JPM-OEt

Name: JPM-OEt
Brand: TargetMol
SKU: T15626
Rating: 4.5 (1 reviews)

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产品编号 T15626Cas号 262381-84-0

JPM-OEt is a broad spectrum cysteine cathepsin inhibitor with antitumor activity. JPM-OEt binds covalently in the active site and irreversibly inhibits the cysteine cathepsin family.

JPM-OEt

还可以

产品编号 T15626Cas号 262381-84-0

JPM-OEt is a broad spectrum cysteine cathepsin inhibitor with antitumor activity. JPM-OEt binds covalently in the active site and irreversibly inhibits the cysteine cathepsin family.

规格	价格	库存
2 mg	¥ 2,660	5日内发货
25 mg	¥ 10,600	6-8周
50 mg	¥ 13,800	6-8周
100 mg	¥ 17,500	6-8周

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产品描述	JPM-OEt is a broad spectrum cysteine cathepsin inhibitor with antitumor activity. JPM-OEt binds covalently in the active site and irreversibly inhibits the cysteine cathepsin family.
体内活性	JPM-OEt (50 mg/kg; i.p.; daily for 30 days) decreases tumor cathepsin B activity obviously[1]. JPM-OEt (50 mg/kg; i.p.; twice daily for 4 weeks) causes tumor regression in the RIP1-Tag2 (RT2) mouse model of pancreatic islet cell tumorigenesis[2]. JPM-OEt (50 mg/kg; i.p.; daily from 63 to 98 days) leads to an obviously delay in the increase of tumor burden during the first 2 weeks of treatment[3].