ARL67156 trisodium salt

Name: ARL67156 trisodium salt
Brand: TargetMol
SKU: T14320
Price: 410 USD
Availability: InStock
Rating: 4.5 (1 reviews)

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产品编号 T14320Cas号 1021868-83-6

ARL 67156 is a weak competitive inhibitor of NTPDase1 (CD39), NTPDase3 and NPP1, with Kis of 11, 18 and 12 μM, respectively[1]. ARL67156 trisodium salt is an inhibitor of ecto-ATPase.

ARL67156 trisodium salt

还可以

产品编号 T14320Cas号 1021868-83-6

ARL 67156 is a weak competitive inhibitor of NTPDase1 (CD39), NTPDase3 and NPP1, with Kis of 11, 18 and 12 μM, respectively[1]. ARL67156 trisodium salt is an inhibitor of ecto-ATPase.

规格	价格	库存	数量
10 mg	¥ 5,280	35日内发货

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产品介绍

生物活性

产品描述	ARL 67156 is a weak competitive inhibitor of NTPDase1 (CD39), NTPDase3 and NPP1, with Kis of 11, 18 and 12 μM, respectively[1]. ARL67156 trisodium salt is an inhibitor of ecto-ATPase.
靶点活性	NTPDase3:18 μM(ki), NPP1:12 μM(ki), NTPDase1:（ki）11 μM
体外活性	ARL67156 is not an effective inhibitor of NTPDase2, NTPDase8, NPP3 and ecto-5′-nucleotidase (CD73). And It also reduces the activity of these enzymes[1]. ARL67156 trisodium salt is also an effective inhibitor of UTP breakdown by superior cervical ganglion cells and to potentiate contractions elicited by this nucleotide in isolated tail artery of rat.

化学信息

分子量	785.05
分子式	C₁₅H₂₁Br₂N₅Na₃O₁₂P₃
CAS No.	1021868-83-6
密度	no data available

储存&溶解度

存储

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.

溶解度信息

H2O: 25 mg/mL (31.72 mM), Sonication is recommended.

溶液配制表

H2O

	1mg	5mg	10mg	50mg
1 mM	1.2738 mL	6.3690 mL	12.7380 mL	63.6902 mL
5 mM	0.2548 mL	1.2738 mL	2.5476 mL	12.7380 mL
10 mM	0.1274 mL	0.6369 mL	1.2738 mL	6.3690 mL
20 mM	0.0637 mL	0.3185 mL	0.6369 mL	3.1845 mL