素。Novobiocin 与 DNA 促旋酶结合并阻断三磷酸腺苷活性。
T5283	NADH disodium salt Disodium NADH,NADH, disodium salt hydrate,beta-烟酰胺腺嘌呤二核苷二钠	Others; Endogenous Metabolite	Metabolism; Others
	NADH disodium salt hydrate是氧化还原酶的辅酶。 NADH在分解代谢过程中起到再生电子供体的作用，包括糖酵解，柠檬酸循环和β-氧化。
TN6774	Emodin 6-O-β-D-glucoside 大黄素-6-O-β-D-葡萄糖苷,Glucoemodin	Others	Others
	Emodin 6-O-β-D-glucoside (Glucoemodin) 是一种从 Reynoutria japonica 中提取的活性化合物。它具有显著的抗炎和屏障保护活性，可用于研究动脉粥样硬化及糖尿病并发症。
T2881	Crustecdysone Commisterone,B-ecdysone,Commisterone,20-Hydroxyecdysone,Ecdysterone,B-ecdysone,β-蜕皮甾酮,Hydroxyecdysone,羟基蜕皮激素	Others; Caspase; Endogenous Metabolite; Autophagy	Apoptosis; Autophagy; Metabolism; Others; Proteases/Proteasome
	Crustecdysone (Hydroxyecdysone) 是来源于露水草的一种蜕皮激素，可调节昆虫的蜕皮或蜕皮过程。它是 Ecdysone 的活性代谢物，通过 20E 核受体复合物 EcR-USP 抑制半胱天冬酶活性并诱导自噬，在心血管系统中具有调节或保护作用。
T6194	Fidaxomicin 非达米星,Tiacumicin B,OPT-80,Clostomicin B1,PAR-101	Apoptosis; DNA/RNA Synthesis; Antibacterial; Antibiotic	Apoptosis; Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
	Fidaxomicin (Tiacumicin B) 是一种大环RNA 聚合酶抑制剂，具有窄谱活性。它选择性地根除致病性艰难梭菌，对构成正常健康肠道菌群的多种细菌影响很小。
T2719	Succinic acid Asuccin,Amber acid,琥珀酸,1,2-Ethanedicarboxylic acid,Wormwood acid,Butanedioic acid,1,4-Butandioic Acid	Endogenous Metabolite	Metabolism
	Succinic acid (1,2-Ethanedicarboxylic acid) 是无氧代谢的发酵产物，也是三羧酸循环的中间产物。
T3417	Amentoflavone Didemethyl-ginkgetin,穗花杉双黄酮,Amenthoflavone,3',8''-Biapigenin	Apoptosis; P450; Phospholipase; Reactive Oxygen Species; Opioid Receptor; COX; Antibacterial; RSV; Antifungal	Apoptosis; Endocrinology/Hormones; GPCR/G Protein; Immunology/Inflammation; Metabolism; Microbiology/Virology; Neuroscience; NF-κB
	Amentoflavone (3',8''-Biapigenin) 是一种具有很多生物活性的双黄酮类天然产物，有抗炎、抗氧化和神经保护等作用。
T2755	Rhoifolin 野漆树苷,Apigenin-7-O-rhamnoglucoside,Apigenin 7-O-neohesperidoside,Rhoifoloside	Others; p38 MAPK; NF-κB; transporter; IGF-1R; Autophagy	Autophagy; MAPK; Metabolism; NF-κB; Others; Tyrosine Kinase/Adaptors
	Rhoifolin (Apigenin 7-O-neohesperidoside) 是从琯溪蜜柚叶子分离的一种黄酮糖苷。它通过 RANKL 诱导的NF-κB 和MAPK 途径改善钛颗粒刺激的骨溶解并减少破骨细胞生成。它通过增强脂联素分泌，胰岛素受体-β的酪氨酸磷酸化和GLUT4易位有助于治疗糖尿病并发症。
T3055	Liensinine Perchlorate	Apoptosis; Others	Apoptosis; Others
	Liensinine Perchlorate 是元莲的成分，可诱导结直肠癌细胞凋亡，具有抗高血压和抗癌活性。
T3912	Saikosaponin B1 柴胡皂苷B1,柴胡皂苷 B1	Others	Others
	Saikosaponin B1 是柴胡的生物活性成分，具有抗癌作用。它能够靶向SMO 抑制 Hedgehog 通路，显著抑制髓母细胞瘤模型中的肿瘤生长。
T0646	5-Aminosalicylic Acid Mesalazine,5-ASA,5-氨基水杨酸,Mesalamine	NF-κB; Lipoxygenase; COX; Glutathione Peroxidase; Endogenous Metabolite; PAK; PPAR	Cytoskeletal Signaling; DNA Damage/DNA Repair; Immunology/Inflammation; Metabolism; Neuroscience; NF-κB
	5-Aminosalicylic Acid (5-ASA) 是一种特异性的PPARγ激动剂，还抑制 p21-激活激酶1(PAK1) 和NF-κB，具有抗炎活性。
T3367	Macranthoidin B 灰毡毛忍冬皂苷乙,金银花,Macranthoiside I	Others	Others
	Macranthoidin B 是一种活性天然皂苷。
T3742	3-Methylcatechol 3-甲基苯邻二酚,3-Methylpyrocatechol,2,3-Toluenediol,3-甲基邻苯二酚,2,3-dihydroxytoluene	Others	Others
	3-Methylcatechol (2,3-Toluenediol) 是由 Pseudomonas putidaMC2 产生，能够用作化学合成中的分子砌块。
T20191	(-)-Camphoric acid (-)-樟脑酸,L-Camphoric acid,Camphoric acid, (-)-	GluR	Neuroscience
	(-)-Camphoric acid (L-Camphoric acid) 是一种活性较低的樟脑酸对映异构体，樟脑酸可诱导 GluR 表达。
T4082	Astragaloside	MMP; ERK; JNK	MAPK; Proteases/Proteasome
	Astragaloside 是黄芪中的主要活性成分之一。
T5556	5a-Pregnane-3,20-dione	Endogenous Metabolite	Metabolism
	5a-Pregnane-3,20-dione 是内源性的孕酮代谢物。
T3848	(Iso)-Isomucronulatol 7-O-glucoside Isomucronulatol 7-O-glucoside,7,2'-dihydroxy-3',4'-dimethoxyisoflavane-7-O-glucoside,黄芪异黄烷苷,7,2′-Dihydroxy-3′,4′-dimethoxyisoflavan 7-O-β-D-glucoside	Others	Others
	Isomucronulatol 7-O-glucoside 是一种具有生物活性的异黄酮，分离自黄芪中。
T3760	2'-Hydroxy-5'-methoxyacetophenone 2'-羟基-5'-甲氧基苯乙酮,5-Methoxy-2-hydroxyacetophenone	Others	Others
	2'-Hydroxy-5'-methoxyacetophenone (5-Methoxy-2-hydroxyacetophenone) 是一种活性生化剂。
T8263	3,4'-Dihydroxyflavone	Influenza Virus	Microbiology/Virology
	3,4'-Dihydroxyflavone 是一种口服活性黄酮类化合物，具有抗甲型流感病毒的抗病毒活性。
T19554	L-Aspartic aicd sodium L-Aspartic acid sodium,Sodium L-aspartate	Others; Sodium Channel; Endogenous Metabolite	Membrane transporter/Ion channel; Metabolism; Others
	L-Aspartic aicd sodium (Sodium L-aspartate) 是一种氨基酸，是一种结肠特异性活性分子输送的前体活性分子，可促进大鼠前脑膜囊泡的 Na+外排。
T3820	Iridin 野鸢尾苷,Lridin	Others	Others
	Iridin (Lridin) 是抑制异黄酮化合物，从Iris milesii 中提取得到。
TN6736	Dihydrolanosterol 24,25-Dihydrolanosterol,Lanostenol,二氢羊毛甾醇	Others	Others
	Dihydrolanosterol 是一种 CYP51 的底物，能够阻碍胆固醇的合成。
TN1927	Methyl Kakuol 1-(6-methoxy-1,3-benzodioxol-5-yl)propan-1-one	TRP/TRPV Channel	Membrane transporter/Ion channel
	Methyl Kakuol 是 TRPA1 的激动剂，EC50 为 0.27 µM，可用于作为 MBST 成分 Asiasari Radix 的活性成分的研究。
T4S1173	Agrimol B 仙鹤草酚B,仙鹤草酚 B	Sirtuin; PPAR	Chromatin/Epigenetic; DNA Damage/DNA Repair; Metabolism
	Agrimol B 是从仙鹤草中分离得到的一种多酚衍生物，可抑制脂肪形成，降低PPARγ的表达，诱导SIRT1易位和表达。
T19398	L-Octanoylcarnitine	Endogenous Metabolite	Metabolism
	L-Octanoylcarnitine 是存在于血浆中的活性辛酰肉碱，是一种乳腺癌的潜在生物标志物。
T6S1652	Benzoylpaeoniflorin	COX	Immunology/Inflammation; Neuroscience
	Benzoylpaeoniflorin 是一种从白芍中提取的天然化合物，可以降低细胞凋亡，对冠心病具有潜在的研究价值。
T3764	1-Triacontanol Myricyl alcohol,1-Triacontanol,三十烷醇,Melissyl alcohol,Well-Bloom,Miraculan,Lithospermoside,triacontan-1-ol	Others	Others
	1-Triacontanol (Melissyl alcohol) 是天然存在的植物生长调节剂。它是饱和长链醇，能够促进许多植物的生长。
T13669	(E)-Cinnamamide trans-Cinnamamide,肉桂酰胺	Others	Others
	(E)-Cinnamamide (trans-Cinnamamide) 是 Cinnamamide 的活性较低的异构体，Cinnamamide 是一种有效的非致命化学驱虫剂，适用于减少鸟类害虫的损害。
T6S1884	Benzoylhypaconine 苯甲酰次乌头碱,Benzoylhypacoitine,苯甲酰次乌头原碱	Others	Others
	Benzoylhypaconine (Benzoylhypacoitine) 是来自 Aconitum 中的一种单酯生物碱，也是Aconitum 的主要药理和毒性成分。
TL0002	Liquiritin apioside	Others	Others
	Liquiritin apioside 是一种从甘草中获得的黄酮，具有镇咳活性。
T3S2197	Polygalic acid Senegenic acid,远志皂甙	Others	Others
	Polygalic acid (Senegenic acid) 是一种三萜皂苷，是远志 (Polygala tenuifolia) 的一种主要活性成分。
T3014	(±)-Abscisic acid Abscisic acid,Dormin,脱落酸,Abscisinsaeure	Others	Others
	(±)-Abscisic acid 是一种口服具有活性的植物激素，也存在与动物中。它可以调节哺乳动物的血糖。
T3227	Danshensu Salvianic acid A,Dan shen suan A,丹参素	Apoptosis; Nrf2; Autophagy	Apoptosis; Autophagy; Immunology/Inflammation
	Danshensu (Dan shen suan A) 是丹参的有效成分，能够激活 Nrf2信号通路，具有保护心血管作用。
TMO2787	Anthraquinone dioxoanthracene,Anthradione,anthracenedione,蒽醌	Virus Protease	Microbiology/Virology
	Anthraquinone (Anthradione) 是常用于缓解便秘的草药中的主要活性成分，可用作染料形成前体。
TQ0070	Luteolin-3-O-beta-D-glucuronide	Others	Others
	Luteolin-3-O-beta-D-glucuronide 是木犀草素葡萄糖醛酸，木犀草素的 3’ 端位置有 β-d-葡萄糖苷酸残基。
T4587	Mirificin BCP10902,Puerarin Apioside,葛根素芹菜糖苷,芹糖葛根素苷	Tyrosinase	Proteases/Proteasome
	Mirificin (BCP10902) 是一种葛根中的异黄酮。它能够抑制酪氨酸酶(Tyrosinase)，IC50=12.66 μM。
T6S0630	Hypaconitine	P450; TNF	Apoptosis; Metabolism
	Hypaconitine 是从乌头属种分离的一种高毒性成分，可研究风湿病。
T21495	Spinosyn A	Others	Others
	Spinosyn A 是聚酮化合物衍生的大环内酯，来自多刺甘蔗多孢菌。Spinosyn A 是有效的杀虫剂。
T4911	α-Arbutin 4-hydroxyphenyl-D-lucopyranoside,alpha-Arbutoside,α-熊果苷,alpha-Arbutin	Tyrosinase	Proteases/Proteasome
	α-Arbutin (4-hydroxyphenyl-D-lucopyranoside) 是一种流行的、有效的皮肤增白剂，也是一种酪氨酸酶 (tyrosinase) 抑制剂。
TN1499	Cimiracemoside C 千层纸素A-7-0-Β-D-葡萄糖醛酸苷,Cimicifugoside M	AMPK	Chromatin/Epigenetic; PI3K/Akt/mTOR signaling
	Cimiracemoside C (Cimicifugoside M) 是在升麻中发现的一种天然产物，可激活 AMPK 并具有抗糖尿病的潜在活性。
TQ0288	Hexahydrocurcumin	Reactive Oxygen Species; ROS; COX	Immunology/Inflammation; Metabolism; Neuroscience; NF-κB
	Hexahydrocurcumin 是一种选择性口服活性COX-2抑制剂，对 COX-1 无活性，是姜黄素的主要代谢产物之一，。它具有抗氧化，抗癌和抗炎作用。
T2S1181	Aloenin Aloenin A,Aloearbonaside,芦荟宁	Beta-Secretase; AChR	Neuroscience
	Aloenin (Aloenin A) A 是一种具有清除过氧自由基作用的天然产物，对 β-分泌酶 (BACE) 具有中等抑制活性。
TN3176L	(2R)-6-Methoxynaringenin
	(2R)-2,3-Dihydro-5,7-dihydroxy-2-(4-hydroxyphenyl)-6-methoxy-4H-1-benzopyran-4-one 是黄芩中的潜在活性成分之一。
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天然产物

Galanthamine N-Oxide

Cat.No: T11351

Target: AChE

Dryocrassin ABBA

Cat.No: T4S1114

Synonym: 东北贯众素,Dryocrassin

Target: Influenza Virus, Antibacterial

macranthoidin A

Cat.No: T3858

Synonym: 灰毡毛忍冬皂苷甲,金银花

Target: Others

Cat.No: T1560

Synonym: 氢化泼尼松,Predonine,Hydroretrocortine,泼尼松龙,Metacortandralone

Target: Glucocorticoid Receptor, Endogenous Metabolite

Cat.No: T5784

Synonym: NSC 609669,拓扑替康,SKF 104864A

Target: Topoisomerase, Autophagy

Cat.No: T1611

Synonym: 13-cis-Retinoic acid,异维A酸

Target: Retinoid Receptor, Endogenous Metabolite, Autophagy

Gentamicin sulfate

Cat.No: T1326

Synonym: SCH9724,Gentamycin sulfate,NSC-82261,硫酸庆大霉素

Target: ribosome, DHFR, Antibacterial, Antibiotic

Novobiocin Sodium

Cat.No: T0974

Synonym: Albamycinsodium,新生霉素钠,Cathomycin,Albamycin

Target: Potassium Channel, DNA gyrase, Topoisomerase, Antibacterial, Antibiotic, ABC, Autophagy

NADH disodium salt

Cat.No: T5283

Synonym: Disodium NADH,NADH, disodium salt hydrate,beta-烟酰胺腺嘌呤二核苷二钠

Target: Others, Endogenous Metabolite

Emodin 6-O-β-D-glucoside

Cat.No: TN6774

Synonym: 大黄素-6-O-β-D-葡萄糖苷,Glucoemodin

Target: Others

Cat.No: T2881

Synonym: Commisterone,B-ecdysone,Commisterone,20-Hydroxyecdysone,Ecdysterone,B-ecdysone,β-蜕皮甾酮,Hydroxyecdysone,羟基蜕皮激素

Target: Others, Caspase, Endogenous Metabolite, Autophagy

Cat.No: T6194

Synonym: 非达米星,Tiacumicin B,OPT-80,Clostomicin B1,PAR-101

Target: Apoptosis, DNA/RNA Synthesis, Antibacterial, Antibiotic

Cat.No: T2719

Synonym: Asuccin,Amber acid,琥珀酸,1,2-Ethanedicarboxylic acid,Wormwood acid,Butanedioic acid,1,4-Butandioic Acid

Target: Endogenous Metabolite

Cat.No: T3417

Synonym: Didemethyl-ginkgetin,穗花杉双黄酮,Amenthoflavone,3',8''-Biapigenin

Target: Apoptosis, P450, Phospholipase, Reactive Oxygen Species, Opioid Receptor, COX, Antibacterial, RSV, Antifungal

Cat.No: T2755

Synonym: 野漆树苷,Apigenin-7-O-rhamnoglucoside,Apigenin 7-O-neohesperidoside,Rhoifoloside

Target: Others, p38 MAPK, NF-κB, transporter, IGF-1R, Autophagy

Liensinine Perchlorate

Cat.No: T3055

Target: Apoptosis, Others

Saikosaponin B1

Cat.No: T3912

Synonym: 柴胡皂苷B1,柴胡皂苷 B1

Target: Others

5-Aminosalicylic Acid

Cat.No: T0646

Synonym: Mesalazine,5-ASA,5-氨基水杨酸,Mesalamine

Target: NF-κB, Lipoxygenase, COX, Glutathione Peroxidase, Endogenous Metabolite, PAK, PPAR

Macranthoidin B

Cat.No: T3367

Synonym: 灰毡毛忍冬皂苷乙,金银花,Macranthoiside I

Target: Others

3-Methylcatechol

Cat.No: T3742

Synonym: 3-甲基苯邻二酚,3-Methylpyrocatechol,2,3-Toluenediol,3-甲基邻苯二酚,2,3-dihydroxytoluene

Target: Others

(-)-Camphoric acid

Cat.No: T20191

Synonym: (-)-樟脑酸,L-Camphoric acid,Camphoric acid, (-)-

Target: GluR

Cat.No: T4082

Target: MMP, ERK, JNK

5a-Pregnane-3,20-dione

Cat.No: T5556

Target: Endogenous Metabolite

(Iso)-Isomucronulatol 7-O-glucoside

Cat.No: T3848

Synonym: Isomucronulatol 7-O-glucoside,7,2'-dihydroxy-3',4'-dimethoxyisoflavane-7-O-glucoside,黄芪异黄烷苷,7,2′-Dihydroxy-3′,4′-dimethoxyisoflavan 7-O-β-D-glucoside

Target: Others

2'-Hydroxy-5'-methoxyacetophenone

Cat.No: T3760

Synonym: 2'-羟基-5'-甲氧基苯乙酮,5-Methoxy-2-hydroxyacetophenone

Target: Others

3,4'-Dihydroxyflavone

Cat.No: T8263

Target: Influenza Virus

L-Aspartic aicd sodium

Cat.No: T19554

Synonym: L-Aspartic acid sodium,Sodium L-aspartate

Target: Others, Sodium Channel, Endogenous Metabolite

Cat.No: T3820

Synonym: 野鸢尾苷,Lridin

Target: Others

Dihydrolanosterol

Cat.No: TN6736

Synonym: 24,25-Dihydrolanosterol,Lanostenol,二氢羊毛甾醇

Target: Others

Cat.No: TN1927

Synonym: 1-(6-methoxy-1,3-benzodioxol-5-yl)propan-1-one

Target: TRP/TRPV Channel

Cat.No: T4S1173

Synonym: 仙鹤草酚B,仙鹤草酚 B

Target: Sirtuin, PPAR

L-Octanoylcarnitine

Cat.No: T19398

Target: Endogenous Metabolite

Benzoylpaeoniflorin

Cat.No: T6S1652

Target: COX

Cat.No: T3764

Synonym: Myricyl alcohol,1-Triacontanol,三十烷醇,Melissyl alcohol,Well-Bloom,Miraculan,Lithospermoside,triacontan-1-ol

Target: Others

(E)-Cinnamamide

Cat.No: T13669

Synonym: trans-Cinnamamide,肉桂酰胺

Target: Others

Benzoylhypaconine

Cat.No: T6S1884

Synonym: 苯甲酰次乌头碱,Benzoylhypacoitine,苯甲酰次乌头原碱

Target: Others

Liquiritin apioside

Cat.No: TL0002

Target: Others

Cat.No: T3S2197

Synonym: Senegenic acid,远志皂甙

Target: Others

(±)-Abscisic acid

Cat.No: T3014

Synonym: Abscisic acid,Dormin,脱落酸,Abscisinsaeure

Target: Others

Cat.No: T3227

Synonym: Salvianic acid A,Dan shen suan A,丹参素

Target: Apoptosis, Nrf2, Autophagy

Cat.No: TMO2787

Synonym: dioxoanthracene,Anthradione,anthracenedione,蒽醌

Target: Virus Protease

Luteolin-3-O-beta-D-glucuronide

Cat.No: TQ0070

Target: Others

Cat.No: T4587

Synonym: BCP10902,Puerarin Apioside,葛根素芹菜糖苷,芹糖葛根素苷

Target: Tyrosinase

Cat.No: T6S0630

Target: P450, TNF

Cat.No: T21495

Target: Others

Cat.No: T4911

Synonym: 4-hydroxyphenyl-D-lucopyranoside,alpha-Arbutoside,α-熊果苷,alpha-Arbutin

Target: Tyrosinase

Cimiracemoside C

Cat.No: TN1499

Synonym: 千层纸素A-7-0-Β-D-葡萄糖醛酸苷,Cimicifugoside M

Target: AMPK

Hexahydrocurcumin

Cat.No: TQ0288

Target: Reactive Oxygen Species, ROS, COX

Cat.No: T2S1181

Synonym: Aloenin A,Aloearbonaside,芦荟宁

Target: Beta-Secretase, AChR

(2R)-6-Methoxynaringenin

Cat.No: TN3176L

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Species：

Expression System：

Tag：

Cat. No.	Product Name	Species	Expression System
TMPK-00539	PLAU/uPA Protein (active form), Cynomolgus, Recombinant (His) URK,ATF,UPA,u-PA,Urokinase,QPD,PLAU,BDPLT5	Cynomolgus	HEK293 Cells
	Plasminogen activator, urokinase (uPA) is a secreted serine protease whose Dysregulation is often accompanied by various cancers. PLAU inhibition could suppress tumor growth. Collectively, PLAU is necessary for tumor progression and can be a diagnostic and prognostic biomarker in HNSCC. PLAU/uPA Protein (active form), Cynomolgus, Recombinant (His) is expressed in HEK293 mammalian cells with C-His tag. The predicted molecular weight is 47.23 kDa and the accession number is A0A2K5WND1.
TMPK-00274	PLAU/uPA Protein (active form), Human, Recombinant (His & Avi), Biotinylated QPD,Urokinase,BDPLT5,UPA,ATF,URK,u-PA,PLAU	Human	HEK293 Cells
	Plasminogen activator, urokinase (uPA) is a secreted serine protease whose Dysregulation is often accompanied by various cancers. PLAU inhibition could suppress tumor growth. Collectively, PLAU is necessary for tumor progression and can be a diagnostic and prognostic biomarker in HNSCC. PLAU/uPA Protein (active form), Human, Recombinant (His & Avi), Biotinylated is expressed in HEK293 mammalian cells with C-His-Avi tag. The predicted molecular weight is 49.3 kDa and the accession number is P0074...
TMPK-00114	C-Reactive Protein /CRP Protein, Human, Recombinant (His) C-reactive protein,MGC88244,PTX1MGC149895,CRP,pentr...	Human	HEK293 Cells
	C-reactive protein (CRP) is a polypeptide molecule belonging to the family of pentraxins. CRP is synthesized primarily by the liver in response to certain pro-inflammatory cytokines. It plays an important role in innate immunity, opsonization by its properties, complement activation and immunoglobulins receptor binding. CRP is a protein of the acute systemic inflammation and is, therefore, a prime marker of inflammation.The CRP is quantified by immunonephelometry or immunoturbidimetry. C-Reactiv...
TMPY-02047	C-Reactive Protein Protein, Rat, Recombinant (His) C-reactive protein, pentraxin-related	Rat	HEK293 Cells
	C-Reactive Protein Protein, Rat, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 24.6 kDa and the accession number is H6X2V1.
TMPY-03363	C-Reactive Protein Protein, Human, Recombinant C-Reactive Protein,C-reactive protein, pen...	Human	HEK293 Cells
	C-Reactive Protein Protein, Human, Recombinant is expressed in HEK293 mammalian cells. The predicted molecular weight is 23 kDa and the accession number is P02741-1.
TMPY-05336	C-Reactive Protein Protein, Human, Recombinant, Biotinylated C-Reactive Protein,PTX1,C-reactive protein...	Human	HEK293 Cells
	C-Reactive Protein Protein, Human, Recombinant, Biotinylated is expressed in HEK293 mammalian cells. The predicted molecular weight is 23 kDa and the accession number is P02741-1.
TMPY-05249	ITK Protein, Human, Recombinant (Actived By LCK, GST) LYK,PSCTK2,LPFS1,IL2-inducible T-cell kinase,EMT	Human	Baculovirus Insect Cells
	ITK Protein, Human, Recombinant (Actived By LCK, GST) is expressed in Baculovirus insect cells with GST tag. The predicted molecular weight is 57.7 kDa and the accession number is Q08881.
TMPY-01581	C-Reactive Protein Protein, Mouse, Recombinant (His) C-reactive protein, pentraxin-related,AI255847	Mouse	HEK293 Cells
	C-Reactive Protein Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 24.4 kDa and the accession number is P14847.
TMPY-06937	C-Reactive Protein Protein, Human, Recombinant (His & Avi), Biotinylated C-Reactive Protein,PTX1,C-reactive protein...	Human	HEK293 Cells
	C-Reactive Protein Protein, Human, Recombinant (His & Avi), Biotinylated is expressed in HEK293 mammalian cells with His and Avi tag. The predicted molecular weight is 26.3 kDa and the accession number is P02741-1.
TMPK-01333	C-Reactive Protein /CRP Protein, Cynomolgus, Recombinant (His) C-reactive protein,pentraxin 1,PTX1,PTX1MGC149895,M...	Cynomolgus	HEK293 Cells
	C-reactive protein (CRP) is a polypeptide molecule belonging to the family of pentraxins. CRP is synthesized primarily by the liver in response to certain pro-inflammatory cytokines. It plays an important role in innate immunity, opsonization by its properties, complement activation and immunoglobulins receptor binding. CRP is a protein of the acute systemic inflammation and is, therefore, a prime marker of inflammation.The CRP is quantified by immunonephelometry or immunoturbidimetry. C-Reactiv...
TMPJ-00254	TGF beta 3 Protein, Human/Mouse/Rat, Recombinant Latency-associated peptide,TGF-beta-3,Transforming growth fa...	Human,Mouse,Rat	HEK293 Cells
	Transforming growth factor beta 3(TGFB3) is a member of a TGF -β superfamily which is defined by theirstructural and functional similarities. TGFB3 is secreted as a complex with LAP. This latent form of TGFB3becomes active upon cleavage by plasmin, matrix metalloproteases, thrombospondin -1, and a subset ofintegrins. It binds with high affinity to TGF- β RII, a type II serine/threonine kinase receptor. TGFB3 is involved incell differentiation, embryogenesis and development.It is believed to regu...
TMPY-05717	Integrin alpha V beta 8 Protein, Human, Recombinant (His) Integrin alpha V β8,Integrin α V β 8	Human	HEK293 Cells
	Integrin alpha V beta 8 is a receptor for fibronectin. It recognizes the sequence R-G-D in its ligands. ITGAVB8 does not appear to assume different activation states; and the cytoplasmic tail does not connect to the cytoskeleton. It binds ligands containing an RGD motif; including vitronectin; fibrin and the latency associated peptide (LAP) of the latent TGF-beta complex. High affinity binding of alpha V beta 8 to LAP allows proteolytic cleavage by MT1-MMP; which releases active TGF-beta. This m...
TMPY-00672	Azurocidin/CAP37 Protein, Human, Recombinant (His) AZU,NAZC,azurocidin 1,hHBP,AZAMP,HUMAZUR,CAP37,HBP,AZU1	Human	HEK293 Cells
	Azurocidin (AZU1), also known as heparin-binding protein (HBP) or cationic antimicrobial protein 37 (CAP37), is an azurophil granule antibiotic protein, with monocyte chemotactic and antibacterial activity. The Azurophil granules, specialized lysosomes of the neutrophil, contain at least 10 proteins implicated in the killing of microorganisms. Azurocidin is a member of the serine protease family that includes Cathepsin G, neutrophil elastase (NE), and proteinase 3 (PR3), however, Azurocidin is n...
TMPY-02585	Acid sphingomyelinase/SMPD1 Protein, Mouse, Recombinant (His) aSMase,ASM,Zn-SMase,A-SMase,sphingomyelin phosphodiesterase ...	Mouse	Baculovirus Insect Cells
	Sphingomyelin phosphodiesterase 1 (SMPD1) , also known as ASM ( acid sphingomyelinase ), is a member of the acid sphingomyelinase family of enzymes. Three isoforms have been identified, isoform 1 is 631 amino acids (aa) in length as the pro form, while Isoform 2 and isoform 3 have lost catalytic activity. The active SMPD1 isoform 1 contains one saposin B-type domain that likely interacts with sphingomyelin, and a catalytic region. Human SMPD1 is 86% aa identical to mouse SMPD1. SMPD1 is a monome...
TMPJ-00137	APRIL/TNFSF13 Protein, Human, Recombinant (Flag & His) TRDL-1,TNF- and APOL-related leukocyte expressed ligand 2,Tu...	Human	HEK293 Cells
	APRIL (a proliferation-inducing ligand), also known as TNFSF13, TALL2, TRDL1, and CD256, is a member of the TNF ligand superfamily. It is synthesized as a 32 kDa proprotein which is cleaved by furin in the Golgi to release the active 17 kDa soluble molecule. Secreted human APRIL, which consists almost entirely of a single TNF homology domain, shares 85% amino acid sequence identity with mouse and rat APRIL. Both APRIL and its close relative BAFF bind and signal through the TNF superfamily recept...
TMPY-02185	Coagulation factor XIII B/F13B Protein, Human, Recombinant (His) Coagulation factor 13,coagulation factor XIII, B polypeptide...	Human	HEK293 Cells
	Coagulation factor XIII B chain, also known as Fibrin-stabilizing factor B subunit, Protein-glutamine gamma-glutamyltransferase B chain, Transglutaminase B chain and F13B, is a secreted protein which contains 1 Sushi ( CCP / SCR ) domains. Coagulation factor XIII is the last zymogen to become activated in the blood coagulation cascade. Plasma factor XIII is a heterotetramer composed of 2 A subunits and 2 B subunits. The A subunits have catalytic function, and the B subunits do not have en...
TMPY-01104	Coagulation factor XI/F11 Protein, Human, Recombinant (His) coagulation factor 11,coagulation factor XI,FXI	Human	HEK293 Cells
	Factor XI (plasma thromboplastin antecedent) is a plasma glycoprotein, and a zymogen acting as a serine protease which participates in blood coagulation as a catalyst in the conversion of factor IX to factor IXa in the presence of calcium ions. It is an unusual dimeric protease, with structural features that distinguish it from vitamin K-dependent coagulation proteases. The factor XI is synthesized in the liver as a single polypeptide chain with a molecular weight estimated between 125 ~160 kDa ...
TMPJ-00897	TPSB2 Protein, Mouse, Recombinant (His) Tryptase-2,Mast cell protease 6,Tryptase beta-2,Tryptase β-2...	Mouse	HEK293 Cells
	Tryptase beta-2(Tpsb2), also known as Mast cell protease 6(mMCP-6), belongs to the peptidase S1 family and Tryptase subfamily. Tryptase is the major neutral protease present in mast cells and is secreted upon the coupled activation-degranulation response of this cell type. It plays a role in innate immunity. Tpsb2 can be detected primarily in skin during embryogenesis. Tpsb2 can not be detected at early embryonic stages but is abundantly expressed in later stages with a peak at E17.5-E18.5. Tryp...
TMPH-03429	DOG1 Protein, S. cerevisiae, Recombinant (His) DOG1,2-DOG-6-P 1,2-deoxyglucose-6-phosphatase 1,2-deoxygluco...	Saccharomyces cerevisiae	P. pastoris (Yeast)
	Active on 2-DOG-6P, also very active on fructose-1P. DOG1 Protein, S. cerevisiae, Recombinant (His) is expressed in yeast with N-6xHis tag. The predicted molecular weight is 29.1 kDa and the accession number is P38774.
TMPH-01629	LOXL1 Protein, Human, Recombinant (His) Lysyl oxidase-like protein 1,LOXL1,Lysyl oxidase homolog 1	Human	E. coli
	Active on elastin and collagen substrates.
TMPH-02825	ACOX1 Protein, Mouse, Recombinant (Myc) AOX,Peroxisomal fatty acyl-CoA oxidase,EC:1.3.3.6,Peroxisoma...	Mouse	E. coli
	Catalyzes the desaturation of acyl-CoAs to 2-trans-enoyl-CoAs. First enzyme of the fatty acid beta-oxidation pathway.; Shows highest activity against medium-chain fatty acyl-CoAs and activity decreases with increasing chain length.; Is active against a much broader range of substrates and shows activity towards very long-chain acyl-CoAs. Is twice as active as isoform 1 against 16-hydroxy-palmitoyl-CoA and is 25% more active against 1,16-hexadecanodioyl-CoA.
TMPH-02474	HAOX1 Protein, Mouse, Recombinant (His) Hao1,Glyoxylate oxidase,Glycolate oxidase,2-Hydroxyacid oxid...	Mouse	E. coli
	Has 2-hydroxyacid oxidase activity. Most active on the 2-carbon substrate glycolate, but is also active on 2-hydroxy fatty acids, with high activity towards 2-hydroxy palmitate and 2-hydroxy octanoate. HAOX1 Protein, Mouse, Recombinant (His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 45.0 kDa and the accession number is Q9WU19.
TMPH-00660	NikR Protein, E. coli, Recombinant (His) nikR,Nickel-responsive regulator	E. coli	E. coli
	Transcriptional repressor of the nikABCDE operon. Is active in the presence of excessive concentrations of intracellular nickel.
TMPH-01628	LOXL1 Protein, Human, Recombinant Lysyl oxidase-like protein 1,Lysyl oxidase homolog 1,LOXL1	Human	E. coli
	Active on elastin and collagen substrates. LOXL1 Protein, Human, Recombinant is expressed in E. coli expression system. The predicted molecular weight is 53.0 kDa and the accession number is Q08397.
TMPH-00655	McjB Protein, E. coli, Recombinant (His & Myc) Microcin J25-processing protein McjB,mcjB	E. coli	E. coli
	Along with McjC, necessary and sufficient to process the inactive microcin J25 (McjA) precursor into the active peptide.
TMPK-01092	OSCAR Protein, Human, Recombinant (hFc) Poly-Ig receptor 3,PIGR3,OSCAR,PIgR-3,MGC33613,mOSCAR	Human	HEK293 Cells
	Osteoclast-associated receptor (OSCAR) is a co-stimulatory receptor in osteoclastogenesis. Synovial tissues from active rheumatoid arthritis (RA) patients express higher levels of OSCAR compared with osteoarthritic and normal patients. OSCAR and tartrate-resistant acid phosphatase (TRAP) expression levels did not differ between the cartilage pannus junction (CPJ) and non-CPJ regions in active RA. OSCAR Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with C-hFc tag. The p...
TMPK-01117	OSCAR Protein, Mouse, Recombinant (hFc) PIgR-3,Poly-Ig receptor 3,OSCAR,MGC33613,mOSCAR,PIGR3	Mouse	HEK293 Cells
	Osteoclast-associated receptor (OSCAR) is a co-stimulatory receptor in osteoclastogenesis. Synovial tissues from active rheumatoid arthritis (RA) patients express higher levels of OSCAR compared with osteoarthritic and normal patients. OSCAR and tartrate-resistant acid phosphatase (TRAP) expression levels did not differ between the cartilage pannus junction (CPJ) and non-CPJ regions in active RA. OSCAR Protein, Mouse, Recombinant (hFc) is expressed in HEK293 mammalian cells with C-hFc tag. The p...
TMPJ-00542	TPSB2 Protein, Human, Recombinant (His) Tryptase-2,Tryptase Beta-2,TPS2,TPSB2,Tryptase II,Tryptase β...	Human	HEK293 Cells
	Tryptases are Trypsin-like Serine Proteases. β-Tryptases are the main isoenzymes in mast cells. Βtryptases form active tetramers with heparin proteoglycan. In the tetramer, the unique arrangement of the active sites facing a narrow central pore, β-Tryptases are resistant to macromolecule protease inhibitors . When mast cells are activated, β-Tryptases are released and participate in provoking inflammatory conditions . β-Tryptases have been implicated as mediators in the pathogenesis of asthma an...
TMPJ-01326	HDHD2 Protein, Human, Recombinant (His) HDHD2,Haloacid Dehalogenase-Like Hydrolase Domain-Containing...	Human	E. coli
	Haloacid Dehalogenase-Like Hydrolase Domain-Containing Protein 22 (HDHD2) is a member of the HAD-like hydrolase superfamily. HDHD2 includes L-2-Haloacid Dehalogenase, Epoxide Hydrolases and Phosphatases. There are two active sites in HDHD2 - an L-2-Haloacid Dehalogenase and a Carboxylate group. The L-2-Haloacid Dehalogenase active site catalyzes the hydrolytic dehalogenation of D- and L-2-Haloalkanoic Acids, producing L- and D-2-Hydroxyalkanoic Acids.
TMPY-02522	OTUB2 Protein, Human, Recombinant (His) OTU deubiquitinase, ubiquitin aldehyde binding 2,OTU2,OTB2,C...	Human	E. coli
	Otubain 2 (OTUB2) is a member of DUBs that belong to the ovarian tumour (OTU) superfamily of proteins which consists of a five-stranded β-sheet sandwiched in between a small helical amino-terminal region consisting of α1 and α2, and a large helical region comprised of α3-α10. Like other DUBs, otubain 2 (OTUB2) cleaves proteins precisely at the ubiquitin-protein bond so that ubiquitylation process can be reversed and regulated. Otubain 2 (OTUB2)'s active-site cleft is sterically occluded by a nov...
TMPH-00596	Colicin-E1 Protein, E. coli, Recombinant (Cell-Free, His & Myc) Colicin-E1,cea	E. coli	E. coli
	This colicin is a channel-forming colicin. This class of transmembrane toxins depolarize the cytoplasmic membrane, leading to dissipation of cellular energy.; Colicins are polypeptide toxins produced by and active against E.coli and closely related bacteria.
TMPH-00597	Colicin-E1 Protein, E. coli, Recombinant (His & Myc) cea,Colicin-E1	E. coli	E. coli
	This colicin is a channel-forming colicin. This class of transmembrane toxins depolarize the cytoplasmic membrane, leading to dissipation of cellular energy.; Colicins are polypeptide toxins produced by and active against E.coli and closely related bacteria.
TMPH-00229	Cathelicidin-4 Protein, Bovine, Recombinant (His & SUMO) Cathelicidin-4,Indolicidin,CATHL4	Bovine	E. coli
	Potent microbicidal activity; active against S.aureus and E.coli. Cathelicidin-4 Protein, Bovine, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 17.9 kDa and the accession number is P33046.
TMPH-01736	PGLYRP2 Protein, Human, Recombinant (His) PGLYRP2,Peptidoglycan recognition protein long,Peptidoglycan...	Human	P. pastoris (Yeast)
	May play a scavenger role by digesting biologically active peptidoglycan (PGN) into biologically inactive fragments. Has no direct bacteriolytic activity. PGLYRP2 Protein, Human, Recombinant (His) is expressed in yeast with N-6xHis tag. The predicted molecular weight is 62.0 kDa and the accession number is Q96PD5.
TMPH-01737	PGLYRP2 Protein, Human, Recombinant (His & SUMO) N-acetylmuramoyl-L-alanine amidase,Peptidoglycan recognition...	Human	E. coli
	May play a scavenger role by digesting biologically active peptidoglycan (PGN) into biologically inactive fragments. Has no direct bacteriolytic activity. PGLYRP2 Protein, Human, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 76.0 kDa and the accession number is Q96PD5.
TMPK-00478	Carbonic Anhydrase 12 Protein, Cynomolgus, Recombinant (His) CA12,CAXII,Carbonic anhydrase,CA-XII,Tumor antigen HOM-RCC-3...	Cynomolgus	HEK293 Cells
	Carbonic anhydrases (CAs) are a family of enzymes involved in the pH regulation of metabolically active cells/tissues. Carbonic anhydrase XII (CA XII) is a key mediator of several signaling pathways that are involved in cancer development.
TMPH-00598	Colicin-E5 Protein, E. coli, Recombinant (His & SUMO) Colicin-E5,col	E. coli	E. coli
	Colicins are polypeptide toxins produced by and active against E.coli and closely related bacteria. This colicin is an endonuclease. Colicin-E5 Protein, E. coli, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 24.8 kDa and the accession number is P18000.
TMPH-03475	MglB Protein, Salmonella typhimurium, Recombinant (His) D-galactose/D-glucose-binding protein,D-galactose-binding pe...	Salmonella typhimurium	P. pastoris (Yeast)
	This protein is involved in the active transport of galactose and glucose. It plays a role in the chemotaxis towards the two sugars by interacting with the trg chemoreceptor. MglB Protein, Salmonella typhimurium, Recombinant (His) is expressed in yeast with N-6xHis tag. The predicted molecular weight is 35.4 kDa and the accession number is P23905.
TMPH-00739	Thioredoxin-1 Protein, E. coli, Recombinant (His) Thioredoxin 1,trxA	E. coli	E. coli
	Participates in various redox reactions through the reversible oxidation of its active center dithiol to a disulfide and catalyzes dithiol-disulfide exchange reactions. Thioredoxin-1 Protein, E. coli, Recombinant (His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 15.7 kDa and the accession number is P0AA25.
TMPY-00821	HGFA Protein (pro form), Human, Recombinant (His) MGC138397,HGFA,RP11-529E1.2,肝细胞生长因子,MGC138395	Human	HEK293 Cells
	HGF activator (HGFA) is a serum-derived serine protease and belongs to the peptidase family S1.HGFA is responsible for the conversion of hepatocyte growth factor (HGF), from the inactive single-chain precursor to the active heterodimeric form, which is a potent mitogen, motogen, and morphogen for liver cells, epithelial cells, and endothelial cells. HGFA is synthesized and secreted by the liver and circulates in the plasma as an inactive single-chain zymogen in normal states. The zymogen is clea...
TMPY-01580	PRSS2 Protein, Mouse, Recombinant (His) Tesp4,protease, serine 2,Try2,Ta,TRY8,TRYP,Prss2	Mouse	HEK293 Cells
	Trypsin-2, also known as Trypsin II, Anionic trypsinogen, Serine protease 2, PRSS2 and TRY2, is a secreted protein that belongs to the trypsin serine protease family including Trypsin, PRSS1, PRSS2 and PRSS3. It consists of a signal peptide (residues 1-15), a pro region (residues 16-23), and a proteolytically active mature chain (residues 24-247). PRSS2 contains one peptidase S1 domain. It is secreted into the duodenum, hydrolysing peptides into their smaller building blocks, which is necessary ...
TMPH-03261	Cathepsin D Protein, Rat, Recombinant (His & Myc) Ctsd,Cathepsin D	Rat	E. coli
	Acid protease active in intracellular protein breakdown. Plays a role in APP processing following cleavage and activation by ADAM30 which leads to APP degradation. Cathepsin D Protein, Rat, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 45.2 kDa and the accession number is P24268.
TMPH-01240	MCM2 Protein, Human, Recombinant (His) DNA replication licensing factor MCM2,Nuclear protein BM28,M...	Human	E. coli
	Acts as component of the MCM2-7 complex (MCM complex) which is the putative replicative helicase essential for 'once per cell cycle' DNA replication initiation and elongation in eukaryotic cells. The active ATPase sites in the MCM2-7 ring are formed through the interaction surfaces of two neighboring subunits such that a critical structure of a conserved arginine finger motif is provided in trans relative to the ATP-binding site of the Walker A box of the adjacent subunit. The six ATPase active ...
TMPH-02254	Trypsin-1 Protein, Human, Recombinant (His & Myc) Trypsin-1,PRSS1,Serine protease 1,Beta-trypsin,Trypsin I,Ani...	Human	E. coli
	Has activity against the synthetic substrates Boc-Phe-Ser-Arg-Mec, Boc-Leu-Thr-Arg-Mec, Boc-Gln-Ala-Arg-Mec and Boc-Val-Pro-Arg-Mec. The single-chain form is more active than the two-chain form against all of these substrates.
TMPH-00516	StxA2 Protein, Enterobacteria phage 933W, Recombinant (E189K, His & Myc) Verotoxin 2 subunit A,Verocytotoxin 2 subunit A,Shiga-like t...	Enterobacteria phage 933W	E. coli
	The A subunit is responsible for inhibiting protein synthesis through the catalytic inactivation of 60S ribosomal subunits. After endocytosis, the A subunit is cleaved by furin in two fragments, A1 and A2: A1 is the catalytically active fragment, and A2 is essential for holotoxin assembly with the B subunits.
TMPH-02408	SPI Protein, Lentinula edodes, Recombinant (His) Serine protease inhibitor	Lentinula edodes	E. coli
	Serine protease inhibitor. Active against beta-trypsin and alpha-chymotrypsin with dissociation constants of 0.35 nM and 40 nM respectively. Inhibits factor XIa, but not other enzymes involved in coagulation and fibrinolysis. Does not inhibit subtilisin, lysyl endopeptidase, arginyl endopeptidase or papain.
TMPH-02195	TXNDC17 Protein, Human, Recombinant (GST) Thioredoxin-like protein 5,Protein 42-9-9,Thioredoxin domain...	Human	E. coli
	Disulfide reductase. May participate in various redox reactions through the reversible oxidation of its active center dithiol to a disulfide and catalyze dithiol-disulfide exchange reactions. Modulates TNF-alpha signaling and NF-kappa-B activation. Has peroxidase activity and may contribute to the elimination of cellular hydrogen peroxide.
TMPH-01246	POLR3A Protein, Human, Recombinant (His) RNA polymerase III subunit C160,RNA polymerase III 155 kDa s...	Human	E. coli
	DNA-dependent RNA polymerase catalyzes the transcription of DNA into RNA using the four ribonucleoside triphosphates as substrates. Largest and catalytic core component of RNA polymerase III which synthesizes small RNAs, such as 5S rRNA and tRNAs. Forms the polymerase active center together with the second largest subunit. A single-stranded DNA template strand of the promoter is positioned within the central active site cleft of Pol III. A bridging helix emanates from RPC1 and crosses the cleft ...
TMPH-00181	Cry1Ia Protein, Bacillus thuringiensis subsp., Recombinant (His & KSI) cryV1,cry1Ia,cryV,81 kDa crystal protein,Insecticidal delta-...	Bacillus thuringiensis subsp. Kurstaki	E. coli
	Promotes colloidosmotic lysis by binding to the midgut epithelial cells of certain coleopteran and lepidopteran species. Active on Plutella xylostella and Bombyx mori. Cry1Ia Protein, Bacillus thuringiensis subsp., Recombinant (His & KSI) is expressed in E. coli expression system with N-6xHis-KSI tag. The predicted molecular weight is 24.9 kDa and the accession number is Q45752.
TMPH-00361	Beta-mammal toxin Cn2 Protein, Centruroides noxius, Recombinant (His) Toxin 2,Beta-mammal toxin Cn2,Toxin II.9.2.2	Centruroides noxius	P. pastoris (Yeast)
	Mammal beta-toxins bind voltage-independently at site-4 of sodium channels (Nav) and shift the activation voltage to more negative potentials. This toxin is active against mammals. Beta-mammal toxin Cn2 Protein, Centruroides noxius, Recombinant (His) is expressed in yeast with N-6xHis tag. The predicted molecular weight is 9.6 kDa and the accession number is P01495.
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重组蛋白

PLAU/uPA Protein (active form), Cynomolgus, Recombinant (His)

Cat.No: TMPK-00539

Species: Cynomolgus

Expression System: HEK293 Cells

PLAU/uPA Protein (active form), Human, Recombinant (His & Avi), Biotinylated

Cat.No: TMPK-00274

Species: Human

Expression System: HEK293 Cells

C-Reactive Protein /CRP Protein, Human, Recombinant (His)

Cat.No: TMPK-00114

Species: Human

Expression System: HEK293 Cells

C-Reactive Protein Protein, Rat, Recombinant (His)

Cat.No: TMPY-02047

Species: Rat

Expression System: HEK293 Cells

C-Reactive Protein Protein, Human, Recombinant

Cat.No: TMPY-03363

Species: Human

Expression System: HEK293 Cells

C-Reactive Protein Protein, Human, Recombinant, Biotinylated

Cat.No: TMPY-05336

Species: Human

Expression System: HEK293 Cells

ITK Protein, Human, Recombinant (Actived By LCK, GST)

Cat.No: TMPY-05249

Species: Human

Expression System: Baculovirus Insect Cells

C-Reactive Protein Protein, Mouse, Recombinant (His)

Cat.No: TMPY-01581

Species: Mouse

Expression System: HEK293 Cells

C-Reactive Protein Protein, Human, Recombinant (His & Avi), Biotinylated

Cat.No: TMPY-06937

Species: Human

Expression System: HEK293 Cells

C-Reactive Protein /CRP Protein, Cynomolgus, Recombinant (His)

Cat.No: TMPK-01333

Species: Cynomolgus

Expression System: HEK293 Cells

TGF beta 3 Protein, Human/Mouse/Rat, Recombinant

Cat.No: TMPJ-00254

Species: Human,Mouse,Rat

Expression System: HEK293 Cells

Integrin alpha V beta 8 Protein, Human, Recombinant (His)

Cat.No: TMPY-05717

Species: Human

Expression System: HEK293 Cells

Azurocidin/CAP37 Protein, Human, Recombinant (His)

Cat.No: TMPY-00672

Species: Human

Expression System: HEK293 Cells

Acid sphingomyelinase/SMPD1 Protein, Mouse, Recombinant (His)

Cat.No: TMPY-02585

Species: Mouse

Expression System: Baculovirus Insect Cells

APRIL/TNFSF13 Protein, Human, Recombinant (Flag & His)

Cat.No: TMPJ-00137

Species: Human

Expression System: HEK293 Cells

Coagulation factor XIII B/F13B Protein, Human, Recombinant (His)

Cat.No: TMPY-02185

Species: Human

Expression System: HEK293 Cells

Coagulation factor XI/F11 Protein, Human, Recombinant (His)

Cat.No: TMPY-01104

Species: Human

Expression System: HEK293 Cells

TPSB2 Protein, Mouse, Recombinant (His)

Cat.No: TMPJ-00897

Species: Mouse

Expression System: HEK293 Cells

DOG1 Protein, S. cerevisiae, Recombinant (His)

Cat.No: TMPH-03429

Species: Saccharomyces cerevisiae

Expression System: P. pastoris (Yeast)

LOXL1 Protein, Human, Recombinant (His)

Cat.No: TMPH-01629

Species: Human

Expression System: E. coli

ACOX1 Protein, Mouse, Recombinant (Myc)

Cat.No: TMPH-02825

Species: Mouse

Expression System: E. coli

HAOX1 Protein, Mouse, Recombinant (His)

Cat.No: TMPH-02474

Species: Mouse

Expression System: E. coli

NikR Protein, E. coli, Recombinant (His)

Cat.No: TMPH-00660

Species: E. coli

Expression System: E. coli

LOXL1 Protein, Human, Recombinant

Cat.No: TMPH-01628

Species: Human

Expression System: E. coli

McjB Protein, E. coli, Recombinant (His & Myc)

Cat.No: TMPH-00655

Species: E. coli

Expression System: E. coli

OSCAR Protein, Human, Recombinant (hFc)

Cat.No: TMPK-01092

Species: Human

Expression System: HEK293 Cells

OSCAR Protein, Mouse, Recombinant (hFc)

Cat.No: TMPK-01117

Species: Mouse

Expression System: HEK293 Cells

TPSB2 Protein, Human, Recombinant (His)

Cat.No: TMPJ-00542

Species: Human

Expression System: HEK293 Cells

HDHD2 Protein, Human, Recombinant (His)

Cat.No: TMPJ-01326

Species: Human

Expression System: E. coli

OTUB2 Protein, Human, Recombinant (His)

Cat.No: TMPY-02522

Species: Human

Expression System: E. coli

Colicin-E1 Protein, E. coli, Recombinant (Cell-Free, His & Myc)

Cat.No: TMPH-00596

Species: E. coli

Expression System: E. coli

Colicin-E1 Protein, E. coli, Recombinant (His & Myc)

Cat.No: TMPH-00597

Species: E. coli

Expression System: E. coli

Cathelicidin-4 Protein, Bovine, Recombinant (His & SUMO)

Cat.No: TMPH-00229

Species: Bovine

Expression System: E. coli

PGLYRP2 Protein, Human, Recombinant (His)

Cat.No: TMPH-01736

Species: Human

Expression System: P. pastoris (Yeast)

PGLYRP2 Protein, Human, Recombinant (His & SUMO)

Cat.No: TMPH-01737

Species: Human

Expression System: E. coli

Carbonic Anhydrase 12 Protein, Cynomolgus, Recombinant (His)

Cat.No: TMPK-00478

Species: Cynomolgus

Expression System: HEK293 Cells

Colicin-E5 Protein, E. coli, Recombinant (His & SUMO)

Cat.No: TMPH-00598

Species: E. coli

Expression System: E. coli

MglB Protein, Salmonella typhimurium, Recombinant (His)

Cat.No: TMPH-03475

Species: Salmonella typhimurium

Expression System: P. pastoris (Yeast)

Thioredoxin-1 Protein, E. coli, Recombinant (His)

Cat.No: TMPH-00739

Species: E. coli

Expression System: E. coli

HGFA Protein (pro form), Human, Recombinant (His)

Cat.No: TMPY-00821

Species: Human

Expression System: HEK293 Cells

PRSS2 Protein, Mouse, Recombinant (His)

Cat.No: TMPY-01580

Species: Mouse

Expression System: HEK293 Cells

Cathepsin D Protein, Rat, Recombinant (His & Myc)

Cat.No: TMPH-03261

Species: Rat

Expression System: E. coli

MCM2 Protein, Human, Recombinant (His)

Cat.No: TMPH-01240

Species: Human

Expression System: E. coli

Trypsin-1 Protein, Human, Recombinant (His & Myc)

Cat.No: TMPH-02254

Species: Human

Expression System: E. coli

StxA2 Protein, Enterobacteria phage 933W, Recombinant (E189K, His & Myc)

Cat.No: TMPH-00516

Species: Enterobacteria phage 933W

Expression System: E. coli

SPI Protein, Lentinula edodes, Recombinant (His)

Cat.No: TMPH-02408

Species: Lentinula edodes

Expression System: E. coli

TXNDC17 Protein, Human, Recombinant (GST)

Cat.No: TMPH-02195

Species: Human

Expression System: E. coli

POLR3A Protein, Human, Recombinant (His)

Cat.No: TMPH-01246

Species: Human

Expression System: E. coli

Cry1Ia Protein, Bacillus thuringiensis subsp., Recombinant (His & KSI)

Cat.No: TMPH-00181

Species: Bacillus thuringiensis subsp. Kurstaki

Expression System: E. coli

Beta-mammal toxin Cn2 Protein, Centruroides noxius, Recombinant (His)

Cat.No: TMPH-00361

Species: Centruroides noxius

Expression System: P. pastoris (Yeast)

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Cat. No.	Product Name	Target	Signaling Pathways
TMIH-0519	Selexipag Active Metabolite-d7
	Selexipag Active Metabolite-d7 是 Selexipag Active Metabolite 的氘代化合物。Selexipag Active Metabolite 的 CAS 号为 475085-57-5。MRE269 是一种口服的长效前列环素受体激动剂前药，是 Selexipag 的活性代谢物，用于治疗肺动脉高压。
TMIH-0315	Lurasidone Inactive Metabolite 14283-d8 5α/6α-Hydroxy Lurasidone-d8 Hydrochloride (Mixture of Diastereomers)
	Lurasidone Inactive Metabolite 14283-d8 是 Lurasidone Inactive Metabolite 14283 的氘代化合物。Lurasidone Inactive Metabolite 14283 的 CAS 号为 186204-31-9。
TMIH-0316	Lurasidone Inactive Metabolite 14326-d8 5β/6β-Hydroxy Lurasidone-d8 Hydrochloride (Mixture of Diastereomers)
	Lurasidone Inactive Metabolite 14326-d8 是 Lurasidone Inactive Metabolite 14326 的氘代化合物。Lurasidone Inactive Metabolite 14326 的 CAS 号为 186204-33-1。
T60016	VV116 GS-621763-d1,JT001	SARS-CoV; RSV	Microbiology/Virology
	VV116 (JT001) 是一种针对呼吸道合胞病毒和 SARS-CoV-2 感染的选择性和口服活性核苷抗病毒剂。
T24046	WNK-IN-11-d3 WNK inhibitor-12,WNKIN12,WNK IN 12,WNK inhibitor 12,WNK-IN-12
	WNK-IN-12 is an effective, selective, and orally active WNK1 kinase inhibitor.
T19305	Eldecalcitol-d6	Others	Others
	Eldecalcitol is an orally active analogue of active vitamin D used in the treatment of osteoporosis. Eldecalcitol-d6 is the deuterium labeled Eldecalcitol.
T10663	Calcitriol-d6 Calcitriol D6,骨化三醇 D6	Others	Others
	Calcitriol D6 is the deuterated form of Calcitriol, which is the hormonally active form of vitamin D. Calcitriol is the active metabolite of vitamin D3 that activates the vitamin D receptor.
T12329	Ospemifene D4 FC-1271a D4	Estrogen/progestogen Receptor	Endocrinology/Hormones
	Ospemifene D4 is a deuterium labeled Ospemifene. Ospemifene is a selective and orally active modulator of estrogen receptor.
T11817	Lansoprazole Sulfide D4	Proton pump	Membrane transporter/Ion channel
	Lansoprazole Sulfide D4 is a deuterium labeled Lansoprazole Sulfide. Lansoprazole Sulfide is an orally active anti-TB (Mycobacterium tuberculosis) agent with IC50 values of 0.59 μM intracellularly and 0.46 μM in broth.Lansoprazole Sulfide is an active metabolite of the proton pump inhibitor Lansoprazole.
T13181	Tolcapone D7 Ro 40-7592 D7	Transferase	Metabolism
	Tolcapone D7 is a deuterium-labeled Tolcapone. Tolcapone is a selective and orally active inhibitor of COMT.
T12638	(R)-Praziquantel-d11 (R)-吡喹酮 D11,(R)-Praziquantel D11	5-HT Receptor	GPCR/G Protein; Neuroscience
	(R)-Praziquantel D11 is the deuterium labeled (R)-Praziquantel. (R)-Praziquantel is the active enantiomer of Praziquantel, is a partial the human 5-HT2B receptor agonist
T12144	N-Desethyl Oxybutynin-d5 hydrochloride N-Desethyl Oxybutynin D5 hydrochloride	Others	Others
	N-Desethyl Oxybutynin D5 hydrochloride is the the active metabolite Oxybutynin, is deuterium labeled N-Desethyl Oxybutynin hydrochloride.
T19489	O-Desmethyl gefitinib D8	EGFR	Angiogenesis; JAK/STAT signaling; Tyrosine Kinase/Adaptors
	O-Desmethyl gefitinib D8 is a deuterium labeled O-Desmethyl gefitinib that is an active metabolite of Gefitinib in human plasma.
TMIJ-0229	Mesalamine-d3
	Mesalamine-d3 是 Mesalamine 的氘代化合物。Mesalamine 的 CAS 号为 89-57-6。5-Aminosalicylic Acid 是一种特异性的PPARγ激动剂，还抑制 p21-激活激酶1 (PAK1) 和NF-κB，具有抗炎活性。
T12355	Palbociclib-d8 PD 0332991 D8,Palbociclib D8	CDK	Cell Cycle/Checkpoint
	Palbociclib D8 is a deuterium labeled Palbociclib. Palbociclib is a selective and orally active inhibitor of CDK4 and CDK6 (IC50s of 11 and 16 nM, respectively).
T13137	TGFβRI-IN-1	TGF-beta/Smad	Stem Cells
	TGFβRI-IN-1 is an oral active and selective inhibitor of TGFβ receptor type I (TGFβRI) kinase(IC50 values of 2 nM and 7.6 μM for TGFβRI and TGFβRII, respectively ).
T10282	Aliskiren D6 Hydrochloride SPP 100 D6 Hydrochloride,CGP60536B D6 Hydrochloride,CGP 60536 D6 Hydrochloride	Others	Others
	Aliskiren (CGP 60536) D6 Hydrochloride is a deuterium-labeled Aliskiren. Aliskiren hemifumarate is a direct and orally active renin inhibitor (IC50: 1.5 nM).
T12210	Netupitant D6 CID-6451149 D6	Others	Others
	Netupitant D6 is the deuterium labeled Netupitant, which is a selective and orally active antagonist of neurokinin-1 receptor.
T13195	Trandolapril D5 RU44570 D5	Others	Others
	Trandolapril D5 is a deuterium labeled Trandolapril. Trandolapril is an orally active inhibitor of angiotensin converting enzyme (ACE) for hypertension and congestive heart failure (CHF).
T19187	Aliskiren D6 hemifumarate CGP 60536 D6 hemifumarate,SPP 100 D6 hemifumarate,CGP60536B D6 hemifumarate	RAAS	Endocrinology/Hormones
	Aliskiren (CGP 60536) D6 hemifumarate is a deuterium-labeled Aliskiren hemifumarate. Aliskiren hemifumarate is a direct and orally active renin inhibitor (IC50: 1.5 nM).
T19273	Debutyldronedarone D7 SR-35021 D7	Others	Others
	Debutyldronedarone D7 is deuterium-labeled Debutyldronedarone, which is the main circulating active metabolite of dronedarone in the body.
TMID-0301	Vitamin-d4-d3
	Vitamin-d4-d3 是 Vitamin 的氘代化合物。Vitamin 的 CAS 号为 511-28-4。
T11585	Hydroxy Itraconazole D8 R-63373 D8	Others	Others
	Hydroxy Itraconazole D8 is the deuterium-labeled Hydroxy Itraconazole. Hydroxy Itraconazole is an active metabolite of Itraconazole, which is a triazole antifungal agent.
TMIJ-0093	Keto Pioglitazone-d4
	Keto Pioglitazone-d4 是 Keto Pioglitazone 的氘代化合物。Keto Pioglitazone 的 CAS 号为 146062-45-5。
T31813	Fludalanine MK641,D-Alanine-2-d, 3-fluoro-,3-Fluoro-D-(2-2H)alanine
	Fludalanine (MK641), an analogue of D-alanine, irreversiably inactivates racemase and also inhibits synthase. When used in combination with cycloserine, it has been found to be more active against a variety of non-mycobacterium organisms than fludalanine
T71984	Enrofloxacin-d5
	Enrofloxacin-d5 is intended for use as an internal standard for the quantification of enrofloxacin by GC- or LC-MS. Enrofloxacin is a fluoroquinolone antibiotic. It is active against panels of Campylobacter, E. coli, and Salmonella isolates (mean MIC50s = 0.06, 0.5, and 0.03 µg/ml, respectively). It is also active against equine isolates of L. intracellularis (MICs = 0.125-0.5 µg/ml). Enrofloxacin inhibits bacterial DNA gyrase. In vivo, enrofloxacin (10 mg/kg) increases survival in a mouse model...
TMID-0300	Vitamin-d4-d5
	Vitamin-d4-d5 是 Vitamin 的氘代化合物。Vitamin 的 CAS 号为 511-28-4。
T10144	4-Hydroxyatomoxetine D3	Others	Others
	4-Hydroxyatomoxetine D3 is a deuterium labeled 4-Hydroxyatomoxetine. 4-Hydroxyatomoxetine is an active metabolite of Atomoxetine. 4-Hydroxyatomoxetine is metabolized by CYP2D6. Atomoxetine is a noradrenaline reuptake inhibitor.
T10149	4-Hydroxypropranolol-d7 hydrochloride (±)-4-hydroxy Propranolol D7 hydrochloride,4-Hydroxypropranolol D7 hydrochloride	Others	Others
	4-Hydroxypropranolol D7 hydrochloride is deuterium-labeled 4-Hydroxypropranolol hydrochloride. 4-Hydroxypropranolol hydrochloride is an active metabolite of Propranolol, with a potency comparable to Propranolol. It inhibits β1- and β2-adrenergic receptors
T12955	Sofosbuvir D6 PSI-7977 D6,GS-7977 D6	Others	Others
	Sofosbuvir D6 is the deuterium labeled Sofosbuvir. Sofosbuvir is an active inhibitor of HCV RNA replication in the HCV replicon assay, demonstrates potent anti-hepatitis C virus (HCV) activity.
TMID-0271	Miloxacin-d3
	Miloxacin-d3 是 Miloxacin 的氘代化合物。Miloxacin 的 CAS 号为 37065-29-5。
T10351	Aprocitentan D4 ACT-132577 D4	Others	Others
	Aprocitentan D4 (ACT-132577 D4) is a deuterium-labeled Aprocitentan. Aprocitentan is a major and pharmacologically active metabolite of Macitentan. Aprocitentan is a dual ETA/ETB antagonist (IC50s: 3.4 nM and 987 nM; pA2s: 6.7 and 5.5).
TMIH-0295	LBQ657-d4
	LBQ657-d4 是 LBQ657 的氘代化合物。LBQ657 的 CAS 号为 149709-44-4。Sacubitrilat 是活性的脑啡肽酶 (NEP) 抑制剂。
TMIJ-0174	Eszopiclone-d8
	Eszopiclone-d8 是 Eszopiclone 的氘代化合物。Eszopiclone 的 CAS 号为 138729-47-2。
T11088	Doxepin D3 Hydrochloride	Histamine Receptor	GPCR/G Protein; Immunology/Inflammation; Neuroscience
	Doxepin D3 Hydrochloride is a deuterium-labeled doxepin hydrochloride.Doxepin hydrochloride is an oral active tricyclic antidepressant used as a sedative.Doxepin hydrochloride is also an effective CYP450 inhibitor, significantly inhibiting CYP450 2C19 and
T36021	Flumequine-13C3 Flumequine-13C3
	Flumequine-13C3is intended for use as an internal standard for the quantification of flumequine by GC- or LC-MS. Flumequine is a fluoroquinolone antibiotic.1It is active againstS. aureus, S. pyogenes, B. subtilis, E. coli, P. aeruginosa, S. faecalis, andK. pneumoniae(MICs = 1-100 μg/ml). Flumequine is also active against field isolates of B. hyodysenteriae (MICs = 6.25-200 μg/ml).2It inhibits DNA gyrase, disrupting supercoiling of bacterial DNA to block transcription and replication.3In vivo, fl...
TMIJ-0141	(S)-Amlodipine-d4
	(S)-Amlodipine-d4 是 (S)-Amlodipine 的氘代化合物。(S)-Amlodipine 的 CAS 号为 103129-82-4。Levamlodipine 是一种二氢吡啶钙通道阻滞剂，具有舒张血管的作用，可用于高血压和心绞痛的研究。
T12521	Ponatinib-d8 AP24534 D8	Others	Others
	Ponatinib D8 is a deuterium labeled Ponatinib. Ponatinib is an orally active inhibitor of multi-targeted kinase(Abl, PDGFRα, VEGFR2, FGFR1, and Src with IC50s of 0.37 nM, 1.1 nM, 1.5 nM, 2.2 nM, and 5.4 nM, respectively).
T11246	Etoricoxib-d4 MK-0663 D4,依托考昔 D4,L-791456 D4,Etoricoxib D4	Others	Others
	Etoricoxib D4 is a non steroidal anti-inflammatory agent, acting as a selective and orally active COX-2 inhibitor, with IC50s of 1.1 μM and 116 μM for COX-2 and COX-1 in human whole blood.Etoricoxib D4 is a deuterium labeled Etoricoxib.
TMID-0079	Norfloxacin-d8
	Norfloxacin-d8 是 Norfloxacin 的氘代化合物。Norfloxacin 的 CAS 号为 70458-96-7。Norfloxacin是广谱抗生素，能通过结合DNA旋转酶抑制革兰氏阳性和阴性菌。
T11197	Enclomiphene D4 hydrochloride (E)-Clomiphene D4 hydrochloride,Enclomifene D4 hydrochloride,trans-Clomiphene D4 hydrochloride	Others	Others
	Enclomiphene D4 hydrochloride ((E)-Clomiphene D4 hydrochloride; trans-Clomiphene D4 hydrochloride; Enclomifene D4 hydrochloride) is a potent and orally active oestrogen receptor antagonist, with antioestrogenic property.Enclomiphene D4 hydrochloride ((E)-Clomiphene D4 hydrochloride; trans-Clomiphene D4 hydrochloride; Enclomifene D4 hydrochloride) is a deuterium labeled Enclomiphene.
TMIJ-0230	Oseltamivir EP Impurity C-d3 HCl
	Oseltamivir EP Impurity C-d3 HCl 是 Oseltamivir EP Impurity C HCl 的氘代化合物。Oseltamivir EP Impurity C HCl 的 CAS 号为 1415963-60-8。
TMID-0217	Norfluoxetine-d5 Hydrochloride
	Norfluoxetine-d5 Hydrochloride 是 Norfluoxetine Hydrochloride 的氘代化合物。Norfluoxetine Hydrochloride 的 CAS 号为 57226-68-3。Norfluoxetine Hydrochloride 是氟西汀的活性代谢物。氟西汀是一种抗抑郁药。
TMIH-0154	Ciprofloxacin-d8
	Ciprofloxacin-d8 是 Ciprofloxacin 的氘代化合物。Ciprofloxacin 的 CAS 号为 85721-33-1。Ciprofloxacin是一种有高抗菌活性的氟喹诺酮类抗生素。
TMIJ-0252	Benazeprilat-d5 Benazepril EP Impurity C-d5
	Benazeprilat-d5 是 Benazeprilat 的氘代化合物。Benazeprilat 的 CAS 号为 86541-78-8。Benazeprilat(CGS 14831) 是一种具有口服活性的贝那普利活性代谢物。Benazeprilat 具有高效的抗血压活性，可与其他其他类别的化合物（包括噻嗪类利尿剂和钙通道阻滞剂）联合使用来减少与心血管风险和继发性终末器官损伤相关的疾病的发生。Benazeprilat 可能用于研究急性左心室衰竭。
TMIH-0394	Nirmatrelvir-d9
	Nirmatrelvir-d9 是 Nirmatrelvir 的氘代化合物。Nirmatrelvir 的 CAS 号为 2628280-40-8。PF-07321332 是一种有效的口服活性SARS-CoV 3CLPRO抑制剂，对 SARS-CoV-2 病毒有针对性，可研究 COVID-19。它是一种胰蛋白酶样蛋白酶抑制剂，可抑制气道上皮钠通道功能。
TMIH-0024	10,11-Dihydro-10-hydroxycarbamazepine-d4 rac-Licarbazepine-d4
	10,11-Dihydro-10-hydroxycarbamazepine-d4 是 10,11-Dihydro-10-hydroxycarbamazepine 的氘代化合物。10,11-Dihydro-10-hydroxycarbamazepine 的 CAS 号为 29331-92-8。Licarbazepine 是一种有效的电压门控钠通道阻滞剂，具有抗惊厥和稳定情绪的功效。
TMIJ-0335	Dehydro aripiprazole-d8
	Dehydro aripiprazole-d8 是 Dehydro aripiprazole 的氘代化合物。Dehydro aripiprazole 的 CAS 号为 129722-25-4。Dehydroaripiprazole 是 Aripiprazole 的活性代谢产物，具有抗精神病活性。Aripiprazole 是也一种抗精神病药。
TMIJ-0271	N-Desethyl Amodiaquine-d5 DiHCl
	N-Desethyl Amodiaquine-d5 DiHCl 是 N-Desethyl Amodiaquine DiHCl 的氘代化合物。N-Desethyl Amodiaquine DiHCl 的 CAS 号为 79352-78-6。N-Desethyl amodiaquine 是一种抗寄生虫剂，是主要的生物活性阿莫地喹代谢物。它对菌株 V1/S 和 3D7 的 IC50值分别为 97 nM 和 25 nM。
TMID-0302	Vitamin K3-d3
	Vitamin K3-d3 是 Vitamin K3 的氘代化合物。Vitamin K3 的 CAS 号为 58-27-5。Menadione是合成的萘醌，能够在体内转化成活性维生素K2。
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同位素标记化合物

Selexipag Active Metabolite-d7

Cat.No: TMIH-0519

Lurasidone Inactive Metabolite 14283-d8

Cat.No: TMIH-0315

Synonym: 5α/6α-Hydroxy Lurasidone-d8 Hydrochloride (Mixture of Diastereomers)

Lurasidone Inactive Metabolite 14326-d8

Cat.No: TMIH-0316

Synonym: 5β/6β-Hydroxy Lurasidone-d8 Hydrochloride (Mixture of Diastereomers)

Cat.No: T60016

Synonym: GS-621763-d1,JT001

Target: SARS-CoV, RSV

Cat.No: T24046

Synonym: WNK inhibitor-12,WNKIN12,WNK IN 12,WNK inhibitor 12,WNK-IN-12

Eldecalcitol-d6

Cat.No: T19305

Target: Others

Cat.No: T10663

Synonym: Calcitriol D6,骨化三醇 D6

Target: Others

Cat.No: T12329

Synonym: FC-1271a D4

Target: Estrogen/progestogen Receptor

Lansoprazole Sulfide D4

Cat.No: T11817

Target: Proton pump

Cat.No: T13181

Synonym: Ro 40-7592 D7

Target: Transferase

(R)-Praziquantel-d11

Cat.No: T12638

Synonym: (R)-吡喹酮 D11,(R)-Praziquantel D11

Target: 5-HT Receptor

N-Desethyl Oxybutynin-d5 hydrochloride

Cat.No: T12144

Synonym: N-Desethyl Oxybutynin D5 hydrochloride

Target: Others

O-Desmethyl gefitinib D8

Cat.No: T19489

Target: EGFR

Cat.No: TMIJ-0229

Cat.No: T12355

Synonym: PD 0332991 D8,Palbociclib D8

Target: CDK

Cat.No: T13137

Target: TGF-beta/Smad

Aliskiren D6 Hydrochloride

Cat.No: T10282

Synonym: SPP 100 D6 Hydrochloride,CGP60536B D6 Hydrochloride,CGP 60536 D6 Hydrochloride

Target: Others

Cat.No: T12210

Synonym: CID-6451149 D6

Target: Others

Trandolapril D5

Cat.No: T13195

Synonym: RU44570 D5

Target: Others

Aliskiren D6 hemifumarate

Cat.No: T19187

Synonym: CGP 60536 D6 hemifumarate,SPP 100 D6 hemifumarate,CGP60536B D6 hemifumarate

Target: RAAS

Debutyldronedarone D7

Cat.No: T19273

Synonym: SR-35021 D7

Target: Others

Cat.No: TMID-0301

Hydroxy Itraconazole D8

Cat.No: T11585

Synonym: R-63373 D8

Target: Others

Keto Pioglitazone-d4

Cat.No: TMIJ-0093

Cat.No: T31813

Synonym: MK641,D-Alanine-2-d, 3-fluoro-,3-Fluoro-D-(2-2H)alanine

Enrofloxacin-d5

Cat.No: T71984

Cat.No: TMID-0300

4-Hydroxyatomoxetine D3

Cat.No: T10144

Target: Others

4-Hydroxypropranolol-d7 hydrochloride

Cat.No: T10149

Synonym: (±)-4-hydroxy Propranolol D7 hydrochloride,4-Hydroxypropranolol D7 hydrochloride

Target: Others

Cat.No: T12955

Synonym: PSI-7977 D6,GS-7977 D6

Target: Others

Cat.No: TMID-0271

Aprocitentan D4

Cat.No: T10351

Synonym: ACT-132577 D4

Target: Others

Cat.No: TMIH-0295

Cat.No: TMIJ-0174

Doxepin D3 Hydrochloride

Cat.No: T11088

Target: Histamine Receptor

Flumequine-13C3

Cat.No: T36021

Synonym: Flumequine-13C3

(S)-Amlodipine-d4

Cat.No: TMIJ-0141

Cat.No: T12521

Synonym: AP24534 D8

Target: Others

Cat.No: T11246

Synonym: MK-0663 D4,依托考昔 D4,L-791456 D4,Etoricoxib D4

Target: Others

Cat.No: TMID-0079

Enclomiphene D4 hydrochloride

Cat.No: T11197

Synonym: (E)-Clomiphene D4 hydrochloride,Enclomifene D4 hydrochloride,trans-Clomiphene D4 hydrochloride

Target: Others

Oseltamivir EP Impurity C-d3 HCl

Cat.No: TMIJ-0230

Norfluoxetine-d5 Hydrochloride

Cat.No: TMID-0217

Ciprofloxacin-d8

Cat.No: TMIH-0154

Benazeprilat-d5

Cat.No: TMIJ-0252

Synonym: Benazepril EP Impurity C-d5

Nirmatrelvir-d9

Cat.No: TMIH-0394

10,11-Dihydro-10-hydroxycarbamazepine-d4

Cat.No: TMIH-0024

Synonym: rac-Licarbazepine-d4

Dehydro aripiprazole-d8

Cat.No: TMIJ-0335

N-Desethyl Amodiaquine-d5 DiHCl

Cat.No: TMIJ-0271

Cat.No: TMID-0302

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