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癌细胞分化化合物库

癌细胞分化化合物库

产品编号 L2140 Cancer Cell Differentiation Compound Library
  库化合物信息   Excel SDF

癌症已经是全球第二大死亡原因,无论在发达国家还是在发展中国家,死亡率和发病率仍不断增高。在癌症中,分化指肿瘤组织与其来源的正常组织相比,相似程度大小。分化良好的癌细胞看起来更像正常细胞,倾向于比低分化或未分化的癌细胞生长和传播的慢。因此分化可用于肿瘤分级系统。

诱导恶性肿瘤细胞分化成熟是恶性肿瘤防治的主要研究方向之一。细胞分化的关键环节是基因调控,故基因表达时间/空间差异性、差异调控下新合成的特异性蛋白质、不同细胞表面抗原以及异常细胞周期、信号传导通路等成为恶性肿瘤细胞分化机制的主要研究点。除了本库中收录的406 个诱导肿瘤细胞分化的小分子外,您也可以参考我们的抗癌分子库,抗癌上市药物库,抗癌临床药物库等。

TargetMol的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
TargetMol Compound Library
规格
1 mg
30 μL * 10 mM (in DMSO)
50 μL * 10 mM (in DMSO)
100 μL * 10 mM (in DMSO)
250 μL * 10 mM (in DMSO)
如果上述化合物库无法满足您的需求,您可发送邮件至tech@targetmol.com咨询我们的技术专员,为您量身定制专属化合物库!
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产品描述

  • 406个诱导肿瘤细胞分化化合物的独特集合,可用于高通量筛选和高内涵筛选;
  • 提供产品的来源、化学信息和生物学信息,为筛选提供理论方向和研究基础;
  • 结构多样,药效显著,可渗透细胞;
  • NMR、HPLC/LCMS检测技术保证产品高纯度和高质量,减少假阳性发生概率。

化合物库定制

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包装和存储

  • 干粉或者DMSO溶液置于带二维码的储存管中,或排列于96孔板/384孔板;
  • 蓝冰运输
获取筛选库化合物信息 (L2140)
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TargetMol Library Books客户使用化合物库发表的文献

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化合物库组成

Autophagy (107)
Apoptosis (93)
PI3K (68)
p38 MAPK (66)
STAT (42)
mTOR (41)
TGF-beta/Smad (41)
HDAC (41)
ERK (34)
Akt (28)
GSK-3 (25)
Wnt/beta-catenin (18)
DNA-PK (18)
NF-κB (16)
ALK (16)
ATM/ATR (15)
CDK (14)
AMPK (14)
Endogenous Metabolite (13)
S6 Kinase (13)
Antibacterial (13)
Parasite (11)
Gamma-secretase (9)
Casein Kinase (8)
Mitophagy (8)
Antibiotic (8)
HIV Protease (7)
PDK (7)
Reactive Oxygen Species (7)
Caspase (6)
Src (6)
PKC (6)
PKA (6)
MEK (6)
BCL (5)
DNA/RNA Synthesis (5)
JAK (5)
Dehydrogenase (5)
MAPK (5)
COX (5)
VEGFR (4)
Virus Protease (4)
PARP (4)
PPAR (4)
Chk (4)
Raf (4)
PDE (4)
Influenza Virus (4)
MMP (3)
HSV (3)
Aurora Kinase (3)
EGFR (3)
FGFR (3)
FLT (3)
TNF (3)
Beta Amyloid (3)
Epigenetic Reader Domain (3)
Antifungal (3)
Carbonic Anhydrase (3)
JNK (3)
Adenosine Receptor (3)
ROCK (3)
AChE (2)
Calcium Channel (2)
TLR (2)
PDGFR (2)
IGF-1R (2)
Drug Metabolite (2)
Porcupine (2)
c-Fms (2)
PI4K (2)
P450 (2)
Phosphatase (2)
CRISPR/Cas9 (2)
P-gp (2)
IκB/IKK (2)
HER (2)
Lipoxygenase (2)
Tyrosine Kinases (2)
Adrenergic Receptor (2)
HBV (2)
Bcr-Abl (2)
IL Receptor (2)
Topoisomerase (2)
DNA (1)
Aromatase (1)
NADPH (1)
MLK (1)
Nrf2 (1)
hCE (1)
BACE (1)
MELK (1)
c-Met/HGFR (1)
Arginase (1)
Retinoid Receptor (1)
Estrogen/progestogen Receptor (1)
HCV Protease (1)
Hck (1)
Potassium Channel (1)
Phospholipase (1)
GABA Receptor (1)
HIF (1)
PLK (1)
DHFR (1)
AChR (1)
c-Kit (1)
Sodium Channel (1)
Ras (1)
Nucleoside Antimetabolite/Analog (1)
HIF/HIF Prolyl-Hydroxylase (1)
FAK (1)
Histamine Receptor (1)
SGK (1)
Hedgehog/Smoothened (1)
Antiviral (1)
Serine Protease (1)
CCR (1)
PTEN (1)
PAD (1)
NOS (1)
Antifolate (1)
Estrogen Receptor/ERR (1)
Isocitrate Dehydrogenase (IDH) (1)
Antioxidant (1)
GluR (1)
MNK (1)
UGT (1)
Fatty Acid Synthase (1)
transporter (1)
Smo (1)
Ferroptosis (1)
YAP (1)
SARS-CoV (1)
CXCR (1)
Integrin (1)
ATPase (1)
c-Myc (1)
5-HT Receptor (1)
RIP kinase (1)
Tie-2 (1)
Beta-Secretase (1)

化合物库信息示例

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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