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TargetMol | Compound Library

神经信号分子库现货

Neuronal Signaling Compound Library

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产品编号 L2600

神经元之间和神经元内部的通信对于神经系统的所有功能至关重要,无论是从发育到衰老,还是从健康到疾病。在过去十年中,我们对神经系统内分子、细胞和系统信号通路的认识取得了巨大进步,在信号通路研究方面取得了重大突破,这些神经信号通路是神经发生、成瘾、自闭症以及情绪障碍的病理生理学和治疗基础。例如:G 蛋白偶联受体(GPCR),包括5-HT 受体、组胺受体、阿片受体等,是研究较多的神经元信号传导途径,GPCR 功能障碍会引起多种神经疾病;Notch 信号途径调节神经干细胞增殖、存活、自我更新和分化,Notch 信号传导异常参与中风、阿尔茨海默病和CNS 肿瘤等疾病中发生的病理过程。因此靶向神经元信号传导,可以用来治疗多种不同CNS 疾病。

TargetMol 神经信号分子库包含2771 种神经信号相关的小分子化合物,主要用于神经系统类疾病的药物研发,可用于高通量、高内涵筛选。

TargetMol 的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
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产品编号 L2600

神经信号分子库

规格

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品描述 产品描述

  • 2771种CNS相关的生物活性小分子化合物的特有集合,用于高通量、高内涵筛选;
  • 靶点包括5-HT receptor、AChR、Histamine receptor、dopamine receptor、Opiod receptor等;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

包装和储存 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
  • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。

包装和储存 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。

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Library Customization | TargetMol 化合物库组成

5-HT Receptor
AChR
COX
Adrenergic Receptor
Dopamine Receptor
Histamine Receptor
Calcium Channel
GABA Receptor
GluR
TRP/TRPV Channel
Cholinesterase (ChE)
Apoptosis
Autophagy
Adenosine Receptor
Endogenous Metabolite
NMDAR
iGluR
Opioid Receptor
MAO
Beta Amyloid
Antibacterial
NF-κB
Potassium Channel
P-gp
Gamma-secretase
Monoamine Oxidase
Cannabinoid Receptor
P2X Receptor
Serotonin Transporter
Norepinephrine
Sodium Channel
Parasite
CaMK
FAAH
Cytochromes P450
Neurokinin receptor
Reactive Oxygen Species
BACE
Neuropeptide Y Receptor
NO Synthase
TNF
P2Y Receptor
PDE
Antibiotic
GPCR
Sigma receptor
Lipoxygenase
OX Receptor
Antioxidant
Influenza Virus
HIV Protease
NOS
PPAR
Beta-Secretase
IL Receptor
Prostaglandin Receptor
Antifungal
ERK
Ferroptosis
ROS
Imidazoline Receptor
Melatonin Receptor
Phospholipase
Akt
Caspase
MT Receptor
Virus Protease
Adenylyl Cyclase
Drug Metabolite
EGFR
GlyT
Mitophagy
p38 MAPK
PGE Synthase
DNA/RNA Synthesis
STAT
AAK1
AMPK
Bcl-2 Family
Carbonic Anhydrase
Dehydrogenase
Estrogen/progestogen Receptor
Glucocorticoid Receptor
HCV Protease
Interleukin
Melanocortin Receptor
PKA
PKC
SARS-CoV
Transferase
Wnt/beta-catenin
CGRP Receptor
Chloride channel
GSK-3
HSV
IκB/IKK
MMP
Monoamine Transporter
MRP
Phosphatase
ABC Transporter
ATPase
Cholecystokinin Receptor
Glutathione Peroxidase
Histone Demethylase
Histone Methyltransferase
PI3K
Serine/threonin kinase
TGF-beta/Smad
TLR
Tyrosinase
Acyltransferase
Antifection
Anti-infection
cAMP
CCR
CDK
Epoxide Hydrolase
HDAC
HIF/HIF Prolyl-Hydroxylase
Immunology/Inflammation related
JNK
MEK
Melanin-concentrating Hormone Receptor (MCHR)
Mitochondrial Metabolism
mTOR
Na+/Ca2+ Exchanger
NADPH
Neurotensin Receptor
PAFR
PARP
RAAS
Reductase
Src
Topoisomerase
transporter
VEGFR
Advanced Glycation End Products
Amino Acids and Derivatives
Androgen Receptor
Arrestin
ATM/ATR
Aurora Kinase
Bcr-Abl
BCRP
DNA
DNA Methyltransferase
DYRK
Epigenetic Reader Domain
Estrogen Receptor/ERR
Gap Junction Protein
GluCls
Glucosidase
GST
HBV
Hydroxylase
IAP
IFNAR
IGF-1R
JAK
LDL
Leukotriene Receptor
Lipase
Microtubule Associated
NOD
Nrf2
p53
Platelet aggregation
Progesterone Receptor
ROCK
RSV
Transaminase
UGT
FOXO3
ACK1
Adenosine Deaminase
Adiponectin Receptor
AhR
Aminopeptidase
Angiotensin-converting Enzyme (ACE)
Anion Exchanger
Annexin A
Antifolate
Antiviral
Aryl Hydrocarbon Receptor
Bombesin Receptor
Casein Kinase
Cell Cycle Arrest
CFTR
c-Met/HGFR
CRISPR/Cas9
Cysteine Protease
FAK
Fatty Acid Synthase
FGFR
FLAP
FLT
Free radical scavengers
FXR
Glucagon Receptor
Glutaminyl Cyclase
gp120/CD4
GPCR19
GTPase
HCN Channel
HMG-CoA Reductase
HSP
Indoleamine 2,3-Dioxygenase (IDO)
Integrin
LIM Kinase
LPL Receptor
LTR
Lysosomal Autophagy
MAGL
MAPK
MicroRNA
Monocarboxylate transporter
Myosin
N-Acetylglucosaminyltransferase
NADPH-oxidase
Neuropeptide W
NMU2R
NOD-like Receptor (NLR)
Nucleoside Antimetabolite/Analog
PAK
Protease-activated Receptor
Proteasome
Raf
Retinoid Receptor
Reverse Transcriptase
ROR
ROS Kinase
S1P Receptor
Somatostatin
Stearoyl-CoA Desaturase (SCD)
STING
Syk
Thrombin