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TargetMol | Compound Library

神经信号分子库现货

Neuronal Signaling Compound Library

产品编号 L2600

神经元之间和神经元内部的通信对于神经系统的所有功能至关重要,无论是从发育到衰老,还是从健康到疾病。在过去十年中,我们对神经系统内分子、细胞和系统信号通路的认识取得了巨大进步,在信号通路研究方面取得了重大突破,这些神经信号通路是神经发生、成瘾、自闭症以及情绪障碍的病理生理学和治疗基础。例如:G 蛋白偶联受体(GPCR),包括5-HT 受体、组胺受体、阿片受体等,是研究较多的神经元信号传导途径,GPCR 功能障碍会引起多种神经疾病;Notch 信号途径调节神经干细胞增殖、存活、自我更新和分化,Notch 信号传导异常参与中风、阿尔茨海默病和CNS 肿瘤等疾病中发生的病理过程。因此靶向神经元信号传导,可以用来治疗多种不同CNS 疾病。 TargetMol 神经信号分子库包含2540 种与中枢神经系统信号传导有关的小分子化合物,主要用于神经系统类疾病的药物研发,可用于高通量、高内涵筛选。

TargetMol的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。

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产品编号 L2600

神经信号分子库
规格
  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品描述 产品描述

  • 2540种CNS相关的生物活性小分子化合物的特有集合,用于高通量、高内涵筛选;
  • 靶点包括5-HT receptor、AChR、Histamine receptor、dopamine receptor、Opiod receptor等;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。

Packaging And Storage | TargetMol 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。

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Library Customization | TargetMol 化合物库定制

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Library Customization | TargetMol 化合物库组成

5-HT Receptor
AChR
COX
Adrenergic Receptor
Dopamine Receptor
Calcium Channel
Histamine Receptor
GABA Receptor
GluR
Autophagy
TRP/TRPV Channel
Apoptosis
Endogenous Metabolite
AChE
iGluR
Adenosine Receptor
NMDAR
Opioid Receptor
MAO
Beta Amyloid
Antibacterial
NF-κB
Monoamine Oxidase
P-gp
Serotonin Transporter
Cannabinoid Receptor
Parasite
Gamma-secretase
Potassium Channel
P2X Receptor
Norepinephrine
Sodium Channel
CaMK
P450
FAAH
Sigma receptor
Reactive Oxygen Species
P2Y Receptor
NO Synthase
Lipoxygenase
GPR
PDE
Neurokinin receptor
HIV Protease
BACE
PPAR
OX Receptor
Influenza Virus
Antibiotic
TNF
Neuropeptide Y Receptor
Ferroptosis
Beta-Secretase
NOS
Antifungal
Mitophagy
Prostaglandin Receptor
ERK
IL Receptor
Antioxidant
Melatonin Receptor
ROS
Phospholipase
Imidazoline Receptor
Virus Protease
Adenylyl cyclase
MT Receptor
DNA/RNA Synthesis
PGE Synthase
HDAC
Chloride channel
Transferase
p38 MAPK
Caspase
PKC
Drug Metabolite
HSV
Akt
SARS-CoV
AMPK
HER
Carbonic Anhydrase
Estrogen/progestogen Receptor
Dehydrogenase
MRP
PKA
Glucocorticoid Receptor
GlyT
Interleukin
EGFR
IκB/IKK
HCV Protease
Glutathione Peroxidase
AAK1 (AP2 associated kinase 1)
BCL
MMP
TGF-beta/Smad
STAT
Melanocortin Receptor
Tyrosinase
Microtubule Associated
ATPase
Histone Methyltransferase
PI3K
NADPH
Histone Demethylase
Phosphatase
GSK-3
Wnt/beta-catenin
Serine/threonin kinase
Immunology/Inflammation related
Monoamine Transporter
TLR
CGRP Receptor
Anti-infection
cholecystokinin
HIF/HIF Prolyl-Hydroxylase
Melanin-concentrating Hormone Receptor (MCHR)
Src
Reductase
Na+/Ca2+ Exchanger
RAAS
JNK
ABC
Neurotensin Receptor
VEGFR
Topoisomerase
Mitochondrial Metabolism
Antifection
CCR
GST
MEK
advanced glycation end products
Transaminase
Amino Acids and Derivatives
Arrestin
IFNAR
DYRK
Lipase
Progesterone Receptor
HBV
Estrogen Receptor/ERR
PARP
Leukotriene Receptor
ROCK
IAP
UGT
Bcr-Abl
PAFR
LDL
CDK
Glucosidase
Guanylate cyclase
PAK
JAK
Epoxide Hydrolase
Aurora Kinase
cAMP
Epigenetic Reader Domain
IGF-1R
DNA
Androgen Receptor
mTOR
BCRP
Acyltransferase
Free radical scavengers
Nrf2
GluCls
RSV
Hydroxylase
Gap Junction Protein
NOD
DNA Methyltransferase
FAK
Proteasome
CAT
Monocarboxylate transporter
ROR
Integrin
LPL Receptor
Neuropeptide W
GTPase
OCT
N-Acetylglucosaminyltransferase
Antifolate
cell cycle arrest
Cysteine Protease
FXR
Aryl Hydrocarbon Receptor
Myosin
Annexin A
FLAP
Adiponectin receptor
GRK
Raf
Glucagon Receptor
Anion Exchanger
MAGL
Fatty Acid Synthase
Bombesin Receptor
Stearoyl-CoA Desaturase (SCD)
Angiotensin-converting Enzyme (ACE)
Somatostatin
PAD
ACK
Indoleamine 2,3-Dioxygenase (IDO)
MAPK
Antiviral
HSP
STING
Trk receptor
Aminopeptidase
GPCR19
Sirtuin
Histone Acetyltransferase
transporter
Casein Kinase
Reverse Transcriptase
Retinoid Receptor
CRISPR/Cas9
Adenosine deaminase
FGFR
NMU2R
Platelet aggregation
FLT
Syk
NADPH-oxidase
S6 Kinase
HMG-CoA Reductase
Protease-activated Receptor
Thrombin
lysosomal autophagy
NOD-like Receptor (NLR)
AhR
ROS Kinase
CFTR
p53
S1P Receptor