首页 工具
登录
购物车

搜索结果

Search Results for " salt "
Targets Recommended: cholecystokinin

1165

抑制剂 & 化合物

189

天然产物

2

TargetMol 试剂盒

6

重组蛋白

46

同位素标记化合物

如果没找到您满意的产品或者您对产品有其他要求,可以联系我们专业顾问为您提供针对性的合理建议。     QQ咨询       网站留言咨询

提交您的定制咨询

点击图片重新获取验证码
Cat. No. Product Name Form Specificity Of Inhibition
C0005 Cell Counting Kit-8 (CCK-8)

Cell Counting Kit-8 (CCK-8)

Solution in bottle
C0052 Penicillin-Streptomycin-Amphotericin B Solution (100×), Sterile

青霉素-链霉素-两性霉素B三抗溶液(100×),灭菌

Solution in bottle

TargetMol 试剂盒

Cell Counting Kit-8 (CCK-8)
Cat.No: C0005
青霉素-链霉素-两性霉素B三抗溶液(100×),灭菌
Cat.No: C0052
Cat. No. Product Name Target Signaling Pathways
T14932L1 Ceruletide Ammonium Salt

Caerulein Ammonium Salt,Ceruletide Ammonium Salt(17650-98-5 Free base),FI-6934 Ammonium Salt,Cerulein Ammonium Salt

cholecystokinin GPCR/G Protein
Ceruletide Ammonium Salt 是一种十肽,起源于热带青蛙的皮肤,是一种有效的胆囊收缩素受体 (cholecystokinin receptor) 激动剂,也是一种安全有效的胆囊收缩剂,对胆囊肌肉和胆管有直接的痉挛性作用。Ceruletide Ammonium Salt 具有镇静活性,可用于研究慢性精神分裂症。
T15024 Silmitasertib sodium salt

CX-4945 sodium salt

Casein Kinase; Autophagy Autophagy; Metabolism; Stem Cells
Silmitasertib sodium salt (CX-4945 sodium salt) 是一种可口服的高度选择性 CK2抑制剂,对 CK2α 和 CK2α' 的 IC50值均为 1 nM。
TP1111L1 Tirzepatide sodium salt

LY-3298176 sodium salt,Tirzepatide sodium salt(2023788-19-2 free base)

Glucagon Receptor GPCR/G Protein
Tirzepatide sodium salt (LY3298176 sodium salt) 是新型 GIP 和 GLP-1 受体双重激动剂,是人类GIP激素的合成肽类似物。Tirzepatide 具有神经保护活性,可以用于预防和治疗 2 型糖尿病和肥胖症。
T11868 Lorglumide sodium salt

CR-1409 sodium salt

cholecystokinin GPCR/G Protein
Lorglumide sodium salt (CR-1409 sodium salt) 是胆囊收缩素受体 (CCK) 的拮抗剂。
T10397 ATN-161 trifluoroacetate salt

ATN-161 TFA salt

Integrin Cytoskeletal Signaling
ATN-161 trifluoroacetate salt (ATN-161 TFA salt) 是一种新型整合素 α5β1 拮抗剂,可在小鼠模型中抑制血管生成和肝转移瘤的生长。
T4200 Sacubitril hemicalcium salt

AHU-377 (hemicalcium salt),LCZ696中间体,AHU377 calcium salt

Neprilysin Metabolism
Sacubitril hemicalcium salt (AHU377 calcium salt) 是一种有效的 NEP 抑制剂,IC50=5 nM。它是研究心力衰竭药物 LCZ696 的组分之一。
T17210L Vaborbactam ammonium salt

RPX7009 ammonium salt,Vaborbactam ammonium salt(1360457-46-0 Free base)

Antibacterial Microbiology/Virology
Vaborbactam ammonium salt 是一种 β-内酰胺酶抑制剂,可以恢复碳青霉烯类药物对 KPC 生产菌株的活性,常与其它药物连用来研究真菌感染。
T76279L1 Retatrutide sodium salt

Retatrutide sodium salt(2381089-83-2 free base),LY3437943 sodium salt

Glucagon Receptor GPCR/G Protein
Retatrutide sodium salt 是一种有效的胰高血糖素受体 (GCGR)、葡萄糖依赖性促胰岛素多肽受体 (GIPR) 和胰高血糖素样肽-1 受体 (GLP-1R) 的三重激动剂肽。Retatrutide sodium salt 可用于研究2型糖尿病和肥胖症。
T33565 NAAD sodium salt

NAAD钠盐,NAAD Na salt,Deamido Nad Sodium Salt,NAAD Na, NaAD

Others Others
NAAD sodium salt (NAAD Na salt) 是烟酰胺腺嘌呤二核苷酸合酶的底物,可用于研究底物的特异性和动力学。
T4535 Etomoxir sodium salt

(R)-(+)-乙莫克舍钠盐,(R)-Etomoxir sodium salt,Na salt,Etomoxir

Apoptosis; Others Apoptosis; Others
Etomoxir sodium salt ((R)-Etomoxir sodium salt) 是一种肉碱棕榈酰转移酶 1a (CPT-1a) 抑制剂,可以阻断脂肪酸合成。Etomoxir sodium salt 具有抗肿瘤活性。
T11315 Fosmidomycin sodium salt

FR-31564 sodium salt

Antibiotic; Parasite Microbiology/Virology
Fosmidomycin sodium salt (FR-31564 sodium salt) 是一种抗感染类抗生素,具有抗疟疾活性,抑制革兰氏阴性菌和革兰氏阳性菌。
T65070 Chenodeoxycholic Acid sodium salt

CDCA sodium salt

FXR Metabolism
Chenodeoxycholic Acid sodium salt (CDCA sodium salt) 是一种人体中的胆汁酸,能够活化核受体 FXR,可挽救痉挛性截瘫 5 型和脑黄瘤病患者诱导多能干细胞衍生神经元的轴突变性,可用于研究胰腺坏死。
T21537L TMC647055 Choline Hydroxide Salt

TMC647055 Choline Hydroxide Salt (1204416-97-6 free base)

HCV Protease Microbiology/Virology; Proteases/Proteasome
TMC647055 Choline Hydroxide Salt 是一种新型有效的 HCV NS5B 聚合酶非核苷抑制剂,可用于治疗 HCV 感染。它具有纳摩尔级细胞效力(EC(50) 为 82 nM),相关细胞毒性较小(CC(50)>20 μM),在大鼠和狗中具有良好的药代动力学特征。 TMC647055 显示出有体外生化、动力学和病毒学特征的前景。
TP1101 Nonapeptide-1 acetate salt (158563-45-2 free base)

Melanostatine-5 acetate salt,Nonapeptide-1 acetate salt

Melanocortin Receptor GPCR/G Protein; Neuroscience
Nonapeptide-1 acetate salt (158563-45-2 free base) (Melanostatine-5 acetate salt) 是一种肽激素,是一种有效的 α-黑色素细胞刺激素 (α-MSH) 拮抗剂,IC50 为 11 nM。
T22592 ATPγS tetralithium salt

ATP-gamma-S tetralithium salt

PERK Apoptosis
ATPγS tetralithium salt 是真核生物翻译起始因子 eIF4A 的核苷酸水解和RNA解链活性的底物,与 p97 突变体和朊病毒相关。
T11511 Guanosine-5'-triphosphate disodium salt

GTP disodium,5'-GTP disodium salt

Others; Endogenous Metabolite Metabolism; Others
Guanosine-5'-triphosphate disodium salt (5'-GTP disodium salt) 是肌原性细胞分化的增强剂,也是翻译和其他重要细胞过程的能量来源。
T15025L CY5 triethylamine salt

CY5 triethylamine salt(146368-11-8 Free base)

Others Others
CY5 triethylamine salt 是一种水溶性染料,激发光波长(nm):649,发射波长(nm):670。
T36688 Deoxyguanosine triphosphate trisodium salt

Deoxyguanosine 5-triphosphate,2'-Deoxyguanosine-5'-triphosphate trisodium salt,dGTP trisodium salt

Nucleoside Antimetabolite/Analog Cell Cycle/Checkpoint; DNA Damage/DNA Repair
Deoxyguanosine triphosphate trisodium salt (2'-Deoxyguanosine-5'-triphosphate trisodium salt) 是细胞中用于 DNA 合成的核苷酸前体,可用于逆转录聚合酶链反应 (RT-PCR) 中以进行 DNA 扩增。
T84284 dITP trisodium salt

2'-Deoxyinosine-5'-triphosphate trisodium salt

Others Others
dITP trisodium salt (2'-Deoxyinosine-5'-triphosphate trisodium salt) 存在于超嗜热细菌 Thermotoga maritima 中,可在诱变PCR中用作突变试剂。
TP1457 BIO-11006 acetate salt (901117-03-1 free base)

BIO-11006 acetate salt

Others Others
BIO-11006 acetate salt (901117-03-1 free base) 是一种多糖基化富含丙氨酸的 C 激酶底物 (MARCKS) 抑制剂,类似于 MANS 肽。
T10851 CMP-Sialic acid sodium salt

CMP-Neu5Ac sodium salt

Endogenous Metabolite Metabolism
CMP-Sialic acid sodium salt (CMP-Neu5Ac sodium salt) 是 UDP-GlcNAc 2-epimerase 的变构抑制剂,是唾液酸的活化形式,广泛存在于动物体内,参与生物体的代谢。
T18910 Acid Yellow 9 monosodium salt

Hydrogen 4-aminoazobenzene-3,4'-disulphonate (sodium salt)

Others Others
Acid Yellow 9 monosodium salt (Hydrogen 4-aminoazobenzene-3,4'-disulphonate (sodium salt)) 是一种可被Pseudomonas fluorescens 降解的含氮染料,是此类菌株碳、氮和能量的唯一来源。
T10759 CEP-28122 mesylate salt (1022958-60-6 free base)

CEP-28122 mesylate salt

ALK Angiogenesis; Tyrosine Kinase/Adaptors
CEP-28122 mesylate salt (1022958-60-6 free base) 是一种高选择性的口服活性 ALK 抑制剂(在基于酶的 TRF 测定中,IC50:1.9 nM)。
T16734L Resorufin sodium salt

试卤灵钠盐,NSC 12097 sodium salt

Others Others
Resorufin sodium salt (NSC-12097 sodium salt) 是高荧光的粉红色染料,可用于 ROS/RNS 和第二种分析物的检测。
T68019L Ursulcholic acid trisodium salt

Ursodeoxycholic acid disulfate trisodium salt,Ursulcholic acid trisodium salt(88426-32-8 Free base)

Others Others
Ursulcholic acid trisodium salt (Ursodeoxycholic acid disulfate trisodium salt) 是 ursodeoxycholic acid 的可溶形式,ursodeoxycholic acid 具有抗高血脂和利胆活性活性。
T33795 3-OMFP Cyclohexylammonium salt

OMFP Cyclohexylammonium salt

Others Others
3-OMFP Cyclohexylammonium salt (OMFP Cyclohexylammonium salt) 是 PTEN 抑制研究的底物,可用来测定CDC25B催化结构域的酶活性。
T11125 Durlobactam sodium salt

杜巴坦,ETX2514 sodium salt,杜洛巴坦

Antibacterial Microbiology/Virology
Durlobactam sodium salt (ETX2514 sodium salt)是一种 β-内酰胺酶抑制剂,针对 A 类 KPC-2、C 类 AmpC 和 D 类 OXA-24,IC50 值分别为 4 nM、14 nM 和 190 nM。 Durlobactam sodium salt 可用于对包括鲍曼不动杆菌在内的耐药革兰氏阴性菌的研究。
T30677L C15AlkOPP t-BA salt

C15AlkOPP t-BA salt(946615-44-7 Free base),C15AlkOPP Tetrabutylamine salt(946615-44-7 Free base)

Others Others
C15AlkOPP Tetrabutylamine salt 是一种"可点击"的farnesyl diphosphate (FPP)的炔烃修饰类似物。
T19820 MOPS sodium salt

MOPS-Na,3-(N-morpholino)propanesulfonic acid sodium salt,3-吗啉丙磺酸钠盐,Sodium 3-Morpholinopropanesulfonate,4-Morpholinepropanesulfonic acid, sodium salt

Others Others
MOPS sodium salt (MOPS-Na) 在生物学中常用作缓冲剂。其中MOPS 缓冲液能使哺乳动物细胞培养基的 pH 值保持稳定。
TP1565L1 Foxy-5 Ammonium Salt

Foxy-5 Ammonium Salt(881188-51-8 Free base)

Wnt/beta-catenin Cytoskeletal Signaling; Stem Cells
Foxy-5 Ammonium Salt是 WNT5A 激动剂,是 WNT5A 的一个模拟肽,是 Wnt 家族的非经典成员。Foxy-5 Ammonium Salt可在不影响 β-catenin 激活的情况下触发胞浆游离钙信号传导,并可抑制上皮癌细胞的迁移和侵袭。Foxy-5 Ammonium Salt在原位小鼠模型中能有效降低 WNT5A 低表达的前列腺癌细胞的转移扩散。
T12705 Reparixin L-lysine salt

REPERTAXIN L-赖氨酸盐,Repertaxin L-lysine salt

CXCR Autophagy; GPCR/G Protein; Immunology/Inflammation
Reparixin L-lysine salt (Repertaxin L-lysine salt) 是趋化因子受体1/2 活化的变构抑制剂。
T1212 Ketorolac tromethamine salt

酮咯酸氨丁三醇,Acular LS,Toradol,Ketorolac tris salt,Acular

COX Immunology/Inflammation; Neuroscience
Ketorolac tromethamine salt (Ketorolac tris salt) 是一种非甾体抗炎剂,是非选择性的 COX 抑制剂,对 COX-1 和 COX-2 的IC50值分别为 20 和 120 nM。
T18949L CY5-SE Ditriethylamine salt

CY5-SE Ditriethylamine salt(146368-14-1 Free base)

Others Others
CY5-SE Ditriethylamine salt 是用于标记寡核苷酸,肽,蛋白质的氨基基团的反应染料。 激发波长 (nm): 649, 发射波长 (nm): 670
TP1545L1 FFAGLDD amine salt

Others Others
FFAGLDD amine salt 是MMP9选择性裂解肽,用于多柔比星(DOX)的胞浆递送,实现时间和空间可控的缓慢药物递送和释放。
T2160 Suramin Sodium Salt

苏拉明钠,BAY-205,Suramin hexasodium salt,苏拉明钠盐,NF-060

Apoptosis; Phosphatase; SARS-CoV; Sirtuin; Reverse Transcriptase; Topoisomerase; Parasite Apoptosis; Chromatin/Epigenetic; DNA Damage/DNA Repair; Metabolism; Microbiology/Virology
Suramin Sodium Salt (BAY-205) 是可逆的竞争性蛋白酪氨酸磷酸酶抑制剂。它抑制 IP5K,是抗寄生虫,抗肿瘤和抗血管生成剂。它是sirtuins 的有效抑制剂,也是 SARS-CoV-2 RNA 依赖性 RNA 聚合酶抑制剂。
T18942L Cy5-N3 triethylamine salt

Cy5-N3 triethylamine salt(1621101-43-6 free base)

Others Others
Cy5-N3 triethylamine salt 是一种花箐类荧光染料。CY5-N3 可用于研究细胞成像。
TP2226 BzATP triethylammonium salt

P2X Receptor Membrane transporter/Ion channel; Neuroscience
BzATP triethylammonium salt 是一种 P2X 受体激动剂,对 P2X1、P2X2、P2X3、P2X2/3、P2X4 和 P2X7 均有效 (pEC50=8.74/5.26/7.10/7.50/6.19/6.31/5.33)。BzATP triethylammonium salt 可以诱导细胞死亡并减少突触传递。
T6747 8-Bromo-cAMP sodium salt

8-Br-Camp sodium salt,8-溴腺苷-3',5'-环单磷酸钠,8-Bromo-cAMP(sodium salt),8-Bromo-cAMP

PKA Tyrosine Kinase/Adaptors
8-Bromo-cAMP sodium salt (8-Br-Camp sodium salt) 是一种环 AMP (cAMP) 类似物,一种 cAMP 依赖性蛋白激酶 (PKA) 的激活剂。8-Bromo-cAMP sodium salt 具有抗肿瘤活性。
T5847 Cloprostenol sodium salt

ICI 80996 sodium salt,DL-Cloprostenol sodium,氯前列烯醇钠,氯前列烯醇纳,Cloprostenol sodium

Prostaglandin Receptor GPCR/G Protein; Immunology/Inflammation
Cloprostenol sodium salt (ICI 80996 sodium salt) 是一种合成的前列腺素类似物,是 PGF2α受体的激动剂,具有黄体溶解性。
T0148L Folinic Acid Calcium Salt Pentahydrate

Folinic acid,亚叶酸钙五水合物,Leucovorin Calcium Pentahydrate,Leucovorin calcium salt pentahydrate

Others; Antifolate Cell Cycle/Checkpoint; Others
Folinic Acid Calcium Salt Pentahydrate (Leucovorin Calcium Pentahydrate) 是一种还原型叶酸,是一种解毒剂,通常与甲氨蝶呤 (MTX) 联用,以降低 MTX 诱导的毒性。
T4251 GJ103 sodium salt

ATM/ATR DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
GJ103 sodium salt 是 GJ072 的活性类似物,它是一种通读化合物 (RTC)。它已被证明可以降低水溶液的表面张力,使分子更容易在溶液中移动。它还被证明可以降低水溶液的粘度,使分子更容易在溶液中移动。此外,它还被证明可以降低水溶液的pH 值,这会对生物体的生化和生理过程产生各种影响。
T72505L CTP Synthetase-IN-1 Ammonium salt

CTPS-IN-1 Ammonium salt,CTP Synthetase-IN-1 Ammonium salt(2338811-71-3 Free base)

Others Others
CTP Synthetase-IN-1 Ammonium salt 是一种具有口服活性和高效性的胞苷 5'-三磷酸合成酶 (CTPS) 抑制剂,具有潜在的抗菌抗炎抗肿瘤活性,可用于研究 SARS-CoV-2病毒感染。
T5878 β-Glycerophosphate disodium salt pentahydrate

五水β-甘油磷酸钠,BETA-GLYCEROL PHOSPHATE DISODIUM SALT,B-甘油磷酸钠五水合物,β-Glycerol phosphate disodium salt pentahydrate

Phosphatase; Endogenous Metabolite Metabolism
β-Glycerophosphate disodium salt pentahydrate 是一种磷酸酶 (phosphatase) 抑制剂。
T39477 Ca-DTPA trisodium salt hydrate

Ca-DTPA trisodium salt hydrate,Calcium trinatrium diethylenetriaminepentaacetic acid hydrate

Others Others
Calcium trinatrium diethylenetriaminepentaacetic acid hydrate (Ca-DTPA trisodium salt hydrate) 是螯合剂和有用的解毒剂,如急性镉中毒。它是一种无毒的 CMV 复制抑制剂。
T38404 MJ33 lithium salt

ROS Immunology/Inflammation
MJ33 lithium salt 是 NADPH 氧化酶 2 型介导的 ROS 生成抑制剂,是一种氟化磷脂类似物,可抑制过氧化物还蛋白 6 (Prdx6) 的磷脂酶 A2 (PLA2) 活性,可用于研究急性肺损伤。
T19596 UDP-GlcNAc Disodium Salt

Uridine 5′-diphospho-N-acetylglucosamine,5′-二磷酸尿嘧啶核苷-N-乙酰半乳糖胺二钠盐,UDP-α-D-N-Acetylglucosamine Disodium Salt

Others Others
UDP-GlcNAc Disodium Salt (UDP-α-D-N-Acetylglucosamine Disodium Salt) 是一种 O-GlcNAc 转移酶 (OGT) 的供体底物。
T13564L2 AZ7550 trimesylate salt

AZ7550 Mesylate,AZ7550 trimesylate salt (1421373-99-0 free base)

MLK MAPK
AZ7550 trimesylate salt (AZ7550 Mesylate) 是奥希替尼的活性代谢产物,AZ7550 trimesylate salt 抑制 IGF1R 活性,可用于研究非小细胞肺癌。
T9306 EST64454 Maleic acid salt

Others Others
EST64454 Maleic acid salt 是EST64454的马来酸盐形式。EST64454是一种用于治疗疼痛的高可溶性σ1受体拮抗剂临床候选药物。
T8855 Polydeoxyribonucleotide(Sodium salt)

Polydeoxyribonucleotide from salmon

Others Others
Polydeoxyribonucleotide(Sodium salt) 可改善大鼠跟腱损伤模型中各种生长因子的分泌,促进胶原蛋白合成,恢复跟腱的拉伸强度。
T30677L1 C15AlkOPP Tetrabutylamine salt (1:2)

C15AlkOPP Tetrabutylamine salt(1:2)(946615-44-7 Free base)

Others Others
C15AlkOPP Tetrabutylamine salt (1:2)是一种FPP 类似物,具有炔基,允许前戊酰化后的蛋白质标记。C15AlkOPP Tetrabutylamine salt (1:2)可用于异戊二烯组学分析。

化合物

Ceruletide Ammonium Salt
Cat.No: T14932L1
Synonym: Caerulein Ammonium Salt,Ceruletide Ammonium Salt(17650-98-5 Free base),FI-6934 Ammonium Salt,Cerulein Ammonium Salt
Target: cholecystokinin
Silmitasertib sodium salt
Cat.No: T15024
Synonym: CX-4945 sodium salt
Target: Casein Kinase, Autophagy
Tirzepatide sodium salt
Cat.No: TP1111L1
Synonym: LY-3298176 sodium salt,Tirzepatide sodium salt(2023788-19-2 free base)
Target: Glucagon Receptor
Lorglumide sodium salt
Cat.No: T11868
Synonym: CR-1409 sodium salt
Target: cholecystokinin
ATN-161 trifluoroacetate salt
Cat.No: T10397
Synonym: ATN-161 TFA salt
Target: Integrin
Sacubitril hemicalcium salt
Cat.No: T4200
Synonym: AHU-377 (hemicalcium salt),LCZ696中间体,AHU377 calcium salt
Target: Neprilysin
Vaborbactam ammonium salt
Cat.No: T17210L
Synonym: RPX7009 ammonium salt,Vaborbactam ammonium salt(1360457-46-0 Free base)
Target: Antibacterial
Retatrutide sodium salt
Cat.No: T76279L1
Synonym: Retatrutide sodium salt(2381089-83-2 free base),LY3437943 sodium salt
Target: Glucagon Receptor
NAAD sodium salt
Cat.No: T33565
Synonym: NAAD钠盐,NAAD Na salt,Deamido Nad Sodium Salt,NAAD Na, NaAD
Target: Others
Etomoxir sodium salt
Cat.No: T4535
Synonym: (R)-(+)-乙莫克舍钠盐,(R)-Etomoxir sodium salt,Na salt,Etomoxir
Target: Apoptosis, Others
Fosmidomycin sodium salt
Cat.No: T11315
Synonym: FR-31564 sodium salt
Target: Antibiotic, Parasite
Chenodeoxycholic Acid sodium salt
Cat.No: T65070
Synonym: CDCA sodium salt
Target: FXR
TMC647055 Choline Hydroxide Salt
Cat.No: T21537L
Synonym: TMC647055 Choline Hydroxide Salt (1204416-97-6 free base)
Target: HCV Protease
Nonapeptide-1 acetate salt (158563-45-2 free base)
Cat.No: TP1101
Synonym: Melanostatine-5 acetate salt,Nonapeptide-1 acetate salt
Target: Melanocortin Receptor
ATPγS tetralithium salt
Cat.No: T22592
Synonym: ATP-gamma-S tetralithium salt
Target: PERK
Guanosine-5'-triphosphate disodium salt
Cat.No: T11511
Synonym: GTP disodium,5'-GTP disodium salt
Target: Others, Endogenous Metabolite
CY5 triethylamine salt
Cat.No: T15025L
Synonym: CY5 triethylamine salt(146368-11-8 Free base)
Target: Others
Deoxyguanosine triphosphate trisodium salt
Cat.No: T36688
Synonym: Deoxyguanosine 5-triphosphate,2'-Deoxyguanosine-5'-triphosphate trisodium salt,dGTP trisodium salt
Target: Nucleoside Antimetabolite/Analog
dITP trisodium salt
Cat.No: T84284
Synonym: 2'-Deoxyinosine-5'-triphosphate trisodium salt
Target: Others
BIO-11006 acetate salt (901117-03-1 free base)
Cat.No: TP1457
Synonym: BIO-11006 acetate salt
Target: Others
CMP-Sialic acid sodium salt
Cat.No: T10851
Synonym: CMP-Neu5Ac sodium salt
Target: Endogenous Metabolite
Acid Yellow 9 monosodium salt
Cat.No: T18910
Synonym: Hydrogen 4-aminoazobenzene-3,4'-disulphonate (sodium salt)
Target: Others
CEP-28122 mesylate salt (1022958-60-6 free base)
Cat.No: T10759
Synonym: CEP-28122 mesylate salt
Target: ALK
Resorufin sodium salt
Cat.No: T16734L
Synonym: 试卤灵钠盐,NSC 12097 sodium salt
Target: Others
Ursulcholic acid trisodium salt
Cat.No: T68019L
Synonym: Ursodeoxycholic acid disulfate trisodium salt,Ursulcholic acid trisodium salt(88426-32-8 Free base)
Target: Others
3-OMFP Cyclohexylammonium salt
Cat.No: T33795
Synonym: OMFP Cyclohexylammonium salt
Target: Others
Durlobactam sodium salt
Cat.No: T11125
Synonym: 杜巴坦,ETX2514 sodium salt,杜洛巴坦
Target: Antibacterial
C15AlkOPP t-BA salt
Cat.No: T30677L
Synonym: C15AlkOPP t-BA salt(946615-44-7 Free base),C15AlkOPP Tetrabutylamine salt(946615-44-7 Free base)
Target: Others
MOPS sodium salt
Cat.No: T19820
Synonym: MOPS-Na,3-(N-morpholino)propanesulfonic acid sodium salt,3-吗啉丙磺酸钠盐,Sodium 3-Morpholinopropanesulfonate,4-Morpholinepropanesulfonic acid, sodium salt
Target: Others
Foxy-5 Ammonium Salt
Cat.No: TP1565L1
Synonym: Foxy-5 Ammonium Salt(881188-51-8 Free base)
Target: Wnt/beta-catenin
Reparixin L-lysine salt
Cat.No: T12705
Synonym: REPERTAXIN L-赖氨酸盐,Repertaxin L-lysine salt
Target: CXCR
Ketorolac tromethamine salt
Cat.No: T1212
Synonym: 酮咯酸氨丁三醇,Acular LS,Toradol,Ketorolac tris salt,Acular
Target: COX
CY5-SE Ditriethylamine salt
Cat.No: T18949L
Synonym: CY5-SE Ditriethylamine salt(146368-14-1 Free base)
Target: Others
FFAGLDD amine salt
Cat.No: TP1545L1
Synonym:
Target: Others
Suramin Sodium Salt
Cat.No: T2160
Synonym: 苏拉明钠,BAY-205,Suramin hexasodium salt,苏拉明钠盐,NF-060
Target: Apoptosis, Phosphatase, SARS-CoV, Sirtuin, Reverse Transcriptase, Topoisomerase, Parasite
Cy5-N3 triethylamine salt
Cat.No: T18942L
Synonym: Cy5-N3 triethylamine salt(1621101-43-6 free base)
Target: Others
BzATP triethylammonium salt
Cat.No: TP2226
Synonym:
Target: P2X Receptor
8-Bromo-cAMP sodium salt
Cat.No: T6747
Synonym: 8-Br-Camp sodium salt,8-溴腺苷-3',5'-环单磷酸钠,8-Bromo-cAMP(sodium salt),8-Bromo-cAMP
Target: PKA
Cloprostenol sodium salt
Cat.No: T5847
Synonym: ICI 80996 sodium salt,DL-Cloprostenol sodium,氯前列烯醇钠,氯前列烯醇纳,Cloprostenol sodium
Target: Prostaglandin Receptor
Folinic Acid Calcium Salt Pentahydrate
Cat.No: T0148L
Synonym: Folinic acid,亚叶酸钙五水合物,Leucovorin Calcium Pentahydrate,Leucovorin calcium salt pentahydrate
Target: Others, Antifolate
GJ103 sodium salt
Cat.No: T4251
Synonym:
Target: ATM/ATR
CTP Synthetase-IN-1 Ammonium salt
Cat.No: T72505L
Synonym: CTPS-IN-1 Ammonium salt,CTP Synthetase-IN-1 Ammonium salt(2338811-71-3 Free base)
Target: Others
β-Glycerophosphate disodium salt pentahydrate
Cat.No: T5878
Synonym: 五水β-甘油磷酸钠,BETA-GLYCEROL PHOSPHATE DISODIUM SALT,B-甘油磷酸钠五水合物,β-Glycerol phosphate disodium salt pentahydrate
Target: Phosphatase, Endogenous Metabolite
Ca-DTPA trisodium salt hydrate
Cat.No: T39477
Synonym: Ca-DTPA trisodium salt hydrate,Calcium trinatrium diethylenetriaminepentaacetic acid hydrate
Target: Others
MJ33 lithium salt
Cat.No: T38404
Synonym:
Target: ROS
UDP-GlcNAc Disodium Salt
Cat.No: T19596
Synonym: Uridine 5′-diphospho-N-acetylglucosamine,5′-二磷酸尿嘧啶核苷-N-乙酰半乳糖胺二钠盐,UDP-α-D-N-Acetylglucosamine Disodium Salt
Target: Others
AZ7550 trimesylate salt
Cat.No: T13564L2
Synonym: AZ7550 Mesylate,AZ7550 trimesylate salt (1421373-99-0 free base)
Target: MLK
EST64454 Maleic acid salt
Cat.No: T9306
Synonym:
Target: Others
Polydeoxyribonucleotide(Sodium salt)
Cat.No: T8855
Synonym: Polydeoxyribonucleotide from salmon
Target: Others
C15AlkOPP Tetrabutylamine salt (1:2)
Cat.No: T30677L1
Synonym: C15AlkOPP Tetrabutylamine salt(1:2)(946615-44-7 Free base)
Target: Others
Cat. No. Product Name Target Signaling Pathways
T8393 Uridine triphosphate trisodium salt

UTP, Trisodium Salt,Uridine 5'-triphosphate trisodium salt,尿苷-5'-三磷酸三钠盐,Uridine triphosphate (trisodium salt)

Others Others
Uridine triphosphate trisodium salt (UTP, Trisodium Salt) 是一种核苷酸,在正常和疾病状态,均能够调节胰腺内分泌和外分泌、通道、增殖、转运体和细胞内信号传导的功能。
T4730 Thymidine-5'-monophosphate disodium salt

胸苷酸二钠,Thymidine 5'-monophosphate disodium salt,TMP DISODIUM SALT

Others; Endogenous Metabolite Metabolism; Others
Thymidine-5'-monophosphate disodium salt (TMP DISODIUM SALT) 是内源性代谢产物的一种。
T3S0156 Atractyloside potassium salt

Atractyloside Dipotassium Salt,苍术苷钾盐,苍术苷二钾盐

Others Others
Atractyloside potassium salt (Atractyloside Dipotassium Salt) 是一种从苍术果实中分离出得到的二萜苷类化合物,具有毒性。它能抑制大鼠心脏线粒体膜的氯离子通道。它是高效、特异性的线粒体 ADP/ATP 转运 (ADP/ATP transport) 抑制剂。
T5079 Adenosine 5'-diphosphate sodium salt

腺苷-5‘-二磷酸钠盐,Adenosine-5'-diphosphate trisodium salt,ADP sodium salt

Others; Endogenous Metabolite Metabolism; Others
Adenosine 5'-diphosphate sodium salt (ADP sodium salt) 是一种核苷二磷酸,是一种 ATP 酶对 ATP 去磷酸化的产物。它通过在 P2T-嘌呤受体上的作用诱导人血小板聚集并抑制刺激的腺苷酸环化酶。
T2944 Danshensu sodium salt

Sodium Danshensu,(±)-DanShenSu sodium salt,丹参素钠,(±)-DanShenSu sodium sal

P450; Autophagy Autophagy; Metabolism
Danshensu sodium salt (Sodium Danshensu) 是从中国草本丹参中提取的一种天然产物,可以抑制去氧肾上腺素和CaCl2 在无Ca2+ 培养基中引起的血管收缩。
T4969 Guanosine 5'-triphosphate trisodium salt

鸟苷-5'-三磷酸三钠盐,GTP Trisodium salt,5'-GTP trisodium salt

Endogenous Metabolite Metabolism
Guanosine 5'-triphosphate trisodium salt (5'-GTP trisodium salt) 为G蛋白(G proteins)信号转导过程中的活化剂。
T19262 D-Glucose 6-phosphate disodium salt

D-​Glucose ​6-​phosphate disodium salt

Endogenous Metabolite Metabolism
D-Glucose 6-phosphate disodium salt 广泛存在于生物提内的化合物,是葡萄糖第 6 号碳经过磷酸化后生成的分子,参与磷酸戊糖途径与糖酵解途径等体内多种多种代谢调节途径。
T1033 Monensin sodium salt

莫能菌素钠盐,Sodium Monensin,Monensin A sodium salt

Sodium Channel; Antibacterial; Antibiotic Membrane transporter/Ion channel; Microbiology/Virology
Monensin sodium salt (Monensin A sodium salt) 是由肉桂链霉菌 分泌的抗生素。它是一种介导Na+/H+交换的离子载体。它引起细胞多泡体 (MVBs) 增大并调节外泌体的分泌。
T21518 Colistin methanesulfonate sodium salt

粘杆菌素甲基磺酸钠,Colistin Methanesulfonate (sodium salt)

Cell wall; Antibacterial Immunology/Inflammation; Microbiology/Virology
Colistin methanesulfonate sodium salt (Colistimethate Sodium) 是一种来自 Bacillus colistinus 的环状多肽抗生素,由多粘菌素 E1 和 E2 组成。
T4743 Uridine 5′-diphosphoglucose disodium salt

二磷酸尿苷葡萄糖二钠盐,UDP-Glucose sodium salt,UDPG sodium salt,UDP-α-D-Glucose sodium salt,Uridine 5'-diphosphoglucose disodium sal

Endogenous Metabolite; P2Y Receptor GPCR/G Protein; Metabolism; Neuroscience
Uridine 5′-diphosphoglucose disodium salt (UDP-Glucose sodium salt) 是一种内源性核苷酸糖,参与代谢中的糖基转移酶反应。它是 P2Y14 受体的激动剂,EC50为 0.35 μM。
T4706 Uridine-5'-diphosphate disodium salt

UDP disodium salt,Uridine 5'-diphosphate disodium salt hyd,尿苷-5'-二磷酸二钠盐

DNA/RNA Synthesis; Endogenous Metabolite; P2Y Receptor Cell Cycle/Checkpoint; DNA Damage/DNA Repair; GPCR/G Protein; Metabolism; Neuroscience
Uridine-5'-diphosphate disodium salt (UDP disodium salt) 是一种选择性 P2Y6受体激动剂,EC50为300 nM,对人 P2Y6受体的 pEC50为6.52。它可刺激炎症介质的产生、吞噬作用和血管收缩,催化多种底物的葡糖醛酸糖化反应,用于核酸生物合成。
T16527 Phytic acid dodecasodium salt hydrate

植酸十二钠盐,myo-Inositol, hexakis(dihydrogen phosphate) dodecasodium salt hydrate,Inositol hexaphosphate dodecasodium salt hydrate

Others; Xanthine Oxidase; Endogenous Metabolite Metabolism; Others
Phytic acid dodecasodium salt hydrate (myo-Inositol, hexakis(dihydrogen phosphate) dodecasodium salt hydrate) 是种子和谷物的磷储存化合物。 Phytic acid dodecasodium salt hydrate 抑制酶促超氧化物源黄嘌呤氧化酶,IC50 为 6 mM,并具有抗氧化、神经保护和抗炎作用。
T5283 NADH disodium salt

Disodium NADH,NADH, disodium salt hydrate,beta-烟酰胺腺嘌呤二核苷二钠

Others; Endogenous Metabolite Metabolism; Others
NADH disodium salt hydrate是氧化还原酶的辅酶。 NADH在分解代谢过程中起到再生电子供体的作用,包括糖酵解,柠檬酸循环和β-氧化。
T22446 NADP disodium salt

Disodium NADP,Triphosphopyridine nucleotide disodium salt,beta-烟酰胺腺嘌呤二核苷酸磷酸二钠盐

Others Others
NADP disodium salt (Disodium NADP) 是一种氧化还原辅助因子,是一种烟酰胺腺嘌呤二核苷酸。它是代谢中电子转移的关键辅因子,可以被交替氧化 (NADP+) 和还原 (NADPH)。
T0958 Penicillin G sodium salt

青霉素钠,Penicillin G Sodium,Benzylpenicillin sodium salt,Benzylpenicillin Sodium

GABA Receptor; Antibacterial; Antibiotic Membrane transporter/Ion channel; Microbiology/Virology; Neuroscience
Penicillin G sodium(Benzylpenicillin sodium) salt 是一种 β-内酰胺类抗生素。
T5258 Dodecanedioic acid diammonium salt

十二烷二酸 二铵盐,1,10-Decanedicarboxylic acid diammonium salt

Others Others
Dodecanedioic acid diammonium salt (1,10-Decanedicarboxylic acid diammonium salt) 是一种二元羧酸,它是水溶性的,并且参与了脂类和碳水化合物的代谢途径中间体。
T65269 L-Aspartic acid potasium salt

Aspartic acid potasium salt,Potassium L-aspartate

Others Others
L-aspartic acid potasium salt(VX-548) 是一种广泛存在于动植物体内的氨基酸。L-aspartic acid potasium salt驱动氮氧化物的产生,从而促进吞噬作用,有助于提高鱼类的成活率。L-aspartic acid potasium salt 可对抗生素产生刺激,刺激作用可能与参与天冬氨酸-4-半醛生物合成的前体有关。
T5693 Pyrroloquinoline quinone disodium salt

吡咯喹啉醌二钠盐,Methoxatin disodium salt

Others; Endogenous Metabolite Metabolism; Others
Pyrroloquinoline quinone disodium salt (Methoxatin disodium salt) 一种阴离子型氧化还原循环原醌,作为氧化还原辅助因子。它是从嗜甲基细菌的培养物中分离的,也存在于哺乳动物的组织。它是哺乳动物的必需营养素,对免疫功能很重要。
T2812 ATP disodium salt hydrate

ATP disodium,ATP disodium salt,Adenosine disodium triphosphate,三磷酸腺苷二钠盐

Others; Endogenous Metabolite Metabolism; Others
ATP disodium salt hydrate (Adenosine disodium triphosphate) 是体内能量储存和代谢的重要物质,为代谢提供能量,同时在细胞中作为辅酶发挥作用。同时,它是也是免疫和炎症中重要的内源性信号分子。
T5087 DL-Isocitric acid trisodium salt

异柠檬酸三钠盐,Isocitric acid trisodium salt

Others; Endogenous Metabolite Metabolism; Others
DL-Isocitric acid trisodium salt 是内源性代谢产物的一种。
T4941 D-Fructose-6-phosphate disodium salt

D-FRUCTOSE 6-PHOSPHATE DISODIUM SALT,D-果糖-6-磷酸二钠

Others; Endogenous Metabolite Metabolism; Others
D-Fructose-6-phosphate disodium salt (D-FRUCTOSE 6-PHOSPHATE DISODIUM SALT) 是内源性代谢产物的一种。
T37984 Fosfructose, sodium salt, hydrate (1:3:8)

D-Fructose-1,6-bisphosphate , sodium salt, hydrate (1:3:8)

Others Others
D-Fructose-1,6-bisphosphate sodium salt hydrate 是碳水化合物代谢的中间体,包括糖酵解和糖异生。在糖酵解过程中,它是由磷酸果糖激酶磷酸化果糖-6-磷酸产生的。由果糖-1,6-二磷酸酶-1介导的逆反应是糖异生的限速步骤之一。同样的反应也发生在植物的叶绿体中,D-Fructose-1,6-bisphosphate sodium salt hydrate 作为还原性戊糖磷酸循环的一部分。由于癌细胞采用糖酵解作为代谢能量产生的主要来源,这一途径已成为癌症化疗的主要靶点。
T21066 Norepinephrine bitartrate salt

Adrenergic Receptor GPCR/G Protein; Neuroscience
Norepinephrine bitartrate salt 是一种肾上腺素能神经递质。
T4713 Phosphorylcholine chloride calcium salt tetrahydrate

Phosphocholine chloride calcium salt tet,胆碱磷酸氯化钙四水,CalciuM Phosphorylcholine Tetrahydrate

Others; Endogenous Metabolite Metabolism; Others
Phosphorylcholine chloride calcium salt tetrahydrate (Phosphocholine chloride calcium salt tet) 是内源性代谢产物的一种。
T1352 ATP disodium salt

Adenosine 5'-triphosphate disodium salt,三磷酸腺苷二钠,ATP,ATP disodium,腺苷-5'-三磷酸二钠盐,Adetide,Adenosine-Triphosphate,Disodium adenosine triphosphate

P2X Receptor; Endogenous Metabolite Membrane transporter/Ion channel; Metabolism; Neuroscience
ATP disodium salt (Adenosine-Triphosphate) 是体内能量储存的重要物质,为代谢提供能量,同时在细胞中作为辅酶发挥作用。Adenosine 5'-triphosphate disodium salt 也是免疫和炎症中重要的内源性信号分子。
T4897 Inosine-5'-triphosphate trisodium salt

ITP,肌苷-5'-三磷酸三钠盐,三磷酸肌苷三钠盐,Inosine 5'-triphosphate trisodium salt

Others; Endogenous Metabolite Metabolism; Others
Inosine-5'-triphosphate trisodium salt (ITP) 是三磷酸核苷,能够作为 ATPases 和 GTPases 的底物。
T4901 5'-Guanylic acid disodium salt

Guanosine 5'-monophosphate disodium salt,5'-鸟苷酸二钠,鸟苷钠5'-单磷酸,GMP-5

Others; Endogenous Metabolite Metabolism; Others
5'-Guanylic acid disodium salt (GMP-5) 由鸟嘌呤,核糖和磷酸组成,是信使 RNA 中的一种核苷酸单体。 鸟苷衍生物参与细胞内信号转导,并已鉴定存在于端粒,核糖体 DNA,免疫球蛋白重链转换区和原癌基因的控制区中的重复基因组序列中。
T5067 Flavin adenine dinucleotide disodium salt

Flavin Adenine Dinucleotide Disodium,黄素腺嘌呤二核苷酸二钠,FAD sodium salt,FAD-Na2

Others; Endogenous Metabolite Metabolism; Others
Flavin adenine dinucleotide disodium salt (FAD sodium salt) 是一种辅酶,作用是促进细胞氧化还原反应中黄素酶的电子转移。
T5068 D-Glucuronic acid sodium salt monohydrate

Sodium D-glucuronate,D-葡糖醛酸钠一水,D-葡萄糖醛酸钠,D(+)-Glucuronic acid sodium salt monohydrate

Others; Endogenous Metabolite Metabolism; Others
D-Glucuronic acid sodium salt monohydrate (Sodium D-glucuronate) 是内源性代谢产物的一种。
TMA2440 Uridine 5'-monophosphate disodium salt

尿苷-5'-单磷酸二钠盐,Disodium UMP,尿苷酸二钠盐,Disodium uridine-5'-monophosphate,5'-UMP disodium salt,Disodium 5'-Uridylate

Others Others
Uridine 5'-monophosphate disodium salt (Disodium UMP) 是合成 RNA 的一种重要成分。
T6674 L-Ascorbic acid sodium salt

(+)-Sodium L-ascorbate,Vitamin C sodium salt,Sodium ascorbate,L-Ascorbic acid sodium,抗坏血酸钠,Sodium L-ascorbate,维生素C钠

Apoptosis; Others; Calcium Channel; Reactive Oxygen Species; Endogenous Metabolite Apoptosis; Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; NF-κB; Others
L-Ascorbic acid sodium salt (Vitamin C sodium salt) 是一种电子供体,是一种内源性抗氧化剂。它还是一种胶原沉积促进剂和弹性生成抑制剂。它选择性抑制 Cav3.2 通道(Cav3.2 channels),IC50为 6.5 μM。
T3551 D-Pantothenic acid hemicalcium salt

泛酸钙,D-Pantothenic Acid Calcium,D-泛酸半钙,Calpanate,Calcium D-pantothenate,Vitamin B5 calcium salt,Calcium pantothenate,Calcium D-Panthotenate

Apoptosis; Endogenous Metabolite Apoptosis; Metabolism
D-Pantothenic acid hemicalcium salt (Calcium pantothenate) 是一种水溶性维生素,能够减少苹果汁中的棒曲霉素。
T19343L Glycerol 3-phosphate biscyclohexylammonium salt

Endogenous Metabolite Metabolism
Glycerol 3-phosphate biscyclohexylammonium salt 是胞质甘油 3-磷酸脱氢酶途径中产生的,即利用 NADH 还原二羟丙酮磷酸的过程。
T4070 Glycocholic Acid Sodium Salt

Glycocholate Sodium,Sodium Glycocholate,甘氨胆酸钠盐

Others Others
Glycocholic Acid Sodium Salt (Sodium Glycocholate) 是一种结合胆汁盐和离子生物去污剂。它参与脂肪的乳化。
T5073 Inosine 5'-monophosphate disodium salt hydrate

Inosine 5'-monophosphate disodium salt,5'-IMP-Na2,肌苷5-单磷酸二钠盐水合物,Disodium 5'-inosinate monohydrate

Others; Endogenous Metabolite Metabolism; Others
Inosine 5'-monophosphate disodium salt hydrate (Inosine 5'-monophosphate disodium salt) 或肌苷酸是次黄嘌呤的核糖核苷酸,是嘌呤合成过程中形成的第一个核苷酸。
TN2349 Taurodeoxycholate sodium salt

Sodium taurodeoxylate,牛磺脱氧胆酸钠

Endogenous Metabolite Metabolism
Taurodeoxycholate sodium salt (Sodium taurodeoxylate) 是胆盐相关的阴离子洗涤剂,用于分离膜蛋白,包括线粒体内膜蛋白。它还可以抑制各种炎症反应。
T4915 β-Glycerophosphate disodium salt hydrate

Phosphatase; Endogenous Metabolite Metabolism
β-Glycerophosphate disodium salt hydrate 是一种磷酸酶抑制剂,是内源性代谢产物的一种。
T5069 D-Glucose 6-phosphate potassium salt

Others Others
在细胞中,当葡萄糖被己糖激酶或葡萄糖激酶磷酸化或在糖原分解过程中通过磷酸葡萄糖变位酶转化葡萄糖 1-磷酸时,会产生D-glucose 6-phosphate (G6P)。 G6P 位于糖酵解和戊糖磷酸途径的起点。当血糖水平高时,它也可以作为糖原储存。
TQ0215 Salinomycin sodium salt

盐霉素钠,Sodium salinomycin,Salinomycin sodium

Apoptosis; Wnt/beta-catenin; Antibacterial; Antibiotic; Autophagy Apoptosis; Autophagy; Cytoskeletal Signaling; Microbiology/Virology; Stem Cells
Salinomycin sodium salt (Sodium salinomycin) 是钾离子载体抗生素,是作用于 Wnt/Fzd/LRP 复合物的Wnt/β-catenin 信号传导抑制剂,能阻断 Wnt 诱导的 LRP6 磷酸化,导致 LRP6 蛋白降解。它选择性抑制人肿瘤干细胞。
T3092 Nigericin sodium salt

尼日利亚菌素,尼日利亚菌素钠盐

Potassium Channel; NOD-like Receptor (NLR); Antibacterial; Antibiotic; NOD Immunology/Inflammation; Membrane transporter/Ion channel; Microbiology/Virology; NF-κB
Nigericin sodium salt 属于抗生素,是一种 NLRP3 激活剂,也是一种阳离子离子载体。Nigericin sodium 可以触发 NALP3 炎性体的激活,可抑制高尔基体功能并抑制革兰氏阳性菌的生长。
T0281 Meclocycline sulfosalicylate salt

磺基水杨酸甲氯环素,Meclutin,Mecloderm,甲环素磺基水杨酸盐,Meclan Cream

Antibacterial; Antibiotic Microbiology/Virology
Meclocycline sulfosalicylate salt (Mecloderm) 是一种具有广谱抗菌活性的四环素抗生素,可预防皮肤细菌感染。
T13528 Acetoacetic acid sodium salt

乙酰乙酸钠,3-氧代丁酸钠盐

Others Others
Acetoacetic acid sodium salt 是一种内源性的非酯化脂肪酸代谢物,与人类糖尿病的发展相关。它诱导氧化应激,抑制牛肝细胞中极低密度脂蛋白的组装。
T5303 Isethionic acid sodium salt

Sodium isethionate,羟乙基磺酸钠

Others; Endogenous Metabolite Metabolism; Others
Isethionic acid sodium salt (Sodium isethionate) 是内源性代谢产物的一种。
T1138 Taurocholic acid sodium salt hydrate

牛胆酸钠,牛磺胆酸钠水合物,Sodium taurocholate hydrate,Taurocholic Acid sodium hydrate

Others; Potassium Channel; Endogenous Metabolite Membrane transporter/Ion channel; Metabolism; Others
Taurocholic acid sodium salt hydrate (Sodium taurocholate hydrate) 是一种胆汁酸钠盐水合物,作用是参与脂肪的乳化。
T8186 Xanthosine 5'-monophosphate sodium salt

XMP,黄苷-5′-单磷酸钠,L-XMP Sodium

Others Others
Xanthosine 5'-monophosphate sodium salt (L-XMP Sodium) 是嘌呤代谢的一种中间体。它可用于研究遗传密码,核酸结构以及 DNA,RNA 和蛋白质合成。
T4727 Taurolithocholic acid sodium salt

牛磺石胆酸钠,Sodium taurolithocholate

Others; Calcium Channel Membrane transporter/Ion channel; Metabolism; Others
Taurolithocholic acid sodium salt (Sodium taurolithocholate) 是抑胆剂和 Ca2+激动剂,可抑制放射性配体与毒蕈碱 M1 结合。
T5584 Phytic acid sodium salt

Sodium phytate hydrate,玉米

Others Others
Phytic acid sodium salt (Sodium phytate hydrate) 源于豆类种子中,具有抗营养活性。它是 [PO4]3-储藏库,是其他肌醇磷酸酯和焦磷酸酯的前体,在植物中被植酸酶逐步水解。
T40814 Colominic acid sodium salt

Polysialic acid sodium salt,Colominic acid sodium salt

Others Others
Colominic acid sodium salt, also known as polysialic acid sodium salt, is naturally isolated from the cell wall of Escherichia coli and animals. It exhibits a red color with an absorption maximum of 530 nm and possesses anti-bacterial activity.
T4922 Uridine 5′-triphosphate tris salt

尿苷-5′-三磷酸酯 三羟甲基氨基甲烷盐,Uridine 5'-triphosphoric acid

Others; Endogenous Metabolite Metabolism; Others
Uridine 5′-triphosphate tris salt (Uridine 5'-triphosphoric acid) 是 P2Y 受体的激动剂,已用于研究细胞内 Ca2+ 的浓度,以及用于体外激酶测定的磷酸盐供体。
T5259 Glycochenodeoxycholic acid sodium salt

GCDCA,甘氨鹅脱氧胆酸钠,Sodium glycochenodeoxycholate

Apoptosis; Others; Endogenous Metabolite Apoptosis; Metabolism; Others
Glycochenodeoxycholic acid sodium salt 是一种从脱氧鹅胆酸和甘氨酸在肝脏中形成的胆汁盐,可诱导肝细胞凋亡。它起到洗涤剂的作用,可溶解脂肪吸收,并本身被吸收。
------------------------ 更多 ------------------------

天然产物

Uridine triphosphate trisodium salt
Cat.No: T8393
Synonym: UTP, Trisodium Salt,Uridine 5'-triphosphate trisodium salt,尿苷-5'-三磷酸三钠盐,Uridine triphosphate (trisodium salt)
Target: Others
Thymidine-5'-monophosphate disodium salt
Cat.No: T4730
Synonym: 胸苷酸二钠,Thymidine 5'-monophosphate disodium salt,TMP DISODIUM SALT
Target: Others, Endogenous Metabolite
Atractyloside potassium salt
Cat.No: T3S0156
Synonym: Atractyloside Dipotassium Salt,苍术苷钾盐,苍术苷二钾盐
Target: Others
Adenosine 5'-diphosphate sodium salt
Cat.No: T5079
Synonym: 腺苷-5‘-二磷酸钠盐,Adenosine-5'-diphosphate trisodium salt,ADP sodium salt
Target: Others, Endogenous Metabolite
Danshensu sodium salt
Cat.No: T2944
Synonym: Sodium Danshensu,(±)-DanShenSu sodium salt,丹参素钠,(±)-DanShenSu sodium sal
Target: P450, Autophagy
Guanosine 5'-triphosphate trisodium salt
Cat.No: T4969
Synonym: 鸟苷-5'-三磷酸三钠盐,GTP Trisodium salt,5'-GTP trisodium salt
Target: Endogenous Metabolite
D-Glucose 6-phosphate disodium salt
Cat.No: T19262
Synonym: D-​Glucose ​6-​phosphate disodium salt
Target: Endogenous Metabolite
Monensin sodium salt
Cat.No: T1033
Synonym: 莫能菌素钠盐,Sodium Monensin,Monensin A sodium salt
Target: Sodium Channel, Antibacterial, Antibiotic
Colistin methanesulfonate sodium salt
Cat.No: T21518
Synonym: 粘杆菌素甲基磺酸钠,Colistin Methanesulfonate (sodium salt)
Target: Cell wall, Antibacterial
Uridine 5′-diphosphoglucose disodium salt
Cat.No: T4743
Synonym: 二磷酸尿苷葡萄糖二钠盐,UDP-Glucose sodium salt,UDPG sodium salt,UDP-α-D-Glucose sodium salt,Uridine 5'-diphosphoglucose disodium sal
Target: Endogenous Metabolite, P2Y Receptor
Uridine-5'-diphosphate disodium salt
Cat.No: T4706
Synonym: UDP disodium salt,Uridine 5'-diphosphate disodium salt hyd,尿苷-5'-二磷酸二钠盐
Target: DNA/RNA Synthesis, Endogenous Metabolite, P2Y Receptor
Phytic acid dodecasodium salt hydrate
Cat.No: T16527
Synonym: 植酸十二钠盐,myo-Inositol, hexakis(dihydrogen phosphate) dodecasodium salt hydrate,Inositol hexaphosphate dodecasodium salt hydrate
Target: Others, Xanthine Oxidase, Endogenous Metabolite
NADH disodium salt
Cat.No: T5283
Synonym: Disodium NADH,NADH, disodium salt hydrate,beta-烟酰胺腺嘌呤二核苷二钠
Target: Others, Endogenous Metabolite
NADP disodium salt
Cat.No: T22446
Synonym: Disodium NADP,Triphosphopyridine nucleotide disodium salt,beta-烟酰胺腺嘌呤二核苷酸磷酸二钠盐
Target: Others
Penicillin G sodium salt
Cat.No: T0958
Synonym: 青霉素钠,Penicillin G Sodium,Benzylpenicillin sodium salt,Benzylpenicillin Sodium
Target: GABA Receptor, Antibacterial, Antibiotic
Dodecanedioic acid diammonium salt
Cat.No: T5258
Synonym: 十二烷二酸 二铵盐,1,10-Decanedicarboxylic acid diammonium salt
Target: Others
L-Aspartic acid potasium salt
Cat.No: T65269
Synonym: Aspartic acid potasium salt,Potassium L-aspartate
Target: Others
Pyrroloquinoline quinone disodium salt
Cat.No: T5693
Synonym: 吡咯喹啉醌二钠盐,Methoxatin disodium salt
Target: Others, Endogenous Metabolite
ATP disodium salt hydrate
Cat.No: T2812
Synonym: ATP disodium,ATP disodium salt,Adenosine disodium triphosphate,三磷酸腺苷二钠盐
Target: Others, Endogenous Metabolite
DL-Isocitric acid trisodium salt
Cat.No: T5087
Synonym: 异柠檬酸三钠盐,Isocitric acid trisodium salt
Target: Others, Endogenous Metabolite
D-Fructose-6-phosphate disodium salt
Cat.No: T4941
Synonym: D-FRUCTOSE 6-PHOSPHATE DISODIUM SALT,D-果糖-6-磷酸二钠
Target: Others, Endogenous Metabolite
Fosfructose, sodium salt, hydrate (1:3:8)
Cat.No: T37984
Synonym: D-Fructose-1,6-bisphosphate , sodium salt, hydrate (1:3:8)
Target: Others
Norepinephrine bitartrate salt
Cat.No: T21066
Synonym:
Target: Adrenergic Receptor
Phosphorylcholine chloride calcium salt tetrahydrate
Cat.No: T4713
Synonym: Phosphocholine chloride calcium salt tet,胆碱磷酸氯化钙四水,CalciuM Phosphorylcholine Tetrahydrate
Target: Others, Endogenous Metabolite
ATP disodium salt
Cat.No: T1352
Synonym: Adenosine 5'-triphosphate disodium salt,三磷酸腺苷二钠,ATP,ATP disodium,腺苷-5'-三磷酸二钠盐,Adetide,Adenosine-Triphosphate,Disodium adenosine triphosphate
Target: P2X Receptor, Endogenous Metabolite
Inosine-5'-triphosphate trisodium salt
Cat.No: T4897
Synonym: ITP,肌苷-5'-三磷酸三钠盐,三磷酸肌苷三钠盐,Inosine 5'-triphosphate trisodium salt
Target: Others, Endogenous Metabolite
5'-Guanylic acid disodium salt
Cat.No: T4901
Synonym: Guanosine 5'-monophosphate disodium salt,5'-鸟苷酸二钠,鸟苷钠5'-单磷酸,GMP-5
Target: Others, Endogenous Metabolite
Flavin adenine dinucleotide disodium salt
Cat.No: T5067
Synonym: Flavin Adenine Dinucleotide Disodium,黄素腺嘌呤二核苷酸二钠,FAD sodium salt,FAD-Na2
Target: Others, Endogenous Metabolite
D-Glucuronic acid sodium salt monohydrate
Cat.No: T5068
Synonym: Sodium D-glucuronate,D-葡糖醛酸钠一水,D-葡萄糖醛酸钠,D(+)-Glucuronic acid sodium salt monohydrate
Target: Others, Endogenous Metabolite
Uridine 5'-monophosphate disodium salt
Cat.No: TMA2440
Synonym: 尿苷-5'-单磷酸二钠盐,Disodium UMP,尿苷酸二钠盐,Disodium uridine-5'-monophosphate,5'-UMP disodium salt,Disodium 5'-Uridylate
Target: Others
L-Ascorbic acid sodium salt
Cat.No: T6674
Synonym: (+)-Sodium L-ascorbate,Vitamin C sodium salt,Sodium ascorbate,L-Ascorbic acid sodium,抗坏血酸钠,Sodium L-ascorbate,维生素C钠
Target: Apoptosis, Others, Calcium Channel, Reactive Oxygen Species, Endogenous Metabolite
D-Pantothenic acid hemicalcium salt
Cat.No: T3551
Synonym: 泛酸钙,D-Pantothenic Acid Calcium,D-泛酸半钙,Calpanate,Calcium D-pantothenate,Vitamin B5 calcium salt,Calcium pantothenate,Calcium D-Panthotenate
Target: Apoptosis, Endogenous Metabolite
Glycerol 3-phosphate biscyclohexylammonium salt
Cat.No: T19343L
Synonym:
Target: Endogenous Metabolite
Glycocholic Acid Sodium Salt
Cat.No: T4070
Synonym: Glycocholate Sodium,Sodium Glycocholate,甘氨胆酸钠盐
Target: Others
Inosine 5'-monophosphate disodium salt hydrate
Cat.No: T5073
Synonym: Inosine 5'-monophosphate disodium salt,5'-IMP-Na2,肌苷5-单磷酸二钠盐水合物,Disodium 5'-inosinate monohydrate
Target: Others, Endogenous Metabolite
Taurodeoxycholate sodium salt
Cat.No: TN2349
Synonym: Sodium taurodeoxylate,牛磺脱氧胆酸钠
Target: Endogenous Metabolite
β-Glycerophosphate disodium salt hydrate
Cat.No: T4915
Synonym:
Target: Phosphatase, Endogenous Metabolite
D-Glucose 6-phosphate potassium salt
Cat.No: T5069
Synonym:
Target: Others
Salinomycin sodium salt
Cat.No: TQ0215
Synonym: 盐霉素钠,Sodium salinomycin,Salinomycin sodium
Target: Apoptosis, Wnt/beta-catenin, Antibacterial, Antibiotic, Autophagy
Nigericin sodium salt
Cat.No: T3092
Synonym: 尼日利亚菌素,尼日利亚菌素钠盐
Target: Potassium Channel, NOD-like Receptor (NLR), Antibacterial, Antibiotic, NOD
Meclocycline sulfosalicylate salt
Cat.No: T0281
Synonym: 磺基水杨酸甲氯环素,Meclutin,Mecloderm,甲环素磺基水杨酸盐,Meclan Cream
Target: Antibacterial, Antibiotic
Acetoacetic acid sodium salt
Cat.No: T13528
Synonym: 乙酰乙酸钠,3-氧代丁酸钠盐
Target: Others
Isethionic acid sodium salt
Cat.No: T5303
Synonym: Sodium isethionate,羟乙基磺酸钠
Target: Others, Endogenous Metabolite
Taurocholic acid sodium salt hydrate
Cat.No: T1138
Synonym: 牛胆酸钠,牛磺胆酸钠水合物,Sodium taurocholate hydrate,Taurocholic Acid sodium hydrate
Target: Others, Potassium Channel, Endogenous Metabolite
Xanthosine 5'-monophosphate sodium salt
Cat.No: T8186
Synonym: XMP,黄苷-5′-单磷酸钠,L-XMP Sodium
Target: Others
Taurolithocholic acid sodium salt
Cat.No: T4727
Synonym: 牛磺石胆酸钠,Sodium taurolithocholate
Target: Others, Calcium Channel
Phytic acid sodium salt
Cat.No: T5584
Synonym: Sodium phytate hydrate,玉米
Target: Others
Colominic acid sodium salt
Cat.No: T40814
Synonym: Polysialic acid sodium salt,Colominic acid sodium salt
Target: Others
Uridine 5′-triphosphate tris salt
Cat.No: T4922
Synonym: 尿苷-5′-三磷酸酯 三羟甲基氨基甲烷盐,Uridine 5'-triphosphoric acid
Target: Others, Endogenous Metabolite
Glycochenodeoxycholic acid sodium salt
Cat.No: T5259
Synonym: GCDCA,甘氨鹅脱氧胆酸钠,Sodium glycochenodeoxycholate
Target: Apoptosis, Others, Endogenous Metabolite
--------- 更多 ---------
Cat. No. Product Name Species Expression System
TMPH-01424 GUCA2B Protein, Human, Recombinant (His)

Guanylate cyclase activator 2B,GUCA2B

Human HEK293 Cells
Endogenous activator of intestinal guanylate cyclase. It stimulates this enzyme through the same receptor binding region as the heat-stable enterotoxins. May be a potent physiological regulator of intestinal fluid and electrolyte transport. May be an autocrine/paracrine regulator of intestinal salt and water transport. GUCA2B Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with N-6xHis tag. The predicted molecular weight is 13.5 kDa and the accession number is Q16661.
TMPY-03353 CEL Protein, Mouse, Recombinant (His)

1810036E18Rik,carboxyl ester lipase,BAL

Mouse Baculovirus Insect Cells
CEL-maturity onset diabetes of the young (MODY), diabetes with pancreatic lipomatosis and exocrine dysfunction, is due to dominant frameshift mutations in the acinar cell carboxyl ester lipase gene (CEL). Bile-salt activated carboxylic ester lipase (CEL) is a major triglyceride, cholesterol ester and vitamin ester hydrolytic enzyme contained within pancreatic and lactating mammary gland secretions. Carboxyl ester lipase is a digestive pancreatic enzyme encoded by the CEL gene. Mutations in CEL c...
TMPJ-00875 NPPB Protein, Human, Recombinant (His)

NPPB,γ-Brain Natriuretic Peptide,Gamma-Brain Natriuretic Pep...

Human E. coli
Human Natriuretic peptides B acts as a cardiac hormone; it is associated with many biological actions, such as diuresis, natriuresis, vasorelaxation, which inhibits the secretion of rennin and aldosterone. It acts as a paracrine antifibrotic factor in the heart. Natriuretic peptides B can help restore the body balance of salt and water, improves the heart function. Natriuretic peptides B binds and stimulates the cGMP production of the NPR1 receptor and binds the clearance receptor NPR3.
TMPJ-01396 PIN4 Protein, Human, Recombinant (His)

Peptidyl-prolyl cis-trans isomerase Pin4,Parvulin-14,Peptidy...

Human E. coli
Peptidyl-prolyl cis-trans isomerase NIMA-interacting 4(PIN4) is a peptidyl-prolyl cis/trans isomerase (PPIase) which interacts with NIMA and is vital for cell cycle regulation. PIN4 has 2 different isoforms: PAR14 and PAR17. Furthermore, PIN4 protein binds to double-stranded DNA under physiological salt conditions. PIN4 is involved as a ribosomal RNA processing factor in ribosome biogenesis. The PAR14 binds to tightly bent AT-rich stretches of double-stranded DNA, but PAR17 binds to double-stran...
TMPY-02133 Carbonic Anhydrase VB Protein, Human, Recombinant (His)

carbonic anhydrase VB, mitochondrial,CA-VB,MGC39962

Human E. coli
Carbonic anhydrase 5B, also known as carbonate dehydratase VB, carbonic anhydrase VB, CA-VB and CA5B, is amember of the alpha-carbonic anhydrase family. The strongest expression of CA5B / CA-VB is in heart, pancreas, kidney, placenta, lung, and skeletal muscle. It is not expressed in liver. Carbonic anhydrases (CAs) are a large family of zinc metalloenzymes first discovered in 1933 that catalyze the reversible hydration of carbon dioxide. CAs participate in a variety of biological process...
TMPY-01877 CA5A Protein, Human, Recombinant (His)

CA5,GS1-21A4.1,CA5AD,carbonic anhydrase VA, mitochondrial,CA...

Human E. coli
Carbonic anhydrase 5A, mitochondrial, also known as Carbonate dehydratase VA, Carbonic anhydrase VA, CA-VA and CA5A, is a member of thealpha-carbonic anhydrase family. Carbonic anhydrases (CAs) are a large family of zinc metalloenzymes first discovered in 1933 that catalyze the reversible hydration of carbon dioxide. CAs participate in a variety of biological processes, including respiration, calcification, acid-base balance, bone resorption, and the formation of aqueous humor, cerebrospi...

重组蛋白

GUCA2B Protein, Human, Recombinant (His)
Cat.No: TMPH-01424
Species: Human
Expression System: HEK293 Cells
CEL Protein, Mouse, Recombinant (His)
Cat.No: TMPY-03353
Species: Mouse
Expression System: Baculovirus Insect Cells
NPPB Protein, Human, Recombinant (His)
Cat.No: TMPJ-00875
Species: Human
Expression System: E. coli
PIN4 Protein, Human, Recombinant (His)
Cat.No: TMPJ-01396
Species: Human
Expression System: E. coli
Carbonic Anhydrase VB Protein, Human, Recombinant (His)
Cat.No: TMPY-02133
Species: Human
Expression System: E. coli
CA5A Protein, Human, Recombinant (His)
Cat.No: TMPY-01877
Species: Human
Expression System: E. coli
Cat. No. Product Name Target Signaling Pathways
TMIH-0511 Sacubitril-d4 calcium salt

AHU-377-d4 calcium salt

Sacubitril-d4 calcium salt 是 Sacubitril calcium salt 的氘代化合物。
TMIH-0504 Rosuvastatin-d6 Calcium Salt

Rosuvastatin-d6 Calcium Salt 是 Rosuvastatin Calcium Salt 的氘代化合物。Rosuvastatin Calcium Salt 的 CAS 号为 147098-20-2。Rosuvastatin calcium 是肝羟甲基戊二酰辅酶 A 还原酶的选择性和竞争性抑制剂,具有抗血脂活性。它降低成熟 hERG 的表达以及热休克蛋白 70 与 hERG 蛋白的相互作用,还降低低密度脂蛋白胆固醇、甘油三酯和 C-反应蛋白水平。它阻断人类醚-a-go-go相关基因电流,延迟心脏复极化,来延长动作电位持续时间和校正 QT 间期间隔。
TMIH-0242 Fluvastatin-d6 Sodium Salt

Fluvastatin-d6 Sodium Salt 是 Fluvastatin Sodium Salt 的氘代化合物。Fluvastatin Sodium Salt 的 CAS 号为 93957-55-2。Fluvastatin sodium salt 是羟甲基戊二酰辅酶 A 还原酶的竞争性抑制剂,IC50为 8 nM。它通过依赖 Nrf2 的抗氧化通路保护血管平滑肌细胞免受氧化应激,是一种常用的降胆固醇剂。
T71205 Fosinopril-d7 sodium salt

Fosinopril-d7 is intended for use as an internal standard for the quantification of fosinopril by GC- or LC-MS. Fosinopril is a prodrug form of the angiotensin-converting enzyme inhibitor fosinoprilat. Oral administration of fosinopril inhibits angiotensin I-induced pressor responses in normotensive rats, dogs, and monkeys when administered at doses of 15, 15, and 10 µmol/kg, respectively. Fosinopril reduces fractional shortening and decreases left ventricular size in a porcine model of congesti...
T71211 Rizatriptan-d6 benzoate salt

Rizatriptan-d6 is intended for use as an internal standard for the quantification of rizatriptan by GC- or LC-MS. Rizatriptan is an agonist of the serotonin receptor subtypes 5-HT1B and 5-HT1D. It is selective for 5-HT1B and 5-HT1D receptors over 5-HT1A receptors. Rizatriptan induces vasoconstriction in isolated human middle meningeal arteries. In vivo, rizatriptan reduces head grooming, the number of oculotemporal strokes, eye blinking, and one-eye closures in a Cacna1a mutant transgenic mou...
T11193 Enalaprilat-d5 sodium

MK-422 D5 Sodium Salt,依那普利拉钠 D5,Enalaprilat D5 Sodium Salt

Others Others
Enalaprilat D5 Sodium Salt is the deuterium labeled Enalaprilat, which is an angiotensin-converting enzyme (ACE) inhibitor.
T70313 Indoxyl Sulfate-d5 potassium salt

Indoxyl sulfate-d5 is intended for use as an internal standard for the quantification of indoxyl sulfate by GC- or LC-MS. Indoxyl sulfate is a uremic toxin and a metabolite of tryptophan. It is formed via sulfation of indole, an intermediate generated from tryptophan by intestinal bacteria, by the sulfotransferase (SULT) isoform 1A1 variant 2 (SULT1A1*2) in the liver. Indoxyl sulfate activates the aryl hydrocarbon receptor (AhR) in HepG2 40/6 hepatoma cells (EC50 = 12.1 nM in a reporter assay). ...
TMIH-0552 Tauroursodeoxycholic Acid-d4 Sodium Salt

Tauroursodeoxycholic Acid-d4 Sodium Salt 是 Tauroursodeoxycholic Acid Sodium Salt 的氘代化合物。Tauroursodeoxycholic Acid Sodium Salt 的 CAS 号为 14605-22-2。Tauroursodeoxycholate,又称 ursodoxicoltaurine,是一种高度亲水性的三级胆汁酸,在人体内以低浓度产生。Tauroursodeoxycholate 是 ursodeoxycholic acid 更亲水的形式,而 ursodeoxycholic acid 是人类体内自然产生的更丰富的胆汁酸。Tauroursodeoxycholate 正在研究用于几种疾病,如原发性胆汁性肝硬化(PBC)、胰岛素抵抗、淀粉样变性、囊性纤维化、胆汁淤滞和肌萎缩性侧索硬化症。
TMIH-0473 rac Metanephrine-d3 Hydrochloride Salt

rac Metanephrine-d3 Hydrochloride Salt 是 rac Metanephrine Hydrochloride Salt 的氘代化合物。
TMIJ-0151 Atorvastatin-d5 Calcium Salt

Atorvastatin-d5 Calcium Salt 是 Atorvastatin Calcium Salt 的氘代化合物。Atorvastatin Calcium Salt 的 CAS 号为 134523-00-5。
TMIH-0010 (S)-Alogliptin Benzoate Salt-13C-d3

(S)-Alogliptin Benzoate Salt-13C-d3 是 (S)-Alogliptin Benzoate Salt 的 13C 和氘代化合物。
TMIJ-0164 Rosuvastatin-d6 Sodium Salt

Rosuvastatin-d6 Sodium Salt 是 Rosuvastatin Sodium Salt 的氘代化合物。Rosuvastatin Sodium Salt 的 CAS 号为 1007871-86-4。
TMID-0273 Promethazine-d6 Hydrochloride Salt

Promethazine-d6 Hydrochloride Salt 是 Promethazine Hydrochloride Salt 的氘代化合物。Promethazine Hydrochloride Salt 的 CAS 号为 1173018-74-0。
TMID-0269 Nafcillin-d5 Sodium Salt

Nafcillin-d5 Sodium Salt 是 Nafcillin Sodium Salt 的氘代化合物。Nafcillin Sodium Salt 的 CAS 号为 985-16-0。
TMIJ-0182 Avibactam sodium salt-13C5

Avibactam sodium salt-13C5 是 Avibactam sodium salt 的 13C 的标记化合物。Avibactam sodium salt 的 CAS 号为 1192491-61-4。Avibactam sodium 是一种可逆的 β-内酰胺酶抑制剂,抑制 TEM-1,P99和KPC-2 β-内酰胺酶,IC50分别为8、80和38 nM。
TMIJ-0119 Pitavastatin-d4 Sodium Salt

Pitavastatin-d4 Sodium Salt 是 Pitavastatin Sodium Salt 的氘代化合物。Pitavastatin Sodium Salt 的 CAS 号为 574705-92-3。
TMIJ-0171 Ceftazidime sodium salt-d6

Ceftazidime sodium salt-d6 是 Ceftazidime sodium salt 的氘代化合物。Ceftazidime sodium salt 的 CAS 号为 73547-61-2。
TMIJ-0301 Esomeprazole-d3 Sodium Salt

Esomeprazole-d3 Sodium Salt 是 Esomeprazole Sodium Salt 的氘代化合物。
TMIJ-0179 Faropenem-d7 Sodium Salt

Faropenem-d7 Sodium Salt 是 Faropenem Sodium Salt 的氘代化合物。Faropenem Sodium Salt 的 CAS 号为 122547-49-3。Faropenem sodium 是一种口服生物可利用的青霉烯类抗生素,能有效杀灭结核分枝杆菌,治疗结核病和社区获得性肺炎。
TMID-0234 Penicillin G-d5 potassium salt

Penicillin G-d5 potassium salt 是 Penicillin G potassium salt 的氘代化合物。Penicillin G potassium salt 的 CAS 号为 113-98-4。Benzylpenicillin potassium是青霉素家族的一种速效抗生素。
TMIJ-0319 Dehydroepiandrosterone Sulfate Sodium Salt-d6

Dehydroepiandrosterone Sulfate Sodium Salt-d6 是 Dehydroepiandrosterone Sulfate Sodium Salt 的氘代化合物。Dehydroepiandrosterone Sulfate Sodium Salt 的 CAS 号为 1099-87-2。
TMID-0294 Taurodeoxycholic Acid-d4 Sodium Salt

Taurodeoxycholic Acid-d4 Sodium Salt 是 Taurodeoxycholic Acid Sodium Salt 的氘代化合物。Taurodeoxycholic Acid Sodium Salt 的 CAS 号为 1180-95-6。Taurodeoxycholate sodium salt 是胆盐相关的阴离子洗涤剂,用于分离膜蛋白,包括线粒体内膜蛋白。它还可以抑制各种炎症反应。
TMIJ-0198 Taurochenodeoxycholic Acid-d5 Sodium Salt

Taurochenodeoxycholic Acid-d5 Sodium Salt 是 Taurochenodeoxycholic Acid Sodium Salt 的氘代化合物。Taurochenodeoxycholic Acid Sodium Salt 的 CAS 号为 6009-98-9。Taurochenodeoxycholic acid sodium 是动物胆汁酸的主要生物活性物质之一。它可诱导细胞凋亡,具有抗炎和免疫调节作用。
TMIH-0434 PHPB-d7

(R/S)-2-(1-hydroxy-n-pentyl)benzoic acid potassium salt-d7

PHPB-d7 是 PHPB 的氘代化合物。
TMIJ-0150 para-Hydroxy Atorvastatin-d5 Calcium Salt

para-Hydroxy Atorvastatin-d5 Calcium Salt 是 para-Hydroxy Atorvastatin Calcium Salt 的氘代化合物。para-Hydroxy Atorvastatin Calcium Salt 的 CAS 号为 214217-88-6。
TMIJ-0152 ortho-Hydroxy Atorvastatin-d5 Calcium Salt

ortho-Hydroxy Atorvastatin-d5 Calcium Salt 是 ortho-Hydroxy Atorvastatin Calcium Salt 的氘代化合物。ortho-Hydroxy Atorvastatin Calcium Salt 的 CAS 号为 265989-47-7。
TMIJ-0256 Estrone-d4 3-Sulfate Sodium Salt

Estrone-d4 3-Sulfate Sodium Salt 是 Estrone 3-Sulfate Sodium Salt 的氘代化合物。Estrone 3-Sulfate Sodium Salt 的 CAS 号为 438-67-5。
TMIJ-0332 Taurolithocholic Acid-d5 Sodium Salt (Major)

Taurolithocholic Acid-d5 Sodium Salt (Major) 是 Taurolithocholic Acid Sodium Salt 的氘代化合物。Taurolithocholic Acid Sodium Salt 的 CAS 号为 6042-32-6。Taurolithocholic acid sodium salt 是抑胆剂和Ca2+激动剂,可抑制放射性配体与毒蕈碱 M1 结合。
TMIJ-0167 Simvastatin EP Impurity A-d6 Sodium Salt

Simvastatin EP Impurity A-d6 Sodium Salt 是 Simvastatin EP Impurity A Sodium Salt 的氘代化合物。Simvastatin EP Impurity A Sodium Salt 的 CAS 号为 101314-97-0。
TMID-0175 DL-α-Hydroxyglutaric acid disodium salt-d4

DL-α-Hydroxyglutaric acid disodium salt-d4 是 DL-α-Hydroxyglutaric acid disodium salt 的氘代化合物。DL-α-Hydroxyglutaric acid disodium salt 的 CAS 号为 40951-21-1。DL-α-Hydroxyglutaric acid disodium salt 是一种 α-羟基酸,由 (R) -5-oxy-2-tetrahydrofuran 羧酸水解形成,在人类神经代谢疾病 D-α-羟基戊二酸尿症中过量产生。DL-α-Hydroxyglutaric acid disodium salt 是α-酮戊二酸 (α-KG)的拮抗剂,可抑制多种α-KG 依赖性双加氧酶。
TMIJ-0219 Cefpodoxime Proxetil EP Impurity A-d3 Sodium Salt

Cefpodoxime Proxetil EP Impurity A-d3 Sodium Salt 是 Cefpodoxime Proxetil EP Impurity A Sodium Salt 的氘代化合物。
T71402 Nicorandil-d4

Nicorandil-d4 is intended for use as an internal standard for the quantification of nicorandil by GC- or LC-MS. Nicorandil is an activator of sulfonylurea receptor 2B (SUR2B) linked to ATP-sensitive potassium channel Kir6.2 (EC50 = ~10 µM) and a nitric oxide (NO) donor. It is selective for SUR2B/Kir6.2 over the SUR2A/Kir6.2 channel (EC50 = >500 µM). Nicorandil activates soluble guanylate cyclase in a cell-free assay and relaxes partially depolarized isolated bovine coronary artery strips (EC50 =...
T19447 N-Demethyl Ivabradine D6 Hydrochloride

Others Others
N-Demethyl Ivabradine D6 Hydrochloride salt is the deuterium labeled N-Demethyl Ivabradine, which is a Ivabradine metabolite.
T70990 ADMA-d6

NG,NG-dimethyl-L-arginine-d6 (ADMA-d6) (hydrochloride) is intended for use as an internal standard for the quantification of NG,NG-dimethyl-L-arginine by GC- or LC-MS. ADMA is an endogenous inhibitor of nitric oxide synthase (NOS). It is formed from arginine by protein arginine methyltransferases (PRMTs) and degraded by dimethylarginine dimethylaminohydrolases (DDAHs) and alanine-glyoxylate aminotransferase 2 (AGXT2). ADMA levels are increased concomitant with an increase in blood pressure in Da...
TMIJ-0037 Sarafloxacin-d8 Hydrochloride

Sarafloxacin-d8 Hydrochloride 是 Sarafloxacin Hydrochloride 的氘代化合物。Sarafloxacin Hydrochloride 的 CAS 号为 91296-87-6。Sarafloxacin hydrochloride是一种抗菌化合物。
T69600 Spermidine-d6

Spermidine-d6 is intended for use as an internal standard for the quantification of spermidine by GC- or LC-MS. Spermidine is an endogenous polyamine. It is formed from putrescine by spermidine synthase. Spermidine (25 µM) inhibits the activity of the human inward-rectifying potassium channel Kir2.3 in a patch-clamp assay. It induces autophagy in HeLa cells when used at a concentration of 100 µM and increases the lifespan of D. melanogaster, yeast, and C. elegans. Spermidine (30 mM in the drinki...
TMIJ-0014 Fenoterol-d6 Hydrobromide

Fenoterol-d6 Hydrobromide 是 Fenoterol Hydrobromide 的氘代化合物。Fenoterol Hydrobromide 的 CAS 号为 1944-12-3。Fenoterol hydrobromide 是一种拟交感神经剂,是一种选择性的,具有口服活性 β2-肾上腺素受体 (β2-adrenoceptor) 激动剂,是一种有效的支气管扩张剂,可用于一种与哮喘、支气管炎和其他阻塞性气道疾病相关的支气管痉挛。
TMIJ-0377 Thiamine Hydrochloride-13C4

Thiamine Hydrochloride-13C4 是 Thiamine Hydrochloride 的 13C 的标记化合物。Thiamine Hydrochloride 的 CAS 号为 67-03-8。Thiamine hydrochloride 是一种必需的微量营养素,是许多中枢代谢酶的辅因子。
TMID-0187 Amitriptyline-d6 Hydrochloride

Amitriptyline-d6 Hydrochloride 是 Amitriptyline Hydrochloride 的氘代化合物。Amitriptyline Hydrochloride 的 CAS 号为 549-18-8。Amitriptyline hydrochloride 是血清素再摄取转运体和去甲肾上腺素再摄取转运体抑制剂,还与多巴胺再摄取转运体结合,其Ki为 2.58 μM。它也抑制肾上腺素能受体、毒蕈碱受体、组胺受体、5-羟色胺受体。它是TrkA和TrkA受体的激动剂,具有强神经营养活性和有抗抑郁作用。
TMID-0258 (±)-Atropine-d3 (N-methyl-d3)

(±)-Atropine-d3 (N-methyl-d3) 是 (±)-Atropine 的氘代化合物。(±)-Atropine 的 CAS 号为 51-55-8。Atropine 是竞争性的毒蕈碱乙酰胆碱受体拮抗剂,有抗近视效果。它是一种从颠茄植物中分离出来的天然生物碱,可阻断乙酰胆碱对心率和收缩力的抑制作用。
TMIJ-0519 Fosaprepitant-d4 Dimeglumine

Fosaprepitant-d4 Dimeglumine 是 Fosaprepitant Dimeglumine 的氘代化合物。Fosaprepitant Dimeglumine 的 CAS 号为 265121-04-8。Fosaprepitant dimeglumine 是 Aprepitant 的前药。它是一种神经激肽 1 受体拮抗剂,可用于预防化疗引起的恶心呕吐。
TMIH-0124 Brivanib Alaninate-d4

Brivanib Alaninate-d4 是 Brivanib Alaninate 的氘代化合物。Brivanib Alaninate 的 CAS 号为 649735-63-7。Brivanib alaninate 是一种血管内皮生长因子受体 2 (VEGFR2) 抑制剂的丙氨酸盐,IC50值为 25 nM,具有潜在的抗肿瘤活性。它对 VEGFR1 和 FGFR1 适度抑制,对 VEGFR2 的选择性是对 PDGFRβ 的 240 倍。
TMIH-0184 Desipramine-d3 HCl

Desipramine-d3 HCl 是 Desipramine HCl 的氘代化合物。Desipramine HCl 的 CAS 号为 58-28-6。Desipramine hydrochloride 是一种二苯并氮杂类衍生物三环类抗抑郁药,可作为选择性去甲肾上腺素再摄取抑制剂。 它还显示出较弱的 5-羟色胺再摄取抑制、α1 阻断、抗组胺和抗胆碱能作用。
TMIH-0512 Salbutamol-d3

Salbutamol-d3 是 Salbutamol 的氘代化合物。Salbutamol 的 CAS 号为 18559-94-9。Salbutamol 是短效的 β2 肾上腺素受体激动剂,用于哮喘和慢性阻塞性肺疾病 (COPD) 引发的支气管痉挛的研究。
TMID-0078 Irinotecan-d10 Hydrochloride

Irinotecan-d10 Hydrochloride 是 Irinotecan Hydrochloride 的氘代化合物。Irinotecan Hydrochloride 的 CAS 号为 100286-90-6。Irinotecan Hydrochloride 是喜树碱半合成衍生物的盐酸盐,是一种拓扑异构酶 I 抑制剂,可研究结肠癌和直肠癌。
TMID-0233 Salbutamol-d9

Salbutamol-d9 是 Salbutamol 的氘代化合物。Salbutamol 的 CAS 号为 18559-94-9。Salbutamol 是短效的 β2 肾上腺素受体激动剂,用于哮喘和慢性阻塞性肺疾病 (COPD) 引发的支气管痉挛的研究。

同位素标记化合物

Sacubitril-d4 calcium salt
Cat.No: TMIH-0511
Synonym: AHU-377-d4 calcium salt
Target:
Rosuvastatin-d6 Calcium Salt
Cat.No: TMIH-0504
Synonym:
Target:
Fluvastatin-d6 Sodium Salt
Cat.No: TMIH-0242
Synonym:
Target:
Fosinopril-d7 sodium salt
Cat.No: T71205
Synonym:
Target:
Rizatriptan-d6 benzoate salt
Cat.No: T71211
Synonym:
Target:
Enalaprilat-d5 sodium
Cat.No: T11193
Synonym: MK-422 D5 Sodium Salt,依那普利拉钠 D5,Enalaprilat D5 Sodium Salt
Target: Others
Indoxyl Sulfate-d5 potassium salt
Cat.No: T70313
Synonym:
Target:
Tauroursodeoxycholic Acid-d4 Sodium Salt
Cat.No: TMIH-0552
Synonym:
Target:
rac Metanephrine-d3 Hydrochloride Salt
Cat.No: TMIH-0473
Synonym:
Target:
Atorvastatin-d5 Calcium Salt
Cat.No: TMIJ-0151
Synonym:
Target:
(S)-Alogliptin Benzoate Salt-13C-d3
Cat.No: TMIH-0010
Synonym:
Target:
Rosuvastatin-d6 Sodium Salt
Cat.No: TMIJ-0164
Synonym:
Target:
Promethazine-d6 Hydrochloride Salt
Cat.No: TMID-0273
Synonym:
Target:
Nafcillin-d5 Sodium Salt
Cat.No: TMID-0269
Synonym:
Target:
Avibactam sodium salt-13C5
Cat.No: TMIJ-0182
Synonym:
Target:
Pitavastatin-d4 Sodium Salt
Cat.No: TMIJ-0119
Synonym:
Target:
Ceftazidime sodium salt-d6
Cat.No: TMIJ-0171
Synonym:
Target:
Esomeprazole-d3 Sodium Salt
Cat.No: TMIJ-0301
Synonym:
Target:
Faropenem-d7 Sodium Salt
Cat.No: TMIJ-0179
Synonym:
Target:
Penicillin G-d5 potassium salt
Cat.No: TMID-0234
Synonym:
Target:
Dehydroepiandrosterone Sulfate Sodium Salt-d6
Cat.No: TMIJ-0319
Synonym:
Target:
Taurodeoxycholic Acid-d4 Sodium Salt
Cat.No: TMID-0294
Synonym:
Target:
Taurochenodeoxycholic Acid-d5 Sodium Salt
Cat.No: TMIJ-0198
Synonym:
Target:
PHPB-d7
Cat.No: TMIH-0434
Synonym: (R/S)-2-(1-hydroxy-n-pentyl)benzoic acid potassium salt-d7
Target:
para-Hydroxy Atorvastatin-d5 Calcium Salt
Cat.No: TMIJ-0150
Synonym:
Target:
ortho-Hydroxy Atorvastatin-d5 Calcium Salt
Cat.No: TMIJ-0152
Synonym:
Target:
Estrone-d4 3-Sulfate Sodium Salt
Cat.No: TMIJ-0256
Synonym:
Target:
Taurolithocholic Acid-d5 Sodium Salt (Major)
Cat.No: TMIJ-0332
Synonym:
Target:
Simvastatin EP Impurity A-d6 Sodium Salt
Cat.No: TMIJ-0167
Synonym:
Target:
DL-α-Hydroxyglutaric acid disodium salt-d4
Cat.No: TMID-0175
Synonym:
Target:
Cefpodoxime Proxetil EP Impurity A-d3 Sodium Salt
Cat.No: TMIJ-0219
Synonym:
Target:
Nicorandil-d4
Cat.No: T71402
Synonym:
Target:
N-Demethyl Ivabradine D6 Hydrochloride
Cat.No: T19447
Synonym:
Target: Others
ADMA-d6
Cat.No: T70990
Synonym:
Target:
Sarafloxacin-d8 Hydrochloride
Cat.No: TMIJ-0037
Synonym:
Target:
Spermidine-d6
Cat.No: T69600
Synonym:
Target:
Fenoterol-d6 Hydrobromide
Cat.No: TMIJ-0014
Synonym:
Target:
Thiamine Hydrochloride-13C4
Cat.No: TMIJ-0377
Synonym:
Target:
Amitriptyline-d6 Hydrochloride
Cat.No: TMID-0187
Synonym:
Target:
(±)-Atropine-d3 (N-methyl-d3)
Cat.No: TMID-0258
Synonym:
Target:
Fosaprepitant-d4 Dimeglumine
Cat.No: TMIJ-0519
Synonym:
Target:
Brivanib Alaninate-d4
Cat.No: TMIH-0124
Synonym:
Target:
Desipramine-d3 HCl
Cat.No: TMIH-0184
Synonym:
Target:
Salbutamol-d3
Cat.No: TMIH-0512
Synonym:
Target:
Irinotecan-d10 Hydrochloride
Cat.No: TMID-0078
Synonym:
Target:
Salbutamol-d9
Cat.No: TMID-0233
Synonym:
Target:
共1165条,每页50条 1 2 3 4 5 ... 24
TargetMol Loading
联系我们
400-820-0310

上海市静安区江场三路238号8楼