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Targets Recommended: Methionine Adenosyltransferase (MAT) Gap Junction Protein DNA Alkylation Immunology/Inflammation related Anion Exchanger Glutathione Peroxidase Anti-infection Antifection Glutathione reductase advanced glycation end products Platelet aggregation Others

721

抑制剂 & 化合物

160

天然产物

30

化合物库

25

TargetMol 试剂盒

160

重组蛋白

27

同位素标记化合物

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Cat. No. Product Name
L2300 离子通道库

931 compounds
931 种与离子通道相关的生物活性小分子化合物的特有集合,用于离子通道相关的疾病和药物研究,可用于高通量筛选和高内涵筛选;
L7110 抗高血压化合物库

678 compounds
678 种高血压相关的小分子,用于高通量和高内涵筛选;
L6750 活血化瘀中药单体库

580 compounds
580种来源于常见活血化瘀中药的单体化合物,是药物开发、药理研究等领域的有效工具。
L3500 组蛋白修饰化合物库

469 compounds
469 个组蛋白修饰相关的小分子化合物的特有集合,用于高通量、高内涵筛选;
L6730 抗病毒中药单体化合物库

268 compounds
268 种具有抗病毒活性的中药单体集合,是药物开发、药理研究的有效工具;
L7700 神经再生化合物库

524 compounds
524 种神经再生相关化合物的独特集合,可用于高通量筛选和高内涵筛选;
L6740 抗结直肠癌中药单体化合物库

382 compounds
382 种抗结直肠癌相关的中药单体集合,是药物开发、药理研究的有效工具;
L7500 凝血与抗凝化合物库

144 compounds
144 个化合物的独特集合,可用于高通量筛选和高内涵筛选;
L6810 中药单体化合物库

2755 compounds
2755 种中药来源的单体化合物,是药物开发、药理研究等领域的有力工具;
L4700 免疫/炎症分子化合物库

4720 compounds
4720 种具有抗炎症活性的化合物的特有集合,可用于高通量筛选和高内涵筛选;
L7810 高溶解性多官能团片段化合物库

1159 compounds
高溶解性多官能团片段库包含1159 种片段分子
L2140 癌细胞分化化合物库

406 compounds
406 个诱导肿瘤细胞分化化合物的独特集合,可用于高通量筛选和高内涵筛选;
L8000 干细胞分化化合物库

1197 compounds
1197 种干细胞分化信号通路相关的生物活性小分子化合物的特有集合,可用于高通量、高内涵筛选;
L2630 神经元分化化合物库

672 compounds
672 种与神经元分化相关的化合物,可以用于神经系统疾病药物研发
L1800 抗感染化合物库

2938 compounds
2938 种具有抗感染活性的化合物的特有集合,包括抗细菌、抗真菌、抗巨细胞病毒、抗HIV、抗SARS、抗流感等活性;
L6710 中药抗炎分子库

1246 compounds
1246 种具有抗炎活性或靶向炎症相关靶点的中药单体集合,是药物开发、药理研究的有效工具;
L2900 氧化还原化合物库

1264 compounds
1264 个活性化合物,已经验证具有一定的抗氧化活性,包括 ROS 清除剂、iNOS、eNOS、及抗氧化的天然产物,是研究疾病机理以及药物研究的优良载体
L8600 泛素化化合物库

210 compounds
210 种泛素化相关的小分子,用于高通量和高内涵筛选;
L6220 蒙药化合物库

950 compounds
950 种蒙药来源的天然产物分子集合,可以用于高通量和高内涵筛选;
L1380 转录因子库

695 compounds
695 种转录因子靶向、结构新颖的化合物;
L6200 瑶药化合物库

221 compounds
221 种瑶药来源的天然产物分子集合,可以用于高通量和高内涵筛选;
L6720 抗COVID-19中药单体库

1147 compounds
根据抗新冠肺炎疫情过程中应用于临床治疗的中药方剂,收集了1147 种相关中药来源的单体化合物,可用于高通量和高内涵筛选,是抗新冠病毒药物研发的良好工具;
L8300 染色质修饰分子库

250 compounds
250 种染色质化学修饰相关的生物活性小分子化合物的特有集合,用于高通量、高内涵筛选;
L3510 甲基化化合物库

128 compounds
128 种甲基化相关的化合物,可以用于高通量和高内涵筛选;
L2800 5-羟色胺分子库

268 compounds
268 种生物活性小分子化合物,用于高通量、高内涵筛选;
L7200 钙通道分子库

140 compounds
140 种钙通道相关化合物的独特集合,可用于高通量筛选和高内涵筛选;
L7300 钾通道分子库

152 compounds
152 种钾通道相关化合物的独特集合,可用于高通量筛选和高内涵筛选;
L7400 钠通道分子库

118 compounds
118 种钠通道相关化合物的独特集合,可用于高通量筛选和高内涵筛选;
L2610 神经递质受体化合物库

1513 compounds
1513 种与神经递质受体相关的化合物,用于高通量、高内涵筛选;
L9600 多肽分子库

791 compounds
791 种多肽类分子,可用于多肽药物开发及信号转导通路和作用机制研究;

化合物库

离子通道库
Cat.No: L2300
Compounds: 931
抗高血压化合物库
Cat.No: L7110
Compounds: 678
活血化瘀中药单体库
Cat.No: L6750
Compounds: 580
组蛋白修饰化合物库
Cat.No: L3500
Compounds: 469
抗病毒中药单体化合物库
Cat.No: L6730
Compounds: 268
神经再生化合物库
Cat.No: L7700
Compounds: 524
抗结直肠癌中药单体化合物库
Cat.No: L6740
Compounds: 382
凝血与抗凝化合物库
Cat.No: L7500
Compounds: 144
中药单体化合物库
Cat.No: L6810
Compounds: 2755
免疫/炎症分子化合物库
Cat.No: L4700
Compounds: 4720
高溶解性多官能团片段化合物库
Cat.No: L7810
Compounds: 1159
癌细胞分化化合物库
Cat.No: L2140
Compounds: 406
干细胞分化化合物库
Cat.No: L8000
Compounds: 1197
神经元分化化合物库
Cat.No: L2630
Compounds: 672
抗感染化合物库
Cat.No: L1800
Compounds: 2938
中药抗炎分子库
Cat.No: L6710
Compounds: 1246
氧化还原化合物库
Cat.No: L2900
Compounds: 1264
泛素化化合物库
Cat.No: L8600
Compounds: 210
蒙药化合物库
Cat.No: L6220
Compounds: 950
转录因子库
Cat.No: L1380
Compounds: 695
瑶药化合物库
Cat.No: L6200
Compounds: 221
抗COVID-19中药单体库
Cat.No: L6720
Compounds: 1147
染色质修饰分子库
Cat.No: L8300
Compounds: 250
甲基化化合物库
Cat.No: L3510
Compounds: 128
5-羟色胺分子库
Cat.No: L2800
Compounds: 268
钙通道分子库
Cat.No: L7200
Compounds: 140
钾通道分子库
Cat.No: L7300
Compounds: 152
钠通道分子库
Cat.No: L7400
Compounds: 118
神经递质受体化合物库
Cat.No: L2610
Compounds: 1513
多肽分子库
Cat.No: L9600
Compounds: 791
Cat. No. Product Name Form Specificity Of Inhibition
C0051 Penicillin-Streptomycin Solution (100×), Sterile

青霉素-链霉素双抗溶液(100×),灭菌

Solut<em>ion</em> in bottle
C0050 BCA Protein Quantification Kit

BCA蛋白浓度测定试剂盒

Solut<em>ion</em> in bottle
C0052 Penicillin-Streptomycin-Amphotericin B Solution (100×), Sterile

青霉素-链霉素-两性霉素B三抗溶液(100×),灭菌

Solut<em>ion</em> in bottle
C0065 Human CD3+ T Cell Isolation Kit (negative selection)

人 CD3+ T 细胞分选试剂盒 (阴选)

Suspens<em>ion</em> in bottle
C0118 HA Tag Immunoprecipitation Kit

HA Tag 免疫沉淀试剂盒

Suspens<em>ion</em> in bottle
C0105 Protein A Immunoprecipitation Kit

Protein A 免疫沉淀试剂盒

Suspens<em>ion</em> in bottle
C0084 Magrose Beads NH2 (10-30 μm, Ultra-suspension)

琼脂糖氨基磁珠 (10-30 μm)

Suspens<em>ion</em> in bottle
C0111 Magrose Beads NTA-Nickel (Ultra-suspension)

His-tag 蛋白纯化磁珠 NTA-Ni

Suspens<em>ion</em> in bottle
C0117 Protein L Immunoprecipitation Kit

Protein L 免疫沉淀试剂盒

Suspens<em>ion</em> in bottle
C0120 Flag Tag Immunoprecipitation Kit

Flag Tag 免疫沉淀试剂盒

Suspens<em>ion</em> in bottle
C0086 Magrose Beads COOH (10-30 μm, Ultra-suspension)

琼脂糖羧基磁珠 (10-30 μm)

Suspens<em>ion</em> in bottle
C0104 Protein A/G Immunoprecipitation Kit

Protein A/G 免疫沉淀试剂盒

Suspens<em>ion</em> in bottle
C0119 MYC Tag Immunoprecipitation Kit

MYC Tag 免疫沉淀试剂盒

Suspens<em>ion</em> in bottle
C0116 Protein G Immunoprecipitation Kit

Protein G 免疫沉淀试剂盒

Suspens<em>ion</em> in bottle
C0068 Mouse CD8+ Cell Isolation Kit (positive selection)

小鼠 CD8+ 细胞分选试剂盒 (阳选)

Suspens<em>ion</em> in bottle
C0062 Mouse CD4+ T Cell Isolation Kit (negative selection)

小鼠 CD4+ T细胞分选试剂盒 (阴选)

Suspens<em>ion</em> in bottle
C0063 Mouse CD8+ T Cell Isolation Kit (negative selection)

小鼠 CD8+ T细胞分选试剂盒 (阴选)

Suspens<em>ion</em> in bottle
C0064 Mouse Neutrophil Cell Isolation Kit (negative selection)

小鼠中性粒细胞分选试剂盒 (阴选)

Suspens<em>ion</em> in bottle
C0121 GST Tag Immunoprecipitation Kit

GST Tag 免疫沉淀试剂盒

Suspens<em>ion</em> in bottle
C0095 Magrose Beads Streptavidin (Ultra-suspension)

琼脂糖链霉亲和素磁珠

Suspens<em>ion</em> in bottle
C0079 Magrose Beads OH (10-30 μm, Ultra-suspension)

琼脂糖羟基磁珠 (10-30 μm)

Suspens<em>ion</em> in bottle
C0067 Mouse CD4+ Cell Isolation Kit (positive selection)

小鼠 CD4+ 细胞分选试剂盒 (阳选)

Suspens<em>ion</em> in bottle
C0066 Human CD34+ Cell Enrichment Kit (positive selection)

人 CD34+ 细胞富集试剂盒 (阴选)

Suspens<em>ion</em> in bottle
C0122 GFP Tag Immunoprecipitation Kit

GFP Tag 免疫沉淀试剂盒

Suspens<em>ion</em> in bottle
C0061 Mouse CD3+ T Cell Isolation Kit (negative selection)

小鼠 CD3+ T细胞分选试剂盒 (阴选)

Suspens<em>ion</em> in bottle

TargetMol 试剂盒

青霉素-链霉素双抗溶液(100×),灭菌
Cat.No: C0051
BCA蛋白浓度测定试剂盒
Cat.No: C0050
青霉素-链霉素-两性霉素B三抗溶液(100×),灭菌
Cat.No: C0052
人 CD3+ T 细胞分选试剂盒 (阴选)
Cat.No: C0065
HA Tag 免疫沉淀试剂盒
Cat.No: C0118
Protein A 免疫沉淀试剂盒
Cat.No: C0105
琼脂糖氨基磁珠 (10-30 μm)
Cat.No: C0084
His-tag 蛋白纯化磁珠 NTA-Ni
Cat.No: C0111
Protein L 免疫沉淀试剂盒
Cat.No: C0117
Flag Tag 免疫沉淀试剂盒
Cat.No: C0120
琼脂糖羧基磁珠 (10-30 μm)
Cat.No: C0086
Protein A/G 免疫沉淀试剂盒
Cat.No: C0104
MYC Tag 免疫沉淀试剂盒
Cat.No: C0119
Protein G 免疫沉淀试剂盒
Cat.No: C0116
小鼠 CD8+ 细胞分选试剂盒 (阳选)
Cat.No: C0068
小鼠 CD4+ T细胞分选试剂盒 (阴选)
Cat.No: C0062
小鼠 CD8+ T细胞分选试剂盒 (阴选)
Cat.No: C0063
小鼠中性粒细胞分选试剂盒 (阴选)
Cat.No: C0064
GST Tag 免疫沉淀试剂盒
Cat.No: C0121
琼脂糖链霉亲和素磁珠
Cat.No: C0095
琼脂糖羟基磁珠 (10-30 μm)
Cat.No: C0079
小鼠 CD4+ 细胞分选试剂盒 (阳选)
Cat.No: C0067
人 CD34+ 细胞富集试剂盒 (阴选)
Cat.No: C0066
GFP Tag 免疫沉淀试剂盒
Cat.No: C0122
小鼠 CD3+ T细胞分选试剂盒 (阴选)
Cat.No: C0061
Cat. No. Product Name Target Signaling Pathways
T32809 L-Lactate ion

L-Lactate,Lactate ion, L-

Others Others
L-Lactate ion is the conjugate base of lactic acid.
T11927 M2 ion channel blocker

Others Others
M2 ion channel blocker ,Antiviral agent, is capable of inhibiting and blocking the activity of M2 ion channel.
T25026 Albitiazolium

Albitiazolium ion

Others Others
Albitiazolium is an antimlarial agent.
T32592 Lauralkonium

Lauralkonium ion,Lauralkonium cation

Others Others
Lauralkonium is a bioactive chemical.
T84763 Ulefnersen

ION-363

Others Others
Ulefnersen是用于肌萎缩侧索硬化(ALS)研究的RNA结合蛋白fused-in sarcoma(FUS)合成抑制剂。
T25640 Laurolinium

Laurolinium ion,Laurolinium cation

Others Others
Laurolinium is an antimicrobial.
T25636 Laudexium

Laudexium ion,Laudexium cation

Others Others
Laudexium is a neuromuscular blocking drug or skeletal muscle relaxant in the category of non-depolarizing neuromuscular-blocking drugs. It is used adjunctively in surgical anesthesia to facilitate endotracheal intubation and to provide skeletal muscle re
T34817 Tetrabutylphosphonium cation

Tetra-n-butylphosphonium,J279H,Tetrabutylphosphonium ion,Tetrabutylphosphonium,Phosphonium, tetrabutyl-

Others Others
Tetrabutylphosphonium cation is a light orange solid and is the salt of the liphilic tetrabutylammonium cation and linear tribromide anion.
T8552 PSEM 89S TFA

AChR Neuroscience
PSEM 89S TFA 是一种脑渗透性和选择性离子通道激动剂,分别对 Q79G 和 L141F 具有正交选择性。
T12421 PF-04885614

Sodium Channel Membrane transporter/Ion channel
PF-04885614是一种有效的NaV1.8抑制剂。PF-04885614有用于神经系统疾病和神经发育疾病研究的潜力。
T16347 NS3623

Potassium Channel Membrane transporter/Ion channel
NS3623 是 hERG1 (KV11.1)钾通道激活剂,激活IKr 和Ito 电流,具有抗心律失常作用。NS3623也是 hERG1 通道抑制剂。
T1814 ICILIN

AG-3-5

TRP/TRPV Channel Membrane transporter/Ion channel
ICILIN (AG-3-5) 是一种有效的的瞬时受体电位 M8 (TRPM8) 离子通道激动剂。 Icilin 激活 EGTA 中的 TRPM8,该激活作用具有剂量依赖性, EC50=1.4 μM。Icilin 通过调节 T 细胞反应减轻自身免疫性神经炎症。
T3171 GSK137647A

GSK 137647

GPR Endocrinology/Hormones; GPCR/G Protein
GSK137647A (GSK 137647) 是一种选择性FFA4激动剂,作用于人类和大小鼠FFA4的pEC50分别为6.3、6.1和6.2。
T10466 BAY-1797

P2X Receptor Membrane transporter/Ion channel; Neuroscience
BAY-1797 是具有口服活性的选择性P2X4高效拮抗剂,对人 P2X4 的IC50为 211 nM,具有抗伤害和抗炎作用。
T2298 ML204

TRP/TRPV Channel Membrane transporter/Ion channel
ML204 是有效的TRPC4/TRPC5通道选择性抑制剂,相比于 TRPC6 ,对TRPC4/TRPC5通道的选择性高出 19 倍,不影响其他的 TRP 通道和电压门控的钠、钾或 Ca2+通道。
T9627 PHD-1-IN-1

HIF/HIF Prolyl-Hydroxylase Chromatin/Epigenetic; Metabolism
PHD-1-IN-1 是口服有效的缺氧诱导因子脯氨酰羟化酶结构域 1抑制剂,IC50为 0.034 μM。它与活性位 Fe2+具有独特的单齿结合相互作用,并诱导形成一个 “Arg367-out” 口袋。
T4585 EGTA

Ethylenebis(oxyethylenenitrilo)tetraacet,乙二醇双(2-氨基乙基醚)四乙酸

Others Others
Ethylenebis(oxyethylenenitrilo)tetraacet 是一种特殊的钙离子螯合剂,能够显著抑制炎性巨噬细胞的底物粘附能力。EGTA (Ethylenebis(oxyethylenenitrilo)tetraacet) 在生理 pH 值(7.4) 下,Kd 为 60.5 nM,对 Ca2+比对 Mg2+有很高的特异性。
T70310 INCB-39110

Others Others
INCB-39110 is a JAK1 inhibitor.
T68783 Stercuronium

Others Others
Stercuronium is an aminosteroid neuromuscular blocking agent which was never marketed. It acts as a competitive antagonist of the nicotinic acetylcholine receptor, and is also reported to be an acetylcholinesterase inhibitor.
T68735 Ciclotropium (free base)

Others Others
Ciclotropium (free base) is quaternary ammonium compound with anticholinergic and parasympatholytic activity. Oral Cyclotropium bromide inhibited fasting and meal-stimulated colonic motility significantly without causing adverse side effects. After cyclotropium bromide, there was a significant correlation between antral contraction amplitude and gastric emptying.
T68502 Dibrospidium Free Base

Others Others
Dibrospidium Free Base is a dispirotripiperazine derivative and alkylating agent with potential antineoplastic and anti-inflammatory activities. The duration of DNA synthesis inhibition in tumor cells was found to correlate with spirobromine antitumor activity. Spirobromin is superior to prospidin by the power of the anti-inflammatory effect. Spyrobromin can diminish the latent period of the development of tumours in the experimental rats at intraperitoneal administration. At intragastric admini...
T2096 Framycetin sulfate

Neomycin Sulphate B,硫酸新霉素B,Framycetin sulphate

Antibacterial; Antibiotic Microbiology/Virology
Framycetin sulfate (Neomycin Sulphate B) 是一种氨基糖苷类抗生素,是 RNase P 裂解活性抑制剂,Ki 为 35 μM。它抑制锤头状核酶,Ki 值为 13.5 μM,可用于肝性脑病和肠致病性大肠杆菌感染的研究。
T40101 (±)-1,2-Diolein

1,2-Dioleoyl-rac-glycerol,甘油1,2-二油酸酯

PKC Chromatin/Epigenetic; Cytoskeletal Signaling
(±)-1,2-Diolein (1,2-Dioleoyl-rac-glycerol) 是一种PKC 激活剂,可以增加肌小管 Ca2+内流。
T40857 Calcium ionophore II

Calcium ionophore II,N,N,N′,N′-Tetracyclohexyl-3-oxapentanediamide

Others Others
Calcium ionophore II (N,N,N′,N′-Tetracyclohexyl-3-oxapentanediamide) 是一种亲脂性离子载体,可用于制备钙离子选择性电极。
T77728 Tubulin polymerization-IN-55

Microtubule Associated Cytoskeletal Signaling
Tubulin polymerization-IN-55 是一种高效的 Tubulin Polymerization 抑制剂,具有潜在的抗血管生成和抗肿瘤活性,对 A549、K562、HepG2、MDA-MB-231 和 HFL-1 显示出抗增殖作用。
T15233 Endovion

NS3728

Chloride channel Membrane transporter/Ion channel
Endovion (NS3728) 是阴离子通道抑制剂 和 Anoctamin-1 (ANO 1) 通道抑制剂,也是特异性的 VRAC/VSOAC 阻断剂。
T1561 Clobetasol propionate

Dermovate,Clobetasol 17-propionate,CGP9555,Temovate,丙酸氯倍他索,CCl 4725

Glucocorticoid Receptor; P450 Endocrinology/Hormones; Metabolism
Clobetasol propionate (CGP9555) 是CYP3A5的选择性抑制剂(IC50:0.206 μM),而对 CYP3A4 或其他主要 CYP 无抑制作用。它是皮质类固醇,对于牛皮癣和其他皮肤病具有潜在的研究价值。
T1234 5,5-Dimethyloxazolidine-2,4-dione

Dimethadion,Dimethadione,二甲双酮,Dimethyloxazolidinedione

Calcium Channel Membrane transporter/Ion channel; Metabolism
5,5-Dimethyloxazolidine-2,4-dione (Dimethadione) 是抗惊厥药,是 TRIMETHADIONE 的活性代谢物。
T6240 Palbociclib Isethionate

Palbociclib (PD0332991) Isethionate,帕博西尼羟乙基磺酸盐,PD 0332991 isethionate,帕布昔利布羟乙基磺酸盐

CDK Cell Cycle/Checkpoint
Palbociclib Isethionate (PD 0332991 isethionate) 是一种高选择性的CDK4/6抑制剂,IC50为11 nM 和16 nM。它对一组 36 种额外的蛋白激酶没有抑制作用。
T9044 SORT-PGRN interaction inhibitor 1

Neurotensin Receptor GPCR/G Protein
SORT-PGRN interaction inhibitor 1 是一种 sortilin-progranulin 相互作用抑制剂,IC50为 2 μM。
T9656 AP-1/NF-κB activation inhibitor 1

NF-κB; DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair; NF-κB
AP-1/NF-κB activation inhibitor 1 是一种有效的 AP-1和 NF-κB 介导的转录激活抑制剂(IC50=1 μM),不阻断 β-actin 启动子驱动的基础转录。AP-1/NF-κB activation inhibitor 1 对受刺激细胞中 IL-2和 IL-8的产生水平有相似的抑制作用。
T40863 Bisdionin C

Antibacterial Microbiology/Virology
Bisdionin C 是一种有效的 GH18 chitinase 抑制剂,对 A. fumigatus ChiB1 的 IC50 为 0.2 μM。 Bisdionin C 抑制人巨噬细胞壳三糖苷酶 (HCHT, IC50 = 8.3 μM) 和酸性哺乳动物几丁质酶 (AMCase, IC50 = 3.4 μM)。
T1127 Beclometasone dipropionate

Beclovent,Beclomethasone dipropionate,二丙酸倍氯米松,丙酸倍氯米松,Beconase,Vancenase

Glucocorticoid Receptor Endocrinology/Hormones
Beclometasone dipropionate (Vancenase) 是具有口服活性的糖皮质激素,具有抗炎和免疫抑制作用。它是Betamethasone 的前体药物,Betamethasone 是 LPS 诱导的炎症及 MMP 释放的抑制剂。
T3189 B7/CD28 interaction inhibitor 1

CTLA-4 inhibitor

Others Others
B7/CD28 interaction inhibitor 1 (CTLA-4 inhibitor) 是B7.1-CD28相互作用抑制剂(IC50:50 nM)。
T34383L 2H-Naphth[2′,1′:4,5]indeno[1,2-d][1,3]dioxole, pregn-4-ene-3,20-dione deriv

Others Others
2H-Naphth[2′,1′:4,5]indeno[1,2-d][1,3]dioxole, pregn-4-ene-3,20-dione deriv在Sprague Dawley大鼠上进行测试时显示出高局部抗炎效力和高肺选择性。
T0283 Trimethadione

三甲双酮,3,5,5,-Trimethyloxazolidine-2,4-dione

Calcium Channel Membrane transporter/Ion channel; Metabolism
Trimethadione (3,5,5,-Trimethyloxazolidine-2,4-dione) 是恶唑烷二酮类抗惊厥剂,也是一种 T 型钙通道阻滞剂,具有抗痛觉过敏作用,可用于研究失神发作。
T1559 Betamethasone dipropionate

Diprolene AF,SCH 11460,二丙酸倍他米松,Betamethasone 17,21-dipropionate,Diprolene,倍他米松二丙酸酯,Diprosone

Glucocorticoid Receptor Endocrinology/Hormones
Betamethasone dipropionate (SCH 11460) 是糖皮质激素类固醇,具有免疫抑制、抗炎作用。
TP1153L Fibronectin Adhesion-promoting Peptide acetate

Fibronectin Adhesion-promoting Peptide acetate(125720-21-0 free base),Heparin Binding Peptide acetate

Others Others
Fibronectin Adhesion-promoting Peptide acetate (Heparin Binding Peptide acetate)(125720-21-0 free base) 是在纤连蛋白的羧基末端肝素结合结构域中发现的肝素结合氨基酸序列之一。
T66154 Paroxypropione

Others Others
It is an inhibitor of the Human Apurinic/apyrimidinic Endonuclease 1 (APE1)
T19528 Propionylcarnitine

Propionyl carnitine

Others Others
Propionylcarnitine (Propionyl carnitine) 是一种被广泛使用的膳食补充剂,有青光眼和难道破裂有关。
T81034L TAT-NSF700 Fusion Peptide acetate

TAT-NSF700 Fusion Peptide acetate 是一种可渗透细胞膜的 N-乙基-马来酰亚胺敏感因子 (NSF) 抑制剂,是一种融合多肽,具有潜在的抗炎活性。TAT-NSF700 Fusion Peptide acetate 与细胞内细胞器相互作用,可用于研究心肌缺血和再灌注损伤。
T0188 Fluticasone (propionate)

丙酸氟替卡松,CCI-187881,氟替卡松丙酸酯,Fluticasone propionate

Glucocorticoid Receptor; Virus Protease; Estrogen/progestogen Receptor; Phospholipase; Endogenous Metabolite; ADC Cytotoxin Antibody-drug Conjugate/ADC Related; Endocrinology/Hormones; Metabolism; Microbiology/Virology
Fluticasone propionate (CCI-187881) 是一种选择性糖皮质激素受体激动剂,是一种局部抗炎激素,亲和力KD 为 0.5 nM。具有抗病毒活性。
T50083 Cell-cell interaction 1

Others Others
12-oxo-N-[1-(propan-2-yl)piperidin-4-yl]-6H,7H,8H,9H,10H,12H-azepino[2,1-b]quinazoline-3-carboxamide 可用作分子结构单元,用于多种化合物的合成。
T7077 2,3-BIS(N-BUTYLTHIO)-1,4-NAPHTHALENEDION

Others Others
2,3-BIS(N-BUTYLTHIO)-1,4-NAPHTHALENEDION 是中间体。
T3560 Desmethylanethol trithione

ADT-OH

VEGFR; Akt Angiogenesis; Cytoskeletal Signaling; PI3K/Akt/mTOR signaling; Tyrosine Kinase/Adaptors
Desmethylanethol trithione (ADT-OH) 是合成硫化氢的供体。它利用上调 FADD 诱导细胞凋亡,并对体内黑色素瘤的形成具有一定的抑制作用,可用于研究癌症疾病。
T65554 cholesterol-absorption inhibitor Intermediate 2

Others Others
cholesterol-absorption inhibitor Intermediate 2 是一种有效且具有口服活性的胆固醇吸收抑制剂,可降低血液中胆固醇含量。
T0830 Bithionol

硫双二氯酚,Actamer,硫氯酚

cAMP; Parasite GPCR/G Protein; Microbiology/Virology
Bithionol (Actamer) 是一种抗寄生虫药物,对若干癌细胞有抑制作用。
T13244 Ubiquitination-IN-1

Others Others
Ubiquitination-IN-1 是一种有效的泛素化和Cksl-Skp2蛋白互作抑制剂 (IC50=0.17 μM) 抑制剂,增加 p27 水平,可通过阻断肿瘤抑制因子的降解发挥作用。
T9978 Glutathione synthesis-IN-1

Others Others
Glutathione synthesis-IN-1 (DC-1)是谷胱甘肽合成抑制剂。
T9228 Propionylpromazine hydrochloride

盐酸丙酰丙嗪,Propiopromazine hydrochloride

Dopamine Receptor GPCR/G Protein; Neuroscience
Propionylpromazine hydrochloride (Propiopromazine hydrochloride) 是多巴胺受体 D2 (DRD2) 拮抗剂,可用于研究帕金森氏病。

化合物

L-Lactate ion
Cat.No: T32809
Synonym: L-Lactate,Lactate ion, L-
Target: Others
M2 ion channel blocker
Cat.No: T11927
Synonym:
Target: Others
Albitiazolium
Cat.No: T25026
Synonym: Albitiazolium ion
Target: Others
Lauralkonium
Cat.No: T32592
Synonym: Lauralkonium ion,Lauralkonium cation
Target: Others
Ulefnersen
Cat.No: T84763
Synonym: ION-363
Target: Others
Laurolinium
Cat.No: T25640
Synonym: Laurolinium ion,Laurolinium cation
Target: Others
Laudexium
Cat.No: T25636
Synonym: Laudexium ion,Laudexium cation
Target: Others
Tetrabutylphosphonium cation
Cat.No: T34817
Synonym: Tetra-n-butylphosphonium,J279H,Tetrabutylphosphonium ion,Tetrabutylphosphonium,Phosphonium, tetrabutyl-
Target: Others
PSEM 89S TFA
Cat.No: T8552
Synonym:
Target: AChR
PF-04885614
Cat.No: T12421
Synonym:
Target: Sodium Channel
NS3623
Cat.No: T16347
Synonym:
Target: Potassium Channel
ICILIN
Cat.No: T1814
Synonym: AG-3-5
Target: TRP/TRPV Channel
GSK137647A
Cat.No: T3171
Synonym: GSK 137647
Target: GPR
BAY-1797
Cat.No: T10466
Synonym:
Target: P2X Receptor
ML204
Cat.No: T2298
Synonym:
Target: TRP/TRPV Channel
PHD-1-IN-1
Cat.No: T9627
Synonym:
Target: HIF/HIF Prolyl-Hydroxylase
EGTA
Cat.No: T4585
Synonym: Ethylenebis(oxyethylenenitrilo)tetraacet,乙二醇双(2-氨基乙基醚)四乙酸
Target: Others
INCB-39110
Cat.No: T70310
Synonym:
Target: Others
Stercuronium
Cat.No: T68783
Synonym:
Target: Others
Ciclotropium (free base)
Cat.No: T68735
Synonym:
Target: Others
Dibrospidium Free Base
Cat.No: T68502
Synonym:
Target: Others
Framycetin sulfate
Cat.No: T2096
Synonym: Neomycin Sulphate B,硫酸新霉素B,Framycetin sulphate
Target: Antibacterial, Antibiotic
(±)-1,2-Diolein
Cat.No: T40101
Synonym: 1,2-Dioleoyl-rac-glycerol,甘油1,2-二油酸酯
Target: PKC
Calcium ionophore II
Cat.No: T40857
Synonym: Calcium ionophore II,N,N,N′,N′-Tetracyclohexyl-3-oxapentanediamide
Target: Others
Tubulin polymerization-IN-55
Cat.No: T77728
Synonym:
Target: Microtubule Associated
Endovion
Cat.No: T15233
Synonym: NS3728
Target: Chloride channel
Clobetasol propionate
Cat.No: T1561
Synonym: Dermovate,Clobetasol 17-propionate,CGP9555,Temovate,丙酸氯倍他索,CCl 4725
Target: Glucocorticoid Receptor, P450
5,5-Dimethyloxazolidine-2,4-dione
Cat.No: T1234
Synonym: Dimethadion,Dimethadione,二甲双酮,Dimethyloxazolidinedione
Target: Calcium Channel
Palbociclib Isethionate
Cat.No: T6240
Synonym: Palbociclib (PD0332991) Isethionate,帕博西尼羟乙基磺酸盐,PD 0332991 isethionate,帕布昔利布羟乙基磺酸盐
Target: CDK
SORT-PGRN interaction inhibitor 1
Cat.No: T9044
Synonym:
Target: Neurotensin Receptor
AP-1/NF-κB activation inhibitor 1
Cat.No: T9656
Synonym:
Target: NF-κB, DNA/RNA Synthesis
Bisdionin C
Cat.No: T40863
Synonym:
Target: Antibacterial
Beclometasone dipropionate
Cat.No: T1127
Synonym: Beclovent,Beclomethasone dipropionate,二丙酸倍氯米松,丙酸倍氯米松,Beconase,Vancenase
Target: Glucocorticoid Receptor
B7/CD28 interaction inhibitor 1
Cat.No: T3189
Synonym: CTLA-4 inhibitor
Target: Others
2H-Naphth[2′,1′:4,5]indeno[1,2-d][1,3]dioxole, pregn-4-ene-3,20-dione deriv
Cat.No: T34383L
Synonym:
Target: Others
Trimethadione
Cat.No: T0283
Synonym: 三甲双酮,3,5,5,-Trimethyloxazolidine-2,4-dione
Target: Calcium Channel
Betamethasone dipropionate
Cat.No: T1559
Synonym: Diprolene AF,SCH 11460,二丙酸倍他米松,Betamethasone 17,21-dipropionate,Diprolene,倍他米松二丙酸酯,Diprosone
Target: Glucocorticoid Receptor
Fibronectin Adhesion-promoting Peptide acetate
Cat.No: TP1153L
Synonym: Fibronectin Adhesion-promoting Peptide acetate(125720-21-0 free base),Heparin Binding Peptide acetate
Target: Others
Paroxypropione
Cat.No: T66154
Synonym:
Target: Others
Propionylcarnitine
Cat.No: T19528
Synonym: Propionyl carnitine
Target: Others
TAT-NSF700 Fusion Peptide acetate
Cat.No: T81034L
Synonym:
Target:
Fluticasone (propionate)
Cat.No: T0188
Synonym: 丙酸氟替卡松,CCI-187881,氟替卡松丙酸酯,Fluticasone propionate
Target: Glucocorticoid Receptor, Virus Protease, Estrogen/progestogen Receptor, Phospholipase, Endogenous Metabolite, ADC Cytotoxin
Cell-cell interaction 1
Cat.No: T50083
Synonym:
Target: Others
2,3-BIS(N-BUTYLTHIO)-1,4-NAPHTHALENEDION
Cat.No: T7077
Synonym:
Target: Others
Desmethylanethol trithione
Cat.No: T3560
Synonym: ADT-OH
Target: VEGFR, Akt
cholesterol-absorption inhibitor Intermediate 2
Cat.No: T65554
Synonym:
Target: Others
Bithionol
Cat.No: T0830
Synonym: 硫双二氯酚,Actamer,硫氯酚
Target: cAMP, Parasite
Ubiquitination-IN-1
Cat.No: T13244
Synonym:
Target: Others
Glutathione synthesis-IN-1
Cat.No: T9978
Synonym:
Target: Others
Propionylpromazine hydrochloride
Cat.No: T9228
Synonym: 盐酸丙酰丙嗪,Propiopromazine hydrochloride
Target: Dopamine Receptor
Cat. No. Product Name Target Signaling Pathways
TQ0192 Senecionine

Aureine,Senecionan-11,16-dione, 12-hydroxy-,千里光宁,Senecionin

Others Others
Senecionine 是一种吡咯里西啶生物碱,从Senecio vulgaris中分离得到,它对动物和人类有毒性。
T8709 Nandrolone phenylpropionate

Nandrolone phenpropionate,苯丙酸诺龙

Androgen Receptor Endocrinology/Hormones
Nandrolone phenylpropionate (Nandrolone phenpropionate) 是一种合成代谢类固醇,是一种 19-nortestosterone 的衍生物。它能够促进蛋白质合成,用于缓解组织分解代谢,可以用于骨质疏松症和特纳综合征的研究。
T5285 3-(Methylthio)propionic acid

3-Methylthiopropionate,3-甲基硫代丙酸,4-Thiapentanoic acid,3-Methylsulfanylpropionic acid

Others; Endogenous Metabolite; Antifungal Metabolism; Microbiology/Virology; Others
3-(Methylthio)propionic acid (4-Thiapentanoic acid) 是methionine 的代谢物,是中间体。
T1165 Ethionamide

Bayer 5312,乙硫异烟胺,2-ethylthioisonicotinamide,Ethinamide

Dehydrogenase; CAT; Antibacterial; Antibiotic Metabolism; Microbiology/Virology; oxidation-reduction
Ethionamide (2-ethylthioisonicotinamide) 是一种抗结核抗生素。
TN7192 7-Bromoquinazoline-2,4(1H,3H)-Dione

7-Bromo-2,4(1H,3H)-quinazolinedione,7-溴喹唑啉-(2,4)二酮,7-Bromo-1H-quinazoline-2,4-dione,7-bromoquinazoline-2,4-diol

Others Others
7-Bromoquinazoline-2,4(1H,3H)-Dione (7-Bromo-2,4(1H,3H)-quinazolinedione) 是一种海洋来源的天然产物,发现于 Pyura sacciformis。
T1285 Anethole trithione

茴三硫,Anetholtrithion

Others; AChR Neuroscience; Others
Anethole trithione (Anetholtrithion) 是硫杂环胆碱,是一种胆汁分泌刺激剂,可增强唾液分泌并增加 mAChR 受体,用于口干症的研究。
T5297 3-Indolepropionic acid

Indolepropionic acid,IPA,indole-3-propionic acid,吲哚-3-丙酸

Antioxidant; Reactive Oxygen Species; Endogenous Metabolite Immunology/Inflammation; Metabolism; NF-κB; oxidation-reduction
3-Indolepropionic acid (Indolepropionic acid) 是强效的抗氧化剂,具有研究阿尔兹海默症的潜能。
T0525 Flopropione

夫洛丙酮,Phloropropiophenone

5-HT Receptor; Transferase GPCR/G Protein; Metabolism; Neuroscience
Flopropione (Phloropropiophenone) 是一种解痉剂,用作 5-HT1A 受体拮抗剂,也是儿茶酚-O-甲基转移酶抑制剂。
T7908 DL-Methionine Methylsulfonium Chloride

DL-蛋氨酸甲基氯化锍,维生素U

Others Others
DL-methionine methylsulfonium chloride 是天然的蛋氨酸衍生物。它能够有效保护胃粘膜,避免其受到乙醇诱导的损伤。
TN7209 3-bromopyrrole-2,5-dione

ZINC13379821,3-溴-1H-吡咯-2,5-二酮,3-Bromo-1H-pyrrole-2,5-dione

Others Others
3-bromopyrrole-2,5-dione (ZINC13379821) 是一种海洋来源的天然产物,存在于 Axinella brevistyla。
T4909 N-Acetyl-DL-methionine

N-乙酰-DL-蛋氨酸,N-乙酰-DL-甲硫氨酸

Others; Endogenous Metabolite Metabolism; Others
N-Acetyl-DL-methionine 是内源性代谢产物的一种。
T4768 Diethyl oxalpropionate

草酰丙酸二乙酯,HYL 2-METHYL-3-OXOSUCCINATE

Others; Endogenous Metabolite Metabolism; Others
Diethyl oxalpropionate (HYL 2-METHYL-3-OXOSUCCINATE) 是一种合成 PDMMLA 的中间体。其中 PDMMLA 的衍生物可用于纳米粒子的合成和研究。
TN6730 Epoxyazadiradione

NF-κB NF-κB
Epoxyazadiradione 是从印楝果实中得到的柠檬苦素。它能够可逆的、非竞争性的抑制人类、约氏疟原虫、疟原虫的互变异构酶活性。它具有抗疟原虫和人类 MIF 诱导的促炎反应的潜力。
TN2064 Physcion 8-O-β-D-glucopyranoside

大黄素甲醚-8-O-Β-D-葡萄糖苷,Physcion 8-O-beta-D-monoglucoside

TNF Apoptosis
Physcion 8-O-β-D-glucopyranoside (Physcion 8-O-beta-D-monoglucoside) 具有抗炎和抗癌活性。Physcion 8-O-β-D-glucopyranoside 可用于常见恶性肿瘤的研究。
T7437 3-(3-Hydroxyphenyl)propionic Acid

m-Hydroxyphenylpropionic acid,3-Hydroxyhydrocinnamic acid,3-(3-羟基苯基)丙酸

Others; Endogenous Metabolite Metabolism; Others
3-(3-Hydroxyphenyl)propionic Acid (m-Hydroxyphenylpropionic acid) 是一种黄酮类代谢产物,由人体微生物区系形成,具有舒张血管的特性。
T8064 Lactobionic acid

Others; Antibacterial Microbiology/Virology; Others
Lactobionic acid 是在里海酸奶中的一种仿生酸,化学上由与半乳糖键合的葡萄糖酸组成。它是具有抗氧化、抗菌和保湿特性的乳糖酸。
T14001 11-Beta-hydroxyandrostenedione

4-雄烯-11β-醇-3,17-二酮,NSC-17102,4-Androsten-11β-ol-3,17-dione

Endogenous Metabolite Metabolism
11-Beta-hydroxyandrostenedione (NSC-17102) 是主要存在于肾上腺的类固醇,也是 11β-羟基类固醇脱氢酶同工酶抑制剂。随着 4-androstenedione 的提高,通过测量血浆中的11-Beta-hydroxyandrostenedione,能够区分高雄激素血症的肾上腺或卵巢起源。
T10939L L-Cystathionine

L-胱硫醚,Cystathionine,ZINC1532680,L-(+)-Cystathionine,Cystathionine, L-

Apoptosis; Endogenous Metabolite Apoptosis; Metabolism
L-Cystathionine (Cystathionine, L-) 是一种与含硫氨基酸的代谢条件有关的关键非蛋白质氨基酸。L-Cystathionine 可用于有关心血管保护的研究。
TJO2742 DL-Methionine

蛋氨酸,methionine,DL-蛋氨酸,Acimetion,Racemethionine

Parasite Microbiology/Virology
DL-Methionine (Acimetion) 存在于肉类、鱼类和奶制品中,是可用于动物的天然饲料,还可杀死马铃薯上的金线虫。它是一种含有硫的必需氨基酸,具有氧化应激防御作用。
T4844 L-Methionine

L(-)-Methionin,L-蛋氨酸,L-Methionin

Endogenous Metabolite Metabolism
L-Methionine (L-Methionin) 是 Methionine 的 L-异构体。Methionine 是必需氨基酸,同时也是肝脏保护剂。
T19397 L-Methionine sulfoxide

L-蛋氨酸亚砜,H-Met(O)-OH

Endogenous Metabolite Metabolism
L-Methionine sulfoxide (H-Met(O)-OH) 是一种甲硫氨酸的代谢产物,能够诱导 M1/classical 巨噬细胞极化,并调节氧化应激和嘌呤能的信号传递参数。
T0449 Menadione

维生素K3,Vitamin K3,甲萘醌

Thrombin; Endogenous Metabolite Metabolism; Proteases/Proteasome
Menadione (Vitamin K3) 是合成的萘醌,能够在体内转化成活性维生素 K2。
T7090 Jionoside A1

焦地黄苯乙醇甙A1,焦地黄苯乙醇苷A1

Others Others
Jionoside A1 分离自Radix Rehmanniae Praeparata 中,具有剂量依赖性免疫增强作用,并对 H2O2处理的 SH-SY5Y 细胞具有中等保护活性。
T1085 L-Glutathione reduced

谷胱甘肽,GSH,Isethion,Glutathione,γ-L-Glutamyl-L-cysteinyl-glycine,Glutathion,还原型谷胱甘肽,Tathion

Ferroptosis; Reactive Oxygen Species; Endogenous Metabolite; Glutathione reductase Apoptosis; Immunology/Inflammation; Metabolism; NF-κB; oxidation-reduction
L-Glutathione reduced (Glutathione) 属于天然三肽,存在与细胞中,是一种内源性抗氧化剂,可以清除氧自由基。L-Glutathione reduced 是某些酶的辅助因子,参与蛋白质二硫键重排并减少过氧化物。
T4857 Pteridine-2,4(1H,3H)-dione

2,4-Dihydroxypteridine,2,4-二羟基蝶啶,Lumazine

Others; Endogenous Metabolite Metabolism; Others
Pteridine-2,4(1H,3H)-dione (Lumazine) 是内源性代谢产物的一种。
T3019 Physcion

大黄素甲醚,Physcione,Parietin,Rheochrysidin

Dehydrogenase; Antibacterial Metabolism; Microbiology/Virology
Physcion (Physcione) 是一种从中药大黄中分离的蒽醌,作为 6-磷酸葡萄糖酸脱氢酶的抑制剂,IC50和 Kd 值分别为 38.5 μM 和 26.0 μM。它具有通便、保肝、抗炎、抗菌、抗增殖、抗肿瘤作用。
TQ0226 Jionoside B1

Glucosidase Metabolism
Jionoside B1 是从熟地黄(Gaertn.)的根中分离出来的,抑制 α-葡萄糖苷酶。
T3411 Curdione

莪术二酮,(+)-Curdione

P450 Metabolism
Curdione ((+)-Curdione) 是一种具有高生物活性的倍半萜类物质,从莪术中分离获得,具有抑制血小板聚集、抵抗血栓形成的作用。
T19418 Methionine sulfoxide

Endogenous Metabolite Metabolism
Methionine sulfoxide 是具有特性氧的甲硫氨酸的氧化产物,能够用作体内氧化应激的生物标记。
T67302 2,3-Pentanedione

Acetylpropionyl

Others Others
2,3-Pentanedione 是一种食品添加剂, 也作为发酵产物自然存在于啤酒、葡萄酒和酸奶中,并在咖啡豆烘焙过程中释放。吸入2,3-Pentanedione 被认为是人严重呼吸道疾病(包括闭塞性细支气管炎)的原因。
T13475 β-Aminopropionitrile

3-氨基丙腈,3-Aminopropionitrile,BAPN

Others; Endogenous Metabolite Metabolism; Others
β-Aminopropionitrile (3-Aminopropionitrile) 是赖氨酰氧化酶的特异性抑制剂。
T4447 S-(5'-Adenosyl)-L-methionine tosylate

S-腺苷蛋氨酸对甲苯磺酸盐,SAMe,S-(5'-Adenosyl)-L-methionine p-toluenesulfonate salt

Others Others
S-(5'-Adenosyl)-L-methionine tosylate (SAMe) 是一种普遍存在的甲基供体,参与多种生物反应,包括由 DNA 和蛋白质甲基转移酶介导的反应。它可改善抑郁、与骨关节炎和纤维肌痛相关的疼痛以及肝毒性。
T5303 Isethionic acid sodium salt

Sodium isethionate,羟乙基磺酸钠

Others; Endogenous Metabolite Metabolism; Others
Isethionic acid sodium salt (Sodium isethionate) 是内源性代谢产物的一种。
T4919 Ureidopropionic acid

Carbamoyl-b-alanine,3-酰脲丙酸,3-Ureidopropionic acid

Endogenous Metabolite Metabolism
Ureidopropionic acid (3-Ureidopropionic acid) 是尿嘧啶代谢的中间体。更具体地说,它是二氢尿嘧啶的分解产物,由二氢嘧啶酶产生。它通过β -脲丙酸酶进一步分解为β -丙氨酸。尿素丙酸本质上是β -丙氨酸的尿素衍生物。高水平的尿丙酸存在于β -尿丙酸酶(UP)缺乏的个体中。嘧啶代谢中的酶缺乏与抗肿瘤药物5-氟尿嘧啶的严重毒性风险有关。
T7931 16a,17a-Epoxy-4-Pregnen-3,20-Dione

Others Others
16a,17a-Epoxy-4-Pregnen-3,20-Dione 是一种合成孕激素,是黄体酮激素的代谢产物,它通过与黄体酮受体结合发挥作用,已被用于研究孕激素对生殖器官的影响,激素对细胞生长和发育的影响,以及激素对免疫系统的影响。
T5215 N-(3-Phenylpropionyl)glycine

N-(3-苯基丙酰基)甘氨酸,Phenylpropionylglycine

Others Others
N-(3-Phenylpropionyl)glycine (Phenylpropionylglycine) 是一种酰基甘氨酸。酰基甘氨酸通常是脂肪酸的次要代谢物。
T5272 3-(3-Methoxyphenyl)propionic acid

3-(3-甲氧基苯基)丙酸,3-Methoxyhydrocinnamic acid

Others; Endogenous Metabolite Metabolism; Others
3-(3-Methoxyphenyl)propionic acid (3-Methoxyhydrocinnamic acid) 是人体自然代谢的有机酸,排泄于尿液中。
TN6737 (25R)-Spirost-4-ene-3,12-dione

Others Others
(25R)-Spirost-4-ene-3,12-dione 是一种天然产物,抑制中性粒细胞超氧阴离子的产生和肥大细胞组胺的释放。
T8059 N-Acetyl-L-methionine

N-Acetylmethionine,N-乙酰-L-蛋氨酸

Others; Endogenous Metabolite Metabolism; Others
N-Acetyl-L-methionine (N-Acetylmethionine) 是人体代谢物,在营养和代谢作用上和 L-methionine 相当。其中 L-methionine 是生长发育并不能够少的氨基酸。
T5556 5a-Pregnane-3,20-dione

Endogenous Metabolite Metabolism
5a-Pregnane-3,20-dione 是内源性的孕酮代谢物。
T3130 Testosterone phenylpropionate

Testosterone hydrocinnamate,苯丙酸睾酮,Retandrol,Testosterone 17-phenylpropionate

Others Others
Testosterone phenylpropionate (Testosterone 17-phenylpropionate) 是一种长效雄激素。d3-Testosterone phenylpropionate 可用作内标物。
T7927 β-Ionone

乙位紫罗兰酮,β-紫罗兰酮,β-lonone

Apoptosis; Others Apoptosis; Others
β-Ionone (β-lonone) 是β-类胡萝卜素的端环类似物,广泛存在于水果和蔬菜中,可有效诱导胃腺癌细胞 SGC7901 凋亡,具有抗增殖、抗转移和抗肿瘤作用。
T6752 S-Adenosyl-L-methionine disulfate tosylate

S-腺苷蛋氨酸对甲苯磺酸硫酸盐,Ademetionine disulfate tosylate

DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
S-Adenosyl-L-methionine disulfate tosylate (Ademetionine disulfate tosylate) 是一种主要生物甲基供体,在所有哺乳动物细胞中合成,但在肝脏中含量较高。
T3381 Lysionotin

岩豆素

Others Others
Lysionotin (Nevadensin) 是一种类黄酮,分离自黄花草药中。它可抑制 α-Toxin (一种成孔蛋白) 的表达,并在体内和体外针对金黄色葡萄球菌显示出显著的保护作用。它可用于研究由金黄色葡萄球菌引起的肺炎。
T5S0691 Shionone

紫菀酮,Shionon

Others Others
Shionone (Shionon) 是一种从Aster tataricus 中分离得到的三萜类化合物,具有独特的六元四环骨架和 3-氧代-4-单甲基结构。它具有镇咳、抗炎作用。
T7285 Ionomycin

Calcium Channel Membrane transporter/Ion channel; Metabolism
Ionomycin 是一种钙离子载体和一种结合钙离子(Ca2+)的抗生素。它是由联合链霉菌(Streptomyces conglobatus)产生的。它在研究中用于提高细胞内钙水平(Ca2+),并作为了解 Ca2+跨生物膜运输的研究工具。Ionomycin 可促进细胞凋亡,诱导蛋白激酶 C (PKC)活化。
T7335 2,3-Diaminopropionic acid

L-2,3-二氨基丙酸,L-2,3-Diaminopropionic acid

Endogenous Metabolite Metabolism
2,3-Diaminopropionic acid (L-2,3-Diaminopropionic acid) 是一种神经毒性氨基酸 b-oxalyl-L-a, b-diaminopropionic acid 的代谢产物。
TN7149 5-[(1H-indol-3-yl)methylidene]imidazolidine-2,4-dione

(4Z)-4-(1H-indol-3-ylmethylidene)-4H-imidazole-2,5-diol,(5Z)-5-(1H-indol-3-ylmethylidene)imidazolidine-2,4-dione

Others Others
5-[(1H-indol-3-yl)methylidene]imidazolidine-2,4-dione ((4Z)-4-(1H-indol-3-ylmethylidene)-4H-imidazole-2,5-diol) 是一种海洋来源的天然产物,存在于Leptopsammia pruvoti。
TN6729 Azadiradione

AZD

Others Others
Azadiradione (AZD) 是 HSF1的一种,是由印楝树中提取得到,具有一定生物活性的柠檬苦素。
T7450 1-Phenylpropane-1,2-dione

1-Phenyl-1,2-propanedione,Acetyl benzoyl,1-苯基-1,2-丙二酮

Others Others
1-Phenylpropane-1,2-dione (Acetyl benzoyl) 是麻黄素生物碱的生物合成前体,分离自从嫩麻黄中。
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天然产物

Senecionine
Cat.No: TQ0192
Synonym: Aureine,Senecionan-11,16-dione, 12-hydroxy-,千里光宁,Senecionin
Target: Others
Nandrolone phenylpropionate
Cat.No: T8709
Synonym: Nandrolone phenpropionate,苯丙酸诺龙
Target: Androgen Receptor
3-(Methylthio)propionic acid
Cat.No: T5285
Synonym: 3-Methylthiopropionate,3-甲基硫代丙酸,4-Thiapentanoic acid,3-Methylsulfanylpropionic acid
Target: Others, Endogenous Metabolite, Antifungal
Ethionamide
Cat.No: T1165
Synonym: Bayer 5312,乙硫异烟胺,2-ethylthioisonicotinamide,Ethinamide
Target: Dehydrogenase, CAT, Antibacterial, Antibiotic
7-Bromoquinazoline-2,4(1H,3H)-Dione
Cat.No: TN7192
Synonym: 7-Bromo-2,4(1H,3H)-quinazolinedione,7-溴喹唑啉-(2,4)二酮,7-Bromo-1H-quinazoline-2,4-dione,7-bromoquinazoline-2,4-diol
Target: Others
Anethole trithione
Cat.No: T1285
Synonym: 茴三硫,Anetholtrithion
Target: Others, AChR
3-Indolepropionic acid
Cat.No: T5297
Synonym: Indolepropionic acid,IPA,indole-3-propionic acid,吲哚-3-丙酸
Target: Antioxidant, Reactive Oxygen Species, Endogenous Metabolite
Flopropione
Cat.No: T0525
Synonym: 夫洛丙酮,Phloropropiophenone
Target: 5-HT Receptor, Transferase
DL-Methionine Methylsulfonium Chloride
Cat.No: T7908
Synonym: DL-蛋氨酸甲基氯化锍,维生素U
Target: Others
3-bromopyrrole-2,5-dione
Cat.No: TN7209
Synonym: ZINC13379821,3-溴-1H-吡咯-2,5-二酮,3-Bromo-1H-pyrrole-2,5-dione
Target: Others
N-Acetyl-DL-methionine
Cat.No: T4909
Synonym: N-乙酰-DL-蛋氨酸,N-乙酰-DL-甲硫氨酸
Target: Others, Endogenous Metabolite
Diethyl oxalpropionate
Cat.No: T4768
Synonym: 草酰丙酸二乙酯,HYL 2-METHYL-3-OXOSUCCINATE
Target: Others, Endogenous Metabolite
Epoxyazadiradione
Cat.No: TN6730
Synonym:
Target: NF-κB
Physcion 8-O-β-D-glucopyranoside
Cat.No: TN2064
Synonym: 大黄素甲醚-8-O-Β-D-葡萄糖苷,Physcion 8-O-beta-D-monoglucoside
Target: TNF
3-(3-Hydroxyphenyl)propionic Acid
Cat.No: T7437
Synonym: m-Hydroxyphenylpropionic acid,3-Hydroxyhydrocinnamic acid,3-(3-羟基苯基)丙酸
Target: Others, Endogenous Metabolite
Lactobionic acid
Cat.No: T8064
Synonym:
Target: Others, Antibacterial
11-Beta-hydroxyandrostenedione
Cat.No: T14001
Synonym: 4-雄烯-11β-醇-3,17-二酮,NSC-17102,4-Androsten-11β-ol-3,17-dione
Target: Endogenous Metabolite
L-Cystathionine
Cat.No: T10939L
Synonym: L-胱硫醚,Cystathionine,ZINC1532680,L-(+)-Cystathionine,Cystathionine, L-
Target: Apoptosis, Endogenous Metabolite
DL-Methionine
Cat.No: TJO2742
Synonym: 蛋氨酸,methionine,DL-蛋氨酸,Acimetion,Racemethionine
Target: Parasite
L-Methionine
Cat.No: T4844
Synonym: L(-)-Methionin,L-蛋氨酸,L-Methionin
Target: Endogenous Metabolite
L-Methionine sulfoxide
Cat.No: T19397
Synonym: L-蛋氨酸亚砜,H-Met(O)-OH
Target: Endogenous Metabolite
Menadione
Cat.No: T0449
Synonym: 维生素K3,Vitamin K3,甲萘醌
Target: Thrombin, Endogenous Metabolite
Jionoside A1
Cat.No: T7090
Synonym: 焦地黄苯乙醇甙A1,焦地黄苯乙醇苷A1
Target: Others
L-Glutathione reduced
Cat.No: T1085
Synonym: 谷胱甘肽,GSH,Isethion,Glutathione,γ-L-Glutamyl-L-cysteinyl-glycine,Glutathion,还原型谷胱甘肽,Tathion
Target: Ferroptosis, Reactive Oxygen Species, Endogenous Metabolite, Glutathione reductase
Pteridine-2,4(1H,3H)-dione
Cat.No: T4857
Synonym: 2,4-Dihydroxypteridine,2,4-二羟基蝶啶,Lumazine
Target: Others, Endogenous Metabolite
Physcion
Cat.No: T3019
Synonym: 大黄素甲醚,Physcione,Parietin,Rheochrysidin
Target: Dehydrogenase, Antibacterial
Jionoside B1
Cat.No: TQ0226
Synonym:
Target: Glucosidase
Curdione
Cat.No: T3411
Synonym: 莪术二酮,(+)-Curdione
Target: P450
Methionine sulfoxide
Cat.No: T19418
Synonym:
Target: Endogenous Metabolite
2,3-Pentanedione
Cat.No: T67302
Synonym: Acetylpropionyl
Target: Others
β-Aminopropionitrile
Cat.No: T13475
Synonym: 3-氨基丙腈,3-Aminopropionitrile,BAPN
Target: Others, Endogenous Metabolite
S-(5'-Adenosyl)-L-methionine tosylate
Cat.No: T4447
Synonym: S-腺苷蛋氨酸对甲苯磺酸盐,SAMe,S-(5'-Adenosyl)-L-methionine p-toluenesulfonate salt
Target: Others
Isethionic acid sodium salt
Cat.No: T5303
Synonym: Sodium isethionate,羟乙基磺酸钠
Target: Others, Endogenous Metabolite
Ureidopropionic acid
Cat.No: T4919
Synonym: Carbamoyl-b-alanine,3-酰脲丙酸,3-Ureidopropionic acid
Target: Endogenous Metabolite
16a,17a-Epoxy-4-Pregnen-3,20-Dione
Cat.No: T7931
Synonym:
Target: Others
N-(3-Phenylpropionyl)glycine
Cat.No: T5215
Synonym: N-(3-苯基丙酰基)甘氨酸,Phenylpropionylglycine
Target: Others
3-(3-Methoxyphenyl)propionic acid
Cat.No: T5272
Synonym: 3-(3-甲氧基苯基)丙酸,3-Methoxyhydrocinnamic acid
Target: Others, Endogenous Metabolite
(25R)-Spirost-4-ene-3,12-dione
Cat.No: TN6737
Synonym:
Target: Others
N-Acetyl-L-methionine
Cat.No: T8059
Synonym: N-Acetylmethionine,N-乙酰-L-蛋氨酸
Target: Others, Endogenous Metabolite
5a-Pregnane-3,20-dione
Cat.No: T5556
Synonym:
Target: Endogenous Metabolite
Testosterone phenylpropionate
Cat.No: T3130
Synonym: Testosterone hydrocinnamate,苯丙酸睾酮,Retandrol,Testosterone 17-phenylpropionate
Target: Others
β-Ionone
Cat.No: T7927
Synonym: 乙位紫罗兰酮,β-紫罗兰酮,β-lonone
Target: Apoptosis, Others
S-Adenosyl-L-methionine disulfate tosylate
Cat.No: T6752
Synonym: S-腺苷蛋氨酸对甲苯磺酸硫酸盐,Ademetionine disulfate tosylate
Target: DNA/RNA Synthesis
Lysionotin
Cat.No: T3381
Synonym: 岩豆素
Target: Others
Shionone
Cat.No: T5S0691
Synonym: 紫菀酮,Shionon
Target: Others
Ionomycin
Cat.No: T7285
Synonym:
Target: Calcium Channel
2,3-Diaminopropionic acid
Cat.No: T7335
Synonym: L-2,3-二氨基丙酸,L-2,3-Diaminopropionic acid
Target: Endogenous Metabolite
5-[(1H-indol-3-yl)methylidene]imidazolidine-2,4-dione
Cat.No: TN7149
Synonym: (4Z)-4-(1H-indol-3-ylmethylidene)-4H-imidazole-2,5-diol,(5Z)-5-(1H-indol-3-ylmethylidene)imidazolidine-2,4-dione
Target: Others
Azadiradione
Cat.No: TN6729
Synonym: AZD
Target: Others
1-Phenylpropane-1,2-dione
Cat.No: T7450
Synonym: 1-Phenyl-1,2-propanedione,Acetyl benzoyl,1-苯基-1,2-丙二酮
Target: Others
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Cat. No. Product Name Species Expression System
TMPH-01863 PIEZO1 Protein, Human, Recombinant (His & Myc)

Protein FAM38A,Membrane protein induced by beta-amyloid trea...

Human E. coli
PIEZO1 Protein, Human, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 33.6 kDa and the accession number is Q92508.
TMPH-01891 KCNE2 Protein, Human, Recombinant (His)

MinK-related peptide 1,Potassium voltage-gated channel subfa...

Human E. coli
KCNE2 Protein, Human, Recombinant (His) is expressed in E. coli expression system with N-10xHis tag. The predicted molecular weight is 17.3 kDa and the accession number is Q9Y6J6.
TMPH-01358 FXYD3 Protein, Human, Recombinant (His & SUMO)

Phospholemman-like,Chloride conductance inducer protein Mat-...

Human E. coli
FXYD3 Protein, Human, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 20.5 kDa and the accession number is Q14802.
TMPY-03236 Human respiratory syncytial virus (RSV) Fusion protein/RSV-F (Strain RSS-2) Protein (His)

F Protein,HRSVgp8

RSV Baculovirus Insect Cells
Human respiratory syncytial virus (RSV) Fusion protein/RSV-F (Strain RSS-2) Protein (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 57.8 kDa and the accession number is P11209.
TMPY-02215 Coagulation factor IX/F9 Protein, Human, Recombinant (His)

FIX,PTC,Coagulation factor 9,coagulation f...

Human HEK293 Cells
Coagulation factor IX/F9 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 50 kDa and the accession number is AAB59620.1.
TMPY-01193 Influenza A H1N1 (A/Brevig Mission/1/1918) Hemagglutinin Protein (His)

Harvey rat sarcoma viral oncogene homolog

H1N1 HEK293 Cells
Influenza A H1N1 (A/Brevig Mission/1/1918) Hemagglutinin Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 37.5 kDa and the accession number is Q9WFX3.
TMPY-01078 Human respiratory syncytial virus (RSV) (A2) Fusion glycoprotein/RSV-F Protein (His)

HRSVgp8,F Protein

RSV Baculovirus Insect Cells
Human respiratory syncytial virus (RSV) (A2) Fusion glycoprotein/RSV-F Protein (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 57.4 kDa and the accession number is P03420.1.
TMPY-04274 Influenza A H1N1 (A/Brevig Mission/1/1918) Nucleoprotein/NP Protein (His)

NP Protein

H1N1 Baculovirus Insect Cells
Influenza A H1N1 (A/Brevig Mission/1/1918) Nucleoprotein/NP Protein (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 57.7 kDa and the accession number is Q5UEW0.1.
TMPY-01101 Coagulation factor X/F10 Protein, Human, Recombinant (His)

FXA,FX,coagulation factor X,coagulation fa...

Human Baculovirus Insect Cells
Coagulation factor X, also known as FX, F10, Eponym Stuart-Prower factor, and thrombokinase, is an enzyme of the coagulation cascade. It is one of the vitamin K-dependent serine proteases, and plays a crucial role in the coagulation cascade and blood clotting, as the first enzyme in the common pathway of thrombus formation. Factor X deficiency is one of the rarest of the inherited coagulation disorders. FX deficiency among the most severe of the rare coagulation defects, typically including hema...
TMPY-01104 Coagulation factor XI/F11 Protein, Human, Recombinant (His)

coagulation factor 11,coagulation factor X...

Human HEK293 Cells
Factor XI (plasma thromboplastin antecedent) is a plasma glycoprotein, and a zymogen acting as a serine protease which participates in blood coagulation as a catalyst in the conversion of factor IX to factor IXa in the presence of calcium ions. It is an unusual dimeric protease, with structural features that distinguish it from vitamin K-dependent coagulation proteases. The factor XI is synthesized in the liver as a single polypeptide chain with a molecular weight estimated between 125 ~160 kDa ...
TMPY-02185 Coagulation factor XIII B/F13B Protein, Human, Recombinant (His)

Coagulation factor 13,coagulation factor X...

Human HEK293 Cells
Coagulation factor XIII B chain, also known as Fibrin-stabilizing factor B subunit, Protein-glutamine gamma-glutamyltransferase B chain, Transglutaminase B chain and F13B, is a secreted protein which contains 1 Sushi ( CCP / SCR ) domains. Coagulation factor XIII is the last zymogen to become activated in the blood coagulation cascade. Plasma factor XIII is a heterotetramer composed of 2 A subunits and 2 B subunits. The A subunits have catalytic function, and the B subunits do not have en...
TMPY-05688 Human respiratory syncytial virus (RSV) Fusion Protein (aa 1-525, His)

HRSVgp8,F Protein

RSV Baculovirus Insect Cells
Human respiratory syncytial virus (RSV) Fusion Protein (aa 1-525, His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 57.12 kDa and the accession number is K7WLI9.
TMPY-05566 Siglec-2/CD22 Protein, Human, Recombinant (His, Solution)

CD22 molecule,SIGLEC-2,SIGLEC2

Human HEK293 Cells
Siglec-2/CD22 Protein, Human, Recombinant (His, Solution) is expressed in HEK293 mammalian cells with His tag. The accession number is P20273-1.
TMPY-01791 Coagulation Factor II Protein, Mouse, Recombinant (His)

Cf-2,coagulation factor II (thrombin),Cf2,FII

Mouse HEK293 Cells
Coagulation Factor II Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 69.3 kDa and the accession number is P19221.
TMPY-06171 SARS-CoV-2 Spike S1+S2 Protein (L18F & D80A & D215G & LAL242-244 deletion & R246I & K417N & E484K & N501Y & D614G & A701V, His), Biotinylated

SARS-CoV-2 Baculovirus Insect Cells
SARS-CoV-2 Spike S1+S2 Protein (L18F & D80A & D215G & LAL242-244 deletion & R246I & K417N & E484K & N501Y & D614G & A701V, His), Biotinylated is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 134 kDa and the accession number is A0A6G7K2L4.
TMPY-06443 SARS-CoV-2 Spike S1 Protein (T19R & T95I & G142D & Y145H & E156G & 157-158 deletion & A222V & L452R & T478K & D614G & P681R, His)

SARS-CoV-2 HEK293 Cells
SARS-CoV-2 Spike S1 Protein (T19R & T95I & G142D & Y145H & E156G & 157-158 deletion & A222V & L452R & T478K & D614G & P681R, His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 76.29 kDa and the accession number is YP_009724390.1.
TMPY-06082 SARS-CoV-2 Spike S1 Protein (HV69-70 deletion & N501Y & D614G, His)

SARS-CoV-2 HEK293 Cells
SARS-CoV-2 Spike S1 Protein (HV69-70 deletion & N501Y & D614G, His) is expressed in HEK293 mammalian cells. The predicted molecular weight is 76.2 kDa and the accession number is A0A6G7K2L4.
TMPY-06129 SARS-CoV-2 Spike S1 Protein (L18F & D80A & D215G & LAL242-244 deletion & R246I & K417N & E484K & N501Y & D614G, His)

SARS-CoV-2 HEK293 Cells
SARS-CoV-2 Spike S1 Protein (L18F & D80A & D215G & LAL242-244 deletion & R246I & K417N & E484K & N501Y & D614G, His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 76 kDa and the accession number is A0A6G7K2L4.
TMPY-00647 Chorionic Gonadotropin/CGA Protein, Human, Recombinant (His)

CG-α,FSH alpha,glycoprotein hormones, alpha polypeptide,FSHA...

Human HEK293 Cells
Chorionic Gonadotropin/CGA Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 11.6 kDa and the accession number is P01215.
TMPY-02923 Chorionic Gonadotropin/CGA Protein, Human, Recombinant (mFc)

HCG,GPHa,CG-ALPHA,glycoprotein hormones, alpha polypeptide,g...

Human HEK293 Cells
Chorionic Gonadotropin/CGA Protein, Human, Recombinant (mFc) is expressed in HEK293 mammalian cells with mFc tag. The predicted molecular weight is 36.6 kDa and the accession number is P01215.
TMPY-06840 Human respiratory syncytial virus (RSV) (A2) Prefusion glycoprotein F/RSV-preF Protein

HRSVgp8,F Protein

RSV CHO Cells
Human respiratory syncytial virus (RSV) (A2) Prefusion glycoprotein F/RSV-preF Protein is expressed in CHO mammalian cells. The predicted molecular weight is 54.5 kDa.
TMPY-05690 Human mastadenovirus B (HAdV-B) encapsidation protein IVa2 Protein (His)

HAdV-B Baculovirus Insect Cells
Human mastadenovirus B (HAdV-B) encapsidation protein IVa2 Protein (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 52.06 kDa and the accession number is YP_002213830.1.
TMPY-06422 SARS-CoV-2 Spike S1 NTD Protein (T19R & T95I & G142D & 156-157 deletion & R158G, His)

SARS-CoV-2 HEK293 Cells
SARS-CoV-2 Spike S1 NTD Protein (T19R & T95I & G142D & 156-157 deletion & R158G, His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 34.10 kDa and the accession number is A0A6G7K2L4.
TMPY-06392 SARS-CoV-2 Spike S1+S2 Protein (Q52R & A67V & 69-70 deletion & Y144 deletion & E484K & D614G & Q677H & F888L, His)

SARS-CoV-2 Baculovirus Insect Cells
SARS-CoV-2 Spike S1+S2 Protein (Q52R & A67V & 69-70 deletion & Y144 deletion & E484K & D614G & Q677H & F888L, His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 133.96 kDa and the accession number is A0A6G7K2L4.
TMPY-06305 SARS-CoV-2 Spike S1 Protein (Q52 & A67V & 69-70 deletion & 144 deletion & E484K & D614G & Q677H, His)

SARS-CoV-2 HEK293 Cells
SARS-CoV-2 Spike S1 Protein (Q52 & A67V & 69-70 deletion & 144 deletion & E484K & D614G & Q677H, His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 76.07 kDa and the accession number is A0A6G7K2L4.
TMPY-06368 Human respiratory syncytial virus (RSV) (A, strain Long) Fusion glycoprotein F0/RSV-F Protein (His)

F Protein,HRSVgp8

RSV Baculovirus Insect Cells
Human respiratory syncytial virus (RSV) (A, strain Long) Fusion glycoprotein F0/RSV-F Protein (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 56.92 kDa and the accession number is P12568.
TMPH-03268 Coagulation factor XI Protein, Rat, Recombinant (His & Myc)

Coagulation factor XI,F11

Rat E. coli
Coagulation factor XI Protein, Rat, Recombinant (His & Myc) is expressed in E. coli.
THMH-00001 CD133/PROM1 Recombinant,Human(Yeast expression,His)

TMPH-00480 Anionic trypsin Protein, Canine, Recombinant (His & SUMO)

Anionic trypsin,EC:3.4.21.4

Canine E. coli
Anionic trypsin Protein, Canine, Recombinant (His & SUMO) is expressed in E. coli.
TMPH-02401 rplL Protein, Legionella pneumophila, Recombinant (His & Myc)

Large ribosomal subunit protein bL12,50S ribosomal protein L...

Legionella pneumophila E. coli
Forms part of the ribosomal stalk which helps the ribosome interact with GTP-bound translation factors. Is thus essential for accurate translation. rplL Protein, Legionella pneumophila, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 20.4 kDa and the accession number is Q5ZYQ1.
TMPH-01798 Nucleolar transcription factor 1 Protein, Human, Recombinant (Cell-Free, His & SUMO)

Nucleolar transcription factor 1,Upstream-binding f...

Human E. coli
Recognizes the ribosomal RNA gene promoter and activates transcription mediated by RNA polymerase I through cooperative interactions with the transcription factor SL1/TIF-IB complex. It binds specifically to the upstream control element. Nucleolar transcription factor 1 Protein, Human, Recombinant (Cell-Free, His & SUMO) is expressed in E. coli expression system with N-10xHis-SUMO tag. The predicted molecular weight is 107.9 kDa and the accession number is P17480.
TMPH-00689 Propionate kinase Protein, E. coli O6:H1, Recombinant (His & Myc)

tdcD,Propionate kinase

E. coli E. coli
Catalyzes the conversion of propionyl phosphate and ADP to propionate and ATP. Propionate kinase Protein, E. coli O6:H1, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 50.4 kDa and the accession number is P59244.
TMPH-00399 RPS13 Protein, Ciona intestinalis, Recombinant (His & Myc)

40S ribosomal protein S13,RPS13,Small ribosomal subunit prot...

Ciona intestinalis E. coli
RPS13 Protein, Ciona intestinalis, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 23.9 kDa and the accession number is Q8I7D6.
TMPH-02452 Measles virus (MeV) (strain Leningrad-16) Fusion glycoprotein F0 (Avi & His)

F,Fusion glycoprotein F0

MeV E. coli
Measles virus (MeV) (strain Leningrad-16) Fusion glycoprotein F0 (Avi & His) is expressed in E. coli expression system with N-10xHis and C-Avi tag. The predicted molecular weight is 61.8 kDa and the accession number is P69356.
TMPH-02399 Pal Protein, Legionella pneumophila, Recombinant (E. coli, His)

pal,19 kDa surface antigen,Peptidoglycan-associated lipoprot...

Legionella pneumophila E. coli
Part of the Tol-Pal system, which plays a role in outer membrane invagination during cell division and is important for maintaining outer membrane integrity. Very strongly associated with the peptidoglycan.
TMPH-01799 Nucleolar transcription factor 1 Protein, Human, Recombinant (E. coli, His & SUMO)

Nucleolar transcription factor 1,Autoantigen NOR-90...

Human E. coli
Recognizes the ribosomal RNA gene promoter and activates transcription mediated by RNA polymerase I through cooperative interactions with the transcription factor SL1/TIF-IB complex. It binds specifically to the upstream control element. Nucleolar transcription factor 1 Protein, Human, Recombinant (E. coli, His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 95.2 kDa and the accession number is P17480.
TMPY-06085 SARS-CoV-2 Spike S1 Protein (HV69-70 deletion & Y453F & D614G, His)

SARS-CoV-2 HEK293 Cells
SARS-CoV-2 Spike S1 Protein (HV69-70 deletion & Y453F & D614G, His) is expressed in HEK293 mammalian cells. The predicted molecular weight is 76.2 kDa and the accession number is A0A6G7K2L4.
TMPY-05355 Coagulation factor IX/F9 Protein, Human, Recombinant (hFc)

P19,Coagulation factor 9,HEMB,FIX,THPH8,Coagulat

Human HEK293 Cells
Coagulation factor IX/F9 Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 75.5 kDa and the accession number is P00740-1.
TMPY-00323 Hepatitis C virus (HCV-1a) NS3 protease/helicase immunodominant region Protein (aa 1356-1459, GST)

NS3

HCV E. coli
HCV NS3 displays three enzymatic activities: serine protease, NTPase, and RNA helicase. HCV NS3 serine protease, in association with NS4A, is responsible for the cleavages of NS3-NS4A, NS4A-NS4B, NS4B-NS5A, and NS5A-NS5B. HCV NS3 RNA helicase binds to RNA and unwinds dsRNA in the 3' to 5' direction, and likely RNA stable secondary structure in the template strand (By similarity). Cleaves and inhibits the host antiviral protein MAVS. NS3/NS4A complex also prevents phosphorylation of human IRF3, t...
TMPY-06406 SARS-CoV-2 Spike S1+S2 Protein (G75V & T76I & R246N & 247, 253 deletion & L452Q & F490S & D614G & T859N, His)

SARS-CoV-2 Baculovirus Insect Cells
SARS-CoV-2 Spike S1+S2 Protein (G75V & T76I & R246N & 247, 253 deletion & L452Q & F490S & D614G & T859N, His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 134.11 kDa and the accession number is A0A6G7K2L4.
TMPY-06444 SARS-CoV-2 Spike S1 Protein (T19R & T95I & E156G & 157-158 deletion & L452R & T478K & D614G & P681R, His)

SARS-CoV-2 HEK293 Cells
SARS-CoV-2 Spike S1 Protein (T19R & T95I & E156G & 157-158 deletion & L452R & T478K & D614G & P681R, His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 76.23 kDa and the accession number is YP_009724390.1.
TMPY-06122 SARS-CoV-2 Spike S1 NTD Protein (L18F & D80A & D215G & LAL242-244 deletion & R246I, His)

SARS-CoV-2 HEK293 Cells
SARS-CoV-2 Spike S1 NTD Protein (L18F & D80A & D215G & LAL242-244 deletion & R246I, His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 33.9 kDa and the accession number is A0A6G7K2L4.
TMPY-06267 SARS-CoV-2 Spike S1 Protein (157-158 deletion & T19R & G142D & E156G & L452R & T478K & D614G & P681R, His & Avi), Biotinylated

SARS-CoV-2 HEK293 Cells
SARS-CoV-2 Spike S1 Protein (157-158 deletion & T19R & G142D & E156G & L452R & T478K & D614G & P681R, His & Avi), Biotinylated is expressed in HEK293 mammalian cells with His and Avi tag. The predicted molecular weight is 78.09 kDa and the accession number is A0A6G7K2L4.
TMPK-00775 PRNP/Prion Protein, Mouse, Recombinant (hFc)

Major prion protein,PrP,ALTPRP,PRIP,PRNP

Mouse HEK293 Cells
Prion protein gene (PRNP) variants determine the susceptibility of humans, sheep and mice to prion diseases, whereas polymorphisms in the open reading frame (ORF) of bovine PRNP seem to be unrelated to the incidence of bovine spongiform encephalopathy (BSE). According to the latest reports, the genetic susceptibility of cattle to BSE is associated with polymorphisms ofthe regulatory region of the PRNP gene and the level ofits expression.
TMPJ-00707 Coagulation factor X/F10 Protein, Mouse, Recombinant (His)

Stuart factor,Coagulation factor X,F10

Mouse HEK293 Cells
Mouse coagulation factor X / F10 a member of the peptidase S1 family. The mature F10 is composed mostly of two EGF-like domains, one Gla gamma-carboxy-glutamate domain and one peptidase S1 domain. Factor Xa is a vitamin K-dependent plasma protease that converts prothrombin to thrombin in the presence of factor Va, calcium and phospholipid during blood clotting. The two chains of F10 are formed from a single-chain precursor by the excision of two Arg residues. A single-chain precursor is initiall...
TMPH-00754 Capsid decoration Protein, Escherichia phage lambda, Recombinant (GST)

Gene product D,Auxiliary protein D,Major capsid protein D,gp...

Escherichia phage lambda E. coli
Stabilizes the expansion of the capsid head shell after genome packaging. The packaging of viral genome in the procapsid triggers a dramatic reconfiguration of the capsid shell, expanding from roughly 50nm to 60nm while the capsid thickness decreases. 415 capsid decoration protein molecules cooperatively bind the expanded capsid, thereby stabilizing the mature capsid shell. Capsid decoration Protein, Escherichia phage lambda, Recombinant (GST) is expressed in E. coli expression system with N-GST...
TMPH-00484 Cationic trypsin Protein, Canine, Recombinant (His & SUMO)

TRP1,Serine protease 1,PRSS1,TRY1,Pretrypsinogen I,Anion...

Canine E. coli
Cationic trypsin Protein, Canine, Recombinant (His & SUMO) is expressed in E. coli.
TMPH-01669 Metallothionein-3/MT3 Protein, Human, Recombinant (His & SUMO)

Metallothionein-III,Metallothionein-3,GIFB...

Human E. coli
Binds heavy metals. Contains three zinc and three copper atoms per polypeptide chain and only a negligible amount of cadmium. Inhibits survival and neurite formation of cortical neurons in vitro.
TMPY-06714 Coagulation factor IX/F9 Protein, Cynomolgus, Recombinant (His)

coagulation factor IX

Cynomolgus HEK293 Cells
Coagulation factor IX/F9 Protein, Cynomolgus, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 50.17 kDa and the accession number is A0A8J8XCV8.
TMPY-06288 SARS-CoV-2 Spike S1+S2 Protein (157-158 deletion & T19R & G142D & E156G & L452R & T478K & D614G & P681R & D950N, His & Avi), Biotinylated

SARS-CoV-2 Baculovirus Insect Cells
SARS-CoV-2 Spike S1+S2 Protein (157-158 deletion & T19R & G142D & E156G & L452R & T478K & D614G & P681R & D950N, His & Avi), Biotinylated is expressed in Baculovirus insect cells with His and Avi tag. The predicted molecular weight is 136.01 kDa and the accession number is A0A6G7K2L4.
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重组蛋白

PIEZO1 Protein, Human, Recombinant (His & Myc)
Cat.No: TMPH-01863
Species: Human
Expression System: E. coli
KCNE2 Protein, Human, Recombinant (His)
Cat.No: TMPH-01891
Species: Human
Expression System: E. coli
FXYD3 Protein, Human, Recombinant (His & SUMO)
Cat.No: TMPH-01358
Species: Human
Expression System: E. coli
Human respiratory syncytial virus (RSV) Fusion protein/RSV-F (Strain RSS-2) Protein (His)
Cat.No: TMPY-03236
Species: RSV
Expression System: Baculovirus Insect Cells
Coagulation factor IX/F9 Protein, Human, Recombinant (His)
Cat.No: TMPY-02215
Species: Human
Expression System: HEK293 Cells
Influenza A H1N1 (A/Brevig Mission/1/1918) Hemagglutinin Protein (His)
Cat.No: TMPY-01193
Species: H1N1
Expression System: HEK293 Cells
Human respiratory syncytial virus (RSV) (A2) Fusion glycoprotein/RSV-F Protein (His)
Cat.No: TMPY-01078
Species: RSV
Expression System: Baculovirus Insect Cells
Influenza A H1N1 (A/Brevig Mission/1/1918) Nucleoprotein/NP Protein (His)
Cat.No: TMPY-04274
Species: H1N1
Expression System: Baculovirus Insect Cells
Coagulation factor X/F10 Protein, Human, Recombinant (His)
Cat.No: TMPY-01101
Species: Human
Expression System: Baculovirus Insect Cells
Coagulation factor XI/F11 Protein, Human, Recombinant (His)
Cat.No: TMPY-01104
Species: Human
Expression System: HEK293 Cells
Coagulation factor XIII B/F13B Protein, Human, Recombinant (His)
Cat.No: TMPY-02185
Species: Human
Expression System: HEK293 Cells
Human respiratory syncytial virus (RSV) Fusion Protein (aa 1-525, His)
Cat.No: TMPY-05688
Species: RSV
Expression System: Baculovirus Insect Cells
Siglec-2/CD22 Protein, Human, Recombinant (His, Solution)
Cat.No: TMPY-05566
Species: Human
Expression System: HEK293 Cells
Coagulation Factor II Protein, Mouse, Recombinant (His)
Cat.No: TMPY-01791
Species: Mouse
Expression System: HEK293 Cells
SARS-CoV-2 Spike S1+S2 Protein (L18F & D80A & D215G & LAL242-244 deletion & R246I & K417N & E484K & N501Y & D614G & A701V, His), Biotinylated
Cat.No: TMPY-06171
Species: SARS-CoV-2
Expression System: Baculovirus Insect Cells
SARS-CoV-2 Spike S1 Protein (T19R & T95I & G142D & Y145H & E156G & 157-158 deletion & A222V & L452R & T478K & D614G & P681R, His)
Cat.No: TMPY-06443
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS-CoV-2 Spike S1 Protein (HV69-70 deletion & N501Y & D614G, His)
Cat.No: TMPY-06082
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS-CoV-2 Spike S1 Protein (L18F & D80A & D215G & LAL242-244 deletion & R246I & K417N & E484K & N501Y & D614G, His)
Cat.No: TMPY-06129
Species: SARS-CoV-2
Expression System: HEK293 Cells
Chorionic Gonadotropin/CGA Protein, Human, Recombinant (His)
Cat.No: TMPY-00647
Species: Human
Expression System: HEK293 Cells
Chorionic Gonadotropin/CGA Protein, Human, Recombinant (mFc)
Cat.No: TMPY-02923
Species: Human
Expression System: HEK293 Cells
Human respiratory syncytial virus (RSV) (A2) Prefusion glycoprotein F/RSV-preF Protein
Cat.No: TMPY-06840
Species: RSV
Expression System: CHO Cells
Human mastadenovirus B (HAdV-B) encapsidation protein IVa2 Protein (His)
Cat.No: TMPY-05690
Species: HAdV-B
Expression System: Baculovirus Insect Cells
SARS-CoV-2 Spike S1 NTD Protein (T19R & T95I & G142D & 156-157 deletion & R158G, His)
Cat.No: TMPY-06422
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS-CoV-2 Spike S1+S2 Protein (Q52R & A67V & 69-70 deletion & Y144 deletion & E484K & D614G & Q677H & F888L, His)
Cat.No: TMPY-06392
Species: SARS-CoV-2
Expression System: Baculovirus Insect Cells
SARS-CoV-2 Spike S1 Protein (Q52 & A67V & 69-70 deletion & 144 deletion & E484K & D614G & Q677H, His)
Cat.No: TMPY-06305
Species: SARS-CoV-2
Expression System: HEK293 Cells
Human respiratory syncytial virus (RSV) (A, strain Long) Fusion glycoprotein F0/RSV-F Protein (His)
Cat.No: TMPY-06368
Species: RSV
Expression System: Baculovirus Insect Cells
Coagulation factor XI Protein, Rat, Recombinant (His & Myc)
Cat.No: TMPH-03268
Species: Rat
Expression System: E. coli
CD133/PROM1 Recombinant,Human(Yeast expression,His)
Cat.No: THMH-00001
Species:
Expression System:
Anionic trypsin Protein, Canine, Recombinant (His & SUMO)
Cat.No: TMPH-00480
Species: Canine
Expression System: E. coli
rplL Protein, Legionella pneumophila, Recombinant (His & Myc)
Cat.No: TMPH-02401
Species: Legionella pneumophila
Expression System: E. coli
Nucleolar transcription factor 1 Protein, Human, Recombinant (Cell-Free, His & SUMO)
Cat.No: TMPH-01798
Species: Human
Expression System: E. coli
Propionate kinase Protein, E. coli O6:H1, Recombinant (His & Myc)
Cat.No: TMPH-00689
Species: E. coli
Expression System: E. coli
RPS13 Protein, Ciona intestinalis, Recombinant (His & Myc)
Cat.No: TMPH-00399
Species: Ciona intestinalis
Expression System: E. coli
Measles virus (MeV) (strain Leningrad-16) Fusion glycoprotein F0 (Avi & His)
Cat.No: TMPH-02452
Species: MeV
Expression System: E. coli
Pal Protein, Legionella pneumophila, Recombinant (E. coli, His)
Cat.No: TMPH-02399
Species: Legionella pneumophila
Expression System: E. coli
Nucleolar transcription factor 1 Protein, Human, Recombinant (E. coli, His & SUMO)
Cat.No: TMPH-01799
Species: Human
Expression System: E. coli
SARS-CoV-2 Spike S1 Protein (HV69-70 deletion & Y453F & D614G, His)
Cat.No: TMPY-06085
Species: SARS-CoV-2
Expression System: HEK293 Cells
Coagulation factor IX/F9 Protein, Human, Recombinant (hFc)
Cat.No: TMPY-05355
Species: Human
Expression System: HEK293 Cells
Hepatitis C virus (HCV-1a) NS3 protease/helicase immunodominant region Protein (aa 1356-1459, GST)
Cat.No: TMPY-00323
Species: HCV
Expression System: E. coli
SARS-CoV-2 Spike S1+S2 Protein (G75V & T76I & R246N & 247, 253 deletion & L452Q & F490S & D614G & T859N, His)
Cat.No: TMPY-06406
Species: SARS-CoV-2
Expression System: Baculovirus Insect Cells
SARS-CoV-2 Spike S1 Protein (T19R & T95I & E156G & 157-158 deletion & L452R & T478K & D614G & P681R, His)
Cat.No: TMPY-06444
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS-CoV-2 Spike S1 NTD Protein (L18F & D80A & D215G & LAL242-244 deletion & R246I, His)
Cat.No: TMPY-06122
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS-CoV-2 Spike S1 Protein (157-158 deletion & T19R & G142D & E156G & L452R & T478K & D614G & P681R, His & Avi), Biotinylated
Cat.No: TMPY-06267
Species: SARS-CoV-2
Expression System: HEK293 Cells
PRNP/Prion Protein, Mouse, Recombinant (hFc)
Cat.No: TMPK-00775
Species: Mouse
Expression System: HEK293 Cells
Coagulation factor X/F10 Protein, Mouse, Recombinant (His)
Cat.No: TMPJ-00707
Species: Mouse
Expression System: HEK293 Cells
Capsid decoration Protein, Escherichia phage lambda, Recombinant (GST)
Cat.No: TMPH-00754
Species: Escherichia phage lambda
Expression System: E. coli
Cationic trypsin Protein, Canine, Recombinant (His & SUMO)
Cat.No: TMPH-00484
Species: Canine
Expression System: E. coli
Metallothionein-3/MT3 Protein, Human, Recombinant (His & SUMO)
Cat.No: TMPH-01669
Species: Human
Expression System: E. coli
Coagulation factor IX/F9 Protein, Cynomolgus, Recombinant (His)
Cat.No: TMPY-06714
Species: Cynomolgus
Expression System: HEK293 Cells
SARS-CoV-2 Spike S1+S2 Protein (157-158 deletion & T19R & G142D & E156G & L452R & T478K & D614G & P681R & D950N, His & Avi), Biotinylated
Cat.No: TMPY-06288
Species: SARS-CoV-2
Expression System: Baculovirus Insect Cells
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Cat. No. Product Name Target Signaling Pathways
TMIH-0475 rac threo-Dihydro Bupropion-d9 Hydrochloride

rac threo-Dihydro Bupropion-d9 Hydrochloride 是 rac threo-Dihydro Bupropion Hydrochloride 的氘代化合物。rac threo-Dihydro Bupropion Hydrochloride 的 CAS 号为 1396889-62-5。
TMIH-0051 3-phenylpropionic acid-d5

3-phenylpropionic acid-d5 是 3-phenylpropionic acid 的氘代化合物。
TMIJ-0084 Propionyl carnitine-d3 HCl

Propionyl carnitine-d3 HCl 是 Propionyl carnitine HCl 的氘代化合物。
TMIJ-0169 erythro-Hydro Bupropion-d9 HCl(enantiomer)

erythro-Hydro Bupropion-d9 HCl(enantiomer) 是 erythro-Hydro Bupropion HCl 的氘代化合物。
TMIJ-0208 Beclomethasone Dipropionate-d6

Beclomethasone Dipropionate-d6 是 Beclomethasone Dipropionate 的氘代化合物。Beclomethasone Dipropionate 的 CAS 号为 5534-09-8。Betamethasone dipropionate是具有口服活性的糖皮质激素,具有抗炎和免疫抑制作用。它是Betamethasone 的前体药物,Betamethasone 是 LPS 诱导的炎症及 MMP 释放的抑制剂。
TMID-0142 4-Androsten-11β-ol-3,17-dione-d7

4-Androsten-11β-ol-3,17-dione-d7 是 4-Androsten-11β-ol-3,17-dione 的氘代化合物。4-Androsten-11β-ol-3,17-dione 的 CAS 号为 382-44-5。11-Beta-hydroxyandrostenedione 是主要存在于肾上腺的类固醇,也是 11β-羟基类固醇脱氢酶同工酶抑制剂。随着 4-androstenedione 的提高,通过测量血浆中的11-Beta-hydroxyandrostenedione,能够区分高雄激素血症的肾上腺或卵巢起源。
TMIJ-0052 Propionicacid-d5

Propionicacid-d5 是 Propionicacid 的氘代化合物。Propionicacid 的 CAS 号为 79-09-4。Propionic acid 被广泛用作食品中的抗真菌剂。它以低水平天然存在于乳制品中,并与其他短链脂肪酸 (SCFA) 一起普遍存在于人类和其他哺乳动物的胃肠道中,作为微生物消化碳水化合物的最终产物。在动物体内有显着的生理活性。
TMIJ-0498 Fluticasone Propionate-d5

Fluticasone Propionate-d5 是 Fluticasone Propionate 的氘代化合物。Fluticasone Propionate 的 CAS 号为 80474-14-2。Fluticasone propionate 是一种选择性糖皮质激素受体激动剂,是一种局部抗炎激素,绝对亲和力KD为 0.5 nM。具有抗病毒活性。
TMIJ-0456 Malathion-d7

Malathion-d7 是 Malathion 的氘代化合物。Malathion 的 CAS 号为 121-75-5。Malathion 是一种杀虫剂,是一种有机磷酸酯的副交感神经药物,不可逆地与胆碱酯酶结合,具有相对较低的人体毒性。
T71893 Clobetasol Propionate-d5

Clobetasol propionate-d5 is intended for use as an internal standard for the quantification of clobetasol propionate by GC- or LC-MS. Clobetasol propionate is a corticosteroid. It binds to glucocorticoid receptors in a cell-free assay and inhibits proliferation of primary human skin fibroblasts when used at a concentration of 5 µg/ml. Topical administration of clobetasol propionate reduces croton oil-induced ear edema in mice. Formulations containing clobetasol propionate have been used in the t...
TMIJ-0054 Propionic-2,2-d2 acid

Propionic-2,2-d2 acid 是 Propionic acid 的氘代化合物。Propionic acid 的 CAS 号为 79-09-4。Propionic acid 被广泛用作食品中的抗真菌剂。它以低水平天然存在于乳制品中,并与其他短链脂肪酸 (SCFA) 一起普遍存在于人类和其他哺乳动物的胃肠道中,作为微生物消化碳水化合物的最终产物。在动物体内有显着的生理活性。
TMID-0148 Nandrolone 17-propionate-d3

Nandrolone 17-propionate-d3 是 Nandrolone 17-propionate 的氘代化合物。Nandrolone 17-propionate 的 CAS 号为 7207-92-3。Nandrolone propionate 是合成代谢类固醇,主要由雄激素和保氮剂组成,具有作用时间相对较长的特点。
TMIH-0040 3-(4-Hydroxyphenyl)propionic acid-d4

HPPA-d4

3-(4-Hydroxyphenyl)propionic acid-d4 是 3-(4-Hydroxyphenyl)propionic acid 的氘代化合物。3-(4-Hydroxyphenyl)propionic acid 的 CAS 号为 501-97-3。Desaminotyrosine 是一种与微生物相关的代谢物,通过增强 I 型干扰素信号传导来预防流感。
TMIH-0330 Mesotrione-d3

Mesotrione-d3 是 Mesotrione 的氘代化合物。Mesotrione 的 CAS 号为 104206-82-8。Mesotrione 是一种苯甲酰环己二酮类除草剂,是一种竞争性羟基苯基丙酮酸双加氧酶酶抑制剂。它对玉米作物具有选择性,它在易感作物中代谢速度快,耐受性较高。
TMIH-0562 Testosterone propionate-d3

Testosterone propionate-d3 是 Testosterone propionate 的氘代化合物。
TMIH-0129 Bupropion Morpholinol-d8

Bupropion Morpholinol-d8 是 Bupropion Morpholinol 的氘代化合物。
TMIH-0089 Androstenedione-d7

Androstenedione-d7 是 Androstenedione 的氘代化合物。Androstenedione 的 CAS 号为 560-62-3。9-hydroxy-4-androstene-3,17-dione 是一种类固醇激素,具有抗肿瘤活性,可以抑制多种癌症细胞的生长,包括乳腺癌、前列腺癌和肺癌细胞。
TMIH-0367 Nandrolone propionat-d3

Nandrolone propionat-d3 是 Nandrolone propionat 的氘代化合物。
TMIJ-0165 Glutathione-(glyucine-13C2-15N) Trifluoroacetate

Glutathione-(glyucine-13C2-15N) Trifluoroacetate 是 Glutathione Trifluoroacetate 的 13C 和 15 N 的标记化合物。
TMIJ-0098 threo-Hydrobupropion-d9 HCl(enantiomer)

threo-Hydrobupropion-d9 HCl(enantiomer) 是 threo-Hydrobupropion HCl 的氘代化合物。
TMIJ-0451 Malathion-d10

Malathion-d10 是 Malathion 的氘代化合物。Malathion 的 CAS 号为 121-75-5。Malathion 是一种杀虫剂,是一种有机磷酸酯的副交感神经药物,不可逆地与胆碱酯酶结合,具有相对较低的人体毒性。
T12442 Phenindione D5

Rectadione D5,苯茚二酮 D5

Others Others
Phenindione D5 is deuterium labeled Phenindione, which functions as a Vitamin K antagonist.
TMIJ-0053 2-Methylpropionic-d7 acid

2-Methylpropionic-d7 acid 是 2-Methylpropionic acid 的氘代化合物。2-Methylpropionic acid 的 CAS 号为 79-31-2。Isobutyric acid 是一种羧酸或短链脂肪酸,具有特征性的汗味。通过微生物(肠道)代谢产生少量异丁酸。在某些食物或发酵饮料中也可能发现少量。
TMIJ-0204 Betamethasone-d10 Dipropionate

Betamethasone-d10 Dipropionate 是 Betamethasone Dipropionate 的氘代化合物。Betamethasone Dipropionate 的 CAS 号为 5593-20-4。Betamethasone dipropionate 是糖皮质激素类固醇,具有免疫抑制、抗炎作用。
TMIJ-0209 Beclomethasone-17-Monopropionate-d3

Beclomethasone-17-Monopropionate-d3 是 Beclomethasone-17-Monopropionate 的氘代化合物。Beclomethasone-17-Monopropionate 的 CAS 号为 5534-18-9。
TMIJ-0481 Fenitrothion-d6 (O,O-dimethyl-d6)

Fenitrothion-d6 (O,O-dimethyl-d6) 是 Fenitrothion 的氘代化合物。Fenitrothion 的 CAS 号为 122-14-5。
T71303 Flufenamic Acid-d4

Flufenamic acid-d4 is intended for use as an internal standard for the quantification of flufenamic acid by GC- or LC-MS. Flufenamic acid is a non-steroidal anti-inflammatory drug (NSAID) and COX inhibitor (IC50s = 3 and 9.3 µM for human COX-1 and COX-2, respectively). Flufenamic acid inhibits TNF-α-induced increases in COX-2 levels and NF-κB activation in HT-29 colon cancer cells in a concentration-dependent manner. It inhibits calcium influx induced by fMLP or A23187 in human polymorphonuclear...

同位素标记化合物

rac threo-Dihydro Bupropion-d9 Hydrochloride
Cat.No: TMIH-0475
Synonym:
Target:
3-phenylpropionic acid-d5
Cat.No: TMIH-0051
Synonym:
Target:
Propionyl carnitine-d3 HCl
Cat.No: TMIJ-0084
Synonym:
Target:
erythro-Hydro Bupropion-d9 HCl(enantiomer)
Cat.No: TMIJ-0169
Synonym:
Target:
Beclomethasone Dipropionate-d6
Cat.No: TMIJ-0208
Synonym:
Target:
4-Androsten-11β-ol-3,17-dione-d7
Cat.No: TMID-0142
Synonym:
Target:
Propionicacid-d5
Cat.No: TMIJ-0052
Synonym:
Target:
Fluticasone Propionate-d5
Cat.No: TMIJ-0498
Synonym:
Target:
Malathion-d7
Cat.No: TMIJ-0456
Synonym:
Target:
Clobetasol Propionate-d5
Cat.No: T71893
Synonym:
Target:
Propionic-2,2-d2 acid
Cat.No: TMIJ-0054
Synonym:
Target:
Nandrolone 17-propionate-d3
Cat.No: TMID-0148
Synonym:
Target:
3-(4-Hydroxyphenyl)propionic acid-d4
Cat.No: TMIH-0040
Synonym: HPPA-d4
Target:
Mesotrione-d3
Cat.No: TMIH-0330
Synonym:
Target:
Testosterone propionate-d3
Cat.No: TMIH-0562
Synonym:
Target:
Bupropion Morpholinol-d8
Cat.No: TMIH-0129
Synonym:
Target:
Androstenedione-d7
Cat.No: TMIH-0089
Synonym:
Target:
Nandrolone propionat-d3
Cat.No: TMIH-0367
Synonym:
Target:
Glutathione-(glyucine-13C2-15N) Trifluoroacetate
Cat.No: TMIJ-0165
Synonym:
Target:
threo-Hydrobupropion-d9 HCl(enantiomer)
Cat.No: TMIJ-0098
Synonym:
Target:
Malathion-d10
Cat.No: TMIJ-0451
Synonym:
Target:
Phenindione D5
Cat.No: T12442
Synonym: Rectadione D5,苯茚二酮 D5
Target: Others
2-Methylpropionic-d7 acid
Cat.No: TMIJ-0053
Synonym:
Target:
Betamethasone-d10 Dipropionate
Cat.No: TMIJ-0204
Synonym:
Target:
Beclomethasone-17-Monopropionate-d3
Cat.No: TMIJ-0209
Synonym:
Target:
Fenitrothion-d6 (O,O-dimethyl-d6)
Cat.No: TMIJ-0481
Synonym:
Target:
Flufenamic Acid-d4
Cat.No: T71303
Synonym:
Target:
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