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BRD4Inhibitor-28(Compound 18)是一款具有口服活性的BRD4抑制剂,其针对BRD40-BD1和BRD40-BD2的IC50值分别为15和55 nM。该化合物同时对BRD2-BD1、BRD3-BD1和BRDT-BD1也表现出抑制作用,对应的IC50值依次为19、25和68 nM。此外,BRD4Inhibitor-28在抗黑色素瘤方面展现出活性。
BRD4Inhibitor-28(Compound 18)是一款具有口服活性的BRD4抑制剂,其针对BRD40-BD1和BRD40-BD2的IC50值分别为15和55 nM。该化合物同时对BRD2-BD1、BRD3-BD1和BRDT-BD1也表现出抑制作用,对应的IC50值依次为19、25和68 nM。此外,BRD4Inhibitor-28在抗黑色素瘤方面展现出活性。
规格 | 价格 | 库存 | 数量 |
---|---|---|---|
25 mg | ¥ 11,700 | 8-10周 | |
50 mg | ¥ 15,300 | 8-10周 | |
100 mg | ¥ 19,500 | 8-10周 |
产品描述 | BRD4 Inhibitor-28 (Compound 18), an orally active molecule, selectively inhibits the bromodomains of BRD4 (BRD4-BD1 and BRD4-BD2) with IC50 values of 15 and 55 nM, respectively. It also demonstrates inhibition of BRD2-BD1, BRD3-BD1, and BRDT-BD1 with IC50 values of 19, 25, and 68 nM, respectively. Furthermore, this compound exhibits anti-melanoma activity [1]. |
分子量 | 387.43 |
分子式 | C23H21N3O3 |
CAS No. | 2468960-80-5 |
存储 | Shipping with blue ice. |
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