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Cat. No. | Product Name | Form | Specificity Of Inhibition |
---|---|---|---|
C0005 |
Cell Counting Kit-8 (CCK-8)
Cell Counting Kit-8 (CCK-8) |
Solution in bottle | |
C0052 |
Penicillin-Streptomycin-Amphotericin B Solution (100×), Sterile
青霉素-链霉素-两性霉素B三抗溶液(100×),灭菌 |
Solution in bottle |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T14932L1 |
Ceruletide Ammonium Salt
Caerulein Ammonium Salt,Ceruletide Ammonium Salt(17650-98-5 Free base),FI-6934 Ammonium Salt,Cerulein Ammonium Salt |
cholecystokinin | GPCR/G Protein |
Ceruletide Ammonium Salt 是一种十肽,起源于热带青蛙的皮肤,是一种有效的胆囊收缩素受体 (cholecystokinin receptor) 激动剂,也是一种安全有效的胆囊收缩剂,对胆囊肌肉和胆管有直接的痉挛性作用。Ceruletide Ammonium Salt 具有镇静活性,可用于研究慢性精神分裂症。 | |||
T15024 |
Silmitasertib sodium salt
CX-4945 sodium salt |
Casein Kinase; Autophagy | Autophagy; Metabolism; Stem Cells |
Silmitasertib sodium salt (CX-4945 sodium salt) 是一种可口服的高度选择性 CK2抑制剂,对 CK2α 和 CK2α' 的 IC50值均为 1 nM。 | |||
TP1111L1 |
Tirzepatide sodium salt
LY-3298176 sodium salt,Tirzepatide sodium salt(2023788-19-2 free base) |
Glucagon Receptor | GPCR/G Protein |
Tirzepatide sodium salt (LY3298176 sodium salt) 是新型 GIP 和 GLP-1 受体双重激动剂,是人类GIP激素的合成肽类似物。Tirzepatide 具有神经保护活性,可以用于预防和治疗 2 型糖尿病和肥胖症。 | |||
T11868 |
Lorglumide sodium salt
CR-1409 sodium salt |
cholecystokinin | GPCR/G Protein |
Lorglumide sodium salt (CR-1409 sodium salt) 是胆囊收缩素受体 (CCK) 的拮抗剂。 | |||
T10397 |
ATN-161 trifluoroacetate salt
ATN-161 TFA salt |
Integrin | Cytoskeletal Signaling |
ATN-161 trifluoroacetate salt (ATN-161 TFA salt) 是一种新型整合素 α5β1 拮抗剂,可在小鼠模型中抑制血管生成和肝转移瘤的生长。 | |||
T4200 |
Sacubitril hemicalcium salt
AHU-377 (hemicalcium salt),LCZ696中间体,AHU377 calcium salt |
Neprilysin | Metabolism |
Sacubitril hemicalcium salt (AHU377 calcium salt) 是一种有效的 NEP 抑制剂,IC50=5 nM。它是研究心力衰竭药物 LCZ696 的组分之一。 | |||
T17210L |
Vaborbactam ammonium salt
RPX7009 ammonium salt,Vaborbactam ammonium salt(1360457-46-0 Free base) |
Antibacterial | Microbiology/Virology |
Vaborbactam ammonium salt 是一种 β-内酰胺酶抑制剂,可以恢复碳青霉烯类药物对 KPC 生产菌株的活性,常与其它药物连用来研究真菌感染。 | |||
T76279L1 |
Retatrutide sodium salt
Retatrutide sodium salt(2381089-83-2 free base),LY3437943 sodium salt |
Glucagon Receptor | GPCR/G Protein |
Retatrutide sodium salt 是一种有效的胰高血糖素受体 (GCGR)、葡萄糖依赖性促胰岛素多肽受体 (GIPR) 和胰高血糖素样肽-1 受体 (GLP-1R) 的三重激动剂肽。Retatrutide sodium salt 可用于研究2型糖尿病和肥胖症。 | |||
T33565 |
NAAD sodium salt
NAAD钠盐,NAAD Na salt,Deamido Nad Sodium Salt,NAAD Na, NaAD |
Others | Others |
NAAD sodium salt (NAAD Na salt) 是烟酰胺腺嘌呤二核苷酸合酶的底物,可用于研究底物的特异性和动力学。 | |||
T4535 |
Etomoxir sodium salt
(R)-(+)-乙莫克舍钠盐,(R)-Etomoxir sodium salt,Na salt,Etomoxir |
Apoptosis; Others | Apoptosis; Others |
Etomoxir sodium salt ((R)-Etomoxir sodium salt) 是一种肉碱棕榈酰转移酶 1a (CPT-1a) 抑制剂,可以阻断脂肪酸合成。Etomoxir sodium salt 具有抗肿瘤活性。 | |||
T11315 |
Fosmidomycin sodium salt
FR-31564 sodium salt |
Antibiotic; Parasite | Microbiology/Virology |
Fosmidomycin sodium salt (FR-31564 sodium salt) 是一种抗感染类抗生素,具有抗疟疾活性,抑制革兰氏阴性菌和革兰氏阳性菌。 | |||
T65070 |
Chenodeoxycholic Acid sodium salt
CDCA sodium salt |
FXR | Metabolism |
Chenodeoxycholic Acid sodium salt (CDCA sodium salt) 是一种人体中的胆汁酸,能够活化核受体 FXR,可挽救痉挛性截瘫 5 型和脑黄瘤病患者诱导多能干细胞衍生神经元的轴突变性,可用于研究胰腺坏死。 | |||
T21537L |
TMC647055 Choline Hydroxide Salt
TMC647055 Choline Hydroxide Salt (1204416-97-6 free base) |
HCV Protease | Microbiology/Virology; Proteases/Proteasome |
TMC647055 Choline Hydroxide Salt 是一种新型有效的 HCV NS5B 聚合酶非核苷抑制剂,可用于治疗 HCV 感染。它具有纳摩尔级细胞效力(EC(50) 为 82 nM),相关细胞毒性较小(CC(50)>20 μM),在大鼠和狗中具有良好的药代动力学特征。 TMC647055 显示出有体外生化、动力学和病毒学特征的前景。 | |||
TP1101 |
Nonapeptide-1 acetate salt (158563-45-2 free base)
Melanostatine-5 acetate salt,Nonapeptide-1 acetate salt |
Melanocortin Receptor | GPCR/G Protein; Neuroscience |
Nonapeptide-1 acetate salt (158563-45-2 free base) (Melanostatine-5 acetate salt) 是一种肽激素,是一种有效的 α-黑色素细胞刺激素 (α-MSH) 拮抗剂,IC50 为 11 nM。 | |||
T22592 |
ATPγS tetralithium salt
ATP-gamma-S tetralithium salt |
PERK | Apoptosis |
ATPγS tetralithium salt 是真核生物翻译起始因子 eIF4A 的核苷酸水解和RNA解链活性的底物,与 p97 突变体和朊病毒相关。 | |||
T11511 |
Guanosine-5'-triphosphate disodium salt
GTP disodium,5'-GTP disodium salt |
Others; Endogenous Metabolite | Metabolism; Others |
Guanosine-5'-triphosphate disodium salt (5'-GTP disodium salt) 是肌原性细胞分化的增强剂,也是翻译和其他重要细胞过程的能量来源。 | |||
T15025L |
CY5 triethylamine salt
CY5 triethylamine salt(146368-11-8 Free base) |
Others | Others |
CY5 triethylamine salt 是一种水溶性染料,激发光波长(nm):649,发射波长(nm):670。 | |||
T36688 |
Deoxyguanosine triphosphate trisodium salt
Deoxyguanosine 5-triphosphate,2'-Deoxyguanosine-5'-triphosphate trisodium salt,dGTP trisodium salt |
Nucleoside Antimetabolite/Analog | Cell Cycle/Checkpoint; DNA Damage/DNA Repair |
Deoxyguanosine triphosphate trisodium salt (2'-Deoxyguanosine-5'-triphosphate trisodium salt) 是细胞中用于 DNA 合成的核苷酸前体,可用于逆转录聚合酶链反应 (RT-PCR) 中以进行 DNA 扩增。 | |||
T84284 |
dITP trisodium salt
2'-Deoxyinosine-5'-triphosphate trisodium salt |
Others | Others |
dITP trisodium salt (2'-Deoxyinosine-5'-triphosphate trisodium salt) 存在于超嗜热细菌 Thermotoga maritima 中,可在诱变PCR中用作突变试剂。 | |||
TP1457 |
BIO-11006 acetate salt (901117-03-1 free base)
BIO-11006 acetate salt |
Others | Others |
BIO-11006 acetate salt (901117-03-1 free base) 是一种多糖基化富含丙氨酸的 C 激酶底物 (MARCKS) 抑制剂,类似于 MANS 肽。 | |||
T10851 |
CMP-Sialic acid sodium salt
CMP-Neu5Ac sodium salt |
Endogenous Metabolite | Metabolism |
CMP-Sialic acid sodium salt (CMP-Neu5Ac sodium salt) 是 UDP-GlcNAc 2-epimerase 的变构抑制剂,是唾液酸的活化形式,广泛存在于动物体内,参与生物体的代谢。 | |||
T18910 |
Acid Yellow 9 monosodium salt
Hydrogen 4-aminoazobenzene-3,4'-disulphonate (sodium salt) |
Others | Others |
Acid Yellow 9 monosodium salt (Hydrogen 4-aminoazobenzene-3,4'-disulphonate (sodium salt)) 是一种可被Pseudomonas fluorescens 降解的含氮染料,是此类菌株碳、氮和能量的唯一来源。 | |||
T10759 |
CEP-28122 mesylate salt (1022958-60-6 free base)
CEP-28122 mesylate salt |
ALK | Angiogenesis; Tyrosine Kinase/Adaptors |
CEP-28122 mesylate salt (1022958-60-6 free base) 是一种高选择性的口服活性 ALK 抑制剂(在基于酶的 TRF 测定中,IC50:1.9 nM)。 | |||
T16734L |
Resorufin sodium salt
试卤灵钠盐,NSC 12097 sodium salt |
Others | Others |
Resorufin sodium salt (NSC-12097 sodium salt) 是高荧光的粉红色染料,可用于 ROS/RNS 和第二种分析物的检测。 | |||
T68019L |
Ursulcholic acid trisodium salt
Ursodeoxycholic acid disulfate trisodium salt,Ursulcholic acid trisodium salt(88426-32-8 Free base) |
Others | Others |
Ursulcholic acid trisodium salt (Ursodeoxycholic acid disulfate trisodium salt) 是 ursodeoxycholic acid 的可溶形式,ursodeoxycholic acid 具有抗高血脂和利胆活性活性。 | |||
T33795 |
3-OMFP Cyclohexylammonium salt
OMFP Cyclohexylammonium salt |
Others | Others |
3-OMFP Cyclohexylammonium salt (OMFP Cyclohexylammonium salt) 是 PTEN 抑制研究的底物,可用来测定CDC25B催化结构域的酶活性。 | |||
T11125 |
Durlobactam sodium salt
杜巴坦,ETX2514 sodium salt,杜洛巴坦 |
Antibacterial | Microbiology/Virology |
Durlobactam sodium salt (ETX2514 sodium salt)是一种 β-内酰胺酶抑制剂,针对 A 类 KPC-2、C 类 AmpC 和 D 类 OXA-24,IC50 值分别为 4 nM、14 nM 和 190 nM。 Durlobactam sodium salt 可用于对包括鲍曼不动杆菌在内的耐药革兰氏阴性菌的研究。 | |||
T30677L |
C15AlkOPP t-BA salt
C15AlkOPP t-BA salt(946615-44-7 Free base),C15AlkOPP Tetrabutylamine salt(946615-44-7 Free base) |
Others | Others |
C15AlkOPP Tetrabutylamine salt 是一种"可点击"的farnesyl diphosphate (FPP)的炔烃修饰类似物。 | |||
T19820 |
MOPS sodium salt
MOPS-Na,3-(N-morpholino)propanesulfonic acid sodium salt,3-吗啉丙磺酸钠盐,Sodium 3-Morpholinopropanesulfonate,4-Morpholinepropanesulfonic acid, sodium salt |
Others | Others |
MOPS sodium salt (MOPS-Na) 在生物学中常用作缓冲剂。其中MOPS 缓冲液能使哺乳动物细胞培养基的 pH 值保持稳定。 | |||
TP1565L1 |
Foxy-5 Ammonium Salt
Foxy-5 Ammonium Salt(881188-51-8 Free base) |
Wnt/beta-catenin | Cytoskeletal Signaling; Stem Cells |
Foxy-5 Ammonium Salt是 WNT5A 激动剂,是 WNT5A 的一个模拟肽,是 Wnt 家族的非经典成员。Foxy-5 Ammonium Salt可在不影响 β-catenin 激活的情况下触发胞浆游离钙信号传导,并可抑制上皮癌细胞的迁移和侵袭。Foxy-5 Ammonium Salt在原位小鼠模型中能有效降低 WNT5A 低表达的前列腺癌细胞的转移扩散。 | |||
T12705 |
Reparixin L-lysine salt
REPERTAXIN L-赖氨酸盐,Repertaxin L-lysine salt |
CXCR | Autophagy; GPCR/G Protein; Immunology/Inflammation |
Reparixin L-lysine salt (Repertaxin L-lysine salt) 是趋化因子受体1/2 活化的变构抑制剂。 | |||
T1212 |
Ketorolac tromethamine salt
酮咯酸氨丁三醇,Acular LS,Toradol,Ketorolac tris salt,Acular |
COX | Immunology/Inflammation; Neuroscience |
Ketorolac tromethamine salt (Ketorolac tris salt) 是一种非甾体抗炎剂,是非选择性的 COX 抑制剂,对 COX-1 和 COX-2 的IC50值分别为 20 和 120 nM。 | |||
T18949L |
CY5-SE Ditriethylamine salt
CY5-SE Ditriethylamine salt(146368-14-1 Free base) |
Others | Others |
CY5-SE Ditriethylamine salt 是用于标记寡核苷酸,肽,蛋白质的氨基基团的反应染料。 激发波长 (nm): 649, 发射波长 (nm): 670 | |||
TP1545L1 |
FFAGLDD amine salt
|
Others | Others |
FFAGLDD amine salt 是MMP9选择性裂解肽,用于多柔比星(DOX)的胞浆递送,实现时间和空间可控的缓慢药物递送和释放。 | |||
T2160 |
Suramin Sodium Salt
苏拉明钠,BAY-205,Suramin hexasodium salt,苏拉明钠盐,NF-060 |
Apoptosis; Phosphatase; SARS-CoV; Sirtuin; Reverse Transcriptase; Topoisomerase; Parasite | Apoptosis; Chromatin/Epigenetic; DNA Damage/DNA Repair; Metabolism; Microbiology/Virology |
Suramin Sodium Salt (BAY-205) 是可逆的竞争性蛋白酪氨酸磷酸酶抑制剂。它抑制 IP5K,是抗寄生虫,抗肿瘤和抗血管生成剂。它是sirtuins 的有效抑制剂,也是 SARS-CoV-2 RNA 依赖性 RNA 聚合酶抑制剂。 | |||
T18942L |
Cy5-N3 triethylamine salt
Cy5-N3 triethylamine salt(1621101-43-6 free base) |
Others | Others |
Cy5-N3 triethylamine salt 是一种花箐类荧光染料。CY5-N3 可用于研究细胞成像。 | |||
TP2226 |
BzATP triethylammonium salt
|
P2X Receptor | Membrane transporter/Ion channel; Neuroscience |
BzATP triethylammonium salt 是一种 P2X 受体激动剂,对 P2X1、P2X2、P2X3、P2X2/3、P2X4 和 P2X7 均有效 (pEC50=8.74/5.26/7.10/7.50/6.19/6.31/5.33)。BzATP triethylammonium salt 可以诱导细胞死亡并减少突触传递。 | |||
T6747 |
8-Bromo-cAMP sodium salt
8-Br-Camp sodium salt,8-溴腺苷-3',5'-环单磷酸钠,8-Bromo-cAMP(sodium salt),8-Bromo-cAMP |
PKA | Tyrosine Kinase/Adaptors |
8-Bromo-cAMP sodium salt (8-Br-Camp sodium salt) 是一种环 AMP (cAMP) 类似物,一种 cAMP 依赖性蛋白激酶 (PKA) 的激活剂。8-Bromo-cAMP sodium salt 具有抗肿瘤活性。 | |||
T5847 |
Cloprostenol sodium salt
ICI 80996 sodium salt,DL-Cloprostenol sodium,氯前列烯醇钠,氯前列烯醇纳,Cloprostenol sodium |
Prostaglandin Receptor | GPCR/G Protein; Immunology/Inflammation |
Cloprostenol sodium salt (ICI 80996 sodium salt) 是一种合成的前列腺素类似物,是 PGF2α受体的激动剂,具有黄体溶解性。 | |||
T0148L |
Folinic Acid Calcium Salt Pentahydrate
Folinic acid,亚叶酸钙五水合物,Leucovorin Calcium Pentahydrate,Leucovorin calcium salt pentahydrate |
Others; Antifolate | Cell Cycle/Checkpoint; Others |
Folinic Acid Calcium Salt Pentahydrate (Leucovorin Calcium Pentahydrate) 是一种还原型叶酸,是一种解毒剂,通常与甲氨蝶呤 (MTX) 联用,以降低 MTX 诱导的毒性。 | |||
T4251 |
GJ103 sodium salt
|
ATM/ATR | DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling |
GJ103 sodium salt 是 GJ072 的活性类似物,它是一种通读化合物 (RTC)。它已被证明可以降低水溶液的表面张力,使分子更容易在溶液中移动。它还被证明可以降低水溶液的粘度,使分子更容易在溶液中移动。此外,它还被证明可以降低水溶液的pH 值,这会对生物体的生化和生理过程产生各种影响。 | |||
T72505L |
CTP Synthetase-IN-1 Ammonium salt
CTPS-IN-1 Ammonium salt,CTP Synthetase-IN-1 Ammonium salt(2338811-71-3 Free base) |
Others | Others |
CTP Synthetase-IN-1 Ammonium salt 是一种具有口服活性和高效性的胞苷 5'-三磷酸合成酶 (CTPS) 抑制剂,具有潜在的抗菌抗炎抗肿瘤活性,可用于研究 SARS-CoV-2病毒感染。 | |||
T5878 |
β-Glycerophosphate disodium salt pentahydrate
五水β-甘油磷酸钠,BETA-GLYCEROL PHOSPHATE DISODIUM SALT,B-甘油磷酸钠五水合物,β-Glycerol phosphate disodium salt pentahydrate |
Phosphatase; Endogenous Metabolite | Metabolism |
β-Glycerophosphate disodium salt pentahydrate 是一种磷酸酶 (phosphatase) 抑制剂。 | |||
T39477 |
Ca-DTPA trisodium salt hydrate
Ca-DTPA trisodium salt hydrate,Calcium trinatrium diethylenetriaminepentaacetic acid hydrate |
Others | Others |
Calcium trinatrium diethylenetriaminepentaacetic acid hydrate (Ca-DTPA trisodium salt hydrate) 是螯合剂和有用的解毒剂,如急性镉中毒。它是一种无毒的 CMV 复制抑制剂。 | |||
T38404 |
MJ33 lithium salt
|
ROS | Immunology/Inflammation |
MJ33 lithium salt 是 NADPH 氧化酶 2 型介导的 ROS 生成抑制剂,是一种氟化磷脂类似物,可抑制过氧化物还蛋白 6 (Prdx6) 的磷脂酶 A2 (PLA2) 活性,可用于研究急性肺损伤。 | |||
T19596 |
UDP-GlcNAc Disodium Salt
Uridine 5′-diphospho-N-acetylglucosamine,5′-二磷酸尿嘧啶核苷-N-乙酰半乳糖胺二钠盐,UDP-α-D-N-Acetylglucosamine Disodium Salt |
Others | Others |
UDP-GlcNAc Disodium Salt (UDP-α-D-N-Acetylglucosamine Disodium Salt) 是一种 O-GlcNAc 转移酶 (OGT) 的供体底物。 | |||
T13564L2 |
AZ7550 trimesylate salt
AZ7550 Mesylate,AZ7550 trimesylate salt (1421373-99-0 free base) |
MLK | MAPK |
AZ7550 trimesylate salt (AZ7550 Mesylate) 是奥希替尼的活性代谢产物,AZ7550 trimesylate salt 抑制 IGF1R 活性,可用于研究非小细胞肺癌。 | |||
T9306 |
EST64454 Maleic acid salt
|
Others | Others |
EST64454 Maleic acid salt 是EST64454的马来酸盐形式。EST64454是一种用于治疗疼痛的高可溶性σ1受体拮抗剂临床候选药物。 | |||
T8855 |
Polydeoxyribonucleotide(Sodium salt)
Polydeoxyribonucleotide from salmon |
Others | Others |
Polydeoxyribonucleotide(Sodium salt) 可改善大鼠跟腱损伤模型中各种生长因子的分泌,促进胶原蛋白合成,恢复跟腱的拉伸强度。 | |||
T30677L1 |
C15AlkOPP Tetrabutylamine salt (1:2)
C15AlkOPP Tetrabutylamine salt(1:2)(946615-44-7 Free base) |
Others | Others |
C15AlkOPP Tetrabutylamine salt (1:2)是一种FPP 类似物,具有炔基,允许前戊酰化后的蛋白质标记。C15AlkOPP Tetrabutylamine salt (1:2)可用于异戊二烯组学分析。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T8393 |
Uridine triphosphate trisodium salt
UTP, Trisodium Salt,Uridine 5'-triphosphate trisodium salt,尿苷-5'-三磷酸三钠盐,Uridine triphosphate (trisodium salt) |
Others | Others |
Uridine triphosphate trisodium salt (UTP, Trisodium Salt) 是一种核苷酸,在正常和疾病状态,均能够调节胰腺内分泌和外分泌、通道、增殖、转运体和细胞内信号传导的功能。 | |||
T4730 |
Thymidine-5'-monophosphate disodium salt
胸苷酸二钠,Thymidine 5'-monophosphate disodium salt,TMP DISODIUM SALT |
Others; Endogenous Metabolite | Metabolism; Others |
Thymidine-5'-monophosphate disodium salt (TMP DISODIUM SALT) 是内源性代谢产物的一种。 | |||
T3S0156 |
Atractyloside potassium salt
Atractyloside Dipotassium Salt,苍术苷钾盐,苍术苷二钾盐 |
Others | Others |
Atractyloside potassium salt (Atractyloside Dipotassium Salt) 是一种从苍术果实中分离出得到的二萜苷类化合物,具有毒性。它能抑制大鼠心脏线粒体膜的氯离子通道。它是高效、特异性的线粒体 ADP/ATP 转运 (ADP/ATP transport) 抑制剂。 | |||
T5079 |
Adenosine 5'-diphosphate sodium salt
腺苷-5‘-二磷酸钠盐,Adenosine-5'-diphosphate trisodium salt,ADP sodium salt |
Others; Endogenous Metabolite | Metabolism; Others |
Adenosine 5'-diphosphate sodium salt (ADP sodium salt) 是一种核苷二磷酸,是一种 ATP 酶对 ATP 去磷酸化的产物。它通过在 P2T-嘌呤受体上的作用诱导人血小板聚集并抑制刺激的腺苷酸环化酶。 | |||
T2944 |
Danshensu sodium salt
Sodium Danshensu,(±)-DanShenSu sodium salt,丹参素钠,(±)-DanShenSu sodium sal |
P450; Autophagy | Autophagy; Metabolism |
Danshensu sodium salt (Sodium Danshensu) 是从中国草本丹参中提取的一种天然产物,可以抑制去氧肾上腺素和CaCl2 在无Ca2+ 培养基中引起的血管收缩。 | |||
T4969 |
Guanosine 5'-triphosphate trisodium salt
鸟苷-5'-三磷酸三钠盐,GTP Trisodium salt,5'-GTP trisodium salt |
Endogenous Metabolite | Metabolism |
Guanosine 5'-triphosphate trisodium salt (5'-GTP trisodium salt) 为G蛋白(G proteins)信号转导过程中的活化剂。 | |||
T19262 |
D-Glucose 6-phosphate disodium salt
D-Glucose 6-phosphate disodium salt |
Endogenous Metabolite | Metabolism |
D-Glucose 6-phosphate disodium salt 广泛存在于生物提内的化合物,是葡萄糖第 6 号碳经过磷酸化后生成的分子,参与磷酸戊糖途径与糖酵解途径等体内多种多种代谢调节途径。 | |||
T1033 |
Monensin sodium salt
莫能菌素钠盐,Sodium Monensin,Monensin A sodium salt |
Sodium Channel; Antibacterial; Antibiotic | Membrane transporter/Ion channel; Microbiology/Virology |
Monensin sodium salt (Monensin A sodium salt) 是由肉桂链霉菌 分泌的抗生素。它是一种介导Na+/H+交换的离子载体。它引起细胞多泡体 (MVBs) 增大并调节外泌体的分泌。 | |||
T21518 |
Colistin methanesulfonate sodium salt
粘杆菌素甲基磺酸钠,Colistin Methanesulfonate (sodium salt) |
Cell wall; Antibacterial | Immunology/Inflammation; Microbiology/Virology |
Colistin methanesulfonate sodium salt (Colistimethate Sodium) 是一种来自 Bacillus colistinus 的环状多肽抗生素,由多粘菌素 E1 和 E2 组成。 | |||
T4743 |
Uridine 5′-diphosphoglucose disodium salt
二磷酸尿苷葡萄糖二钠盐,UDP-Glucose sodium salt,UDPG sodium salt,UDP-α-D-Glucose sodium salt,Uridine 5'-diphosphoglucose disodium sal |
Endogenous Metabolite; P2Y Receptor | GPCR/G Protein; Metabolism; Neuroscience |
Uridine 5′-diphosphoglucose disodium salt (UDP-Glucose sodium salt) 是一种内源性核苷酸糖,参与代谢中的糖基转移酶反应。它是 P2Y14 受体的激动剂,EC50为 0.35 μM。 | |||
T4706 |
Uridine-5'-diphosphate disodium salt
UDP disodium salt,Uridine 5'-diphosphate disodium salt hyd,尿苷-5'-二磷酸二钠盐 |
DNA/RNA Synthesis; Endogenous Metabolite; P2Y Receptor | Cell Cycle/Checkpoint; DNA Damage/DNA Repair; GPCR/G Protein; Metabolism; Neuroscience |
Uridine-5'-diphosphate disodium salt (UDP disodium salt) 是一种选择性 P2Y6受体激动剂,EC50为300 nM,对人 P2Y6受体的 pEC50为6.52。它可刺激炎症介质的产生、吞噬作用和血管收缩,催化多种底物的葡糖醛酸糖化反应,用于核酸生物合成。 | |||
T16527 |
Phytic acid dodecasodium salt hydrate
植酸十二钠盐,myo-Inositol, hexakis(dihydrogen phosphate) dodecasodium salt hydrate,Inositol hexaphosphate dodecasodium salt hydrate |
Others; Xanthine Oxidase; Endogenous Metabolite | Metabolism; Others |
Phytic acid dodecasodium salt hydrate (myo-Inositol, hexakis(dihydrogen phosphate) dodecasodium salt hydrate) 是种子和谷物的磷储存化合物。 Phytic acid dodecasodium salt hydrate 抑制酶促超氧化物源黄嘌呤氧化酶,IC50 为 6 mM,并具有抗氧化、神经保护和抗炎作用。 | |||
T5283 |
NADH disodium salt
Disodium NADH,NADH, disodium salt hydrate,beta-烟酰胺腺嘌呤二核苷二钠 |
Others; Endogenous Metabolite | Metabolism; Others |
NADH disodium salt hydrate是氧化还原酶的辅酶。 NADH在分解代谢过程中起到再生电子供体的作用,包括糖酵解,柠檬酸循环和β-氧化。 | |||
T22446 |
NADP disodium salt
Disodium NADP,Triphosphopyridine nucleotide disodium salt,beta-烟酰胺腺嘌呤二核苷酸磷酸二钠盐 |
Others | Others |
NADP disodium salt (Disodium NADP) 是一种氧化还原辅助因子,是一种烟酰胺腺嘌呤二核苷酸。它是代谢中电子转移的关键辅因子,可以被交替氧化 (NADP+) 和还原 (NADPH)。 | |||
T0958 |
Penicillin G sodium salt
青霉素钠,Penicillin G Sodium,Benzylpenicillin sodium salt,Benzylpenicillin Sodium |
GABA Receptor; Antibacterial; Antibiotic | Membrane transporter/Ion channel; Microbiology/Virology; Neuroscience |
Penicillin G sodium(Benzylpenicillin sodium) salt 是一种 β-内酰胺类抗生素。 | |||
T5258 |
Dodecanedioic acid diammonium salt
十二烷二酸 二铵盐,1,10-Decanedicarboxylic acid diammonium salt |
Others | Others |
Dodecanedioic acid diammonium salt (1,10-Decanedicarboxylic acid diammonium salt) 是一种二元羧酸,它是水溶性的,并且参与了脂类和碳水化合物的代谢途径中间体。 | |||
T65269 |
L-Aspartic acid potasium salt
Aspartic acid potasium salt,Potassium L-aspartate |
Others | Others |
L-aspartic acid potasium salt(VX-548) 是一种广泛存在于动植物体内的氨基酸。L-aspartic acid potasium salt驱动氮氧化物的产生,从而促进吞噬作用,有助于提高鱼类的成活率。L-aspartic acid potasium salt 可对抗生素产生刺激,刺激作用可能与参与天冬氨酸-4-半醛生物合成的前体有关。 | |||
T5693 |
Pyrroloquinoline quinone disodium salt
吡咯喹啉醌二钠盐,Methoxatin disodium salt |
Others; Endogenous Metabolite | Metabolism; Others |
Pyrroloquinoline quinone disodium salt (Methoxatin disodium salt) 一种阴离子型氧化还原循环原醌,作为氧化还原辅助因子。它是从嗜甲基细菌的培养物中分离的,也存在于哺乳动物的组织。它是哺乳动物的必需营养素,对免疫功能很重要。 | |||
T2812 |
ATP disodium salt hydrate
ATP disodium,ATP disodium salt,Adenosine disodium triphosphate,三磷酸腺苷二钠盐 |
Others; Endogenous Metabolite | Metabolism; Others |
ATP disodium salt hydrate (Adenosine disodium triphosphate) 是体内能量储存和代谢的重要物质,为代谢提供能量,同时在细胞中作为辅酶发挥作用。同时,它是也是免疫和炎症中重要的内源性信号分子。 | |||
T5087 |
DL-Isocitric acid trisodium salt
异柠檬酸三钠盐,Isocitric acid trisodium salt |
Others; Endogenous Metabolite | Metabolism; Others |
DL-Isocitric acid trisodium salt 是内源性代谢产物的一种。 | |||
T4941 |
D-Fructose-6-phosphate disodium salt
D-FRUCTOSE 6-PHOSPHATE DISODIUM SALT,D-果糖-6-磷酸二钠 |
Others; Endogenous Metabolite | Metabolism; Others |
D-Fructose-6-phosphate disodium salt (D-FRUCTOSE 6-PHOSPHATE DISODIUM SALT) 是内源性代谢产物的一种。 | |||
T37984 |
Fosfructose, sodium salt, hydrate (1:3:8)
D-Fructose-1,6-bisphosphate , sodium salt, hydrate (1:3:8) |
Others | Others |
D-Fructose-1,6-bisphosphate sodium salt hydrate 是碳水化合物代谢的中间体,包括糖酵解和糖异生。在糖酵解过程中,它是由磷酸果糖激酶磷酸化果糖-6-磷酸产生的。由果糖-1,6-二磷酸酶-1介导的逆反应是糖异生的限速步骤之一。同样的反应也发生在植物的叶绿体中,D-Fructose-1,6-bisphosphate sodium salt hydrate 作为还原性戊糖磷酸循环的一部分。由于癌细胞采用糖酵解作为代谢能量产生的主要来源,这一途径已成为癌症化疗的主要靶点。 | |||
T21066 |
Norepinephrine bitartrate salt
|
Adrenergic Receptor | GPCR/G Protein; Neuroscience |
Norepinephrine bitartrate salt 是一种肾上腺素能神经递质。 | |||
T4713 |
Phosphorylcholine chloride calcium salt tetrahydrate
Phosphocholine chloride calcium salt tet,胆碱磷酸氯化钙四水,CalciuM Phosphorylcholine Tetrahydrate |
Others; Endogenous Metabolite | Metabolism; Others |
Phosphorylcholine chloride calcium salt tetrahydrate (Phosphocholine chloride calcium salt tet) 是内源性代谢产物的一种。 | |||
T1352 |
ATP disodium salt
Adenosine 5'-triphosphate disodium salt,三磷酸腺苷二钠,ATP,ATP disodium,腺苷-5'-三磷酸二钠盐,Adetide,Adenosine-Triphosphate,Disodium adenosine triphosphate |
P2X Receptor; Endogenous Metabolite | Membrane transporter/Ion channel; Metabolism; Neuroscience |
ATP disodium salt (Adenosine-Triphosphate) 是体内能量储存的重要物质,为代谢提供能量,同时在细胞中作为辅酶发挥作用。Adenosine 5'-triphosphate disodium salt 也是免疫和炎症中重要的内源性信号分子。 | |||
T4897 |
Inosine-5'-triphosphate trisodium salt
ITP,肌苷-5'-三磷酸三钠盐,三磷酸肌苷三钠盐,Inosine 5'-triphosphate trisodium salt |
Others; Endogenous Metabolite | Metabolism; Others |
Inosine-5'-triphosphate trisodium salt (ITP) 是三磷酸核苷,能够作为 ATPases 和 GTPases 的底物。 | |||
T4901 |
5'-Guanylic acid disodium salt
Guanosine 5'-monophosphate disodium salt,5'-鸟苷酸二钠,鸟苷钠5'-单磷酸,GMP-5 |
Others; Endogenous Metabolite | Metabolism; Others |
5'-Guanylic acid disodium salt (GMP-5) 由鸟嘌呤,核糖和磷酸组成,是信使 RNA 中的一种核苷酸单体。 鸟苷衍生物参与细胞内信号转导,并已鉴定存在于端粒,核糖体 DNA,免疫球蛋白重链转换区和原癌基因的控制区中的重复基因组序列中。 | |||
T5067 |
Flavin adenine dinucleotide disodium salt
Flavin Adenine Dinucleotide Disodium,黄素腺嘌呤二核苷酸二钠,FAD sodium salt,FAD-Na2 |
Others; Endogenous Metabolite | Metabolism; Others |
Flavin adenine dinucleotide disodium salt (FAD sodium salt) 是一种辅酶,作用是促进细胞氧化还原反应中黄素酶的电子转移。 | |||
T5068 |
D-Glucuronic acid sodium salt monohydrate
Sodium D-glucuronate,D-葡糖醛酸钠一水,D-葡萄糖醛酸钠,D(+)-Glucuronic acid sodium salt monohydrate |
Others; Endogenous Metabolite | Metabolism; Others |
D-Glucuronic acid sodium salt monohydrate (Sodium D-glucuronate) 是内源性代谢产物的一种。 | |||
TMA2440 |
Uridine 5'-monophosphate disodium salt
尿苷-5'-单磷酸二钠盐,Disodium UMP,尿苷酸二钠盐,Disodium uridine-5'-monophosphate,5'-UMP disodium salt,Disodium 5'-Uridylate |
Others | Others |
Uridine 5'-monophosphate disodium salt (Disodium UMP) 是合成 RNA 的一种重要成分。 | |||
T6674 |
L-Ascorbic acid sodium salt
(+)-Sodium L-ascorbate,Vitamin C sodium salt,Sodium ascorbate,L-Ascorbic acid sodium,抗坏血酸钠,Sodium L-ascorbate,维生素C钠 |
Apoptosis; Others; Calcium Channel; Reactive Oxygen Species; Endogenous Metabolite | Apoptosis; Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; NF-κB; Others |
L-Ascorbic acid sodium salt (Vitamin C sodium salt) 是一种电子供体,是一种内源性抗氧化剂。它还是一种胶原沉积促进剂和弹性生成抑制剂。它选择性抑制 Cav3.2 通道(Cav3.2 channels),IC50为 6.5 μM。 | |||
T3551 |
D-Pantothenic acid hemicalcium salt
泛酸钙,D-Pantothenic Acid Calcium,D-泛酸半钙,Calpanate,Calcium D-pantothenate,Vitamin B5 calcium salt,Calcium pantothenate,Calcium D-Panthotenate |
Apoptosis; Endogenous Metabolite | Apoptosis; Metabolism |
D-Pantothenic acid hemicalcium salt (Calcium pantothenate) 是一种水溶性维生素,能够减少苹果汁中的棒曲霉素。 | |||
T19343L |
Glycerol 3-phosphate biscyclohexylammonium salt
|
Endogenous Metabolite | Metabolism |
Glycerol 3-phosphate biscyclohexylammonium salt 是胞质甘油 3-磷酸脱氢酶途径中产生的,即利用 NADH 还原二羟丙酮磷酸的过程。 | |||
T4070 |
Glycocholic Acid Sodium Salt
Glycocholate Sodium,Sodium Glycocholate,甘氨胆酸钠盐 |
Others | Others |
Glycocholic Acid Sodium Salt (Sodium Glycocholate) 是一种结合胆汁盐和离子生物去污剂。它参与脂肪的乳化。 | |||
T5073 |
Inosine 5'-monophosphate disodium salt hydrate
Inosine 5'-monophosphate disodium salt,5'-IMP-Na2,肌苷5-单磷酸二钠盐水合物,Disodium 5'-inosinate monohydrate |
Others; Endogenous Metabolite | Metabolism; Others |
Inosine 5'-monophosphate disodium salt hydrate (Inosine 5'-monophosphate disodium salt) 或肌苷酸是次黄嘌呤的核糖核苷酸,是嘌呤合成过程中形成的第一个核苷酸。 | |||
TN2349 |
Taurodeoxycholate sodium salt
Sodium taurodeoxylate,牛磺脱氧胆酸钠 |
Endogenous Metabolite | Metabolism |
Taurodeoxycholate sodium salt (Sodium taurodeoxylate) 是胆盐相关的阴离子洗涤剂,用于分离膜蛋白,包括线粒体内膜蛋白。它还可以抑制各种炎症反应。 | |||
T4915 |
β-Glycerophosphate disodium salt hydrate
|
Phosphatase; Endogenous Metabolite | Metabolism |
β-Glycerophosphate disodium salt hydrate 是一种磷酸酶抑制剂,是内源性代谢产物的一种。 | |||
T5069 |
D-Glucose 6-phosphate potassium salt
|
Others | Others |
在细胞中,当葡萄糖被己糖激酶或葡萄糖激酶磷酸化或在糖原分解过程中通过磷酸葡萄糖变位酶转化葡萄糖 1-磷酸时,会产生D-glucose 6-phosphate (G6P)。 G6P 位于糖酵解和戊糖磷酸途径的起点。当血糖水平高时,它也可以作为糖原储存。 | |||
TQ0215 |
Salinomycin sodium salt
盐霉素钠,Sodium salinomycin,Salinomycin sodium |
Apoptosis; Wnt/beta-catenin; Antibacterial; Antibiotic; Autophagy | Apoptosis; Autophagy; Cytoskeletal Signaling; Microbiology/Virology; Stem Cells |
Salinomycin sodium salt (Sodium salinomycin) 是钾离子载体抗生素,是作用于 Wnt/Fzd/LRP 复合物的Wnt/β-catenin 信号传导抑制剂,能阻断 Wnt 诱导的 LRP6 磷酸化,导致 LRP6 蛋白降解。它选择性抑制人肿瘤干细胞。 | |||
T3092 |
Nigericin sodium salt
尼日利亚菌素,尼日利亚菌素钠盐 |
Potassium Channel; NOD-like Receptor (NLR); Antibacterial; Antibiotic; NOD | Immunology/Inflammation; Membrane transporter/Ion channel; Microbiology/Virology; NF-κB |
Nigericin sodium salt 属于抗生素,是一种 NLRP3 激活剂,也是一种阳离子离子载体。Nigericin sodium 可以触发 NALP3 炎性体的激活,可抑制高尔基体功能并抑制革兰氏阳性菌的生长。 | |||
T0281 |
Meclocycline sulfosalicylate salt
磺基水杨酸甲氯环素,Meclutin,Mecloderm,甲环素磺基水杨酸盐,Meclan Cream |
Antibacterial; Antibiotic | Microbiology/Virology |
Meclocycline sulfosalicylate salt (Mecloderm) 是一种具有广谱抗菌活性的四环素抗生素,可预防皮肤细菌感染。 | |||
T13528 |
Acetoacetic acid sodium salt
乙酰乙酸钠,3-氧代丁酸钠盐 |
Others | Others |
Acetoacetic acid sodium salt 是一种内源性的非酯化脂肪酸代谢物,与人类糖尿病的发展相关。它诱导氧化应激,抑制牛肝细胞中极低密度脂蛋白的组装。 | |||
T5303 |
Isethionic acid sodium salt
Sodium isethionate,羟乙基磺酸钠 |
Others; Endogenous Metabolite | Metabolism; Others |
Isethionic acid sodium salt (Sodium isethionate) 是内源性代谢产物的一种。 | |||
T1138 |
Taurocholic acid sodium salt hydrate
牛胆酸钠,牛磺胆酸钠水合物,Sodium taurocholate hydrate,Taurocholic Acid sodium hydrate |
Others; Potassium Channel; Endogenous Metabolite | Membrane transporter/Ion channel; Metabolism; Others |
Taurocholic acid sodium salt hydrate (Sodium taurocholate hydrate) 是一种胆汁酸钠盐水合物,作用是参与脂肪的乳化。 | |||
T8186 |
Xanthosine 5'-monophosphate sodium salt
XMP,黄苷-5′-单磷酸钠,L-XMP Sodium |
Others | Others |
Xanthosine 5'-monophosphate sodium salt (L-XMP Sodium) 是嘌呤代谢的一种中间体。它可用于研究遗传密码,核酸结构以及 DNA,RNA 和蛋白质合成。 | |||
T4727 |
Taurolithocholic acid sodium salt
牛磺石胆酸钠,Sodium taurolithocholate |
Others; Calcium Channel | Membrane transporter/Ion channel; Metabolism; Others |
Taurolithocholic acid sodium salt (Sodium taurolithocholate) 是抑胆剂和 Ca2+激动剂,可抑制放射性配体与毒蕈碱 M1 结合。 | |||
T5584 |
Phytic acid sodium salt
Sodium phytate hydrate,玉米 |
Others | Others |
Phytic acid sodium salt (Sodium phytate hydrate) 源于豆类种子中,具有抗营养活性。它是 [PO4]3-储藏库,是其他肌醇磷酸酯和焦磷酸酯的前体,在植物中被植酸酶逐步水解。 | |||
T40814 |
Colominic acid sodium salt
Polysialic acid sodium salt,Colominic acid sodium salt |
Others | Others |
Colominic acid sodium salt, also known as polysialic acid sodium salt, is naturally isolated from the cell wall of Escherichia coli and animals. It exhibits a red color with an absorption maximum of 530 nm and possesses anti-bacterial activity. | |||
T4922 |
Uridine 5′-triphosphate tris salt
尿苷-5′-三磷酸酯 三羟甲基氨基甲烷盐,Uridine 5'-triphosphoric acid |
Others; Endogenous Metabolite | Metabolism; Others |
Uridine 5′-triphosphate tris salt (Uridine 5'-triphosphoric acid) 是 P2Y 受体的激动剂,已用于研究细胞内 Ca2+ 的浓度,以及用于体外激酶测定的磷酸盐供体。 | |||
T5259 |
Glycochenodeoxycholic acid sodium salt
GCDCA,甘氨鹅脱氧胆酸钠,Sodium glycochenodeoxycholate |
Apoptosis; Others; Endogenous Metabolite | Apoptosis; Metabolism; Others |
Glycochenodeoxycholic acid sodium salt 是一种从脱氧鹅胆酸和甘氨酸在肝脏中形成的胆汁盐,可诱导肝细胞凋亡。它起到洗涤剂的作用,可溶解脂肪吸收,并本身被吸收。 | |||
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Cat. No. | Product Name | Species | Expression System |
---|---|---|---|
TMPH-01424 |
GUCA2B Protein, Human, Recombinant (His)
Guanylate cyclase activator 2B,GUCA2B |
Human | HEK293 Cells |
Endogenous activator of intestinal guanylate cyclase. It stimulates this enzyme through the same receptor binding region as the heat-stable enterotoxins. May be a potent physiological regulator of intestinal fluid and electrolyte transport. May be an autocrine/paracrine regulator of intestinal salt and water transport. GUCA2B Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with N-6xHis tag. The predicted molecular weight is 13.5 kDa and the accession number is Q16661. | |||
TMPY-03353 |
CEL Protein, Mouse, Recombinant (His)
1810036E18Rik,carboxyl ester lipase,BAL |
Mouse | Baculovirus Insect Cells |
CEL-maturity onset diabetes of the young (MODY), diabetes with pancreatic lipomatosis and exocrine dysfunction, is due to dominant frameshift mutations in the acinar cell carboxyl ester lipase gene (CEL). Bile-salt activated carboxylic ester lipase (CEL) is a major triglyceride, cholesterol ester and vitamin ester hydrolytic enzyme contained within pancreatic and lactating mammary gland secretions. Carboxyl ester lipase is a digestive pancreatic enzyme encoded by the CEL gene. Mutations in CEL c... | |||
TMPJ-00875 |
NPPB Protein, Human, Recombinant (His)
NPPB,γ-Brain Natriuretic Peptide,Gamma-Brain Natriuretic Pep... |
Human | E. coli |
Human Natriuretic peptides B acts as a cardiac hormone; it is associated with many biological actions, such as diuresis, natriuresis, vasorelaxation, which inhibits the secretion of rennin and aldosterone. It acts as a paracrine antifibrotic factor in the heart. Natriuretic peptides B can help restore the body balance of salt and water, improves the heart function. Natriuretic peptides B binds and stimulates the cGMP production of the NPR1 receptor and binds the clearance receptor NPR3. | |||
TMPJ-01396 |
PIN4 Protein, Human, Recombinant (His)
Peptidyl-prolyl cis-trans isomerase Pin4,Parvulin-14,Peptidy... |
Human | E. coli |
Peptidyl-prolyl cis-trans isomerase NIMA-interacting 4(PIN4) is a peptidyl-prolyl cis/trans isomerase (PPIase) which interacts with NIMA and is vital for cell cycle regulation. PIN4 has 2 different isoforms: PAR14 and PAR17. Furthermore, PIN4 protein binds to double-stranded DNA under physiological salt conditions. PIN4 is involved as a ribosomal RNA processing factor in ribosome biogenesis. The PAR14 binds to tightly bent AT-rich stretches of double-stranded DNA, but PAR17 binds to double-stran... | |||
TMPY-02133 |
Carbonic Anhydrase VB Protein, Human, Recombinant (His)
carbonic anhydrase VB, mitochondrial,CA-VB,MGC39962 |
Human | E. coli |
Carbonic anhydrase 5B, also known as carbonate dehydratase VB, carbonic anhydrase VB, CA-VB and CA5B, is amember of the alpha-carbonic anhydrase family. The strongest expression of CA5B / CA-VB is in heart, pancreas, kidney, placenta, lung, and skeletal muscle. It is not expressed in liver. Carbonic anhydrases (CAs) are a large family of zinc metalloenzymes first discovered in 1933 that catalyze the reversible hydration of carbon dioxide. CAs participate in a variety of biological process... | |||
TMPY-01877 |
CA5A Protein, Human, Recombinant (His)
CA5,GS1-21A4.1,CA5AD,carbonic anhydrase VA, mitochondrial,CA... |
Human | E. coli |
Carbonic anhydrase 5A, mitochondrial, also known as Carbonate dehydratase VA, Carbonic anhydrase VA, CA-VA and CA5A, is a member of thealpha-carbonic anhydrase family. Carbonic anhydrases (CAs) are a large family of zinc metalloenzymes first discovered in 1933 that catalyze the reversible hydration of carbon dioxide. CAs participate in a variety of biological processes, including respiration, calcification, acid-base balance, bone resorption, and the formation of aqueous humor, cerebrospi... |
Cat. No. | Product Name | Target | Signaling Pathways |
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TMIH-0511 |
Sacubitril-d4 calcium salt
AHU-377-d4 calcium salt |
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Sacubitril-d4 calcium salt 是 Sacubitril calcium salt 的氘代化合物。 | |||
TMIH-0504 |
Rosuvastatin-d6 Calcium Salt
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Rosuvastatin-d6 Calcium Salt 是 Rosuvastatin Calcium Salt 的氘代化合物。Rosuvastatin Calcium Salt 的 CAS 号为 147098-20-2。Rosuvastatin calcium 是肝羟甲基戊二酰辅酶 A 还原酶的选择性和竞争性抑制剂,具有抗血脂活性。它降低成熟 hERG 的表达以及热休克蛋白 70 与 hERG 蛋白的相互作用,还降低低密度脂蛋白胆固醇、甘油三酯和 C-反应蛋白水平。它阻断人类醚-a-go-go相关基因电流,延迟心脏复极化,来延长动作电位持续时间和校正 QT 间期间隔。 | |||
TMIH-0242 |
Fluvastatin-d6 Sodium Salt
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Fluvastatin-d6 Sodium Salt 是 Fluvastatin Sodium Salt 的氘代化合物。Fluvastatin Sodium Salt 的 CAS 号为 93957-55-2。Fluvastatin sodium salt 是羟甲基戊二酰辅酶 A 还原酶的竞争性抑制剂,IC50为 8 nM。它通过依赖 Nrf2 的抗氧化通路保护血管平滑肌细胞免受氧化应激,是一种常用的降胆固醇剂。 | |||
T71205 |
Fosinopril-d7 sodium salt
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Fosinopril-d7 is intended for use as an internal standard for the quantification of fosinopril by GC- or LC-MS. Fosinopril is a prodrug form of the angiotensin-converting enzyme inhibitor fosinoprilat. Oral administration of fosinopril inhibits angiotensin I-induced pressor responses in normotensive rats, dogs, and monkeys when administered at doses of 15, 15, and 10 µmol/kg, respectively. Fosinopril reduces fractional shortening and decreases left ventricular size in a porcine model of congesti... | |||
T71211 |
Rizatriptan-d6 benzoate salt
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Rizatriptan-d6 is intended for use as an internal standard for the quantification of rizatriptan by GC- or LC-MS. Rizatriptan is an agonist of the serotonin receptor subtypes 5-HT1B and 5-HT1D. It is selective for 5-HT1B and 5-HT1D receptors over 5-HT1A receptors. Rizatriptan induces vasoconstriction in isolated human middle meningeal arteries. In vivo, rizatriptan reduces head grooming, the number of oculotemporal strokes, eye blinking, and one-eye closures in a Cacna1a mutant transgenic mou... | |||
T11193 |
Enalaprilat-d5 sodium
MK-422 D5 Sodium Salt,依那普利拉钠 D5,Enalaprilat D5 Sodium Salt |
Others | Others |
Enalaprilat D5 Sodium Salt is the deuterium labeled Enalaprilat, which is an angiotensin-converting enzyme (ACE) inhibitor. | |||
T70313 |
Indoxyl Sulfate-d5 potassium salt
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Indoxyl sulfate-d5 is intended for use as an internal standard for the quantification of indoxyl sulfate by GC- or LC-MS. Indoxyl sulfate is a uremic toxin and a metabolite of tryptophan. It is formed via sulfation of indole, an intermediate generated from tryptophan by intestinal bacteria, by the sulfotransferase (SULT) isoform 1A1 variant 2 (SULT1A1*2) in the liver. Indoxyl sulfate activates the aryl hydrocarbon receptor (AhR) in HepG2 40/6 hepatoma cells (EC50 = 12.1 nM in a reporter assay). ... | |||
TMIH-0552 |
Tauroursodeoxycholic Acid-d4 Sodium Salt
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Tauroursodeoxycholic Acid-d4 Sodium Salt 是 Tauroursodeoxycholic Acid Sodium Salt 的氘代化合物。Tauroursodeoxycholic Acid Sodium Salt 的 CAS 号为 14605-22-2。Tauroursodeoxycholate,又称 ursodoxicoltaurine,是一种高度亲水性的三级胆汁酸,在人体内以低浓度产生。Tauroursodeoxycholate 是 ursodeoxycholic acid 更亲水的形式,而 ursodeoxycholic acid 是人类体内自然产生的更丰富的胆汁酸。Tauroursodeoxycholate 正在研究用于几种疾病,如原发性胆汁性肝硬化(PBC)、胰岛素抵抗、淀粉样变性、囊性纤维化、胆汁淤滞和肌萎缩性侧索硬化症。 | |||
TMIH-0473 |
rac Metanephrine-d3 Hydrochloride Salt
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rac Metanephrine-d3 Hydrochloride Salt 是 rac Metanephrine Hydrochloride Salt 的氘代化合物。 | |||
TMIJ-0151 |
Atorvastatin-d5 Calcium Salt
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Atorvastatin-d5 Calcium Salt 是 Atorvastatin Calcium Salt 的氘代化合物。Atorvastatin Calcium Salt 的 CAS 号为 134523-00-5。 | |||
TMIH-0010 |
(S)-Alogliptin Benzoate Salt-13C-d3
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(S)-Alogliptin Benzoate Salt-13C-d3 是 (S)-Alogliptin Benzoate Salt 的 13C 和氘代化合物。 | |||
TMIJ-0164 |
Rosuvastatin-d6 Sodium Salt
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Rosuvastatin-d6 Sodium Salt 是 Rosuvastatin Sodium Salt 的氘代化合物。Rosuvastatin Sodium Salt 的 CAS 号为 1007871-86-4。 | |||
TMID-0273 |
Promethazine-d6 Hydrochloride Salt
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Promethazine-d6 Hydrochloride Salt 是 Promethazine Hydrochloride Salt 的氘代化合物。Promethazine Hydrochloride Salt 的 CAS 号为 1173018-74-0。 | |||
TMID-0269 |
Nafcillin-d5 Sodium Salt
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Nafcillin-d5 Sodium Salt 是 Nafcillin Sodium Salt 的氘代化合物。Nafcillin Sodium Salt 的 CAS 号为 985-16-0。 | |||
TMIJ-0182 |
Avibactam sodium salt-13C5
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Avibactam sodium salt-13C5 是 Avibactam sodium salt 的 13C 的标记化合物。Avibactam sodium salt 的 CAS 号为 1192491-61-4。Avibactam sodium 是一种可逆的 β-内酰胺酶抑制剂,抑制 TEM-1,P99和KPC-2 β-内酰胺酶,IC50分别为8、80和38 nM。 | |||
TMIJ-0119 |
Pitavastatin-d4 Sodium Salt
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Pitavastatin-d4 Sodium Salt 是 Pitavastatin Sodium Salt 的氘代化合物。Pitavastatin Sodium Salt 的 CAS 号为 574705-92-3。 | |||
TMIJ-0171 |
Ceftazidime sodium salt-d6
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Ceftazidime sodium salt-d6 是 Ceftazidime sodium salt 的氘代化合物。Ceftazidime sodium salt 的 CAS 号为 73547-61-2。 | |||
TMIJ-0301 |
Esomeprazole-d3 Sodium Salt
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Esomeprazole-d3 Sodium Salt 是 Esomeprazole Sodium Salt 的氘代化合物。 | |||
TMIJ-0179 |
Faropenem-d7 Sodium Salt
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Faropenem-d7 Sodium Salt 是 Faropenem Sodium Salt 的氘代化合物。Faropenem Sodium Salt 的 CAS 号为 122547-49-3。Faropenem sodium 是一种口服生物可利用的青霉烯类抗生素,能有效杀灭结核分枝杆菌,治疗结核病和社区获得性肺炎。 | |||
TMID-0234 |
Penicillin G-d5 potassium salt
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Penicillin G-d5 potassium salt 是 Penicillin G potassium salt 的氘代化合物。Penicillin G potassium salt 的 CAS 号为 113-98-4。Benzylpenicillin potassium是青霉素家族的一种速效抗生素。 | |||
TMIJ-0319 |
Dehydroepiandrosterone Sulfate Sodium Salt-d6
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Dehydroepiandrosterone Sulfate Sodium Salt-d6 是 Dehydroepiandrosterone Sulfate Sodium Salt 的氘代化合物。Dehydroepiandrosterone Sulfate Sodium Salt 的 CAS 号为 1099-87-2。 | |||
TMID-0294 |
Taurodeoxycholic Acid-d4 Sodium Salt
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Taurodeoxycholic Acid-d4 Sodium Salt 是 Taurodeoxycholic Acid Sodium Salt 的氘代化合物。Taurodeoxycholic Acid Sodium Salt 的 CAS 号为 1180-95-6。Taurodeoxycholate sodium salt 是胆盐相关的阴离子洗涤剂,用于分离膜蛋白,包括线粒体内膜蛋白。它还可以抑制各种炎症反应。 | |||
TMIJ-0198 |
Taurochenodeoxycholic Acid-d5 Sodium Salt
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Taurochenodeoxycholic Acid-d5 Sodium Salt 是 Taurochenodeoxycholic Acid Sodium Salt 的氘代化合物。Taurochenodeoxycholic Acid Sodium Salt 的 CAS 号为 6009-98-9。Taurochenodeoxycholic acid sodium 是动物胆汁酸的主要生物活性物质之一。它可诱导细胞凋亡,具有抗炎和免疫调节作用。 | |||
TMIH-0434 |
PHPB-d7
(R/S)-2-(1-hydroxy-n-pentyl)benzoic acid potassium salt-d7 |
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PHPB-d7 是 PHPB 的氘代化合物。 | |||
TMIJ-0150 |
para-Hydroxy Atorvastatin-d5 Calcium Salt
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para-Hydroxy Atorvastatin-d5 Calcium Salt 是 para-Hydroxy Atorvastatin Calcium Salt 的氘代化合物。para-Hydroxy Atorvastatin Calcium Salt 的 CAS 号为 214217-88-6。 | |||
TMIJ-0152 |
ortho-Hydroxy Atorvastatin-d5 Calcium Salt
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ortho-Hydroxy Atorvastatin-d5 Calcium Salt 是 ortho-Hydroxy Atorvastatin Calcium Salt 的氘代化合物。ortho-Hydroxy Atorvastatin Calcium Salt 的 CAS 号为 265989-47-7。 | |||
TMIJ-0256 |
Estrone-d4 3-Sulfate Sodium Salt
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Estrone-d4 3-Sulfate Sodium Salt 是 Estrone 3-Sulfate Sodium Salt 的氘代化合物。Estrone 3-Sulfate Sodium Salt 的 CAS 号为 438-67-5。 | |||
TMIJ-0332 |
Taurolithocholic Acid-d5 Sodium Salt (Major)
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Taurolithocholic Acid-d5 Sodium Salt (Major) 是 Taurolithocholic Acid Sodium Salt 的氘代化合物。Taurolithocholic Acid Sodium Salt 的 CAS 号为 6042-32-6。Taurolithocholic acid sodium salt 是抑胆剂和Ca2+激动剂,可抑制放射性配体与毒蕈碱 M1 结合。 | |||
TMIJ-0167 |
Simvastatin EP Impurity A-d6 Sodium Salt
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Simvastatin EP Impurity A-d6 Sodium Salt 是 Simvastatin EP Impurity A Sodium Salt 的氘代化合物。Simvastatin EP Impurity A Sodium Salt 的 CAS 号为 101314-97-0。 | |||
TMID-0175 |
DL-α-Hydroxyglutaric acid disodium salt-d4
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DL-α-Hydroxyglutaric acid disodium salt-d4 是 DL-α-Hydroxyglutaric acid disodium salt 的氘代化合物。DL-α-Hydroxyglutaric acid disodium salt 的 CAS 号为 40951-21-1。DL-α-Hydroxyglutaric acid disodium salt 是一种 α-羟基酸,由 (R) -5-oxy-2-tetrahydrofuran 羧酸水解形成,在人类神经代谢疾病 D-α-羟基戊二酸尿症中过量产生。DL-α-Hydroxyglutaric acid disodium salt 是α-酮戊二酸 (α-KG)的拮抗剂,可抑制多种α-KG 依赖性双加氧酶。 | |||
TMIJ-0219 |
Cefpodoxime Proxetil EP Impurity A-d3 Sodium Salt
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Cefpodoxime Proxetil EP Impurity A-d3 Sodium Salt 是 Cefpodoxime Proxetil EP Impurity A Sodium Salt 的氘代化合物。 | |||
T71402 |
Nicorandil-d4
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Nicorandil-d4 is intended for use as an internal standard for the quantification of nicorandil by GC- or LC-MS. Nicorandil is an activator of sulfonylurea receptor 2B (SUR2B) linked to ATP-sensitive potassium channel Kir6.2 (EC50 = ~10 µM) and a nitric oxide (NO) donor. It is selective for SUR2B/Kir6.2 over the SUR2A/Kir6.2 channel (EC50 = >500 µM). Nicorandil activates soluble guanylate cyclase in a cell-free assay and relaxes partially depolarized isolated bovine coronary artery strips (EC50 =... | |||
T19447 |
N-Demethyl Ivabradine D6 Hydrochloride
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Others | Others |
N-Demethyl Ivabradine D6 Hydrochloride salt is the deuterium labeled N-Demethyl Ivabradine, which is a Ivabradine metabolite. | |||
T70990 |
ADMA-d6
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NG,NG-dimethyl-L-arginine-d6 (ADMA-d6) (hydrochloride) is intended for use as an internal standard for the quantification of NG,NG-dimethyl-L-arginine by GC- or LC-MS. ADMA is an endogenous inhibitor of nitric oxide synthase (NOS). It is formed from arginine by protein arginine methyltransferases (PRMTs) and degraded by dimethylarginine dimethylaminohydrolases (DDAHs) and alanine-glyoxylate aminotransferase 2 (AGXT2). ADMA levels are increased concomitant with an increase in blood pressure in Da... | |||
TMIJ-0037 |
Sarafloxacin-d8 Hydrochloride
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Sarafloxacin-d8 Hydrochloride 是 Sarafloxacin Hydrochloride 的氘代化合物。Sarafloxacin Hydrochloride 的 CAS 号为 91296-87-6。Sarafloxacin hydrochloride是一种抗菌化合物。 | |||
T69600 |
Spermidine-d6
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Spermidine-d6 is intended for use as an internal standard for the quantification of spermidine by GC- or LC-MS. Spermidine is an endogenous polyamine. It is formed from putrescine by spermidine synthase. Spermidine (25 µM) inhibits the activity of the human inward-rectifying potassium channel Kir2.3 in a patch-clamp assay. It induces autophagy in HeLa cells when used at a concentration of 100 µM and increases the lifespan of D. melanogaster, yeast, and C. elegans. Spermidine (30 mM in the drinki... | |||
TMIJ-0014 |
Fenoterol-d6 Hydrobromide
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Fenoterol-d6 Hydrobromide 是 Fenoterol Hydrobromide 的氘代化合物。Fenoterol Hydrobromide 的 CAS 号为 1944-12-3。Fenoterol hydrobromide 是一种拟交感神经剂,是一种选择性的,具有口服活性 β2-肾上腺素受体 (β2-adrenoceptor) 激动剂,是一种有效的支气管扩张剂,可用于一种与哮喘、支气管炎和其他阻塞性气道疾病相关的支气管痉挛。 | |||
TMIJ-0377 |
Thiamine Hydrochloride-13C4
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Thiamine Hydrochloride-13C4 是 Thiamine Hydrochloride 的 13C 的标记化合物。Thiamine Hydrochloride 的 CAS 号为 67-03-8。Thiamine hydrochloride 是一种必需的微量营养素,是许多中枢代谢酶的辅因子。 | |||
TMID-0187 |
Amitriptyline-d6 Hydrochloride
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Amitriptyline-d6 Hydrochloride 是 Amitriptyline Hydrochloride 的氘代化合物。Amitriptyline Hydrochloride 的 CAS 号为 549-18-8。Amitriptyline hydrochloride 是血清素再摄取转运体和去甲肾上腺素再摄取转运体抑制剂,还与多巴胺再摄取转运体结合,其Ki为 2.58 μM。它也抑制肾上腺素能受体、毒蕈碱受体、组胺受体、5-羟色胺受体。它是TrkA和TrkA受体的激动剂,具有强神经营养活性和有抗抑郁作用。 | |||
TMID-0258 |
(±)-Atropine-d3 (N-methyl-d3)
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(±)-Atropine-d3 (N-methyl-d3) 是 (±)-Atropine 的氘代化合物。(±)-Atropine 的 CAS 号为 51-55-8。Atropine 是竞争性的毒蕈碱乙酰胆碱受体拮抗剂,有抗近视效果。它是一种从颠茄植物中分离出来的天然生物碱,可阻断乙酰胆碱对心率和收缩力的抑制作用。 | |||
TMIJ-0519 |
Fosaprepitant-d4 Dimeglumine
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Fosaprepitant-d4 Dimeglumine 是 Fosaprepitant Dimeglumine 的氘代化合物。Fosaprepitant Dimeglumine 的 CAS 号为 265121-04-8。Fosaprepitant dimeglumine 是 Aprepitant 的前药。它是一种神经激肽 1 受体拮抗剂,可用于预防化疗引起的恶心呕吐。 | |||
TMIH-0124 |
Brivanib Alaninate-d4
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Brivanib Alaninate-d4 是 Brivanib Alaninate 的氘代化合物。Brivanib Alaninate 的 CAS 号为 649735-63-7。Brivanib alaninate 是一种血管内皮生长因子受体 2 (VEGFR2) 抑制剂的丙氨酸盐,IC50值为 25 nM,具有潜在的抗肿瘤活性。它对 VEGFR1 和 FGFR1 适度抑制,对 VEGFR2 的选择性是对 PDGFRβ 的 240 倍。 | |||
TMIH-0184 |
Desipramine-d3 HCl
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Desipramine-d3 HCl 是 Desipramine HCl 的氘代化合物。Desipramine HCl 的 CAS 号为 58-28-6。Desipramine hydrochloride 是一种二苯并氮杂类衍生物三环类抗抑郁药,可作为选择性去甲肾上腺素再摄取抑制剂。 它还显示出较弱的 5-羟色胺再摄取抑制、α1 阻断、抗组胺和抗胆碱能作用。 | |||
TMIH-0512 |
Salbutamol-d3
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Salbutamol-d3 是 Salbutamol 的氘代化合物。Salbutamol 的 CAS 号为 18559-94-9。Salbutamol 是短效的 β2 肾上腺素受体激动剂,用于哮喘和慢性阻塞性肺疾病 (COPD) 引发的支气管痉挛的研究。 | |||
TMID-0078 |
Irinotecan-d10 Hydrochloride
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Irinotecan-d10 Hydrochloride 是 Irinotecan Hydrochloride 的氘代化合物。Irinotecan Hydrochloride 的 CAS 号为 100286-90-6。Irinotecan Hydrochloride 是喜树碱半合成衍生物的盐酸盐,是一种拓扑异构酶 I 抑制剂,可研究结肠癌和直肠癌。 | |||
TMID-0233 |
Salbutamol-d9
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Salbutamol-d9 是 Salbutamol 的氘代化合物。Salbutamol 的 CAS 号为 18559-94-9。Salbutamol 是短效的 β2 肾上腺素受体激动剂,用于哮喘和慢性阻塞性肺疾病 (COPD) 引发的支气管痉挛的研究。 |