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Tyk2-IN-5 is a selective and orally active inhibitor of Tyk2 JH2 (Ki: 0.086 nM for Tyk2 JH2; IC50: 25 nM for IFNα).
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Tyk2-IN-5 is a selective and orally active inhibitor of Tyk2 JH2 (Ki: 0.086 nM for Tyk2 JH2; IC50: 25 nM for IFNα).
规格 | 价格 | 库存 | 数量 |
---|---|---|---|
2 mg | ¥ 3,190 | 5日内发货 | |
5 mg | ¥ 3,730 | 5日内发货 | |
25 mg | ¥ 11,700 | 6-8周 | |
50 mg | ¥ 15,300 | 6-8周 | |
100 mg | ¥ 19,500 | 6-8周 | |
1 mL x 10 mM (in DMSO) | ¥ 4,120 | 5日内发货 |
产品描述 | Tyk2-IN-5 is a selective and orally active inhibitor of Tyk2 JH2 (Ki: 0.086 nM for Tyk2 JH2; IC50: 25 nM for IFNα). |
靶点活性 | IFN-α:25 nM, TYK2 JH1:0.086 nM (ki) |
分子量 | 434.43 |
分子式 | C21H19FN8O2 |
CAS No. | 1797432-62-2 |
密度 | 1.58 g/cm3 (Predicted) |
存储 | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | ||||||||||||||||||||||||||||||
溶解度信息 | DMSO: 43.33 mg/mL (99.74 mM), Sonication is recommended. | ||||||||||||||||||||||||||||||
溶液配制表 | |||||||||||||||||||||||||||||||
DMSO
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