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A-893 是一个具有细胞活性的,甲基转移酶SMYD2的抑制剂,IC50值为 2.8 nM。
A-893 是一个具有细胞活性的,甲基转移酶SMYD2的抑制剂,IC50值为 2.8 nM。
规格 | 价格 | 库存 | 数量 |
---|---|---|---|
25 mg | ¥ 10,600 | 10-14周 | |
50 mg | ¥ 13,800 | 10-14周 | |
100 mg | ¥ 17,500 | 10-14周 |
产品描述 | A-893 is a cell-active inhibitor of Methyltransferase SMYD2 (IC 50 = 2.8 nM) . |
体外活性 | As expected, the ratio of p53K370me1 to overall p53 levels is reduced by treatment with either A-893 or AZ505. While this unexpectedly depicts a more robust response with AZ505, further dissection of the data provides clarity into the origin of this. While overall p53 levels are unaffected by A-893, a surprising >3-fold increase is observed with AZ505. Analysis of p53K370me1 levels reveals that inhibitor A-893 exhibited 42% reduction in the methyl mark, while AZ-505 is slightly less effective at 28% reduction [1]. |
分子量 | 577.54 |
分子式 | C29H38Cl2N4O4 |
CAS No. | 1868232-32-9 |
密度 | 1.32 g/cm3 (Predicted) |
存储 | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
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