721
160
30
25
160
27
Cat. No. | Product Name | ||
---|---|---|---|
L2300 | 离子通道库 | 931 compounds | |
931 种与离子通道相关的生物活性小分子化合物的特有集合,用于离子通道相关的疾病和药物研究,可用于高通量筛选和高内涵筛选; | |||
L7110 | 抗高血压化合物库 | 678 compounds | |
678 种高血压相关的小分子,用于高通量和高内涵筛选; | |||
L6750 | 活血化瘀中药单体库 | 580 compounds | |
580种来源于常见活血化瘀中药的单体化合物,是药物开发、药理研究等领域的有效工具。 | |||
L3500 | 组蛋白修饰化合物库 | 469 compounds | |
469 个组蛋白修饰相关的小分子化合物的特有集合,用于高通量、高内涵筛选; | |||
L6730 | 抗病毒中药单体化合物库 | 268 compounds | |
268 种具有抗病毒活性的中药单体集合,是药物开发、药理研究的有效工具; | |||
L7700 | 神经再生化合物库 | 524 compounds | |
524 种神经再生相关化合物的独特集合,可用于高通量筛选和高内涵筛选; | |||
L6740 | 抗结直肠癌中药单体化合物库 | 382 compounds | |
382 种抗结直肠癌相关的中药单体集合,是药物开发、药理研究的有效工具; | |||
L7500 | 凝血与抗凝化合物库 | 144 compounds | |
144 个化合物的独特集合,可用于高通量筛选和高内涵筛选; | |||
L6810 | 中药单体化合物库 | 2755 compounds | |
2755 种中药来源的单体化合物,是药物开发、药理研究等领域的有力工具; | |||
L4700 | 免疫/炎症分子化合物库 | 4720 compounds | |
4720 种具有抗炎症活性的化合物的特有集合,可用于高通量筛选和高内涵筛选; | |||
L7810 | 高溶解性多官能团片段化合物库 | 1159 compounds | |
高溶解性多官能团片段库包含1159 种片段分子 | |||
L2140 | 癌细胞分化化合物库 | 406 compounds | |
406 个诱导肿瘤细胞分化化合物的独特集合,可用于高通量筛选和高内涵筛选; | |||
L8000 | 干细胞分化化合物库 | 1197 compounds | |
1197 种干细胞分化信号通路相关的生物活性小分子化合物的特有集合,可用于高通量、高内涵筛选; | |||
L2630 | 神经元分化化合物库 | 672 compounds | |
672 种与神经元分化相关的化合物,可以用于神经系统疾病药物研发 | |||
L1800 | 抗感染化合物库 | 2938 compounds | |
2938 种具有抗感染活性的化合物的特有集合,包括抗细菌、抗真菌、抗巨细胞病毒、抗HIV、抗SARS、抗流感等活性; | |||
L6710 | 中药抗炎分子库 | 1246 compounds | |
1246 种具有抗炎活性或靶向炎症相关靶点的中药单体集合,是药物开发、药理研究的有效工具; | |||
L2900 | 氧化还原化合物库 | 1264 compounds | |
1264 个活性化合物,已经验证具有一定的抗氧化活性,包括 ROS 清除剂、iNOS、eNOS、及抗氧化的天然产物,是研究疾病机理以及药物研究的优良载体 | |||
L8600 | 泛素化化合物库 | 210 compounds | |
210 种泛素化相关的小分子,用于高通量和高内涵筛选; | |||
L6220 | 蒙药化合物库 | 950 compounds | |
950 种蒙药来源的天然产物分子集合,可以用于高通量和高内涵筛选; | |||
L1380 | 转录因子库 | 695 compounds | |
695 种转录因子靶向、结构新颖的化合物; | |||
L6200 | 瑶药化合物库 | 221 compounds | |
221 种瑶药来源的天然产物分子集合,可以用于高通量和高内涵筛选; | |||
L6720 | 抗COVID-19中药单体库 | 1147 compounds | |
根据抗新冠肺炎疫情过程中应用于临床治疗的中药方剂,收集了1147 种相关中药来源的单体化合物,可用于高通量和高内涵筛选,是抗新冠病毒药物研发的良好工具; | |||
L8300 | 染色质修饰分子库 | 250 compounds | |
250 种染色质化学修饰相关的生物活性小分子化合物的特有集合,用于高通量、高内涵筛选; | |||
L3510 | 甲基化化合物库 | 128 compounds | |
128 种甲基化相关的化合物,可以用于高通量和高内涵筛选; | |||
L2800 | 5-羟色胺分子库 | 268 compounds | |
268 种生物活性小分子化合物,用于高通量、高内涵筛选; | |||
L7200 | 钙通道分子库 | 140 compounds | |
140 种钙通道相关化合物的独特集合,可用于高通量筛选和高内涵筛选; | |||
L7300 | 钾通道分子库 | 152 compounds | |
152 种钾通道相关化合物的独特集合,可用于高通量筛选和高内涵筛选; | |||
L7400 | 钠通道分子库 | 118 compounds | |
118 种钠通道相关化合物的独特集合,可用于高通量筛选和高内涵筛选; | |||
L2610 | 神经递质受体化合物库 | 1513 compounds | |
1513 种与神经递质受体相关的化合物,用于高通量、高内涵筛选; | |||
L9600 | 多肽分子库 | 791 compounds | |
791 种多肽类分子,可用于多肽药物开发及信号转导通路和作用机制研究; |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T32809 |
L-Lactate ion
L-Lactate,Lactate ion, L- |
Others | Others |
L-Lactate ion is the conjugate base of lactic acid. | |||
T11927 |
M2 ion channel blocker
|
Others | Others |
M2 ion channel blocker ,Antiviral agent, is capable of inhibiting and blocking the activity of M2 ion channel. | |||
T25026 |
Albitiazolium
Albitiazolium ion |
Others | Others |
Albitiazolium is an antimlarial agent. | |||
T32592 |
Lauralkonium
Lauralkonium ion,Lauralkonium cation |
Others | Others |
Lauralkonium is a bioactive chemical. | |||
T84763 |
Ulefnersen
ION-363 |
Others | Others |
Ulefnersen是用于肌萎缩侧索硬化(ALS)研究的RNA结合蛋白fused-in sarcoma(FUS)合成抑制剂。 | |||
T25640 |
Laurolinium
Laurolinium ion,Laurolinium cation |
Others | Others |
Laurolinium is an antimicrobial. | |||
T25636 |
Laudexium
Laudexium ion,Laudexium cation |
Others | Others |
Laudexium is a neuromuscular blocking drug or skeletal muscle relaxant in the category of non-depolarizing neuromuscular-blocking drugs. It is used adjunctively in surgical anesthesia to facilitate endotracheal intubation and to provide skeletal muscle re | |||
T34817 |
Tetrabutylphosphonium cation
Tetra-n-butylphosphonium,J279H,Tetrabutylphosphonium ion,Tetrabutylphosphonium,Phosphonium, tetrabutyl- |
Others | Others |
Tetrabutylphosphonium cation is a light orange solid and is the salt of the liphilic tetrabutylammonium cation and linear tribromide anion. | |||
T8552 |
PSEM 89S TFA
|
AChR | Neuroscience |
PSEM 89S TFA 是一种脑渗透性和选择性离子通道激动剂,分别对 Q79G 和 L141F 具有正交选择性。 | |||
T12421 |
PF-04885614
|
Sodium Channel | Membrane transporter/Ion channel |
PF-04885614是一种有效的NaV1.8抑制剂。PF-04885614有用于神经系统疾病和神经发育疾病研究的潜力。 | |||
T16347 |
NS3623
|
Potassium Channel | Membrane transporter/Ion channel |
NS3623 是 hERG1 (KV11.1)钾通道激活剂,激活IKr 和Ito 电流,具有抗心律失常作用。NS3623也是 hERG1 通道抑制剂。 | |||
T1814 |
ICILIN
AG-3-5 |
TRP/TRPV Channel | Membrane transporter/Ion channel |
ICILIN (AG-3-5) 是一种有效的的瞬时受体电位 M8 (TRPM8) 离子通道激动剂。 Icilin 激活 EGTA 中的 TRPM8,该激活作用具有剂量依赖性, EC50=1.4 μM。Icilin 通过调节 T 细胞反应减轻自身免疫性神经炎症。 | |||
T3171 |
GSK137647A
GSK 137647 |
GPR | Endocrinology/Hormones; GPCR/G Protein |
GSK137647A (GSK 137647) 是一种选择性FFA4激动剂,作用于人类和大小鼠FFA4的pEC50分别为6.3、6.1和6.2。 | |||
T10466 |
BAY-1797
|
P2X Receptor | Membrane transporter/Ion channel; Neuroscience |
BAY-1797 是具有口服活性的选择性P2X4高效拮抗剂,对人 P2X4 的IC50为 211 nM,具有抗伤害和抗炎作用。 | |||
T2298 |
ML204
|
TRP/TRPV Channel | Membrane transporter/Ion channel |
ML204 是有效的TRPC4/TRPC5通道选择性抑制剂,相比于 TRPC6 ,对TRPC4/TRPC5通道的选择性高出 19 倍,不影响其他的 TRP 通道和电压门控的钠、钾或 Ca2+通道。 | |||
T9627 |
PHD-1-IN-1
|
HIF/HIF Prolyl-Hydroxylase | Chromatin/Epigenetic; Metabolism |
PHD-1-IN-1 是口服有效的缺氧诱导因子脯氨酰羟化酶结构域 1抑制剂,IC50为 0.034 μM。它与活性位 Fe2+具有独特的单齿结合相互作用,并诱导形成一个 “Arg367-out” 口袋。 | |||
T4585 |
EGTA
Ethylenebis(oxyethylenenitrilo)tetraacet,乙二醇双(2-氨基乙基醚)四乙酸 |
Others | Others |
Ethylenebis(oxyethylenenitrilo)tetraacet 是一种特殊的钙离子螯合剂,能够显著抑制炎性巨噬细胞的底物粘附能力。EGTA (Ethylenebis(oxyethylenenitrilo)tetraacet) 在生理 pH 值(7.4) 下,Kd 为 60.5 nM,对 Ca2+比对 Mg2+有很高的特异性。 | |||
T70310 |
INCB-39110
|
Others | Others |
INCB-39110 is a JAK1 inhibitor. | |||
T68783 |
Stercuronium
|
Others | Others |
Stercuronium is an aminosteroid neuromuscular blocking agent which was never marketed. It acts as a competitive antagonist of the nicotinic acetylcholine receptor, and is also reported to be an acetylcholinesterase inhibitor. | |||
T68735 |
Ciclotropium (free base)
|
Others | Others |
Ciclotropium (free base) is quaternary ammonium compound with anticholinergic and parasympatholytic activity. Oral Cyclotropium bromide inhibited fasting and meal-stimulated colonic motility significantly without causing adverse side effects. After cyclotropium bromide, there was a significant correlation between antral contraction amplitude and gastric emptying. | |||
T68502 |
Dibrospidium Free Base
|
Others | Others |
Dibrospidium Free Base is a dispirotripiperazine derivative and alkylating agent with potential antineoplastic and anti-inflammatory activities. The duration of DNA synthesis inhibition in tumor cells was found to correlate with spirobromine antitumor activity. Spirobromin is superior to prospidin by the power of the anti-inflammatory effect. Spyrobromin can diminish the latent period of the development of tumours in the experimental rats at intraperitoneal administration. At intragastric admini... | |||
T2096 |
Framycetin sulfate
Neomycin Sulphate B,硫酸新霉素B,Framycetin sulphate |
Antibacterial; Antibiotic | Microbiology/Virology |
Framycetin sulfate (Neomycin Sulphate B) 是一种氨基糖苷类抗生素,是 RNase P 裂解活性抑制剂,Ki 为 35 μM。它抑制锤头状核酶,Ki 值为 13.5 μM,可用于肝性脑病和肠致病性大肠杆菌感染的研究。 | |||
T40101 |
(±)-1,2-Diolein
1,2-Dioleoyl-rac-glycerol,甘油1,2-二油酸酯 |
PKC | Chromatin/Epigenetic; Cytoskeletal Signaling |
(±)-1,2-Diolein (1,2-Dioleoyl-rac-glycerol) 是一种PKC 激活剂,可以增加肌小管 Ca2+内流。 | |||
T40857 |
Calcium ionophore II
Calcium ionophore II,N,N,N′,N′-Tetracyclohexyl-3-oxapentanediamide |
Others | Others |
Calcium ionophore II (N,N,N′,N′-Tetracyclohexyl-3-oxapentanediamide) 是一种亲脂性离子载体,可用于制备钙离子选择性电极。 | |||
T77728 |
Tubulin polymerization-IN-55
|
Microtubule Associated | Cytoskeletal Signaling |
Tubulin polymerization-IN-55 是一种高效的 Tubulin Polymerization 抑制剂,具有潜在的抗血管生成和抗肿瘤活性,对 A549、K562、HepG2、MDA-MB-231 和 HFL-1 显示出抗增殖作用。 | |||
T15233 |
Endovion
NS3728 |
Chloride channel | Membrane transporter/Ion channel |
Endovion (NS3728) 是阴离子通道抑制剂 和 Anoctamin-1 (ANO 1) 通道抑制剂,也是特异性的 VRAC/VSOAC 阻断剂。 | |||
T1561 |
Clobetasol propionate
Dermovate,Clobetasol 17-propionate,CGP9555,Temovate,丙酸氯倍他索,CCl 4725 |
Glucocorticoid Receptor; P450 | Endocrinology/Hormones; Metabolism |
Clobetasol propionate (CGP9555) 是CYP3A5的选择性抑制剂(IC50:0.206 μM),而对 CYP3A4 或其他主要 CYP 无抑制作用。它是皮质类固醇,对于牛皮癣和其他皮肤病具有潜在的研究价值。 | |||
T1234 |
5,5-Dimethyloxazolidine-2,4-dione
Dimethadion,Dimethadione,二甲双酮,Dimethyloxazolidinedione |
Calcium Channel | Membrane transporter/Ion channel; Metabolism |
5,5-Dimethyloxazolidine-2,4-dione (Dimethadione) 是抗惊厥药,是 TRIMETHADIONE 的活性代谢物。 | |||
T6240 |
Palbociclib Isethionate
Palbociclib (PD0332991) Isethionate,帕博西尼羟乙基磺酸盐,PD 0332991 isethionate,帕布昔利布羟乙基磺酸盐 |
CDK | Cell Cycle/Checkpoint |
Palbociclib Isethionate (PD 0332991 isethionate) 是一种高选择性的CDK4/6抑制剂,IC50为11 nM 和16 nM。它对一组 36 种额外的蛋白激酶没有抑制作用。 | |||
T9044 |
SORT-PGRN interaction inhibitor 1
|
Neurotensin Receptor | GPCR/G Protein |
SORT-PGRN interaction inhibitor 1 是一种 sortilin-progranulin 相互作用抑制剂,IC50为 2 μM。 | |||
T9656 |
AP-1/NF-κB activation inhibitor 1
|
NF-κB; DNA/RNA Synthesis | Cell Cycle/Checkpoint; DNA Damage/DNA Repair; NF-κB |
AP-1/NF-κB activation inhibitor 1 是一种有效的 AP-1和 NF-κB 介导的转录激活抑制剂(IC50=1 μM),不阻断 β-actin 启动子驱动的基础转录。AP-1/NF-κB activation inhibitor 1 对受刺激细胞中 IL-2和 IL-8的产生水平有相似的抑制作用。 | |||
T40863 |
Bisdionin C
|
Antibacterial | Microbiology/Virology |
Bisdionin C 是一种有效的 GH18 chitinase 抑制剂,对 A. fumigatus ChiB1 的 IC50 为 0.2 μM。 Bisdionin C 抑制人巨噬细胞壳三糖苷酶 (HCHT, IC50 = 8.3 μM) 和酸性哺乳动物几丁质酶 (AMCase, IC50 = 3.4 μM)。 | |||
T1127 |
Beclometasone dipropionate
Beclovent,Beclomethasone dipropionate,二丙酸倍氯米松,丙酸倍氯米松,Beconase,Vancenase |
Glucocorticoid Receptor | Endocrinology/Hormones |
Beclometasone dipropionate (Vancenase) 是具有口服活性的糖皮质激素,具有抗炎和免疫抑制作用。它是Betamethasone 的前体药物,Betamethasone 是 LPS 诱导的炎症及 MMP 释放的抑制剂。 | |||
T3189 |
B7/CD28 interaction inhibitor 1
CTLA-4 inhibitor |
Others | Others |
B7/CD28 interaction inhibitor 1 (CTLA-4 inhibitor) 是B7.1-CD28相互作用抑制剂(IC50:50 nM)。 | |||
T34383L |
2H-Naphth[2′,1′:4,5]indeno[1,2-d][1,3]dioxole, pregn-4-ene-3,20-dione deriv
|
Others | Others |
2H-Naphth[2′,1′:4,5]indeno[1,2-d][1,3]dioxole, pregn-4-ene-3,20-dione deriv在Sprague Dawley大鼠上进行测试时显示出高局部抗炎效力和高肺选择性。 | |||
T0283 |
Trimethadione
三甲双酮,3,5,5,-Trimethyloxazolidine-2,4-dione |
Calcium Channel | Membrane transporter/Ion channel; Metabolism |
Trimethadione (3,5,5,-Trimethyloxazolidine-2,4-dione) 是恶唑烷二酮类抗惊厥剂,也是一种 T 型钙通道阻滞剂,具有抗痛觉过敏作用,可用于研究失神发作。 | |||
T1559 |
Betamethasone dipropionate
Diprolene AF,SCH 11460,二丙酸倍他米松,Betamethasone 17,21-dipropionate,Diprolene,倍他米松二丙酸酯,Diprosone |
Glucocorticoid Receptor | Endocrinology/Hormones |
Betamethasone dipropionate (SCH 11460) 是糖皮质激素类固醇,具有免疫抑制、抗炎作用。 | |||
TP1153L |
Fibronectin Adhesion-promoting Peptide acetate
Fibronectin Adhesion-promoting Peptide acetate(125720-21-0 free base),Heparin Binding Peptide acetate |
Others | Others |
Fibronectin Adhesion-promoting Peptide acetate (Heparin Binding Peptide acetate)(125720-21-0 free base) 是在纤连蛋白的羧基末端肝素结合结构域中发现的肝素结合氨基酸序列之一。 | |||
T66154 |
Paroxypropione
|
Others | Others |
It is an inhibitor of the Human Apurinic/apyrimidinic Endonuclease 1 (APE1) | |||
T19528 |
Propionylcarnitine
Propionyl carnitine |
Others | Others |
Propionylcarnitine (Propionyl carnitine) 是一种被广泛使用的膳食补充剂,有青光眼和难道破裂有关。 | |||
T81034L |
TAT-NSF700 Fusion Peptide acetate
|
||
TAT-NSF700 Fusion Peptide acetate 是一种可渗透细胞膜的 N-乙基-马来酰亚胺敏感因子 (NSF) 抑制剂,是一种融合多肽,具有潜在的抗炎活性。TAT-NSF700 Fusion Peptide acetate 与细胞内细胞器相互作用,可用于研究心肌缺血和再灌注损伤。 | |||
T0188 |
Fluticasone (propionate)
丙酸氟替卡松,CCI-187881,氟替卡松丙酸酯,Fluticasone propionate |
Glucocorticoid Receptor; Virus Protease; Estrogen/progestogen Receptor; Phospholipase; Endogenous Metabolite; ADC Cytotoxin | Antibody-drug Conjugate/ADC Related; Endocrinology/Hormones; Metabolism; Microbiology/Virology |
Fluticasone propionate (CCI-187881) 是一种选择性糖皮质激素受体激动剂,是一种局部抗炎激素,亲和力KD 为 0.5 nM。具有抗病毒活性。 | |||
T50083 |
Cell-cell interaction 1
|
Others | Others |
12-oxo-N-[1-(propan-2-yl)piperidin-4-yl]-6H,7H,8H,9H,10H,12H-azepino[2,1-b]quinazoline-3-carboxamide 可用作分子结构单元,用于多种化合物的合成。 | |||
T7077 |
2,3-BIS(N-BUTYLTHIO)-1,4-NAPHTHALENEDION
|
Others | Others |
2,3-BIS(N-BUTYLTHIO)-1,4-NAPHTHALENEDION 是中间体。 | |||
T3560 |
Desmethylanethol trithione
ADT-OH |
VEGFR; Akt | Angiogenesis; Cytoskeletal Signaling; PI3K/Akt/mTOR signaling; Tyrosine Kinase/Adaptors |
Desmethylanethol trithione (ADT-OH) 是合成硫化氢的供体。它利用上调 FADD 诱导细胞凋亡,并对体内黑色素瘤的形成具有一定的抑制作用,可用于研究癌症疾病。 | |||
T65554 |
cholesterol-absorption inhibitor Intermediate 2
|
Others | Others |
cholesterol-absorption inhibitor Intermediate 2 是一种有效且具有口服活性的胆固醇吸收抑制剂,可降低血液中胆固醇含量。 | |||
T0830 |
Bithionol
硫双二氯酚,Actamer,硫氯酚 |
cAMP; Parasite | GPCR/G Protein; Microbiology/Virology |
Bithionol (Actamer) 是一种抗寄生虫药物,对若干癌细胞有抑制作用。 | |||
T13244 |
Ubiquitination-IN-1
|
Others | Others |
Ubiquitination-IN-1 是一种有效的泛素化和Cksl-Skp2蛋白互作抑制剂 (IC50=0.17 μM) 抑制剂,增加 p27 水平,可通过阻断肿瘤抑制因子的降解发挥作用。 | |||
T9978 |
Glutathione synthesis-IN-1
|
Others | Others |
Glutathione synthesis-IN-1 (DC-1)是谷胱甘肽合成抑制剂。 | |||
T9228 |
Propionylpromazine hydrochloride
盐酸丙酰丙嗪,Propiopromazine hydrochloride |
Dopamine Receptor | GPCR/G Protein; Neuroscience |
Propionylpromazine hydrochloride (Propiopromazine hydrochloride) 是多巴胺受体 D2 (DRD2) 拮抗剂,可用于研究帕金森氏病。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TQ0192 |
Senecionine
Aureine,Senecionan-11,16-dione, 12-hydroxy-,千里光宁,Senecionin |
Others | Others |
Senecionine 是一种吡咯里西啶生物碱,从Senecio vulgaris中分离得到,它对动物和人类有毒性。 | |||
T8709 |
Nandrolone phenylpropionate
Nandrolone phenpropionate,苯丙酸诺龙 |
Androgen Receptor | Endocrinology/Hormones |
Nandrolone phenylpropionate (Nandrolone phenpropionate) 是一种合成代谢类固醇,是一种 19-nortestosterone 的衍生物。它能够促进蛋白质合成,用于缓解组织分解代谢,可以用于骨质疏松症和特纳综合征的研究。 | |||
T5285 |
3-(Methylthio)propionic acid
3-Methylthiopropionate,3-甲基硫代丙酸,4-Thiapentanoic acid,3-Methylsulfanylpropionic acid |
Others; Endogenous Metabolite; Antifungal | Metabolism; Microbiology/Virology; Others |
3-(Methylthio)propionic acid (4-Thiapentanoic acid) 是methionine 的代谢物,是中间体。 | |||
T1165 |
Ethionamide
Bayer 5312,乙硫异烟胺,2-ethylthioisonicotinamide,Ethinamide |
Dehydrogenase; CAT; Antibacterial; Antibiotic | Metabolism; Microbiology/Virology; oxidation-reduction |
Ethionamide (2-ethylthioisonicotinamide) 是一种抗结核抗生素。 | |||
TN7192 |
7-Bromoquinazoline-2,4(1H,3H)-Dione
7-Bromo-2,4(1H,3H)-quinazolinedione,7-溴喹唑啉-(2,4)二酮,7-Bromo-1H-quinazoline-2,4-dione,7-bromoquinazoline-2,4-diol |
Others | Others |
7-Bromoquinazoline-2,4(1H,3H)-Dione (7-Bromo-2,4(1H,3H)-quinazolinedione) 是一种海洋来源的天然产物,发现于 Pyura sacciformis。 | |||
T1285 |
Anethole trithione
茴三硫,Anetholtrithion |
Others; AChR | Neuroscience; Others |
Anethole trithione (Anetholtrithion) 是硫杂环胆碱,是一种胆汁分泌刺激剂,可增强唾液分泌并增加 mAChR 受体,用于口干症的研究。 | |||
T5297 |
3-Indolepropionic acid
Indolepropionic acid,IPA,indole-3-propionic acid,吲哚-3-丙酸 |
Antioxidant; Reactive Oxygen Species; Endogenous Metabolite | Immunology/Inflammation; Metabolism; NF-κB; oxidation-reduction |
3-Indolepropionic acid (Indolepropionic acid) 是强效的抗氧化剂,具有研究阿尔兹海默症的潜能。 | |||
T0525 |
Flopropione
夫洛丙酮,Phloropropiophenone |
5-HT Receptor; Transferase | GPCR/G Protein; Metabolism; Neuroscience |
Flopropione (Phloropropiophenone) 是一种解痉剂,用作 5-HT1A 受体拮抗剂,也是儿茶酚-O-甲基转移酶抑制剂。 | |||
T7908 |
DL-Methionine Methylsulfonium Chloride
DL-蛋氨酸甲基氯化锍,维生素U |
Others | Others |
DL-methionine methylsulfonium chloride 是天然的蛋氨酸衍生物。它能够有效保护胃粘膜,避免其受到乙醇诱导的损伤。 | |||
TN7209 |
3-bromopyrrole-2,5-dione
ZINC13379821,3-溴-1H-吡咯-2,5-二酮,3-Bromo-1H-pyrrole-2,5-dione |
Others | Others |
3-bromopyrrole-2,5-dione (ZINC13379821) 是一种海洋来源的天然产物,存在于 Axinella brevistyla。 | |||
T4909 |
N-Acetyl-DL-methionine
N-乙酰-DL-蛋氨酸,N-乙酰-DL-甲硫氨酸 |
Others; Endogenous Metabolite | Metabolism; Others |
N-Acetyl-DL-methionine 是内源性代谢产物的一种。 | |||
T4768 |
Diethyl oxalpropionate
草酰丙酸二乙酯,HYL 2-METHYL-3-OXOSUCCINATE |
Others; Endogenous Metabolite | Metabolism; Others |
Diethyl oxalpropionate (HYL 2-METHYL-3-OXOSUCCINATE) 是一种合成 PDMMLA 的中间体。其中 PDMMLA 的衍生物可用于纳米粒子的合成和研究。 | |||
TN6730 |
Epoxyazadiradione
|
NF-κB | NF-κB |
Epoxyazadiradione 是从印楝果实中得到的柠檬苦素。它能够可逆的、非竞争性的抑制人类、约氏疟原虫、疟原虫的互变异构酶活性。它具有抗疟原虫和人类 MIF 诱导的促炎反应的潜力。 | |||
TN2064 |
Physcion 8-O-β-D-glucopyranoside
大黄素甲醚-8-O-Β-D-葡萄糖苷,Physcion 8-O-beta-D-monoglucoside |
TNF | Apoptosis |
Physcion 8-O-β-D-glucopyranoside (Physcion 8-O-beta-D-monoglucoside) 具有抗炎和抗癌活性。Physcion 8-O-β-D-glucopyranoside 可用于常见恶性肿瘤的研究。 | |||
T7437 |
3-(3-Hydroxyphenyl)propionic Acid
m-Hydroxyphenylpropionic acid,3-Hydroxyhydrocinnamic acid,3-(3-羟基苯基)丙酸 |
Others; Endogenous Metabolite | Metabolism; Others |
3-(3-Hydroxyphenyl)propionic Acid (m-Hydroxyphenylpropionic acid) 是一种黄酮类代谢产物,由人体微生物区系形成,具有舒张血管的特性。 | |||
T8064 |
Lactobionic acid
|
Others; Antibacterial | Microbiology/Virology; Others |
Lactobionic acid 是在里海酸奶中的一种仿生酸,化学上由与半乳糖键合的葡萄糖酸组成。它是具有抗氧化、抗菌和保湿特性的乳糖酸。 | |||
T14001 |
11-Beta-hydroxyandrostenedione
4-雄烯-11β-醇-3,17-二酮,NSC-17102,4-Androsten-11β-ol-3,17-dione |
Endogenous Metabolite | Metabolism |
11-Beta-hydroxyandrostenedione (NSC-17102) 是主要存在于肾上腺的类固醇,也是 11β-羟基类固醇脱氢酶同工酶抑制剂。随着 4-androstenedione 的提高,通过测量血浆中的11-Beta-hydroxyandrostenedione,能够区分高雄激素血症的肾上腺或卵巢起源。 | |||
T10939L |
L-Cystathionine
L-胱硫醚,Cystathionine,ZINC1532680,L-(+)-Cystathionine,Cystathionine, L- |
Apoptosis; Endogenous Metabolite | Apoptosis; Metabolism |
L-Cystathionine (Cystathionine, L-) 是一种与含硫氨基酸的代谢条件有关的关键非蛋白质氨基酸。L-Cystathionine 可用于有关心血管保护的研究。 | |||
TJO2742 |
DL-Methionine
蛋氨酸,methionine,DL-蛋氨酸,Acimetion,Racemethionine |
Parasite | Microbiology/Virology |
DL-Methionine (Acimetion) 存在于肉类、鱼类和奶制品中,是可用于动物的天然饲料,还可杀死马铃薯上的金线虫。它是一种含有硫的必需氨基酸,具有氧化应激防御作用。 | |||
T4844 |
L-Methionine
L(-)-Methionin,L-蛋氨酸,L-Methionin |
Endogenous Metabolite | Metabolism |
L-Methionine (L-Methionin) 是 Methionine 的 L-异构体。Methionine 是必需氨基酸,同时也是肝脏保护剂。 | |||
T19397 |
L-Methionine sulfoxide
L-蛋氨酸亚砜,H-Met(O)-OH |
Endogenous Metabolite | Metabolism |
L-Methionine sulfoxide (H-Met(O)-OH) 是一种甲硫氨酸的代谢产物,能够诱导 M1/classical 巨噬细胞极化,并调节氧化应激和嘌呤能的信号传递参数。 | |||
T0449 |
Menadione
维生素K3,Vitamin K3,甲萘醌 |
Thrombin; Endogenous Metabolite | Metabolism; Proteases/Proteasome |
Menadione (Vitamin K3) 是合成的萘醌,能够在体内转化成活性维生素 K2。 | |||
T7090 |
Jionoside A1
焦地黄苯乙醇甙A1,焦地黄苯乙醇苷A1 |
Others | Others |
Jionoside A1 分离自Radix Rehmanniae Praeparata 中,具有剂量依赖性免疫增强作用,并对 H2O2处理的 SH-SY5Y 细胞具有中等保护活性。 | |||
T1085 |
L-Glutathione reduced
谷胱甘肽,GSH,Isethion,Glutathione,γ-L-Glutamyl-L-cysteinyl-glycine,Glutathion,还原型谷胱甘肽,Tathion |
Ferroptosis; Reactive Oxygen Species; Endogenous Metabolite; Glutathione reductase | Apoptosis; Immunology/Inflammation; Metabolism; NF-κB; oxidation-reduction |
L-Glutathione reduced (Glutathione) 属于天然三肽,存在与细胞中,是一种内源性抗氧化剂,可以清除氧自由基。L-Glutathione reduced 是某些酶的辅助因子,参与蛋白质二硫键重排并减少过氧化物。 | |||
T4857 |
Pteridine-2,4(1H,3H)-dione
2,4-Dihydroxypteridine,2,4-二羟基蝶啶,Lumazine |
Others; Endogenous Metabolite | Metabolism; Others |
Pteridine-2,4(1H,3H)-dione (Lumazine) 是内源性代谢产物的一种。 | |||
T3019 |
Physcion
大黄素甲醚,Physcione,Parietin,Rheochrysidin |
Dehydrogenase; Antibacterial | Metabolism; Microbiology/Virology |
Physcion (Physcione) 是一种从中药大黄中分离的蒽醌,作为 6-磷酸葡萄糖酸脱氢酶的抑制剂,IC50和 Kd 值分别为 38.5 μM 和 26.0 μM。它具有通便、保肝、抗炎、抗菌、抗增殖、抗肿瘤作用。 | |||
TQ0226 |
Jionoside B1
|
Glucosidase | Metabolism |
Jionoside B1 是从熟地黄(Gaertn.)的根中分离出来的,抑制 α-葡萄糖苷酶。 | |||
T3411 |
Curdione
莪术二酮,(+)-Curdione |
P450 | Metabolism |
Curdione ((+)-Curdione) 是一种具有高生物活性的倍半萜类物质,从莪术中分离获得,具有抑制血小板聚集、抵抗血栓形成的作用。 | |||
T19418 |
Methionine sulfoxide
|
Endogenous Metabolite | Metabolism |
Methionine sulfoxide 是具有特性氧的甲硫氨酸的氧化产物,能够用作体内氧化应激的生物标记。 | |||
T67302 |
2,3-Pentanedione
Acetylpropionyl |
Others | Others |
2,3-Pentanedione 是一种食品添加剂, 也作为发酵产物自然存在于啤酒、葡萄酒和酸奶中,并在咖啡豆烘焙过程中释放。吸入2,3-Pentanedione 被认为是人严重呼吸道疾病(包括闭塞性细支气管炎)的原因。 | |||
T13475 |
β-Aminopropionitrile
3-氨基丙腈,3-Aminopropionitrile,BAPN |
Others; Endogenous Metabolite | Metabolism; Others |
β-Aminopropionitrile (3-Aminopropionitrile) 是赖氨酰氧化酶的特异性抑制剂。 | |||
T4447 |
S-(5'-Adenosyl)-L-methionine tosylate
S-腺苷蛋氨酸对甲苯磺酸盐,SAMe,S-(5'-Adenosyl)-L-methionine p-toluenesulfonate salt |
Others | Others |
S-(5'-Adenosyl)-L-methionine tosylate (SAMe) 是一种普遍存在的甲基供体,参与多种生物反应,包括由 DNA 和蛋白质甲基转移酶介导的反应。它可改善抑郁、与骨关节炎和纤维肌痛相关的疼痛以及肝毒性。 | |||
T5303 |
Isethionic acid sodium salt
Sodium isethionate,羟乙基磺酸钠 |
Others; Endogenous Metabolite | Metabolism; Others |
Isethionic acid sodium salt (Sodium isethionate) 是内源性代谢产物的一种。 | |||
T4919 |
Ureidopropionic acid
Carbamoyl-b-alanine,3-酰脲丙酸,3-Ureidopropionic acid |
Endogenous Metabolite | Metabolism |
Ureidopropionic acid (3-Ureidopropionic acid) 是尿嘧啶代谢的中间体。更具体地说,它是二氢尿嘧啶的分解产物,由二氢嘧啶酶产生。它通过β -脲丙酸酶进一步分解为β -丙氨酸。尿素丙酸本质上是β -丙氨酸的尿素衍生物。高水平的尿丙酸存在于β -尿丙酸酶(UP)缺乏的个体中。嘧啶代谢中的酶缺乏与抗肿瘤药物5-氟尿嘧啶的严重毒性风险有关。 | |||
T7931 |
16a,17a-Epoxy-4-Pregnen-3,20-Dione
|
Others | Others |
16a,17a-Epoxy-4-Pregnen-3,20-Dione 是一种合成孕激素,是黄体酮激素的代谢产物,它通过与黄体酮受体结合发挥作用,已被用于研究孕激素对生殖器官的影响,激素对细胞生长和发育的影响,以及激素对免疫系统的影响。 | |||
T5215 |
N-(3-Phenylpropionyl)glycine
N-(3-苯基丙酰基)甘氨酸,Phenylpropionylglycine |
Others | Others |
N-(3-Phenylpropionyl)glycine (Phenylpropionylglycine) 是一种酰基甘氨酸。酰基甘氨酸通常是脂肪酸的次要代谢物。 | |||
T5272 |
3-(3-Methoxyphenyl)propionic acid
3-(3-甲氧基苯基)丙酸,3-Methoxyhydrocinnamic acid |
Others; Endogenous Metabolite | Metabolism; Others |
3-(3-Methoxyphenyl)propionic acid (3-Methoxyhydrocinnamic acid) 是人体自然代谢的有机酸,排泄于尿液中。 | |||
TN6737 |
(25R)-Spirost-4-ene-3,12-dione
|
Others | Others |
(25R)-Spirost-4-ene-3,12-dione 是一种天然产物,抑制中性粒细胞超氧阴离子的产生和肥大细胞组胺的释放。 | |||
T8059 |
N-Acetyl-L-methionine
N-Acetylmethionine,N-乙酰-L-蛋氨酸 |
Others; Endogenous Metabolite | Metabolism; Others |
N-Acetyl-L-methionine (N-Acetylmethionine) 是人体代谢物,在营养和代谢作用上和 L-methionine 相当。其中 L-methionine 是生长发育并不能够少的氨基酸。 | |||
T5556 |
5a-Pregnane-3,20-dione
|
Endogenous Metabolite | Metabolism |
5a-Pregnane-3,20-dione 是内源性的孕酮代谢物。 | |||
T3130 |
Testosterone phenylpropionate
Testosterone hydrocinnamate,苯丙酸睾酮,Retandrol,Testosterone 17-phenylpropionate |
Others | Others |
Testosterone phenylpropionate (Testosterone 17-phenylpropionate) 是一种长效雄激素。d3-Testosterone phenylpropionate 可用作内标物。 | |||
T7927 |
β-Ionone
乙位紫罗兰酮,β-紫罗兰酮,β-lonone |
Apoptosis; Others | Apoptosis; Others |
β-Ionone (β-lonone) 是β-类胡萝卜素的端环类似物,广泛存在于水果和蔬菜中,可有效诱导胃腺癌细胞 SGC7901 凋亡,具有抗增殖、抗转移和抗肿瘤作用。 | |||
T6752 |
S-Adenosyl-L-methionine disulfate tosylate
S-腺苷蛋氨酸对甲苯磺酸硫酸盐,Ademetionine disulfate tosylate |
DNA/RNA Synthesis | Cell Cycle/Checkpoint; DNA Damage/DNA Repair |
S-Adenosyl-L-methionine disulfate tosylate (Ademetionine disulfate tosylate) 是一种主要生物甲基供体,在所有哺乳动物细胞中合成,但在肝脏中含量较高。 | |||
T3381 |
Lysionotin
岩豆素 |
Others | Others |
Lysionotin (Nevadensin) 是一种类黄酮,分离自黄花草药中。它可抑制 α-Toxin (一种成孔蛋白) 的表达,并在体内和体外针对金黄色葡萄球菌显示出显著的保护作用。它可用于研究由金黄色葡萄球菌引起的肺炎。 | |||
T5S0691 |
Shionone
紫菀酮,Shionon |
Others | Others |
Shionone (Shionon) 是一种从Aster tataricus 中分离得到的三萜类化合物,具有独特的六元四环骨架和 3-氧代-4-单甲基结构。它具有镇咳、抗炎作用。 | |||
T7285 |
Ionomycin
|
Calcium Channel | Membrane transporter/Ion channel; Metabolism |
Ionomycin 是一种钙离子载体和一种结合钙离子(Ca2+)的抗生素。它是由联合链霉菌(Streptomyces conglobatus)产生的。它在研究中用于提高细胞内钙水平(Ca2+),并作为了解 Ca2+跨生物膜运输的研究工具。Ionomycin 可促进细胞凋亡,诱导蛋白激酶 C (PKC)活化。 | |||
T7335 |
2,3-Diaminopropionic acid
L-2,3-二氨基丙酸,L-2,3-Diaminopropionic acid |
Endogenous Metabolite | Metabolism |
2,3-Diaminopropionic acid (L-2,3-Diaminopropionic acid) 是一种神经毒性氨基酸 b-oxalyl-L-a, b-diaminopropionic acid 的代谢产物。 | |||
TN7149 |
5-[(1H-indol-3-yl)methylidene]imidazolidine-2,4-dione
(4Z)-4-(1H-indol-3-ylmethylidene)-4H-imidazole-2,5-diol,(5Z)-5-(1H-indol-3-ylmethylidene)imidazolidine-2,4-dione |
Others | Others |
5-[(1H-indol-3-yl)methylidene]imidazolidine-2,4-dione ((4Z)-4-(1H-indol-3-ylmethylidene)-4H-imidazole-2,5-diol) 是一种海洋来源的天然产物,存在于Leptopsammia pruvoti。 | |||
TN6729 |
Azadiradione
AZD |
Others | Others |
Azadiradione (AZD) 是 HSF1的一种,是由印楝树中提取得到,具有一定生物活性的柠檬苦素。 | |||
T7450 |
1-Phenylpropane-1,2-dione
1-Phenyl-1,2-propanedione,Acetyl benzoyl,1-苯基-1,2-丙二酮 |
Others | Others |
1-Phenylpropane-1,2-dione (Acetyl benzoyl) 是麻黄素生物碱的生物合成前体,分离自从嫩麻黄中。 | |||
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Cat. No. | Product Name | Species | Expression System |
---|---|---|---|
TMPH-01863 |
PIEZO1 Protein, Human, Recombinant (His & Myc)
Protein FAM38A,Membrane protein induced by beta-amyloid trea... |
Human | E. coli |
PIEZO1 Protein, Human, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 33.6 kDa and the accession number is Q92508. | |||
TMPH-01891 |
KCNE2 Protein, Human, Recombinant (His)
MinK-related peptide 1,Potassium voltage-gated channel subfa... |
Human | E. coli |
KCNE2 Protein, Human, Recombinant (His) is expressed in E. coli expression system with N-10xHis tag. The predicted molecular weight is 17.3 kDa and the accession number is Q9Y6J6. | |||
TMPH-01358 |
FXYD3 Protein, Human, Recombinant (His & SUMO)
Phospholemman-like,Chloride conductance inducer protein Mat-... |
Human | E. coli |
FXYD3 Protein, Human, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 20.5 kDa and the accession number is Q14802. | |||
TMPY-03236 |
Human respiratory syncytial virus (RSV) Fusion protein/RSV-F (Strain RSS-2) Protein (His)
F Protein,HRSVgp8 |
RSV | Baculovirus Insect Cells |
Human respiratory syncytial virus (RSV) Fusion protein/RSV-F (Strain RSS-2) Protein (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 57.8 kDa and the accession number is P11209. | |||
TMPY-02215 |
Coagulation factor IX/F9 Protein, Human, Recombinant (His)
FIX,PTC,Coagulation factor 9,coagulation f... |
Human | HEK293 Cells |
Coagulation factor IX/F9 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 50 kDa and the accession number is AAB59620.1. | |||
TMPY-01193 |
Influenza A H1N1 (A/Brevig Mission/1/1918) Hemagglutinin Protein (His)
Harvey rat sarcoma viral oncogene homolog |
H1N1 | HEK293 Cells |
Influenza A H1N1 (A/Brevig Mission/1/1918) Hemagglutinin Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 37.5 kDa and the accession number is Q9WFX3. | |||
TMPY-01078 |
Human respiratory syncytial virus (RSV) (A2) Fusion glycoprotein/RSV-F Protein (His)
HRSVgp8,F Protein |
RSV | Baculovirus Insect Cells |
Human respiratory syncytial virus (RSV) (A2) Fusion glycoprotein/RSV-F Protein (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 57.4 kDa and the accession number is P03420.1. | |||
TMPY-04274 |
Influenza A H1N1 (A/Brevig Mission/1/1918) Nucleoprotein/NP Protein (His)
NP Protein |
H1N1 | Baculovirus Insect Cells |
Influenza A H1N1 (A/Brevig Mission/1/1918) Nucleoprotein/NP Protein (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 57.7 kDa and the accession number is Q5UEW0.1. | |||
TMPY-01101 |
Coagulation factor X/F10 Protein, Human, Recombinant (His)
FXA,FX,coagulation factor X,coagulation fa... |
Human | Baculovirus Insect Cells |
Coagulation factor X, also known as FX, F10, Eponym Stuart-Prower factor, and thrombokinase, is an enzyme of the coagulation cascade. It is one of the vitamin K-dependent serine proteases, and plays a crucial role in the coagulation cascade and blood clotting, as the first enzyme in the common pathway of thrombus formation. Factor X deficiency is one of the rarest of the inherited coagulation disorders. FX deficiency among the most severe of the rare coagulation defects, typically including hema... | |||
TMPY-01104 |
Coagulation factor XI/F11 Protein, Human, Recombinant (His)
coagulation factor 11,coagulation factor X... |
Human | HEK293 Cells |
Factor XI (plasma thromboplastin antecedent) is a plasma glycoprotein, and a zymogen acting as a serine protease which participates in blood coagulation as a catalyst in the conversion of factor IX to factor IXa in the presence of calcium ions. It is an unusual dimeric protease, with structural features that distinguish it from vitamin K-dependent coagulation proteases. The factor XI is synthesized in the liver as a single polypeptide chain with a molecular weight estimated between 125 ~160 kDa ... | |||
TMPY-02185 |
Coagulation factor XIII B/F13B Protein, Human, Recombinant (His)
Coagulation factor 13,coagulation factor X... |
Human | HEK293 Cells |
Coagulation factor XIII B chain, also known as Fibrin-stabilizing factor B subunit, Protein-glutamine gamma-glutamyltransferase B chain, Transglutaminase B chain and F13B, is a secreted protein which contains 1 Sushi ( CCP / SCR ) domains. Coagulation factor XIII is the last zymogen to become activated in the blood coagulation cascade. Plasma factor XIII is a heterotetramer composed of 2 A subunits and 2 B subunits. The A subunits have catalytic function, and the B subunits do not have en... | |||
TMPY-05688 |
Human respiratory syncytial virus (RSV) Fusion Protein (aa 1-525, His)
HRSVgp8,F Protein |
RSV | Baculovirus Insect Cells |
Human respiratory syncytial virus (RSV) Fusion Protein (aa 1-525, His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 57.12 kDa and the accession number is K7WLI9. | |||
TMPY-05566 |
Siglec-2/CD22 Protein, Human, Recombinant (His, Solution)
CD22 molecule,SIGLEC-2,SIGLEC2 |
Human | HEK293 Cells |
Siglec-2/CD22 Protein, Human, Recombinant (His, Solution) is expressed in HEK293 mammalian cells with His tag. The accession number is P20273-1. | |||
TMPY-01791 |
Coagulation Factor II Protein, Mouse, Recombinant (His)
Cf-2,coagulation factor II (thrombin),Cf2,FII |
Mouse | HEK293 Cells |
Coagulation Factor II Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 69.3 kDa and the accession number is P19221. | |||
TMPY-06171 |
SARS-CoV-2 Spike S1+S2 Protein (L18F & D80A & D215G & LAL242-244 deletion & R246I & K417N & E484K & N501Y & D614G & A701V, His), Biotinylated
|
SARS-CoV-2 | Baculovirus Insect Cells |
SARS-CoV-2 Spike S1+S2 Protein (L18F & D80A & D215G & LAL242-244 deletion & R246I & K417N & E484K & N501Y & D614G & A701V, His), Biotinylated is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 134 kDa and the accession number is A0A6G7K2L4. | |||
TMPY-06443 |
SARS-CoV-2 Spike S1 Protein (T19R & T95I & G142D & Y145H & E156G & 157-158 deletion & A222V & L452R & T478K & D614G & P681R, His)
|
SARS-CoV-2 | HEK293 Cells |
SARS-CoV-2 Spike S1 Protein (T19R & T95I & G142D & Y145H & E156G & 157-158 deletion & A222V & L452R & T478K & D614G & P681R, His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 76.29 kDa and the accession number is YP_009724390.1. | |||
TMPY-06082 |
SARS-CoV-2 Spike S1 Protein (HV69-70 deletion & N501Y & D614G, His)
|
SARS-CoV-2 | HEK293 Cells |
SARS-CoV-2 Spike S1 Protein (HV69-70 deletion & N501Y & D614G, His) is expressed in HEK293 mammalian cells. The predicted molecular weight is 76.2 kDa and the accession number is A0A6G7K2L4. | |||
TMPY-06129 |
SARS-CoV-2 Spike S1 Protein (L18F & D80A & D215G & LAL242-244 deletion & R246I & K417N & E484K & N501Y & D614G, His)
|
SARS-CoV-2 | HEK293 Cells |
SARS-CoV-2 Spike S1 Protein (L18F & D80A & D215G & LAL242-244 deletion & R246I & K417N & E484K & N501Y & D614G, His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 76 kDa and the accession number is A0A6G7K2L4. | |||
TMPY-00647 |
Chorionic Gonadotropin/CGA Protein, Human, Recombinant (His)
CG-α,FSH alpha,glycoprotein hormones, alpha polypeptide,FSHA... |
Human | HEK293 Cells |
Chorionic Gonadotropin/CGA Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 11.6 kDa and the accession number is P01215. | |||
TMPY-02923 |
Chorionic Gonadotropin/CGA Protein, Human, Recombinant (mFc)
HCG,GPHa,CG-ALPHA,glycoprotein hormones, alpha polypeptide,g... |
Human | HEK293 Cells |
Chorionic Gonadotropin/CGA Protein, Human, Recombinant (mFc) is expressed in HEK293 mammalian cells with mFc tag. The predicted molecular weight is 36.6 kDa and the accession number is P01215. | |||
TMPY-06840 |
Human respiratory syncytial virus (RSV) (A2) Prefusion glycoprotein F/RSV-preF Protein
HRSVgp8,F Protein |
RSV | CHO Cells |
Human respiratory syncytial virus (RSV) (A2) Prefusion glycoprotein F/RSV-preF Protein is expressed in CHO mammalian cells. The predicted molecular weight is 54.5 kDa. | |||
TMPY-05690 |
Human mastadenovirus B (HAdV-B) encapsidation protein IVa2 Protein (His)
|
HAdV-B | Baculovirus Insect Cells |
Human mastadenovirus B (HAdV-B) encapsidation protein IVa2 Protein (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 52.06 kDa and the accession number is YP_002213830.1. | |||
TMPY-06422 |
SARS-CoV-2 Spike S1 NTD Protein (T19R & T95I & G142D & 156-157 deletion & R158G, His)
|
SARS-CoV-2 | HEK293 Cells |
SARS-CoV-2 Spike S1 NTD Protein (T19R & T95I & G142D & 156-157 deletion & R158G, His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 34.10 kDa and the accession number is A0A6G7K2L4. | |||
TMPY-06392 |
SARS-CoV-2 Spike S1+S2 Protein (Q52R & A67V & 69-70 deletion & Y144 deletion & E484K & D614G & Q677H & F888L, His)
|
SARS-CoV-2 | Baculovirus Insect Cells |
SARS-CoV-2 Spike S1+S2 Protein (Q52R & A67V & 69-70 deletion & Y144 deletion & E484K & D614G & Q677H & F888L, His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 133.96 kDa and the accession number is A0A6G7K2L4. | |||
TMPY-06305 |
SARS-CoV-2 Spike S1 Protein (Q52 & A67V & 69-70 deletion & 144 deletion & E484K & D614G & Q677H, His)
|
SARS-CoV-2 | HEK293 Cells |
SARS-CoV-2 Spike S1 Protein (Q52 & A67V & 69-70 deletion & 144 deletion & E484K & D614G & Q677H, His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 76.07 kDa and the accession number is A0A6G7K2L4. | |||
TMPY-06368 |
Human respiratory syncytial virus (RSV) (A, strain Long) Fusion glycoprotein F0/RSV-F Protein (His)
F Protein,HRSVgp8 |
RSV | Baculovirus Insect Cells |
Human respiratory syncytial virus (RSV) (A, strain Long) Fusion glycoprotein F0/RSV-F Protein (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 56.92 kDa and the accession number is P12568. | |||
TMPH-03268 |
Coagulation factor XI Protein, Rat, Recombinant (His & Myc)
Coagulation factor XI,F11 |
Rat | E. coli |
Coagulation factor XI Protein, Rat, Recombinant (His & Myc) is expressed in E. coli. | |||
THMH-00001 |
CD133/PROM1 Recombinant,Human(Yeast expression,His)
|
||
TMPH-00480 |
Anionic trypsin Protein, Canine, Recombinant (His & SUMO)
Anionic trypsin,EC:3.4.21.4 |
Canine | E. coli |
Anionic trypsin Protein, Canine, Recombinant (His & SUMO) is expressed in E. coli. | |||
TMPH-02401 |
rplL Protein, Legionella pneumophila, Recombinant (His & Myc)
Large ribosomal subunit protein bL12,50S ribosomal protein L... |
Legionella pneumophila | E. coli |
Forms part of the ribosomal stalk which helps the ribosome interact with GTP-bound translation factors. Is thus essential for accurate translation. rplL Protein, Legionella pneumophila, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 20.4 kDa and the accession number is Q5ZYQ1. | |||
TMPH-01798 |
Nucleolar transcription factor 1 Protein, Human, Recombinant (Cell-Free, His & SUMO)
Nucleolar transcription factor 1,Upstream-binding f... |
Human | E. coli |
Recognizes the ribosomal RNA gene promoter and activates transcription mediated by RNA polymerase I through cooperative interactions with the transcription factor SL1/TIF-IB complex. It binds specifically to the upstream control element. Nucleolar transcription factor 1 Protein, Human, Recombinant (Cell-Free, His & SUMO) is expressed in E. coli expression system with N-10xHis-SUMO tag. The predicted molecular weight is 107.9 kDa and the accession number is P17480. | |||
TMPH-00689 |
Propionate kinase Protein, E. coli O6:H1, Recombinant (His & Myc)
tdcD,Propionate kinase |
E. coli | E. coli |
Catalyzes the conversion of propionyl phosphate and ADP to propionate and ATP. Propionate kinase Protein, E. coli O6:H1, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 50.4 kDa and the accession number is P59244. | |||
TMPH-00399 |
RPS13 Protein, Ciona intestinalis, Recombinant (His & Myc)
40S ribosomal protein S13,RPS13,Small ribosomal subunit prot... |
Ciona intestinalis | E. coli |
RPS13 Protein, Ciona intestinalis, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 23.9 kDa and the accession number is Q8I7D6. | |||
TMPH-02452 |
Measles virus (MeV) (strain Leningrad-16) Fusion glycoprotein F0 (Avi & His)
F,Fusion glycoprotein F0 |
MeV | E. coli |
Measles virus (MeV) (strain Leningrad-16) Fusion glycoprotein F0 (Avi & His) is expressed in E. coli expression system with N-10xHis and C-Avi tag. The predicted molecular weight is 61.8 kDa and the accession number is P69356. | |||
TMPH-02399 |
Pal Protein, Legionella pneumophila, Recombinant (E. coli, His)
pal,19 kDa surface antigen,Peptidoglycan-associated lipoprot... |
Legionella pneumophila | E. coli |
Part of the Tol-Pal system, which plays a role in outer membrane invagination during cell division and is important for maintaining outer membrane integrity. Very strongly associated with the peptidoglycan. | |||
TMPH-01799 |
Nucleolar transcription factor 1 Protein, Human, Recombinant (E. coli, His & SUMO)
Nucleolar transcription factor 1,Autoantigen NOR-90... |
Human | E. coli |
Recognizes the ribosomal RNA gene promoter and activates transcription mediated by RNA polymerase I through cooperative interactions with the transcription factor SL1/TIF-IB complex. It binds specifically to the upstream control element. Nucleolar transcription factor 1 Protein, Human, Recombinant (E. coli, His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 95.2 kDa and the accession number is P17480. | |||
TMPY-06085 |
SARS-CoV-2 Spike S1 Protein (HV69-70 deletion & Y453F & D614G, His)
|
SARS-CoV-2 | HEK293 Cells |
SARS-CoV-2 Spike S1 Protein (HV69-70 deletion & Y453F & D614G, His) is expressed in HEK293 mammalian cells. The predicted molecular weight is 76.2 kDa and the accession number is A0A6G7K2L4. | |||
TMPY-05355 |
Coagulation factor IX/F9 Protein, Human, Recombinant (hFc)
P19,Coagulation factor 9,HEMB,FIX,THPH8,Coagulat |
Human | HEK293 Cells |
Coagulation factor IX/F9 Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 75.5 kDa and the accession number is P00740-1. | |||
TMPY-00323 |
Hepatitis C virus (HCV-1a) NS3 protease/helicase immunodominant region Protein (aa 1356-1459, GST)
NS3 |
HCV | E. coli |
HCV NS3 displays three enzymatic activities: serine protease, NTPase, and RNA helicase. HCV NS3 serine protease, in association with NS4A, is responsible for the cleavages of NS3-NS4A, NS4A-NS4B, NS4B-NS5A, and NS5A-NS5B. HCV NS3 RNA helicase binds to RNA and unwinds dsRNA in the 3' to 5' direction, and likely RNA stable secondary structure in the template strand (By similarity). Cleaves and inhibits the host antiviral protein MAVS. NS3/NS4A complex also prevents phosphorylation of human IRF3, t... | |||
TMPY-06406 |
SARS-CoV-2 Spike S1+S2 Protein (G75V & T76I & R246N & 247, 253 deletion & L452Q & F490S & D614G & T859N, His)
|
SARS-CoV-2 | Baculovirus Insect Cells |
SARS-CoV-2 Spike S1+S2 Protein (G75V & T76I & R246N & 247, 253 deletion & L452Q & F490S & D614G & T859N, His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 134.11 kDa and the accession number is A0A6G7K2L4. | |||
TMPY-06444 |
SARS-CoV-2 Spike S1 Protein (T19R & T95I & E156G & 157-158 deletion & L452R & T478K & D614G & P681R, His)
|
SARS-CoV-2 | HEK293 Cells |
SARS-CoV-2 Spike S1 Protein (T19R & T95I & E156G & 157-158 deletion & L452R & T478K & D614G & P681R, His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 76.23 kDa and the accession number is YP_009724390.1. | |||
TMPY-06122 |
SARS-CoV-2 Spike S1 NTD Protein (L18F & D80A & D215G & LAL242-244 deletion & R246I, His)
|
SARS-CoV-2 | HEK293 Cells |
SARS-CoV-2 Spike S1 NTD Protein (L18F & D80A & D215G & LAL242-244 deletion & R246I, His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 33.9 kDa and the accession number is A0A6G7K2L4. | |||
TMPY-06267 |
SARS-CoV-2 Spike S1 Protein (157-158 deletion & T19R & G142D & E156G & L452R & T478K & D614G & P681R, His & Avi), Biotinylated
|
SARS-CoV-2 | HEK293 Cells |
SARS-CoV-2 Spike S1 Protein (157-158 deletion & T19R & G142D & E156G & L452R & T478K & D614G & P681R, His & Avi), Biotinylated is expressed in HEK293 mammalian cells with His and Avi tag. The predicted molecular weight is 78.09 kDa and the accession number is A0A6G7K2L4. | |||
TMPK-00775 |
PRNP/Prion Protein, Mouse, Recombinant (hFc)
Major prion protein,PrP,ALTPRP,PRIP,PRNP |
Mouse | HEK293 Cells |
Prion protein gene (PRNP) variants determine the susceptibility of humans, sheep and mice to prion diseases, whereas polymorphisms in the open reading frame (ORF) of bovine PRNP seem to be unrelated to the incidence of bovine spongiform encephalopathy (BSE). According to the latest reports, the genetic susceptibility of cattle to BSE is associated with polymorphisms ofthe regulatory region of the PRNP gene and the level ofits expression. | |||
TMPJ-00707 |
Coagulation factor X/F10 Protein, Mouse, Recombinant (His)
Stuart factor,Coagulation factor X,F10 |
Mouse | HEK293 Cells |
Mouse coagulation factor X / F10 a member of the peptidase S1 family. The mature F10 is composed mostly of two EGF-like domains, one Gla gamma-carboxy-glutamate domain and one peptidase S1 domain. Factor Xa is a vitamin K-dependent plasma protease that converts prothrombin to thrombin in the presence of factor Va, calcium and phospholipid during blood clotting. The two chains of F10 are formed from a single-chain precursor by the excision of two Arg residues. A single-chain precursor is initiall... | |||
TMPH-00754 |
Capsid decoration Protein, Escherichia phage lambda, Recombinant (GST)
Gene product D,Auxiliary protein D,Major capsid protein D,gp... |
Escherichia phage lambda | E. coli |
Stabilizes the expansion of the capsid head shell after genome packaging. The packaging of viral genome in the procapsid triggers a dramatic reconfiguration of the capsid shell, expanding from roughly 50nm to 60nm while the capsid thickness decreases. 415 capsid decoration protein molecules cooperatively bind the expanded capsid, thereby stabilizing the mature capsid shell. Capsid decoration Protein, Escherichia phage lambda, Recombinant (GST) is expressed in E. coli expression system with N-GST... | |||
TMPH-00484 |
Cationic trypsin Protein, Canine, Recombinant (His & SUMO)
TRP1,Serine protease 1,PRSS1,TRY1,Pretrypsinogen I,Anion... |
Canine | E. coli |
Cationic trypsin Protein, Canine, Recombinant (His & SUMO) is expressed in E. coli. | |||
TMPH-01669 |
Metallothionein-3/MT3 Protein, Human, Recombinant (His & SUMO)
Metallothionein-III,Metallothionein-3,GIFB... |
Human | E. coli |
Binds heavy metals. Contains three zinc and three copper atoms per polypeptide chain and only a negligible amount of cadmium. Inhibits survival and neurite formation of cortical neurons in vitro. | |||
TMPY-06714 |
Coagulation factor IX/F9 Protein, Cynomolgus, Recombinant (His)
coagulation factor IX |
Cynomolgus | HEK293 Cells |
Coagulation factor IX/F9 Protein, Cynomolgus, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 50.17 kDa and the accession number is A0A8J8XCV8. | |||
TMPY-06288 |
SARS-CoV-2 Spike S1+S2 Protein (157-158 deletion & T19R & G142D & E156G & L452R & T478K & D614G & P681R & D950N, His & Avi), Biotinylated
|
SARS-CoV-2 | Baculovirus Insect Cells |
SARS-CoV-2 Spike S1+S2 Protein (157-158 deletion & T19R & G142D & E156G & L452R & T478K & D614G & P681R & D950N, His & Avi), Biotinylated is expressed in Baculovirus insect cells with His and Avi tag. The predicted molecular weight is 136.01 kDa and the accession number is A0A6G7K2L4. | |||
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Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TMIH-0475 |
rac threo-Dihydro Bupropion-d9 Hydrochloride
|
||
rac threo-Dihydro Bupropion-d9 Hydrochloride 是 rac threo-Dihydro Bupropion Hydrochloride 的氘代化合物。rac threo-Dihydro Bupropion Hydrochloride 的 CAS 号为 1396889-62-5。 | |||
TMIH-0051 |
3-phenylpropionic acid-d5
|
||
3-phenylpropionic acid-d5 是 3-phenylpropionic acid 的氘代化合物。 | |||
TMIJ-0084 |
Propionyl carnitine-d3 HCl
|
||
Propionyl carnitine-d3 HCl 是 Propionyl carnitine HCl 的氘代化合物。 | |||
TMIJ-0169 |
erythro-Hydro Bupropion-d9 HCl(enantiomer)
|
||
erythro-Hydro Bupropion-d9 HCl(enantiomer) 是 erythro-Hydro Bupropion HCl 的氘代化合物。 | |||
TMIJ-0208 |
Beclomethasone Dipropionate-d6
|
||
Beclomethasone Dipropionate-d6 是 Beclomethasone Dipropionate 的氘代化合物。Beclomethasone Dipropionate 的 CAS 号为 5534-09-8。Betamethasone dipropionate是具有口服活性的糖皮质激素,具有抗炎和免疫抑制作用。它是Betamethasone 的前体药物,Betamethasone 是 LPS 诱导的炎症及 MMP 释放的抑制剂。 | |||
TMID-0142 |
4-Androsten-11β-ol-3,17-dione-d7
|
||
4-Androsten-11β-ol-3,17-dione-d7 是 4-Androsten-11β-ol-3,17-dione 的氘代化合物。4-Androsten-11β-ol-3,17-dione 的 CAS 号为 382-44-5。11-Beta-hydroxyandrostenedione 是主要存在于肾上腺的类固醇,也是 11β-羟基类固醇脱氢酶同工酶抑制剂。随着 4-androstenedione 的提高,通过测量血浆中的11-Beta-hydroxyandrostenedione,能够区分高雄激素血症的肾上腺或卵巢起源。 | |||
TMIJ-0052 |
Propionicacid-d5
|
||
Propionicacid-d5 是 Propionicacid 的氘代化合物。Propionicacid 的 CAS 号为 79-09-4。Propionic acid 被广泛用作食品中的抗真菌剂。它以低水平天然存在于乳制品中,并与其他短链脂肪酸 (SCFA) 一起普遍存在于人类和其他哺乳动物的胃肠道中,作为微生物消化碳水化合物的最终产物。在动物体内有显着的生理活性。 | |||
TMIJ-0498 |
Fluticasone Propionate-d5
|
||
Fluticasone Propionate-d5 是 Fluticasone Propionate 的氘代化合物。Fluticasone Propionate 的 CAS 号为 80474-14-2。Fluticasone propionate 是一种选择性糖皮质激素受体激动剂,是一种局部抗炎激素,绝对亲和力KD为 0.5 nM。具有抗病毒活性。 | |||
TMIJ-0456 |
Malathion-d7
|
||
Malathion-d7 是 Malathion 的氘代化合物。Malathion 的 CAS 号为 121-75-5。Malathion 是一种杀虫剂,是一种有机磷酸酯的副交感神经药物,不可逆地与胆碱酯酶结合,具有相对较低的人体毒性。 | |||
T71893 |
Clobetasol Propionate-d5
|
||
Clobetasol propionate-d5 is intended for use as an internal standard for the quantification of clobetasol propionate by GC- or LC-MS. Clobetasol propionate is a corticosteroid. It binds to glucocorticoid receptors in a cell-free assay and inhibits proliferation of primary human skin fibroblasts when used at a concentration of 5 µg/ml. Topical administration of clobetasol propionate reduces croton oil-induced ear edema in mice. Formulations containing clobetasol propionate have been used in the t... | |||
TMIJ-0054 |
Propionic-2,2-d2 acid
|
||
Propionic-2,2-d2 acid 是 Propionic acid 的氘代化合物。Propionic acid 的 CAS 号为 79-09-4。Propionic acid 被广泛用作食品中的抗真菌剂。它以低水平天然存在于乳制品中,并与其他短链脂肪酸 (SCFA) 一起普遍存在于人类和其他哺乳动物的胃肠道中,作为微生物消化碳水化合物的最终产物。在动物体内有显着的生理活性。 | |||
TMID-0148 |
Nandrolone 17-propionate-d3
|
||
Nandrolone 17-propionate-d3 是 Nandrolone 17-propionate 的氘代化合物。Nandrolone 17-propionate 的 CAS 号为 7207-92-3。Nandrolone propionate 是合成代谢类固醇,主要由雄激素和保氮剂组成,具有作用时间相对较长的特点。 | |||
TMIH-0040 |
3-(4-Hydroxyphenyl)propionic acid-d4
HPPA-d4 |
||
3-(4-Hydroxyphenyl)propionic acid-d4 是 3-(4-Hydroxyphenyl)propionic acid 的氘代化合物。3-(4-Hydroxyphenyl)propionic acid 的 CAS 号为 501-97-3。Desaminotyrosine 是一种与微生物相关的代谢物,通过增强 I 型干扰素信号传导来预防流感。 | |||
TMIH-0330 |
Mesotrione-d3
|
||
Mesotrione-d3 是 Mesotrione 的氘代化合物。Mesotrione 的 CAS 号为 104206-82-8。Mesotrione 是一种苯甲酰环己二酮类除草剂,是一种竞争性羟基苯基丙酮酸双加氧酶酶抑制剂。它对玉米作物具有选择性,它在易感作物中代谢速度快,耐受性较高。 | |||
TMIH-0562 |
Testosterone propionate-d3
|
||
Testosterone propionate-d3 是 Testosterone propionate 的氘代化合物。 | |||
TMIH-0129 |
Bupropion Morpholinol-d8
|
||
Bupropion Morpholinol-d8 是 Bupropion Morpholinol 的氘代化合物。 | |||
TMIH-0089 |
Androstenedione-d7
|
||
Androstenedione-d7 是 Androstenedione 的氘代化合物。Androstenedione 的 CAS 号为 560-62-3。9-hydroxy-4-androstene-3,17-dione 是一种类固醇激素,具有抗肿瘤活性,可以抑制多种癌症细胞的生长,包括乳腺癌、前列腺癌和肺癌细胞。 | |||
TMIH-0367 |
Nandrolone propionat-d3
|
||
Nandrolone propionat-d3 是 Nandrolone propionat 的氘代化合物。 | |||
TMIJ-0165 |
Glutathione-(glyucine-13C2-15N) Trifluoroacetate
|
||
Glutathione-(glyucine-13C2-15N) Trifluoroacetate 是 Glutathione Trifluoroacetate 的 13C 和 15 N 的标记化合物。 | |||
TMIJ-0098 |
threo-Hydrobupropion-d9 HCl(enantiomer)
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threo-Hydrobupropion-d9 HCl(enantiomer) 是 threo-Hydrobupropion HCl 的氘代化合物。 | |||
TMIJ-0451 |
Malathion-d10
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Malathion-d10 是 Malathion 的氘代化合物。Malathion 的 CAS 号为 121-75-5。Malathion 是一种杀虫剂,是一种有机磷酸酯的副交感神经药物,不可逆地与胆碱酯酶结合,具有相对较低的人体毒性。 | |||
T12442 |
Phenindione D5
Rectadione D5,苯茚二酮 D5 |
Others | Others |
Phenindione D5 is deuterium labeled Phenindione, which functions as a Vitamin K antagonist. | |||
TMIJ-0053 |
2-Methylpropionic-d7 acid
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2-Methylpropionic-d7 acid 是 2-Methylpropionic acid 的氘代化合物。2-Methylpropionic acid 的 CAS 号为 79-31-2。Isobutyric acid 是一种羧酸或短链脂肪酸,具有特征性的汗味。通过微生物(肠道)代谢产生少量异丁酸。在某些食物或发酵饮料中也可能发现少量。 | |||
TMIJ-0204 |
Betamethasone-d10 Dipropionate
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Betamethasone-d10 Dipropionate 是 Betamethasone Dipropionate 的氘代化合物。Betamethasone Dipropionate 的 CAS 号为 5593-20-4。Betamethasone dipropionate 是糖皮质激素类固醇,具有免疫抑制、抗炎作用。 | |||
TMIJ-0209 |
Beclomethasone-17-Monopropionate-d3
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Beclomethasone-17-Monopropionate-d3 是 Beclomethasone-17-Monopropionate 的氘代化合物。Beclomethasone-17-Monopropionate 的 CAS 号为 5534-18-9。 | |||
TMIJ-0481 |
Fenitrothion-d6 (O,O-dimethyl-d6)
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Fenitrothion-d6 (O,O-dimethyl-d6) 是 Fenitrothion 的氘代化合物。Fenitrothion 的 CAS 号为 122-14-5。 | |||
T71303 |
Flufenamic Acid-d4
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Flufenamic acid-d4 is intended for use as an internal standard for the quantification of flufenamic acid by GC- or LC-MS. Flufenamic acid is a non-steroidal anti-inflammatory drug (NSAID) and COX inhibitor (IC50s = 3 and 9.3 µM for human COX-1 and COX-2, respectively). Flufenamic acid inhibits TNF-α-induced increases in COX-2 levels and NF-κB activation in HT-29 colon cancer cells in a concentration-dependent manner. It inhibits calcium influx induced by fMLP or A23187 in human polymorphonuclear... |