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规格 | 价格 | 库存 | 数量 |
---|---|---|---|
1 mg | ¥ 798 | 现货 | |
5 mg | ¥ 1,990 | 现货 | |
10 mg | ¥ 2,920 | 现货 | |
25 mg | ¥ 4,590 | 现货 | |
50 mg | ¥ 5,920 | 现货 | |
100 mg | ¥ 8,330 | 现货 | |
200 mg | ¥ 11,200 | 现货 |
产品描述 | CALP3 acetate is a potent Ca2+ channel blocker that activates EF hand motifs of Ca2+-binding proteins. CALP3 acetate can functionally mimic increased [Ca2+]i by modulating the activity of Calmodulin (CaM), Ca2+ channels and pumps. |
体外活性 | CALP3以剂量依赖的方式抑制了谷氨酸引起的长时间大幅度增加Fura-2负载神经细胞中的[Ca2+]i(IC50=37.25 μM)。同样,CALP3以剂量依赖的方式抑制了谷氨酸诱导的大鼠新皮质神经元培养细胞的细胞毒性(IC50=50.97 μM),以及剂量依赖性抑制细胞凋亡(IC50=33.41 μM)。CALP3(100 μM)抑制由HIV gp120和SAg在人T细胞中诱导的细胞凋亡。此外,CALP3(100 μM;15分钟预处理)降低了棉酚引起的坏死,提高了活细胞的比例[1][2]。 |
分子量 | 941.12 |
分子式 | C46H72N10O11 |
CAS No. |
存储 | keep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
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