p38α inhibitor 2

Name: p38α inhibitor 2
Brand: TargetMol
SKU: T36012
Price: 197 USD
Availability: InStock
Rating: 4.5 (1 reviews)

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产品编号 T36012Cas号 1095003-80-7

p38α inhibitor 2 is a highly potent and selective p38α MAPK inhibitor, with a pIC50 of 9.6. p38α inhibitor 2 inhibits the hERG ion channel (IC50=27 μM) and shows a promising selectivity profile when tested in a panel of 51 other protein kinases (<30% inhibition at 10 μM concentration) and a panel of 141 other biological targets[1].

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p38α inhibitor 2

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产品编号 T36012Cas号 1095003-80-7

规格	价格	库存
2 mg	¥ 2,480	5日内发货
5 mg	¥ 2,890	5日内发货
25 mg	¥ 10,800	6-8周
50 mg	¥ 14,100	6-8周
100 mg	¥ 19,500	6-8周
1 mL x 10 mM (in DMSO)	¥ 2,970	5日内发货

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TargetMol 的所有产品仅用作科学研究或药证申报，不能被用于人体，我们不向个人提供产品和服务。请您遵守承诺用途，不得违反法律法规规定用于任何其他用途。

产品介绍

生物活性

产品描述

P38α Inhibitor 2, a potent and selective inhibitor of p38α MAPK, exhibits a pIC50 value of 9.6. It also demonstrates inhibition of the hERG ion channel (IC50=27 μM) and maintains promising selectivity, with <30% inhibition across a panel of 51 protein kinases at a 10 μM concentration and a broad specificity against 141 other biological targets[1].

化学信息

分子量	475.58
分子式	C₂₇H₃₃N₅O₃
CAS No.	1095003-80-7
密度	1.23 g/cm3 (Predicted)

储存&溶解度

存储

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.

溶解度信息

DMSO: 250 mg/mL (525.67 mM), Sonication is recommended.

溶液配制表

DMSO

	1mg	5mg	10mg	50mg
1 mM	2.1027 mL	10.5135 mL	21.0270 mL	105.1348 mL
5 mM	0.4205 mL	2.1027 mL	4.2054 mL	21.0270 mL
10 mM	0.2103 mL	1.0513 mL	2.1027 mL	10.5135 mL
20 mM	0.1051 mL	0.5257 mL	1.0513 mL	5.2567 mL
50 mM	0.0421 mL	0.2103 mL	0.4205 mL	2.1027 mL
100 mM	0.0210 mL	0.1051 mL	0.2103 mL	1.0513 mL