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Search Results for " calcium channel "
Targets Recommended: Calcium Channel Calcium Channel

329

抑制剂 & 化合物

45

天然产物

1

化合物库

19

重组蛋白

21

同位素标记化合物

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Cat. No. Product Name
L7200 钙通道分子库

140 compounds
140 种钙通道相关化合物的独特集合,可用于高通量筛选和高内涵筛选;

化合物库

钙通道分子库
Cat.No: L7200
Compounds: 140
Cat. No. Product Name Target Signaling Pathways
T77710 Calcium Channel antagonist 2

WAY-327363

Calcium Channel Membrane transporter/Ion channel; Metabolism
Calcium Channel antagonist 2是一种 calcium channel 拮抗剂 (IC50=5-20 μM),可用于研究像疼痛和糖尿病等由于 Ca2+ 通道造成的疾病。
T10101 Calcium channel-modulator-1

Others; Calcium Channel Membrane transporter/Ion channel; Metabolism; Others
Calcium channel-modulator-1是钙离子通道调节剂(IC50:0.8 μM),具有阻塞主动脉收缩的专业化。
T77711 Calcium Channel antagonist 4

Calcium Channel Membrane transporter/Ion channel; Metabolism
Calcium Channel antagonist 4 是一种电压门控钙通道抑制剂(IC50 : 5-20μM)。
T77712 Calcium Channel antagonist 3

Calcium Channel Membrane transporter/Ion channel; Metabolism
Calcium Channel antagonist 3 是一种电压门控钙通道抑制剂(IC50 : 5-20μM)。
T12153 N-type calcium channel blocker-1

Calcium Channel Membrane transporter/Ion channel; Metabolism
N-type calcium channel blocker-1 is an orally active analgesic agent,shows high affinity to functionally block N-type calcium channels.
T2519 Lercanidipine

乐卡地平,Masnidipine

Calcium Channel Membrane transporter/Ion channel; Metabolism
Lercanidipine (Masnidipine) 是二氢吡啶类的钙通道阻滞剂,具有持久的降压作用和肾脏保护作用。
T10659 Ca2+ channel agonist 1

Calcium Channel; CDK Cell Cycle/Checkpoint; Membrane transporter/Ion channel; Metabolism
Ca2+channel agonist 1 是 N-型钙离子通道激动剂和Cdk2的抑制剂,EC50分别为 14.23 μM 和 3.34 μM,可用作运动神经末梢功能障碍的潜在治疗方法。
T12015 Methyl homoveratrate

Others Others
Methyl homoveratrate 是血浆、尿液和粪便提取物中 McN5691 的代谢物,是电压依赖性钙通道阻滞剂。
T1530 Mitiglinide calcium hydrate

KAD-1229 calcium hydrate,米格列奈钙,Mitiglinide calcium,S-21403 calcium hydrate

Potassium Channel Membrane transporter/Ion channel
Mitiglinide calcium hydrate (S-21403 calcium hydrate) 是一种 ATP 敏感的 K+通道 (KATPchannel) 拮抗剂, 属于促胰岛素化合物。它对 Kir6.2/SUR1 复合物 (胰腺-细胞 KATP 通道) 具有高度特异性,在 2 型糖尿病中有研究价值。
T7603 Pinaverium bromide

Calcium Channel Membrane transporter/Ion channel; Metabolism
Pinaverium bromide 是一种具有解痉作用的钙通道阻滞剂,可有效缓解疼痛、腹泻和肠道不适。
T8944 TTA-A2

Calcium Channel Membrane transporter/Ion channel; Metabolism
TTA-A2 是一种选择性 T 型钙通道拮抗剂,是一种有效的抗惊厥药,可减少孕烷 X 受体的激活。它对 Cav3.1 (a1G) 和 Cav3.2 (a1H) 通道在 -80 mV 和- 100 mV 保持电位上具有同样的作用,IC50 值分别为 89 和 92 nM。它可用于多种人类神经系统疾病的研究,包括睡眠障碍和癫痫。
T11353 Gallopamil

Methoxyverapamil,戈洛帕米

Calcium Channel Membrane transporter/Ion channel; Metabolism
Gallopamil (Methoxyverapamil) 是一种苯烷基胺钙拮抗剂,以浓度依赖性方式抑制酸分泌 (IC50 = 10.9 μM)。Gallopamil 显示出抗心律失常和血管扩张剂的功效。
T0283 Trimethadione

三甲双酮,3,5,5,-Trimethyloxazolidine-2,4-dione

Calcium Channel Membrane transporter/Ion channel; Metabolism
Trimethadione (3,5,5,-Trimethyloxazolidine-2,4-dione) 是恶唑烷二酮类抗惊厥剂,也是一种 T 型钙通道阻滞剂,具有抗痛觉过敏作用,可用于研究失神发作。
T23280 Ruthenium Red

钌红,Ammoniated ruthenium oxychloride

Calcium Channel Membrane transporter/Ion channel; Metabolism
Ruthenium Red (Ammoniated ruthenium oxychloride) 是一种 L 型钙电流 (ICa) 阻断剂,是一种聚阳离子染料,广泛用于电子显微镜 (EM) 下细胞、组织和营养细菌的观察。它能与磷脂和脂肪酸反应强烈,并与酸性粘多糖结合。
T0957 Isradipine

PN 200-110,伊拉地平

Calcium Channel; Autophagy Autophagy; Membrane transporter/Ion channel; Metabolism
Isradipine (PN 200-110) 是一种二氢吡啶类钙通道阻滞剂,具有抗高血压和血管扩张活性。它是一种具有口服活性的 L 型钙通道阻滞剂,也是一种潜在可行的帕金森病神经保护剂。
T15423 GSK-7975A

Calcium Channel Membrane transporter/Ion channel; Metabolism
GSK-7975A 是具有口服活性的高效CRAC 通道抑制剂。
T8863 VK-II-36

Others Others
VK-II-36 是 carvedilol 的类似物,能够在不阻断 β 受体的情况下抑制肌浆网钙释放。它能够抑制早期和延迟后去极化诱发的触发活动,可用于局灶性室性心律失常的研究。
T11353L Gallopamil hydrochloride

Methoxyverapamil hydrochloride

Calcium Channel Membrane transporter/Ion channel; Metabolism
Gallopamil hydrochloride (Methoxyverapamil hydrochloride) 是苯烷基胺钙的拮抗剂。Gallopamil hydrochloride 可用于抗心律失常和血管扩张剂研究。
T10690 Cav 2.2 blocker 1

Calcium Channel Membrane transporter/Ion channel; Metabolism
Cav 2.2 blocker 1 是一种N 型钙离子通道 (Cav 2.2) 的阻断剂,IC50值为 1 nM,可用于治疗疼痛。
T5023 Propiverine hydrochloride

Others; Calcium Channel; AChR Membrane transporter/Ion channel; Metabolism; Neuroscience; Others
Propiverine hydrochloride 是一种痉挛剂,具有钙拮抗和抗胆碱能特性,用于研究膀胱过度活动和尿失禁。
T0119 Nitrendipine

BAY-E-5009,Bayotensin,尼群地平

Calcium Channel; Autophagy Autophagy; Membrane transporter/Ion channel; Metabolism
Nitrendipine (BAY-E-5009) 是 Nifedipine 的类似物,是一种钙通道阻滞剂,具有显着的血管扩张作用。它是一种有效的抗高血压药且不会降低肾小球滤过率,并且具有轻微的利钠作用。
T6874 Lercanidipine hydrochloride

Corifeo,Carmen,Cardiovasc,乐卡地平盐酸盐,盐酸乐卡地平

Calcium Channel Membrane transporter/Ion channel; Metabolism
Lercanidipine hydrochloride (Corifeo) 是亲脂性二氢吡啶-钙通道阻滞剂,具有持久的降压作用和保护肾脏作用。
T11517 GV-58

Calcium Channel Membrane transporter/Ion channel; Metabolism
GV-58 是选择性 N 型和 P/Q 型 Ca2+ 通道激动剂,EC50值分别为7.21和8.81uM。它对 CDK 激酶活性的抑制作用减少了 20 倍。
T7373 CDN1163

Calcium Channel Membrane transporter/Ion channel; Metabolism
CDN1163 是肌膜/内质网 Ca2+-ATPase (SERCA)的变构激活剂,可改善 Ca2+稳态,可减轻糖尿病和代谢紊乱。
T8674 SR33805

Calcium Channel Membrane transporter/Ion channel; Metabolism
SR33805 是钙通道拮抗剂,在去极化和极化条件下的 EC50值分别为 4.1 和 33 nM。它阻止 L 型 Ca2+通道,可用于研究急性或慢性心脏衰竭。
T13047 Synta66

Calcium Channel Membrane transporter/Ion channel; Metabolism
Synta66 是一种钙池操纵钙离子通道 Orai 抑制剂,用于神经系统疾病的研究。
T12608 QX-314 chloride

Sodium Channel Membrane transporter/Ion channel
QX-314 chloride 是钠离子通道电荷阻滞剂,具有膜不渗透性。
T3703 ABT-639

ABT 639

Calcium Channel Membrane transporter/Ion channel; Metabolism
ABT-639 是一种有效的选择性 T 型钙通道阻滞剂。
T16014 Mavatrep

JNJ-39439335

TRP/TRPV Channel Membrane transporter/Ion channel
Mavatrep (JNJ-39439335) 是一种特异性的 TRPV1 拮抗剂,Ki 为 6.5 nM,可用于炎症性疼痛的研究。
T0030 Bupivacaine hydrochloride

Vivacaine,Bupivacaine HCl,盐酸布比卡因

Sodium Channel Membrane transporter/Ion channel
Bupivacaine hydrochloride (Vivacaine) 是NMDA 受体抑制剂,可用于慢性疼痛的研究。它可阻断钠、L-钙和钾通道,还阻断SCN5A 通道,IC50为 69.5 μM。
T0916 Butamben

Butyl 4-aminobenzoate,4-氨基苯甲酸丁酯

Potassium Channel; Calcium Channel; Sodium Channel Membrane transporter/Ion channel; Metabolism
Butamben (Butyl 4-aminobenzoate) 是一种长效局部麻醉剂,用于治疗慢性疼痛。
T0343 Nimodipine

尼莫地平,BAY-e 9736

Glucocorticoid Receptor; AhR; Calcium Channel; Autophagy Autophagy; Endocrinology/Hormones; Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism
Nimodipine (BAY-e 9736) 是一种具有口服活性,耐受性良好的光敏二氢吡啶钙拮抗剂。它可研究脑血管疾病。
T22788 FPL64176

FPL 64176

Calcium Channel Membrane transporter/Ion channel; Metabolism
FPL64176 是一种非二氢吡啶类L 型钙通道激动剂,EC50值为 16 nM。
T3543 NS-638

NS 638

Calcium Channel Membrane transporter/Ion channel; Metabolism
NS-638 是一种 Ca2+ 通道阻滞剂,可阻断 K+ 刺激的细胞内 Ca2+ 升高,IC50值为3.4 μM。
T1198 Tetracaine hydrochloride

盐酸丁卡因,Amethocaine hydrochloride,Amethocalne HCl,Tetracaine HCl

Calcium Channel; Sodium Channel Membrane transporter/Ion channel; Metabolism
Tetracaine hydrochloride (Amethocalne HCl) 是一种钙通道蛋白抑制剂,可阻断肌浆网中 Ca2+的电压敏感释放。它主要用作眼科的止痒剂和局部用药,可用于表面和脊髓麻醉。
T0388 Cilnidipine

FRC-8653,西尼地平

Calcium Channel Membrane transporter/Ion channel; Metabolism
Cilnidipine (FRC-8653) 是二氢吡啶类Ca2+通道阻断剂,可作用于 L 和 N 型 Ca2+通道,具有抗高血压活性。
T7216 Mirogabalin

DS5565

Calcium Channel Membrane transporter/Ion channel; Metabolism
Mirogabalin (DS5565) 是一种高效的、选择性的 α2δ-1 配体,作用于电压敏感性钙通道复合体的α2δ-1亚基。
T6848 GSK1016790A

GSK101

Calcium Channel; TRP/TRPV Channel Membrane transporter/Ion channel; Metabolism
GSK1016790A (GSK101) 是选择性瞬时受体电位香草酸 4 通道激活剂,可引起 HEK 细胞中 Ca2+流入并升高细胞内 Ca2+。
T29201 Z944

Z 944,Z-944

Calcium Channel Membrane transporter/Ion channel; Metabolism
Z944 是有效的 T 型钙通道拮抗剂,对跨模态和视觉识别记忆障碍有缓解作用。
T0858 Flufenamic acid

Arlef,Nichisedan,氟灭酸,氟芬那酸,Achless

Potassium Channel; Calcium Channel; Chloride channel; COX; AMPK; Parasite Chromatin/Epigenetic; Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; Microbiology/Virology; Neuroscience; PI3K/Akt/mTOR signaling
Flufenamic acid (Arlef) 是一种非甾体类抗炎剂,是一种邻氨基苯甲酸衍生物,具有镇痛、抗炎和解热的特性。 它用于肌肉骨骼和关节疾病。
T5632 Suvecaltamide

MK-8998

Calcium Channel Membrane transporter/Ion channel; Metabolism
Suvecaltamide (MK-8998) 是一种选择性的 T 型钙通道抑制剂。
T1510 Rosuvastatin calcium

ZD 4522 Calcium,ZD4522,Rosuvastatin hemicalcium,瑞舒伐他汀钙

Potassium Channel; HMG-CoA Reductase; Autophagy Autophagy; Membrane transporter/Ion channel; Metabolism
Rosuvastatin calcium (ZD4522) 是肝羟甲基戊二酰辅酶 A 还原酶的选择性和竞争性抑制剂,具有抗血脂活性。它降低成熟 hERG 的表达以及热休克蛋白 70 与 hERG 蛋白的相互作用,还降低低密度脂蛋白胆固醇、甘油三酯和 C-反应蛋白水平。它阻断人类醚-a-go-go 相关基因电流,延迟心脏复极化,来延长动作电位持续时间和校正 QT 间期间隔。
T6577 Manidipine

Iperten,Franidipine,Artedil,马尼地平

Calcium Channel Membrane transporter/Ion channel; Metabolism
Manidipine (Iperten) 是一种二氢吡啶类钙通道阻滞剂,有降压作用。
T0702 Gabapentin

Neurontin,Gabapentine,加巴喷丁,Aclonium

Calcium Channel; GABA Receptor Membrane transporter/Ion channel; Metabolism; Neuroscience
Gabapentin (Neurontin) 是GABA 类似物,是一种抗癫痫药,可用于缓解神经性疼痛。
T0327 Fendiline hydrochloride

Fendiline HCl,盐酸芬他林

Calcium Channel Membrane transporter/Ion channel; Metabolism
Fendiline hydrochloride (Fendiline HCl) 是一种非选择性钙通道抑制剂。
T10885 CRAC intermediate 2

Others; Calcium Channel Membrane transporter/Ion channel; Metabolism; Others
CRAC intermediate 2是CRAC 抑制剂合成的中间体化合物。
T5376 Aranidipine

阿雷地平,MPC1304

Calcium Channel Membrane transporter/Ion channel; Metabolism
Aranidipine (MPC1304) 是一种钙通道拮抗剂,具有强效和持久的抗高血压作用。
T8815 Azumolene

阿珠莫林,EU4093 free base

Calcium Channel Membrane transporter/Ion channel; Metabolism
Azumolene (EU4093 free base) 是一种 Dantrolene 的类似物,是一种肌肉松弛剂,可用于恶性高热研究。它是一种 ryanodine 受体调节剂,并通过 ryanodine 受体抑制钙释放。
T16571 Pranidipine

普拉地平,OPC-13340

Calcium Channel Membrane transporter/Ion channel; Metabolism
Pranidipine (OPC-13340) 是一种高效且长效的 1,4-二氢吡啶钙通道阻滞剂,可延长乙酰胆碱诱导的内皮松弛以及硝酸甘油诱导的内皮松弛,具有抗高血压作用。
T0163 Nisoldipine

尼索地平,BAY-k 5552

Calcium Channel; Reactive Oxygen Species Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; NF-κB
Nisoldipine (BAY-k 5552) 是一种高效特异的L 型Cav1.2通道阻断剂,IC50=10 nM。

化合物

Calcium Channel antagonist 2
Cat.No: T77710
Synonym: WAY-327363
Target: Calcium Channel
Calcium channel-modulator-1
Cat.No: T10101
Synonym:
Target: Others, Calcium Channel
Calcium Channel antagonist 4
Cat.No: T77711
Synonym:
Target: Calcium Channel
Calcium Channel antagonist 3
Cat.No: T77712
Synonym:
Target: Calcium Channel
N-type calcium channel blocker-1
Cat.No: T12153
Synonym:
Target: Calcium Channel
Lercanidipine
Cat.No: T2519
Synonym: 乐卡地平,Masnidipine
Target: Calcium Channel
Ca2+ channel agonist 1
Cat.No: T10659
Synonym:
Target: Calcium Channel, CDK
Methyl homoveratrate
Cat.No: T12015
Synonym:
Target: Others
Mitiglinide calcium hydrate
Cat.No: T1530
Synonym: KAD-1229 calcium hydrate,米格列奈钙,Mitiglinide calcium,S-21403 calcium hydrate
Target: Potassium Channel
Pinaverium bromide
Cat.No: T7603
Synonym:
Target: Calcium Channel
TTA-A2
Cat.No: T8944
Synonym:
Target: Calcium Channel
Gallopamil
Cat.No: T11353
Synonym: Methoxyverapamil,戈洛帕米
Target: Calcium Channel
Trimethadione
Cat.No: T0283
Synonym: 三甲双酮,3,5,5,-Trimethyloxazolidine-2,4-dione
Target: Calcium Channel
Ruthenium Red
Cat.No: T23280
Synonym: 钌红,Ammoniated ruthenium oxychloride
Target: Calcium Channel
Isradipine
Cat.No: T0957
Synonym: PN 200-110,伊拉地平
Target: Calcium Channel, Autophagy
GSK-7975A
Cat.No: T15423
Synonym:
Target: Calcium Channel
VK-II-36
Cat.No: T8863
Synonym:
Target: Others
Gallopamil hydrochloride
Cat.No: T11353L
Synonym: Methoxyverapamil hydrochloride
Target: Calcium Channel
Cav 2.2 blocker 1
Cat.No: T10690
Synonym:
Target: Calcium Channel
Propiverine hydrochloride
Cat.No: T5023
Synonym:
Target: Others, Calcium Channel, AChR
Nitrendipine
Cat.No: T0119
Synonym: BAY-E-5009,Bayotensin,尼群地平
Target: Calcium Channel, Autophagy
Lercanidipine hydrochloride
Cat.No: T6874
Synonym: Corifeo,Carmen,Cardiovasc,乐卡地平盐酸盐,盐酸乐卡地平
Target: Calcium Channel
GV-58
Cat.No: T11517
Synonym:
Target: Calcium Channel
CDN1163
Cat.No: T7373
Synonym:
Target: Calcium Channel
SR33805
Cat.No: T8674
Synonym:
Target: Calcium Channel
Synta66
Cat.No: T13047
Synonym:
Target: Calcium Channel
QX-314 chloride
Cat.No: T12608
Synonym:
Target: Sodium Channel
ABT-639
Cat.No: T3703
Synonym: ABT 639
Target: Calcium Channel
Mavatrep
Cat.No: T16014
Synonym: JNJ-39439335
Target: TRP/TRPV Channel
Bupivacaine hydrochloride
Cat.No: T0030
Synonym: Vivacaine,Bupivacaine HCl,盐酸布比卡因
Target: Sodium Channel
Butamben
Cat.No: T0916
Synonym: Butyl 4-aminobenzoate,4-氨基苯甲酸丁酯
Target: Potassium Channel, Calcium Channel, Sodium Channel
Nimodipine
Cat.No: T0343
Synonym: 尼莫地平,BAY-e 9736
Target: Glucocorticoid Receptor, AhR, Calcium Channel, Autophagy
FPL64176
Cat.No: T22788
Synonym: FPL 64176
Target: Calcium Channel
NS-638
Cat.No: T3543
Synonym: NS 638
Target: Calcium Channel
Tetracaine hydrochloride
Cat.No: T1198
Synonym: 盐酸丁卡因,Amethocaine hydrochloride,Amethocalne HCl,Tetracaine HCl
Target: Calcium Channel, Sodium Channel
Cilnidipine
Cat.No: T0388
Synonym: FRC-8653,西尼地平
Target: Calcium Channel
Mirogabalin
Cat.No: T7216
Synonym: DS5565
Target: Calcium Channel
GSK1016790A
Cat.No: T6848
Synonym: GSK101
Target: Calcium Channel, TRP/TRPV Channel
Z944
Cat.No: T29201
Synonym: Z 944,Z-944
Target: Calcium Channel
Flufenamic acid
Cat.No: T0858
Synonym: Arlef,Nichisedan,氟灭酸,氟芬那酸,Achless
Target: Potassium Channel, Calcium Channel, Chloride channel, COX, AMPK, Parasite
Suvecaltamide
Cat.No: T5632
Synonym: MK-8998
Target: Calcium Channel
Rosuvastatin calcium
Cat.No: T1510
Synonym: ZD 4522 Calcium,ZD4522,Rosuvastatin hemicalcium,瑞舒伐他汀钙
Target: Potassium Channel, HMG-CoA Reductase, Autophagy
Manidipine
Cat.No: T6577
Synonym: Iperten,Franidipine,Artedil,马尼地平
Target: Calcium Channel
Gabapentin
Cat.No: T0702
Synonym: Neurontin,Gabapentine,加巴喷丁,Aclonium
Target: Calcium Channel, GABA Receptor
Fendiline hydrochloride
Cat.No: T0327
Synonym: Fendiline HCl,盐酸芬他林
Target: Calcium Channel
CRAC intermediate 2
Cat.No: T10885
Synonym:
Target: Others, Calcium Channel
Aranidipine
Cat.No: T5376
Synonym: 阿雷地平,MPC1304
Target: Calcium Channel
Azumolene
Cat.No: T8815
Synonym: 阿珠莫林,EU4093 free base
Target: Calcium Channel
Pranidipine
Cat.No: T16571
Synonym: 普拉地平,OPC-13340
Target: Calcium Channel
Nisoldipine
Cat.No: T0163
Synonym: 尼索地平,BAY-k 5552
Target: Calcium Channel, Reactive Oxygen Species
Cat. No. Product Name Target Signaling Pathways
T8206 Cycleanine

Others Others
Cycleanine 是一种高效血管选择性Ca- 拮抗剂,具有缓解疼痛、肌肉松弛和抗炎作用。它还具有有效的抗菌、抗真菌、抗疟原虫和细胞毒活性。
TN2322 Yangambin

Calcium Channel; PAFR GPCR/G Protein; Membrane transporter/Ion channel; Metabolism
Yangambin 是从诸如番荔枝科植物中分离出来的呋喃木脂素,是选择性PAF 受体拮抗剂,通过调控Ca2+通道抑制 Ca2+流入,导致 [Ca2+]i 在血管平滑肌细胞和随后的外周血管舒张中减少,具有降压作用。
T6S1418 Praeruptorin C

Antioxidant; Calcium Channel Membrane transporter/Ion channel; Metabolism; oxidation-reduction
Praeruptorin C 是白花前胡中的一种主要成分,是钙拮抗剂,pD2′值为 5.7。
T11665 Ionomycin calcium

SQ23377 calcium,罗红霉素钙盐(链霉菌属载体)

Apoptosis; Calcium Channel; Antibacterial; Antibiotic; PKC Apoptosis; Chromatin/Epigenetic; Cytoskeletal Signaling; Membrane transporter/Ion channel; Metabolism; Microbiology/Virology
Ionomycin calcium (SQ23377 calcium) 是选择性钙离子载体,也是一种由 Streptomyces conglobatus 产生的抗生素。它对二价阳离子具有高度特异性,还诱导蛋白激酶 C 激活。Ionomycin 促进细胞凋亡。
T8787 Drotaverine hydrochloride

PDE Metabolism
Drotaverine hydrochloride 是磷酸二酯酶 4 (PDE4)的抑制剂,也是 L 型电压依赖钙通道(L-VDCC)的阻滞剂,可阻断3',5'-环腺苷单磷酸的降解。它在体内有抗痉挛效果,但无抗胆碱能的效果。
T0728 Ethosuximide

Zarontin,乙琥胺

Calcium Channel Membrane transporter/Ion channel; Metabolism
Ethosuximide (Zarontin) 是一种抗癫痫药物,可改善多种神经退行性疾病模型的表型,且阻断低电压激活的 T 型钙通道。
T3904 Gomisin J

Calcium Channel; AMPK Chromatin/Epigenetic; Membrane transporter/Ion channel; Metabolism; PI3K/Akt/mTOR signaling
Gomisin J 是在五味子中发现的小分子量木脂素,具有血管舒张活性,在非酒精性脂肪性肝病方面有研究潜力。 它通过激活 AMPK、LKB1 和 Ca2+/钙调蛋白依赖性蛋白激酶 II 以及抑制 HepG2 细胞中的胎球蛋白 A 来调节脂肪生成酶和脂肪分解酶以及炎症分子的表达,从而抑制脂质积累。
TN1008 Psoralenoside

CaMK; Calcium Channel; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; Neuroscience
Psoralenoside 是源于补骨脂中的苯并呋喃苷,具有抗肿瘤、抗菌、促进成骨细胞增殖和雌激素样活性。它对组胺 H1、钙调素和电压门控 l 型钙通道具有较高的亲和力。
T5723 Menthol

薄荷脑,DL-Menthol

Others; Calcium Channel Membrane transporter/Ion channel; Metabolism; Others
Menthol (DL-Menthol) 是从薄荷或薄荷油中得到的一种天然产物,具有调味和局部麻醉特性。它通过抑制神经元细胞膜的 Ca++电流,刺激冷感受器,从而产生清凉的感觉。
T15027 Cyclopiazonic acid

环匹阿尼酸,环二氮酸

Calcium Channel Membrane transporter/Ion channel; Metabolism
Cyclopiazonic acid 是一种神经毒性次级代谢产物 (SM),源于A. flavus,是一种纳摩尔内质网钙 ATP 酶抑制剂 (Ca2+ATPase; SERCA),是植物细胞死亡的有效诱导剂。
T4S1422 Praeruptorin E

白花前胡素 E,白花前胡素E

Others; Calcium Channel Membrane transporter/Ion channel; Metabolism; Others
Praeruptorin E 是白花前胡中的一种主要成分,是钙拮抗剂,pD2′值为 5.2。
TQ0302 Thapsigargin

毒胡萝卜素

Apoptosis; SARS-CoV; Calcium Channel Apoptosis; Membrane transporter/Ion channel; Metabolism; Microbiology/Virology
Thapsigargin 属于天然产物,是一种肌/内质网 Ca2+ ATP 酶 (SERCA) 的抑制剂,也是一种内质网应激诱导剂。Thapsigargin 通过阻断细胞将钙泵入肌浆和内质网的能力来提高胞浆钙浓度。
T3013 Catharanthine tartrate

Catharanthine hemitartrate,酒石酸长春质碱

Others; Calcium Channel Membrane transporter/Ion channel; Metabolism; Others
Catharanthine tartrate (Catharanthine hemitartrate) 是长春花中的一种生物碱,可抑制电压门控 L 型钙离子通道,具有抗肿瘤和降血压活性。
T2782 Catharanthine

(+)-3, 4-Didehydrocoronaridine,长春质碱,(+)-3,4-Didehydrocoronaridine

Calcium Channel; AChR Membrane transporter/Ion channel; Metabolism; Neuroscience
Catharanthine ((+)-3,4-Didehydrocoronaridine) 是长春花中的一种生物碱,可抑制电压门控 L 型钙离子通道,具有抗肿瘤和降血压活性。
T4590 (+)-Kavain

醉椒素,Kavain,L-KAWAIN,(R)-KAWAIN

Calcium Channel; GABA Receptor; Sodium Channel; Monoamine Transporter Membrane transporter/Ion channel; Metabolism; Neuroscience
(+)-Kavain ((R)-KAWAIN) 是从卡瓦胡椒中提取的一种主要的卡瓦内酯,可通过电压依赖性的 Na+和 Ca2+通道相互作用,减弱血管平滑肌的收缩,具有抗惊厥作用。它可与α4β2δ GABAA 受体结合,加强 GABA 的功效,用于炎症疾病研究。
T6S1500 Ginsenoside Rf

人参皂苷 Rf,Ginsenoside-Rf,Panaxoside Rf

Calcium Channel; Endogenous Metabolite Membrane transporter/Ion channel; Metabolism
Ginsenoside Rf (Panaxoside Rf) 是人参根的微量成分,可抑制 N 型 Ca2+通道。
T10024 1-Octanol

Octanol,正辛醇

Calcium Channel; Endogenous Metabolite Membrane transporter/Ion channel; Metabolism
1-Octanol (Octanol) 是一种饱和脂肪醇,是一种 T 型钙通道抑制剂,对天然 T 电流的IC50为 4 μM。它是一种具有类似柴油特性的极具吸引力的生物燃料。
TN7108 Urolithin C

Apoptosis; Calcium Channel; Reactive Oxygen Species; IGF-1R; Endogenous Metabolite Apoptosis; Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; NF-κB; Tyrosine Kinase/Adaptors
Urolithin C 属于多酚类,是鞣花酸的肠道微生物代谢产物,具有胰岛素分泌的葡萄糖依赖性激活活性。Urolithin C 是 L 型 Ca2+通道开放剂,可增强 Ca2+的流入。它通过线粒体介导的途径诱导细胞凋亡,并刺激活性氧的形成。
T4727 Taurolithocholic acid sodium salt

牛磺石胆酸钠,Sodium taurolithocholate

Others; Calcium Channel Membrane transporter/Ion channel; Metabolism; Others
Taurolithocholic acid sodium salt (Sodium taurolithocholate) 是抑胆剂和 Ca2+激动剂,可抑制放射性配体与毒蕈碱 M1 结合。
T3S1916 Heteroclitin D

异型南五味子丁素,异南五味子丁素;异型南五味子丁素

Calcium Channel Membrane transporter/Ion channel; Metabolism
Heteroclitin D 是异形南五味子中的一种木脂素,可抑制 L 型钙通道,具有抗脂质过氧化作用。
T5701 OPHIOPOGONIN D

麦冬皂苷 D,麦冬皂苷D

RAAS; Calcium Channel; NF-κB; PPAR DNA Damage/DNA Repair; Endocrinology/Hormones; Membrane transporter/Ion channel; Metabolism; NF-κB
Ophiopogonin D 是从麦冬的块茎中分离的一种天然产物,是罕见的天然存在的 C29甾体糖苷。它是一种 CYP2J3 诱导剂,用于炎症和心血管疾病的相关研究。
T2996 Tetrandrine

NSC-77037,d-Tetrandrine,Hanfangchin A,粉防己碱,Fanchinine,Sinomenine A,汉防己甲素

Potassium Channel; Calcium Channel Membrane transporter/Ion channel; Metabolism
Tetrandrine (Sinomenine A) 是来自粉防己的一种双苯基异喹啉生物碱,可抑制电压门控钙离子通道 (ICa) 和 Ca2+激活的钾离子通道。
T7056 Dronedarone

决奈达隆,SR 33589

P450; Potassium Channel; Calcium Channel; Sodium Channel; Adrenergic Receptor; AChR; Autophagy Autophagy; GPCR/G Protein; Membrane transporter/Ion channel; Metabolism; Neuroscience
Dronedarone (SR 33589) 是一种胺碘酮类似物,对治疗心房颤动可能有效。它是CYP3A4的底物和中度抑制剂。它是多种离子电流的有效阻滞剂,通过非竞争性结合到肾上腺素能受体显示出抗肾上腺素能的效果。
T4S1419 (±)-Praeruptorin A

Praeruptorin A,(±)-白花前胡甲素,白花前胡甲素,(-)-Praeruptorin A

p38 MAPK; Calcium Channel; Akt Cytoskeletal Signaling; MAPK; Membrane transporter/Ion channel; Metabolism; PI3K/Akt/mTOR signaling
(±)-Praeruptorin A 是来自白花前胡的干燥根中的一种主要成分,用于研究伴有厚痰和呼吸困难的咳嗽,非天生性咳嗽和上呼吸道感染。它是顺式-内酯 (CKL) 的二酯化产物,可作为 Ca2+-反流阻滞剂,用于高血压的研究。
T1221 Acetylcholine chloride

ACh chloride,Pilofrin,氯化乙酰胆碱

Calcium Channel; Endogenous Metabolite; AChR Membrane transporter/Ion channel; Metabolism; Neuroscience
Acetylcholine chloride (Pilofrin) 是一种神经递质,是胆碱能激动剂,通过刺激烟碱乙酰胆碱受体调节多巴胺能神经元活性,在体外抑制 p53 突变肽的聚集。
T8288 14-Deoxyandrographolide

去氧穿心莲内酯,14-去氧穿心莲内酯

Apoptosis; Others Apoptosis; Others
14-Deoxyandrographolide 是穿心莲中的一种天然产物,是一种钙通道阻断剂,具有保肝功效。它通过诱导 TNFRSF1A 的释放,使肝细胞对 TNF-α 介导的凋亡脱敏。
T6856 Halofuginone

卤夫酮,常山酮,Tempostatin,empostatin,RU-19110

Calcium Channel; DNA/RNA Synthesis; Sodium Channel; Parasite; TGF-beta/Smad Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Membrane transporter/Ion channel; Metabolism; Microbiology/Virology; Stem Cells
Halofuginone (RU-19110) 是Febrifugine 的衍生物,是一种竞争性脯氨酰-tRNA 合成酶抑制剂。它也是肺血管扩张剂,可激活Kv 通道并阻断电压门控、受体操作和存储操作的钙离子通道。它具有抗炎、抗癌、抗疟疾和抗纤维化作用。
T5S2059 Glaucine

Calcium Channel; Dopamine Receptor; Influenza Virus; Adrenergic Receptor; PDE GPCR/G Protein; Membrane transporter/Ion channel; Metabolism; Microbiology/Virology; Neuroscience
Glaucine 是从海罂粟中分离的一种生物碱,具有镇咳、抗炎和支气管扩张作用。它是具有口服活性的磷酸二酯酶 4 选择性抑制剂。它还是非选择性的 α-肾上腺素受体拮抗剂,具有抗氧化和抗病毒活性。
T0928 L-Ascorbic acid

维生素C,Vitamin C,Ascorbic acid,L(+)-Ascorbic acid,抗坏血酸,L-Ascorbate

Apoptosis; Calcium Channel; Reactive Oxygen Species; Endogenous Metabolite Apoptosis; Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; NF-κB
L-Ascorbic acid (Vitamin C) 属于天然产物,是一种强效的还原剂和抗氧化剂。L-Ascorbic acid 具有抗细菌感染、解毒反应和胶原蛋白形成的作用。L-Ascorbic acid 被用于治疗坏血病。
T3524 Halofuginone hydrobromide

卤夫酮溴氢酸盐,Tempostatin,RU-19110 (hydrobromide),Stenorol,常山酮溴酸盐

Others; Calcium Channel; DNA/RNA Synthesis; Sodium Channel; Parasite; TGF-beta/Smad Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Membrane transporter/Ion channel; Metabolism; Microbiology/Virology; Others; Stem Cells
Halofuginone hydrobromid 是Febrifugine 的衍生物,是竞争性脯氨酰-tRNA 合成酶抑制剂。它是 I 型胶原合成的特异性抑制剂,并通过抑制TGF-β活性可减轻骨关节炎。它具有抗疟疾、抗炎、抗癌、抗纤维化作用。
T3915 Ginsenoside Ro

人参皂苷Ro,Chikusetsusaponin 5,Polysciasaponin P3,人参皂苷 Ro,Chikusetsusaponin V

Calcium Channel; Reductase; Prostaglandin Receptor Endocrinology/Hormones; GPCR/G Protein; Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism
Ginsenoside Ro (Chikusetsusaponin V) 能降低 TXA2产量,较弱降低 COX-1 和 TXAS 活性,具有 Ca2+拮抗剂的抗血小板作用,IC50为 155 μM。
T2878 Ginsenoside Rd

Panaxoside Rd,Sanchinoside Rd,人参皂苷Rd,人参皂苷 Rd,Gypenoside VIII

P450; Calcium Channel; NF-κB; COX; Endogenous Metabolite Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; Neuroscience; NF-κB
Ginsenoside Rd (Gypenoside VIII) 抑制 TNFα 诱导的NF-κB 转录活性,还抑制COX-2和iNOSmRNA 的表达。它抑制CYP2D6、CYP1A2、CYP3A4和CYP2C9,也抑制Ca2+内流,有可能抑制或阻止肿瘤生长。
T3377 L-Phenylalanine

L-苯丙氨酸,(S)-2-Amino-3-phenylpropionic acid,phenylalanine,3-Phenyl-L-alanine

Calcium Channel; Endogenous Metabolite; iGluR Membrane transporter/Ion channel; Metabolism; Neuroscience
L-Phenylalanine (3-Phenyl-L-alanine) 是分离自大肠杆菌的必需氨基酸,是 NMDARs(KB573 μM) 和非 NMDARs 的甘氨酸和谷氨酸结合位点的竞争性拮抗剂,用于食品香料和药品的生产中。它是一种电压依赖性 α2δ 亚基 Ca2+通道拮抗剂,Ki 为 980 nM。
T2946 Tanshinone IIA sulfonate sodium

丹参酮IIA磺酸盐,丹参酮IIA-磺酸钠,Tanshinone IIA sulfonate,Sodium Tanshinone IIA sulfonate,Tanshinone IIA sodium sulfonate,sodium

CaMK; P450; Calcium Channel Membrane transporter/Ion channel; Metabolism; Neuroscience
Tanshinone IIA sulfonate sodium (Tanshinone IIA sodium sulfonate) 是从丹参中提取的丹参酮IIA 的水溶性衍生物,是SOCE 抑制剂,用于心血管疾病的研究。
T6674 L-Ascorbic acid sodium salt

(+)-Sodium L-ascorbate,Vitamin C sodium salt,Sodium ascorbate,L-Ascorbic acid sodium,抗坏血酸钠,Sodium L-ascorbate,维生素C钠

Apoptosis; Others; Calcium Channel; Reactive Oxygen Species; Endogenous Metabolite Apoptosis; Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; NF-κB; Others
L-Ascorbic acid sodium salt (Vitamin C sodium salt) 是一种电子供体,是一种内源性抗氧化剂。它还是一种胶原沉积促进剂和弹性生成抑制剂。它选择性抑制 Cav3.2 通道(Cav3.2 channels),IC50为 6.5 μM。
T23735 Jamaicin

An-Co-A4,AnCoA-4,An Co A4,AnCoA4

Calcium Channel Membrane transporter/Ion channel; Metabolism
Jamaicin (AnCoA4) 是一种从鸡血藤植物中提取的异黄酮,是一种 STIM1-Orai1 通道的抑制剂,可阻断钙离子流入,减少其与 STIM1 的相互作用,抑制 T 细胞的活化。
T0792 (-)-Sparteine sulfate pentahydrate

(-)-Sparteine Sulfate,Lupinidine sulfate pentahydrate,(-)-Sparteine sulfate salt,sulfate pentahydrate,五水合硫酸司巴丁

Sodium Channel Membrane transporter/Ion channel
(-)-Sparteine sulfate pentahydrate ((-)-Sparteine Sulfate) 是一种生物碱,是钠通道抑制剂,属于1a 类抗心律失常药。
T3S0807 Berbamine

CaMK; NF-κB; Autophagy Autophagy; Neuroscience; NF-κB
Berbamine 是从黄柏中提取的一种天然产物,是钙通道阻滞剂,具有抗肿瘤、免疫调节和心血管作用。
T75429 (±)-Liquiritigenin

(±)-4',7-Dihydroxyflavanone

Apoptosis; Calcium Channel Apoptosis; Membrane transporter/Ion channel; Metabolism
(±)-Liquiritigenin ((±)-4',7-Dihydroxyflavanone) 是从 Angelica keiskei 提取得到的类黄酮,抑制钙活化的氯离子通道TMEM16A。(±)-Liquiritigenin 诱导细胞凋亡增加和 Caspase3 活性增强。(±)-Liquiritigenin 可用于研究乳腺癌。
T3929 Kaurenoic acid

Kauren-19-Oic Acid,异贝壳杉烯酸,kaurenoate,kaur-16-en-18-oic acid

Others Others
Kaurenoic acid (kaurenoate) 是一种二萜,来源于 Sphagneticola trilobata 中,可以抑制细胞因子的产生和激活 NO–cyclic GMP–PKG–ATP- 敏感型钾通道信号通路,并抑制炎症疼痛。
T3S0209 Vincristine

ERK; p38 MAPK; NF-κB; Akt; JNK; mTOR Cytoskeletal Signaling; MAPK; NF-κB; PI3K/Akt/mTOR signaling
Vincristine 属于生物碱类天然产物,可与微管蛋白结合并抑制微管的形成,从而抑制肿瘤细胞的有丝分裂。Vincristine 可用作微管去稳定剂,用于研究治疗血液系统肿瘤,如白血病和淋巴瘤以及儿童肉瘤的相关研究。
T2163 Dihydrocapsaicin

CCRIS1589,二氢辣椒素,6,7-Dihydrocapsaicin,8-Methyl-N-vanillylnonanamide

Others; TRP/TRPV Channel Membrane transporter/Ion channel; Others
Dihydrocapsaicin (CCRIS1589) 是一种天然来源的辣椒素,是TRPV1的选择性激动剂,同时可以增加 p-Akt 水平。它可以增强低温诱导的神经保护。
TMA0763 Methyl 3,4,5-trimethoxycinnamate

Potassium Channel; Calcium Channel Membrane transporter/Ion channel; Metabolism
Methyl 3,4,5-trimethoxycinnamate may protect the heart from arrhythmias via its inhibitory effect on calcium channel.
T3029 Sparteine sulfate

硫酸司巴丁,Depasan,Tocosimplex,Actospar

Others; Sodium Channel Membrane transporter/Ion channel; Others
Sparteine sulfate (Tocosimplex) 是一种 1a 类抗心律失常药和钠通道阻滞剂。它可以螯合二价钙和镁。
T27564 Hymenidin

5-HT Receptor GPCR/G Protein; Neuroscience
Hymenidin是一种从冲绳海绵Hymeniacidon sp。中分离出的生物碱,是一种5-羟色胺能受体拮抗剂和电压门控钾通道抑制剂,具有潜在的抗原生动物作用,可选择性结合 FOXO1 DNA ,可降低去极化诱导的细胞钙升高。

天然产物

Cycleanine
Cat.No: T8206
Synonym:
Target: Others
Yangambin
Cat.No: TN2322
Synonym:
Target: Calcium Channel, PAFR
Praeruptorin C
Cat.No: T6S1418
Synonym:
Target: Antioxidant, Calcium Channel
Ionomycin calcium
Cat.No: T11665
Synonym: SQ23377 calcium,罗红霉素钙盐(链霉菌属载体)
Target: Apoptosis, Calcium Channel, Antibacterial, Antibiotic, PKC
Drotaverine hydrochloride
Cat.No: T8787
Synonym:
Target: PDE
Ethosuximide
Cat.No: T0728
Synonym: Zarontin,乙琥胺
Target: Calcium Channel
Gomisin J
Cat.No: T3904
Synonym:
Target: Calcium Channel, AMPK
Psoralenoside
Cat.No: TN1008
Synonym:
Target: CaMK, Calcium Channel, Histamine Receptor
Menthol
Cat.No: T5723
Synonym: 薄荷脑,DL-Menthol
Target: Others, Calcium Channel
Cyclopiazonic acid
Cat.No: T15027
Synonym: 环匹阿尼酸,环二氮酸
Target: Calcium Channel
Praeruptorin E
Cat.No: T4S1422
Synonym: 白花前胡素 E,白花前胡素E
Target: Others, Calcium Channel
Thapsigargin
Cat.No: TQ0302
Synonym: 毒胡萝卜素
Target: Apoptosis, SARS-CoV, Calcium Channel
Catharanthine tartrate
Cat.No: T3013
Synonym: Catharanthine hemitartrate,酒石酸长春质碱
Target: Others, Calcium Channel
Catharanthine
Cat.No: T2782
Synonym: (+)-3, 4-Didehydrocoronaridine,长春质碱,(+)-3,4-Didehydrocoronaridine
Target: Calcium Channel, AChR
(+)-Kavain
Cat.No: T4590
Synonym: 醉椒素,Kavain,L-KAWAIN,(R)-KAWAIN
Target: Calcium Channel, GABA Receptor, Sodium Channel, Monoamine Transporter
Ginsenoside Rf
Cat.No: T6S1500
Synonym: 人参皂苷 Rf,Ginsenoside-Rf,Panaxoside Rf
Target: Calcium Channel, Endogenous Metabolite
1-Octanol
Cat.No: T10024
Synonym: Octanol,正辛醇
Target: Calcium Channel, Endogenous Metabolite
Urolithin C
Cat.No: TN7108
Synonym:
Target: Apoptosis, Calcium Channel, Reactive Oxygen Species, IGF-1R, Endogenous Metabolite
Taurolithocholic acid sodium salt
Cat.No: T4727
Synonym: 牛磺石胆酸钠,Sodium taurolithocholate
Target: Others, Calcium Channel
Heteroclitin D
Cat.No: T3S1916
Synonym: 异型南五味子丁素,异南五味子丁素;异型南五味子丁素
Target: Calcium Channel
OPHIOPOGONIN D
Cat.No: T5701
Synonym: 麦冬皂苷 D,麦冬皂苷D
Target: RAAS, Calcium Channel, NF-κB, PPAR
Tetrandrine
Cat.No: T2996
Synonym: NSC-77037,d-Tetrandrine,Hanfangchin A,粉防己碱,Fanchinine,Sinomenine A,汉防己甲素
Target: Potassium Channel, Calcium Channel
Dronedarone
Cat.No: T7056
Synonym: 决奈达隆,SR 33589
Target: P450, Potassium Channel, Calcium Channel, Sodium Channel, Adrenergic Receptor, AChR, Autophagy
(±)-Praeruptorin A
Cat.No: T4S1419
Synonym: Praeruptorin A,(±)-白花前胡甲素,白花前胡甲素,(-)-Praeruptorin A
Target: p38 MAPK, Calcium Channel, Akt
Acetylcholine chloride
Cat.No: T1221
Synonym: ACh chloride,Pilofrin,氯化乙酰胆碱
Target: Calcium Channel, Endogenous Metabolite, AChR
14-Deoxyandrographolide
Cat.No: T8288
Synonym: 去氧穿心莲内酯,14-去氧穿心莲内酯
Target: Apoptosis, Others
Halofuginone
Cat.No: T6856
Synonym: 卤夫酮,常山酮,Tempostatin,empostatin,RU-19110
Target: Calcium Channel, DNA/RNA Synthesis, Sodium Channel, Parasite, TGF-beta/Smad
Glaucine
Cat.No: T5S2059
Synonym:
Target: Calcium Channel, Dopamine Receptor, Influenza Virus, Adrenergic Receptor, PDE
L-Ascorbic acid
Cat.No: T0928
Synonym: 维生素C,Vitamin C,Ascorbic acid,L(+)-Ascorbic acid,抗坏血酸,L-Ascorbate
Target: Apoptosis, Calcium Channel, Reactive Oxygen Species, Endogenous Metabolite
Halofuginone hydrobromide
Cat.No: T3524
Synonym: 卤夫酮溴氢酸盐,Tempostatin,RU-19110 (hydrobromide),Stenorol,常山酮溴酸盐
Target: Others, Calcium Channel, DNA/RNA Synthesis, Sodium Channel, Parasite, TGF-beta/Smad
Ginsenoside Ro
Cat.No: T3915
Synonym: 人参皂苷Ro,Chikusetsusaponin 5,Polysciasaponin P3,人参皂苷 Ro,Chikusetsusaponin V
Target: Calcium Channel, Reductase, Prostaglandin Receptor
Ginsenoside Rd
Cat.No: T2878
Synonym: Panaxoside Rd,Sanchinoside Rd,人参皂苷Rd,人参皂苷 Rd,Gypenoside VIII
Target: P450, Calcium Channel, NF-κB, COX, Endogenous Metabolite
L-Phenylalanine
Cat.No: T3377
Synonym: L-苯丙氨酸,(S)-2-Amino-3-phenylpropionic acid,phenylalanine,3-Phenyl-L-alanine
Target: Calcium Channel, Endogenous Metabolite, iGluR
Tanshinone IIA sulfonate sodium
Cat.No: T2946
Synonym: 丹参酮IIA磺酸盐,丹参酮IIA-磺酸钠,Tanshinone IIA sulfonate,Sodium Tanshinone IIA sulfonate,Tanshinone IIA sodium sulfonate,sodium
Target: CaMK, P450, Calcium Channel
L-Ascorbic acid sodium salt
Cat.No: T6674
Synonym: (+)-Sodium L-ascorbate,Vitamin C sodium salt,Sodium ascorbate,L-Ascorbic acid sodium,抗坏血酸钠,Sodium L-ascorbate,维生素C钠
Target: Apoptosis, Others, Calcium Channel, Reactive Oxygen Species, Endogenous Metabolite
Jamaicin
Cat.No: T23735
Synonym: An-Co-A4,AnCoA-4,An Co A4,AnCoA4
Target: Calcium Channel
(-)-Sparteine sulfate pentahydrate
Cat.No: T0792
Synonym: (-)-Sparteine Sulfate,Lupinidine sulfate pentahydrate,(-)-Sparteine sulfate salt,sulfate pentahydrate,五水合硫酸司巴丁
Target: Sodium Channel
Berbamine
Cat.No: T3S0807
Synonym:
Target: CaMK, NF-κB, Autophagy
(±)-Liquiritigenin
Cat.No: T75429
Synonym: (±)-4',7-Dihydroxyflavanone
Target: Apoptosis, Calcium Channel
Kaurenoic acid
Cat.No: T3929
Synonym: Kauren-19-Oic Acid,异贝壳杉烯酸,kaurenoate,kaur-16-en-18-oic acid
Target: Others
Vincristine
Cat.No: T3S0209
Synonym:
Target: ERK, p38 MAPK, NF-κB, Akt, JNK, mTOR
Dihydrocapsaicin
Cat.No: T2163
Synonym: CCRIS1589,二氢辣椒素,6,7-Dihydrocapsaicin,8-Methyl-N-vanillylnonanamide
Target: Others, TRP/TRPV Channel
Methyl 3,4,5-trimethoxycinnamate
Cat.No: TMA0763
Synonym:
Target: Potassium Channel, Calcium Channel
Sparteine sulfate
Cat.No: T3029
Synonym: 硫酸司巴丁,Depasan,Tocosimplex,Actospar
Target: Others, Sodium Channel
Hymenidin
Cat.No: T27564
Synonym:
Target: 5-HT Receptor
Cat. No. Product Name Species Expression System
TMPH-01279 CRACR2B Protein, Human, Recombinant (His)

CRACR2B,EFCAB4A,EF-hand calcium-binding domain-cont...

Human E. coli
Plays a role in store-operated Ca(2+) entry (SOCE).
TMPH-00780 CACNA1C Protein, Guinea Pig, Recombinant (His)

CACNA1C,CACNL1A1,CACH2,CACN2,Voltage-dependent L-type ca...

Guinea pig E. coli
Pore-forming, alpha-1C subunit of the voltage-gated calcium channel that gives rise to L-type calcium currents. Mediates influx of calcium ions into the cytoplasm, and thereby triggers calcium release from the sarcoplasm. Plays an important role in excitation-contraction coupling in the heart. Required for normal heart development and normal regulation of heart rhythm. Required for normal contraction of smooth muscle cells in blood vessels and in the intestine. Essential for normal blood pressur...
TMPH-02308 CACNA2D1 Protein, Human, Recombinant (His & SUMO)

MHS3,Voltage-dependent calcium channel sub...

Human E. coli
The alpha-2/delta subunit of voltage-dependent calcium channels regulates calcium current density and activation/inactivation kinetics of the calcium channel. Plays an important role in excitation-contraction coupling.
TMPH-01028 KCNMA1 Protein, Human, Recombinant

K(VCA)alpha,Calcium-activated potassium channel...

Human E. coli
KCNMA1 Protein, Human, Recombinant is expressed in E. coli expression system. The predicted molecular weight is 17.2 kDa and the accession number is Q12791.
TMPH-03750 SLC7A11 Protein, Human, Recombinant (His)

SLC7A11,Calcium channel blocker resistance...

Human E. coli
Sodium-independent, high-affinity exchange of anionic amino acids with high specificity for anionic form of cystine and glutamate.
TMPH-02551 CD20 Protein, Mouse, Recombinant (His)

Membrane-spanning 4-domains subfamily A member 1,CD20,B-lymp...

Mouse P. pastoris (Yeast)
B-lymphocyte-specific membrane protein that plays a role in the regulation of cellular calcium influx necessary for the development, differentiation, and activation of B-lymphocytes. Functions as a store-operated calcium (SOC) channel component promoting calcium influx after activation by the B-cell receptor/BCR. CD20 Protein, Mouse, Recombinant (His) is expressed in yeast with N-6xHis tag. The predicted molecular weight is 22.3 kDa and the accession number is P19437.
TMPY-03615 CSEN Protein, Human, Recombinant (His)

Kv channel interacting protein 3, calsenilin,DREAM,...

Human E. coli
KCNIP3 (Potassium Voltage-Gated Channel Interacting Protein 3, also known as CSEN) is a Protein Coding gene. CSEN is a member of the family of voltage-gated potassium (Kv) channel-interacting proteins, which belong to the recoverin branch of the EF-hand superfamily. Members of this family are integral subunit components of native Kv4 channel complexes that may regulate A-type currents, and hence neuronal excitability, in response to changes in intracellular calcium. CSEN also functions as a calc...
TMPH-00344 CD20 Protein, Canine, Recombinant (His & Myc)

MS4A1,Membrane-spanning 4-domains subfamily A member 1,CD20,...

Canine E. coli
B-lymphocyte-specific membrane protein that plays a role in the regulation of cellular calcium influx necessary for the development, differentiation, and activation of B-lymphocytes. Functions as a store-operated calcium (SOC) channel component promoting calcium influx after activation by the B-cell receptor/BCR. CD20 Protein, Canine, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 17.4 kDa and the accession number ...
TMPJ-00888 ANXA7 Protein, Human, Recombinant

Annexin A7,Annexin-7,Synexin,ANXA7,Annexin VII,SNX,ANX7

Human E. coli
Annexin A7 (ANXA7) is a member of the annexin family of calcium-dependent phospholipid binding proteins. Annexin A7 has a unique, highly hydrophobic N-terminal domain and a conserved C-terminal region. The C-terminal region is composed of alternating hydrophobic and hydrophilic segments. Annexin A7 is a calcium/phospholipid-binding protein with diverse properties including voltage-sensitive calcium channel activity and promotes membrane fusion and is also involved in exocytosis.
TMPH-02905 TRPC1 Protein, Mouse, Recombinant (His)

Transient receptor protein 1,Short transient receptor potent...

Mouse E. coli
Thought to form a receptor-activated non-selective calcium permeant cation channel. Probably is operated by a phosphatidylinositol second messenger system activated by receptor tyrosine kinases or G-protein coupled receptors. Seems to be also activated by intracellular calcium store depletion. TRPC1 Protein, Mouse, Recombinant (His) is expressed in E. coli expression system with N-10xHis tag. The predicted molecular weight is 94.0 kDa and the accession number is Q61056.
TMPH-01394 GRIN1 Protein, Human, Recombinant (His)

N-methyl-D-aspartate receptor subunit NR1,Glutamate [NMDA] r...

Human E. coli
Component of NMDA receptor complexes that function as heterotetrameric, ligand-gated ion channels with high calcium permeability and voltage-dependent sensitivity to magnesium. Channel activation requires binding of the neurotransmitter glutamate to the epsilon subunit, glycine binding to the zeta subunit, plus membrane depolarization to eliminate channel inhibition by Mg(2+). Sensitivity to glutamate and channel kinetics depend on the subunit composition. GRIN1 Protein, Human, Recombinant (His)...
TMPH-02336 TAS2R10 Protein, Human, Recombinant (His & KSI)

Taste receptor family B member 2,Taste receptor type 2 membe...

Human E. coli
Gustducin-coupled strychnine receptor implicated in the perception of bitter compounds in the oral cavity and the gastrointestinal tract. Signals through PLCB2 and the calcium-regulated cation channel TRPM5. TAS2R10 Protein, Human, Recombinant (His & KSI) is expressed in E. coli expression system with N-6xHis-KSI tag. The predicted molecular weight is 19.6 kDa and the accession number is Q9NYW0.
TMPY-03438 Calsequestrin 1 Protein, Human, Recombinant

CASQ,PDIB1,VMCQA,calsequestrin 1 (fast-twitch, skeletal musc...

Human E. coli
Calsequestrin-1 is an isoform of calsequestrin. Calsequestrin is a calcium-binding protein of the sarcoplasmic reticulum. It helps hold calcium in the cisterna of the sarcoplasmic reticulum after a muscle contraction, even though the concentration of calcium in the sarcoplasmic reticulum is much higher than in the cytosol. Two forms of calsequestrin have been identified: Calsequestrin-2 and Calsequestrin-1. Calsequestrin-1 is found in fast skeletal muscle. The release of calsequestrin-boun...
TMPY-02955 CABP5 Protein, Human, Recombinant (His)

calcium binding protein 5,CABP3

Human E. coli
CABP3, also known as CABP5, belongs to a subfamily of calcium binding proteins, which share similarity to calmodulin. Calcium binding proteins are an important component of calcium mediated cellular signal transduction. Expression of CABP3 gene is retina-specific. The mouse homolog of CABP3 has been shown to express in the inner nuclear layer of the retina, suggested its role in neuronal functioning. The specific function of CABP3 gene is unknown. Study of the transcripts and genomic structure r...
TMPH-03390 TRPV2 Protein, Rat, Recombinant (His)

Transient receptor potential cation channel subfami...

Rat E. coli
Calcium-permeable, non-selective cation channel with an outward rectification. Seems to be regulated, at least in part, by growth factors, like IGF1, PDGF and morphogenetic neuropeptide/head activator. May transduce physical stimuli in mast cells. Activated by temperatures higher than 52 degrees Celsius; is not activated by vanilloids and acidic pH. TRPV2 Protein, Rat, Recombinant (His) is expressed in E. coli expression system with N-10xHis tag. The predicted molecular weight is 88.2 kDa and th...
TMPJ-00666 CLIC2 Protein, Human, Recombinant (His)

CLIC2,XAP121,Chloride Intracellular Channel Protein...

Human E. coli
Chloride Intracellular Channel Protein 2 (CLIC2) is a critical component of all living cells; it regulatescellular traffic of Chloride ion and it can be inserted into membranes anf form chloride ion channels. Membrane insertion seems to be redox-regulated and may occur only under oxydizing conditions, channel activity depends on the pH. CLIC2 is involved in regulating membrane potential and organic solute transport. CLIC2 modulates the activity of RYR2 and inhibits Calcium influx. CLIC2 can be d...
TMPJ-01074 PKCE Protein, Human, Recombinant (His)

PRKCE,PKCE,nPKC-ε,nPKC-Epsilon,Protein Kinase C Epsilon Type...

Human E. coli
Protein Kinase C Epsilon type is a member of the serine- and threonine-specific protein kinase family that can be activated by calcium and the second messenger diacylglycerol. Protein Kinase C Epsilon contains these domains: one AGC-kinase C-terminal domain, one C2 domain, one protein kinase domain and two phorbol-ester/DAG-type zinc fingers. Protein Kinase C Epsilon phosphorylate a variety of protein targets and has been identified to participate in diverse cellular signaling pathways. It has m...
TMPY-01605 STIM1 Protein, Human, Recombinant (His)

stromal interaction molecule 1,TAM1,GOK,STRMK,IMD10,D11S4896...

Human HEK293 Cells
Stromal interaction molecule 1, also known as STIM1 and GOK, is a cell membrane, a single-pass type I membrane protein and a endoplasmic reticulum membrane protein. STIM1 / GOK is ubiquitously expressed in various human primary cells and tumor cell lines. It contains one EF-hand domain and one SAM (sterile alpha motif) domain. STIM1 / GOK plays a role in mediating Ca2+influx following depletion of intracellular Ca2+stores. It acts as Ca2+sensor in the endoplasmic reticulum via its EF-hand domain...
TMPH-03753 MYLK Protein, Human, Recombinant (His)

MYLK,Myosin light chain kinase, smooth muscle,Telokin,Kinase...

Human E. coli
Calcium/calmodulin-dependent myosin light chain kinase implicated in smooth muscle contraction via phosphorylation of myosin light chains (MLC). Also regulates actin-myosin interaction through a non-kinase activity. Phosphorylates PTK2B/PYK2 and myosin light-chains. Involved in the inflammatory response (e.g. apoptosis, vascular permeability, leukocyte diapedesis), cell motility and morphology, airway hyperreactivity and other activities relevant to asthma. Required for tonic airway smooth muscl...

重组蛋白

CRACR2B Protein, Human, Recombinant (His)
Cat.No: TMPH-01279
Species: Human
Expression System: E. coli
CACNA1C Protein, Guinea Pig, Recombinant (His)
Cat.No: TMPH-00780
Species: Guinea pig
Expression System: E. coli
CACNA2D1 Protein, Human, Recombinant (His & SUMO)
Cat.No: TMPH-02308
Species: Human
Expression System: E. coli
KCNMA1 Protein, Human, Recombinant
Cat.No: TMPH-01028
Species: Human
Expression System: E. coli
SLC7A11 Protein, Human, Recombinant (His)
Cat.No: TMPH-03750
Species: Human
Expression System: E. coli
CD20 Protein, Mouse, Recombinant (His)
Cat.No: TMPH-02551
Species: Mouse
Expression System: P. pastoris (Yeast)
CSEN Protein, Human, Recombinant (His)
Cat.No: TMPY-03615
Species: Human
Expression System: E. coli
CD20 Protein, Canine, Recombinant (His & Myc)
Cat.No: TMPH-00344
Species: Canine
Expression System: E. coli
ANXA7 Protein, Human, Recombinant
Cat.No: TMPJ-00888
Species: Human
Expression System: E. coli
TRPC1 Protein, Mouse, Recombinant (His)
Cat.No: TMPH-02905
Species: Mouse
Expression System: E. coli
GRIN1 Protein, Human, Recombinant (His)
Cat.No: TMPH-01394
Species: Human
Expression System: E. coli
TAS2R10 Protein, Human, Recombinant (His & KSI)
Cat.No: TMPH-02336
Species: Human
Expression System: E. coli
Calsequestrin 1 Protein, Human, Recombinant
Cat.No: TMPY-03438
Species: Human
Expression System: E. coli
CABP5 Protein, Human, Recombinant (His)
Cat.No: TMPY-02955
Species: Human
Expression System: E. coli
TRPV2 Protein, Rat, Recombinant (His)
Cat.No: TMPH-03390
Species: Rat
Expression System: E. coli
CLIC2 Protein, Human, Recombinant (His)
Cat.No: TMPJ-00666
Species: Human
Expression System: E. coli
PKCE Protein, Human, Recombinant (His)
Cat.No: TMPJ-01074
Species: Human
Expression System: E. coli
STIM1 Protein, Human, Recombinant (His)
Cat.No: TMPY-01605
Species: Human
Expression System: HEK293 Cells
MYLK Protein, Human, Recombinant (His)
Cat.No: TMPH-03753
Species: Human
Expression System: E. coli
Cat. No. Product Name Target Signaling Pathways
T40376 L-Phenylalanine-15N

L-苯丙氨酸 15N,(S)-2-Amino-3-phenylpropionic acid-15N,L-Phenylalanine-15N

Calcium Channel Membrane transporter/Ion channel; Metabolism
L-Phenylalanine-15N ((S)-2-Amino-3-phenylpropionic acid-15N) 是 15N 标记的 L-Phenylalanine。L-Phenylalanine 是从大肠杆菌中分离出来的一种必需氨基酸。 L-Phenylalanine 广泛用于食品香精和药物的生产。
T12222 Nifedipine-d6

硝苯地平 D6,Nifedipine D6,BAY-a-1040 D6

Others Others
Nifedipine D6 is deuterium labeled nifedipine which is a potent blocker of calcium channel.
T10439 Azelnidipine D7

CS-905 D7

Others Others
Azelnidipine D7 is a deuterium-labeled Azelnidipine. Azelnidipine is an L-type calcium channel blocker.
T10816 Cinnarizine D8

Others Others
Cinnarizine D8 is a deuterium-labeled Cinnarizine which is an antihistamine and a calcium channel blocker.
T12625 (R)-Lercanidipine-d3 hydrochloride

(R)-Lercanidipine D3 hydrochloride

Calcium Channel Membrane transporter/Ion channel; Metabolism
(R)-lercanidipine D3 hydrochloride is a deuterium labeled (R)-Lercanidipine hydrochloride. (R)-Lercanidipine D3 (hydrochloride) is a calcium channel blocker.
T12243 Norverapamil-d7

D591 D7,(±)-Norverapamil D7

Others Others
Norverapamil D7 is a deuterium labeled Norverapamil . Norverapamil is a blocker of L-type calcium channel and an inhibitor of P-glycoprotein (P-gp) function .
TMIH-0087 Amlodipine-d4 Maleate (Racemic)

Amlodipine-d4 Maleate (Racemic) 是 Amlodipine Maleate (Racemic) 的氘代化合物。Amlodipine Maleate (Racemic) 的 CAS 号为 88150-47-4。Amlodipine maleate是一种具有口服活性的二氢吡啶类钙通道阻滞剂,通过阻滞电压依赖性L型钙通道,从而抑制钙离子内流。Amlodipine maleate可用于研究高血压和癌症。
TMIH-0107 Barnidipine-d5

Barnidipine-d5 是 Barnidipine 的氘代化合物。Barnidipine 的 CAS 号为 104713-75-9。Barnidipine 是一种二氢吡啶类钙通道阻滞剂,对 CaA 受体具有选择性作用。它是一种抗高血压药物,通过减少其血管扩张作用继发的外周血管阻力起作用。
TMIJ-0095 Nimodipine-d7

Nimodipine-d7 是 Nimodipine 的氘代化合物。Nimodipine 的 CAS 号为 66085-59-4。Nimodipine 是一种具有口服活性,耐受性良好的光敏二氢吡啶钙拮抗剂。它可研究脑血管疾病。
TMIJ-0187 Lercanidipine-13C-d3 HCl

Lercanidipine-13C-d3 HCl 是 Lercanidipine HCl 的 13C 和氘代化合物。Lercanidipine HCl 的 CAS 号为 132866-11-6。Lercanidipine hydrochloride 是亲脂性二氢吡啶-钙通道阻滞剂,具有持久的降压作用和保护肾脏作用。
TMIH-0002 (+/-)-Verapamil hydrochloride-d7

(+/-)-Verapamil hydrochloride-d7 是 (+/-)-Verapamil hydrochloride 的氘代化合物。(+/-)-Verapamil hydrochloride 的 CAS 号为 152-11-4。Verapamil hydrochloride 是一种钙通道阻滞剂,是一种可口服的 P 糖蛋白 (P-gp) 抑制剂,可抑制CYP3A4,用于高血压、心律不齐和心绞痛的研究。
TMIJ-0140 Felodipine-d5

Felodipine-d5 是 Felodipine 的氘代化合物。Felodipine 的 CAS 号为 72509-76-3。Felodipine 是一种长效的 1, 4-二氢吡啶钙通道抑制剂,可跨越血脑屏障,可诱导自噬,具有抗高血压活性。它通过选择性作用于血管平滑肌,尤其是阻力血管来降低血压。
TMIJ-0285 Verapamil-d7 Hydrochloride

Verapamil-d7 Hydrochloride 是 Verapamil Hydrochloride 的氘代化合物。Verapamil Hydrochloride 的 CAS 号为 152-11-4。Verapamil hydrochloride 是一种钙通道阻滞剂,是一种可口服的 P 糖蛋白 (P-gp) 抑制剂,可抑制CYP3A4,用于高血压、心律不齐和心绞痛的研究。
TMIJ-0270 Pinaverium-d4 Bromide (Mixture of Diastereomers)

Pinaverium-d4 Bromide (Mixture of Diastereomers) 是 Pinaverium Bromide 的氘代化合物。Pinaverium Bromide 的 CAS 号为 53251-94-8。Pinaverium bromide 是一种具有解痉作用的钙通道阻滞剂,可有效缓解疼痛、腹泻和肠道不适。
TMIH-0399 Norverapamil-d7 HCl

Norverapamil-d7 HCl 是 Norverapamil HCl 的氘代化合物。Norverapamil HCl 的 CAS 号为 67812-42-4。Norverapamil hydrochloride是 Verapamil 的 N-去甲基代谢物,是L型钙通道阻滞剂和 P-糖蛋白 (P-gp) 功能抑制剂。
TMIJ-0077 Clevidipine-d7

Clevidipine-d7 是 Clevidipine 的氘代化合物。Clevidipine 的 CAS 号为 167221-71-8。Clevidipine butyrate 是一种二氢吡啶 L 型钙通道阻滞剂,IC50为7.1 nM。它对血管平滑肌有选择性,可用于降低血压。
T71303 Flufenamic Acid-d4

Flufenamic acid-d4 is intended for use as an internal standard for the quantification of flufenamic acid by GC- or LC-MS. Flufenamic acid is a non-steroidal anti-inflammatory drug (NSAID) and COX inhibitor (IC50s = 3 and 9.3 µM for human COX-1 and COX-2, respectively). Flufenamic acid inhibits TNF-α-induced increases in COX-2 levels and NF-κB activation in HT-29 colon cancer cells in a concentration-dependent manner. It inhibits calcium influx induced by fMLP or A23187 in human polymorphonuclear...
TMIJ-0141 (S)-Amlodipine-d4

(S)-Amlodipine-d4 是 (S)-Amlodipine 的氘代化合物。(S)-Amlodipine 的 CAS 号为 103129-82-4。Levamlodipine 是一种二氢吡啶钙通道阻滞剂,具有舒张血管的作用,可用于高血压和心绞痛的研究。
TMIJ-0252 Benazeprilat-d5

Benazepril EP Impurity C-d5

Benazeprilat-d5 是 Benazeprilat 的氘代化合物。Benazeprilat 的 CAS 号为 86541-78-8。Benazeprilat(CGS 14831) 是一种具有口服活性的贝那普利活性代谢物。Benazeprilat 具有高效的抗血压活性,可与其他其他类别的化合物(包括噻嗪类利尿剂和钙通道阻滞剂)联合使用来减少与心血管风险和继发性终末器官损伤相关的疾病的发生。Benazeprilat 可能用于研究急性左心室衰竭。
TMID-0299 Zonisamide-d4

Zonisamide-d4 是 Zonisamide 的氘代化合物。Zonisamide 的 CAS 号为 68291-97-4。Zonisamide 是锌酶碳酸酐酶 (carbonic anhydrase) 的有效抑制剂,对人类线粒体同工酶 hCA II 和 hCA V 作用的Ki值分别为 35.2 nM 和 20.6 nM。Zonisamide 具有抗癫痫活性,在癫痫、癫痫发作和帕金森病的研究中具有价值。
T37847 Zonisamide-13C2,15N

Zonisamide-13C2,15N

Zonisamide-13C2,15N is intended for use as an internal standard for the quantification of zonisamide by GC- or LC-MS. Zonisamide is an antiepileptic agent.1 It selectively inhibits the repeated firing of sodium channels (IC50 = 2 μg/ml) in mouse embryo spinal cord neurons and inhibits spontaneous channel firing when used at concentrations greater than 10 μg/ml.2 In rat cerebral cortex neurons, zonisamide (1-1,000 μM) inhibits T-type calcium channels with a maximum reduction of 60% of the calcium...

同位素标记化合物

L-Phenylalanine-15N
Cat.No: T40376
Synonym: L-苯丙氨酸 15N,(S)-2-Amino-3-phenylpropionic acid-15N,L-Phenylalanine-15N
Target: Calcium Channel
Nifedipine-d6
Cat.No: T12222
Synonym: 硝苯地平 D6,Nifedipine D6,BAY-a-1040 D6
Target: Others
Azelnidipine D7
Cat.No: T10439
Synonym: CS-905 D7
Target: Others
Cinnarizine D8
Cat.No: T10816
Synonym:
Target: Others
(R)-Lercanidipine-d3 hydrochloride
Cat.No: T12625
Synonym: (R)-Lercanidipine D3 hydrochloride
Target: Calcium Channel
Norverapamil-d7
Cat.No: T12243
Synonym: D591 D7,(±)-Norverapamil D7
Target: Others
Amlodipine-d4 Maleate (Racemic)
Cat.No: TMIH-0087
Synonym:
Target:
Barnidipine-d5
Cat.No: TMIH-0107
Synonym:
Target:
Nimodipine-d7
Cat.No: TMIJ-0095
Synonym:
Target:
Lercanidipine-13C-d3 HCl
Cat.No: TMIJ-0187
Synonym:
Target:
(+/-)-Verapamil hydrochloride-d7
Cat.No: TMIH-0002
Synonym:
Target:
Felodipine-d5
Cat.No: TMIJ-0140
Synonym:
Target:
Verapamil-d7 Hydrochloride
Cat.No: TMIJ-0285
Synonym:
Target:
Pinaverium-d4 Bromide (Mixture of Diastereomers)
Cat.No: TMIJ-0270
Synonym:
Target:
Norverapamil-d7 HCl
Cat.No: TMIH-0399
Synonym:
Target:
Clevidipine-d7
Cat.No: TMIJ-0077
Synonym:
Target:
Flufenamic Acid-d4
Cat.No: T71303
Synonym:
Target:
(S)-Amlodipine-d4
Cat.No: TMIJ-0141
Synonym:
Target:
Benazeprilat-d5
Cat.No: TMIJ-0252
Synonym: Benazepril EP Impurity C-d5
Target:
Zonisamide-d4
Cat.No: TMID-0299
Synonym:
Target:
Zonisamide-13C2,15N
Cat.No: T37847
Synonym: Zonisamide-13C2,15N
Target:
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