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Targets Recommended: Amino Acids and Derivatives Aminopeptidase Others PROTAC Linker

2998

抑制剂 & 化合物

271

天然产物

12

化合物库

407

重组蛋白

43

同位素标记化合物

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Cat. No. Product Name
L2550 谷氨酰胺代谢化合物库

565 compounds
565 种谷氨酰胺代谢相关的分子,可以用于高通量和高内涵筛选;
L2400 内分泌激素分子库

784 compounds
784 种与内分泌系统相关的生物活性小分子化合物的特有集合,用于高通量、高内涵筛选;
L9610 环肽库

80 compounds
80 种环肽分子,可用于高通量和高内涵筛选;
L1600 激酶抑制剂库

2720 compounds
2720 种激酶抑制剂/调节剂的独特集合,用于特定靶向激酶,可用于高通量筛选和高内涵筛选;
L2800 5-羟色胺分子库

268 compounds
268 种生物活性小分子化合物,用于高通量、高内涵筛选;
L2130 抗癌细胞代谢库

1268 compounds
1268 种癌细胞代谢相关的生物活性小分子化合物的特有集合,用于肿瘤相关的研究以及抗肿瘤药物的筛选,用于高通量、高内涵筛选;
L2501 人内源代谢化合物库 Plus

1283 compounds
1283种内源性生物活性化合物的独特集合,用于高通量、高内涵筛选。
L3300 组胺&褪黑色素化合物库

153 compounds
153 种生物活性小分子化合物,用于高通量、高内涵筛选;
L9600 多肽分子库

791 compounds
791 种多肽类分子,可用于多肽药物开发及信号转导通路和作用机制研究;
L2570 人代谢物化合物库

4454 compounds
4454 种人代谢物的独特集合,用于高通量、高内涵筛选;
L7600 趋化因子抑制剂库

59 compounds
59 种趋化因子或其受体抑制剂的独特集合,可用于高通量筛选和高内涵筛选;
DO2200 共价抑制剂库CD

12000 compounds
数量多:超过12000种共价结合化合物,并且数量在持续增加;

化合物库

谷氨酰胺代谢化合物库
Cat.No: L2550
Compounds: 565
内分泌激素分子库
Cat.No: L2400
Compounds: 784
环肽库
Cat.No: L9610
Compounds: 80
激酶抑制剂库
Cat.No: L1600
Compounds: 2720
5-羟色胺分子库
Cat.No: L2800
Compounds: 268
抗癌细胞代谢库
Cat.No: L2130
Compounds: 1268
人内源代谢化合物库 Plus
Cat.No: L2501
Compounds: 1283
组胺&褪黑色素化合物库
Cat.No: L3300
Compounds: 153
多肽分子库
Cat.No: L9600
Compounds: 791
人代谢物化合物库
Cat.No: L2570
Compounds: 4454
趋化因子抑制剂库
Cat.No: L7600
Compounds: 59
共价抑制剂库CD
Cat.No: DO2200
Compounds: 12000
Cat. No. Product Name Target Signaling Pathways
T17548 Biotin-C5-amino-C5-amino

Others; PROTAC Linker Others; PROTAC
Biotin-C5-amino-C5-amino 是一种属于 alkyl chain 类的 PROTAC linker,可用于 PROTAC 分子的合成。
T21017 5'-Amino-5'-deoxyadenosine

5' Amino 5' deoxyadenosine,5'Amino5'deoxyadenosine,Nsc 238990,NH2dAdo

Apoptosis; Adenosine Receptor Apoptosis; GPCR/G Protein; Neuroscience
5'-Amino-5'-deoxyadenosine (NH2dAdo) 是一种针对惰性淋巴系统恶性肿瘤的腺苷激酶抑制剂,具有抗肿瘤和抗癌作用。5'-Amino-5'-deoxyadenosine 的抗癌机制通过抑制 DNA 合成,诱导细胞凋亡 (apoptosis) 等来实现。
T17405 Amino-PEG12-acid

Others; PROTAC Linker Others; PROTAC
Amino-PEG12-acid 是一种属于 PEG 类的 PROTAC linker,可用于 PROTAC 分子的合成。
T17402 Amino-PEG10-acid

Others; PROTAC Linker Others; PROTAC
Amino-PEG10-acid 是一种属于 PEG 类的 PROTAC linker,可用于 PROTAC 分子的合成。
T17408 Amino-PEG12-Boc

Others; PROTAC Linker Others; PROTAC
Amino-PEG12-Boc 是一种属于 PEG 类的 PROTAC linker,可用于 PROTAC 分子的合成。
T17406 Amino-PEG12-alcohol

Others; PROTAC Linker Others; PROTAC
Amino-PEG12-alcohol 是一种属于 PEG 类的 PROTAC linker,可用于 PROTAC 分子的合成。
T17411 Amino-PEG13-amine

H2N-PEG13-CH2CH2NH2

Others; PROTAC Linker Others; PROTAC
Amino-PEG13-amine (H2N-PEG13-CH2CH2NH2) 是一种属于 PEG 类的 PROTAC linker,可用于 PROTAC 分子的合成。
T14250 Amino-PEG8-amine

Others Others
Amino-PEG8-amine 是一种以聚乙二醇为基础的 PROTAC 连接剂,可用于PROTACs 的合成,是一种含有两个氨基(NH2)基团的共轭PEG 衍生物。
T9323 4-Amino-6-(trifluoromethyl)benzene-1,3-disulfonamide

4-氨基-6-(三氟甲基)苯-1,3-二磺酰胺,4-Amino-6-(trifluoromethyl)benzene-1,3-d,2,4-Disulfamyl-5-trifluoromethylaniline,2-amino-4-trifluoromethyl-1,5-benzendisulfonamide

Carbonic Anhydrase Metabolism
4-Amino-6-(trifluoromethyl)benzene-1,3-disulfonamide (4-Amino-6-(trifluoromethyl)benzene-1,3-d) 是一种碳酸酐酶抑制剂,用作潜在的抗肿瘤和抗青光眼药物。
T17441 Amino-PEG9-alcohol

胺基-九聚乙二醇

Others; PROTAC Linker Others; PROTAC
Amino-PEG9-alcohol 是一种基于 PEG 的 PROTAC 接头,可用于 PROTAC 的合成。
T7542 Amino Tadalafil

氨基他达那非,氨基他达拉非

PDE Metabolism
Amino Tadalafil 是一种 Tadalafil 的类似物,是一种磷酸二酯酶 5 抑制剂,可用于多种疾病,如勃起功能障碍,肺动脉高压和下尿路功能障碍。
T17440 Amino-PEG7-acid

氨基-七聚乙二醇-羧酸

Others; PROTAC Linker Others; PROTAC
Amino-PEG7-acid 是一种属于 PEG 类的 PROTAC linker,可用于 PROTAC 分子的合成。
T1370 2-Amino-5-Fluorophenol

Others Others
2-Amino-5-Fluorophenol(2-AF)用于合成各种药物和化合物,包括抗癌药、抗炎药和其他药物,以及抗微生物、抗真菌和抗病毒的化合物。
T9344 3-Amino-2-oxazolidinone

Others; Endogenous Metabolite Metabolism; Others
3-Amino-2-oxazolidinone 是一种呋喃唑烷酮的代谢物 (metabolite),可用作检测呋喃唑烷酮残留的一个指标。
T14226 Amino-PEG11-amine

氨基-十二聚乙二醇-氨基

Others; PROTAC Linker Others; PROTAC
Amino-PEG11-amine 是一种基于 PEG(12 个单位)的 PROTAC 接头,能够结合两种基于单乙基雌酚的配体,是制备用于乳腺癌内分泌治疗的更具选择性和活性的 ER 拮抗剂的替代策略。
T0644 3-Amino-5-methylisoxazole

Others Others
3-Amino-5-methylisoxazole 是医药中间体,用于生产磺胺类药物。
T1722 5-Amino-4-imidazolecarboxamide

Others Others
5-Amino-4-imidazolecarboxamide 是一种咪唑衍生物。
T1685 2-Amino-5-chlorobenzophenone

Others Others
2-Amino-5-chlorobenzophenone 用作医药中间体。
T9441 2-Amino-p-cresol

Others Others
2-Amino-p-cresol 是合成多种化合物的中间体,包括药物、染料等;还被用作合成各种聚合物的试剂和酶的抑制剂。
T7234 5-Amino-2-chloropyridine

Others Others
5-Amino-2-chloropyridine 是吡啶中间体。
T0526 2-Amino-5-nitrobenzophenone

Others Others
2-Amino-5-nitrobenzophenone 用作工业和有机中间体。
T8826 3-AMINO-1,2,4-TRIAZINE

Others Others
3-AMINO-1,2,4-TRIAZINE 是一种芳香族生物活性化合物,已用于合成各种药物,包括抗真菌药物氟康唑、抗炎药物布洛芬和抗癌药物紫杉醇;也被用于设计新药,如抗艾滋病药物齐多夫定和抗疟疾药物青蒿素;以及用于合成各种其他化合物,如抗糖尿病药物二甲双胍和抗高血压药物赖诺普利。
T14238 Amino-PEG4-Boc

15-氨基-4,7,10,13-四氧杂十五烷酸叔丁酯

PROTAC Linker PROTAC
Amino-PEG4-Boc 是一种属于 PEG 类的 PROTAC linker,可用于 PROTAC 分子的合成。
T17413 Amino-PEG14-alcohol

氨基十四聚乙二醇羟基,H2N-PEG14-OH

Others; PROTAC Linker Others; PROTAC
Amino-PEG14-alcohol (H2N-PEG14-OH) 是一种属于 PEG 类的 PROTAC linker,可用于 PROTAC 分子的合成。
TQ0018 6-Amino-5-azacytidine

Antibacterial Microbiology/Virology
6-Amino-5-azacytidine 对大肠杆菌的生长有抑制作用。
T21524 4-amino-1,8-Naphthalimide

PARP Chromatin/Epigenetic; DNA Damage/DNA Repair
4-amino-1,8-Naphthalimide 是PARP 抑制剂,可增强癌细胞对 γ 辐射诱导的细胞毒性的敏感度。
T17407 Amino-PEG12-amine

H2N-PEG12-CH2CH2NH2,PEODA13,氨基十三聚乙二醇氨基

Others; PROTAC Linker Others; PROTAC
Amino-PEG12-amine (H2N-PEG12-CH2CH2NH2) 是一种属于 PEG 类的 PROTAC linker,可用于 PROTAC 分子的合成。
T9234 Tocainide hydrochloride

2-amino-n-(2,6-dimethylphenyl)propanamide hydrochloride

Sodium Channel Membrane transporter/Ion channel
Tocainide hydrochloride (2-amino-n-(2,6-dimethylphenyl)propanamide hydrochloride) 是利多卡因的伯胺类似物,是钠通道阻滞剂,在产生疼痛的病灶中(神经膜上) 阻断钠通道。Tocainide hydrochloride 具有用于心律不齐研究的价值。
T0567 2-Amino-5-chlorobenzoic acid

Others; Amino Acids and Derivatives Metabolism; Others
2-Amino-5-chlorobenzoic acid 是杀虫剂 Chlordimeform 的代谢物。可用于制备缓解疾病的抗风湿药(DMARDs)。
T1376 2-Amino-5-methyl-3-thiophenecarbonitrile

COX Immunology/Inflammation; Neuroscience
2-Amino-5-methyl-3-thiophenecarbonitrile 常用于合成 Olanzapine。
T50016 2-amino-4-methyl-1,3-thiazole-5-carbohydrazide

Others Others
2-amino-4-methyl-1,3-thiazole-5-carbohydrazide (AMTCH)具有抗肿瘤活性,通过诱导细胞凋亡或细胞程序性死亡抑制癌细胞的生长,也具有抗细菌和真菌活性。
T9462 2-Amino-6-cyclopropylamino-9H-purine

Others Others
2-Amino-6-cyclopropylamino-9H-purine 是阿巴卡韦(abacavir) 的关键中间体,以氰基乙酸乙酯为原料,经亚硝化、盐酸胍在 EtONa 存在下环合、还原得到2,4,5-三氨基-6-羟基嘧啶
T9085 JFD01307SC

[(1,1-DIOXIDOTETRAHYDROTHIEN-3-YL)AMINO]

Antibacterial Microbiology/Virology
JFD01307SC ([(1,1-DIOXIDOTETRAHYDROTHIEN-3-YL)AMINO]) 是一种谷氨酰胺合成酶抑制剂。 它是抗结核剂,可作为 L-谷氨酸盐的模拟物,靶向参与谷氨酰胺生物合成的酶。
T85257 (S)-3'-amino Blebbistatin

meta-amino Blebbistatin,(−)-3'-amino Blebbistatin,m-amino Blebbistatin

Others Others
"(S)-3'-amino Blebbistatin, retaining the active stereochemistry of the less stable and more phototoxic (–)-blebbistatin, serves as a refined selective cell-permeable inhibitor of non-muscle myosin II ATPases. This compound efficaciously inhibits the Mg-ATPase activity and in vitro motility of non-muscle myosin IIA and IIB across several species with IC50s ranging from 0.5-5 µM, and exhibits minimal inhibition against smooth muscle myosin (IC50= 80 µM). Its primary functions include obstructing ...
T7401 (S)-3-AMino-2-Methylpropanoic acid-HCl

Others Others
(S)-3-AMino-2-Methylpropanoic acid-HCl 是一种氨基酸衍生物,是兴奋性神经递质谷氨酸的激动剂,影响神经系统。
T8760 NNMTi

5-Amino-1-methylquinolinium

Others Others
NNMTi (5-Amino-1-methylquinolinium) 是烟酰胺 N -甲基转移酶的抑制剂 (IC50=1.2 μM),可选择性地结合 NNMT 底物结合位点残基。它能诱导体外成肌细胞分化,提高老年小鼠肌肉干细胞融合和再生能力。
T8910 2-AMINO-5-PHENYL-THIOPHENE-3-CARBOXYLIC

IκB/IKK NF-κB
2-AMINO-5-PHENYL-THIOPHENE-3-CARBOXYLIC 是 IKKβ 的抑制剂。
T5445 2-Amino-4-hydroxypyrrolo[2,3- d]pyrimidi

Others Others
2-Amino-4-hydroxypyrrolo[2,3- d]pyrimidi 用作中间体。
T9828 N-[1-(Aminocarbonyl)-4-[(2-chloro-1-iminoethyl)amino]butyl]benzamide

PAD Chromatin/Epigenetic
N-[1-(Aminocarbonyl)-4-[(2-chloro-1-iminoethyl)amino]butyl]benzamide 是Cl-amidine (S 构型)的消旋形式。Cl-amidine 口服有效的 PAD 抑制剂。
T9838 2-Amino-3-(2-chlorophenyl)propanoic acid

2-Chloro-DL-Phenylalanine

Amino Acids and Derivatives Metabolism
2-Amino-3-(2-chlorophenyl)propanoic acid (2-Chloro-DL-Phenylalanine) 是一种苯丙氨酸衍生物,参与生物代谢。
T9287 Hydroxychloroquine

2-[[4-[(7-Chloroquinolin-4-yl)amino]pentyl](ethyl)amino]ethanol,羟氯喹

SARS-CoV; TLR; Parasite; Autophagy Autophagy; Immunology/Inflammation; Microbiology/Virology
Hydroxychloroquine (2-[[4-[(7-Chloroquinolin-4-yl)amino]pentyl](ethyl)amino]ethanol) 是一种合成抗疟疾剂,有效抑制SARS-CoV-2感染,也抑制 Toll 样受体 7/9 信号传导。
T9042 Teriflunomide impurity 3

4-Amino-N-(4-trifluoromethylphenyl)benzamide

COX Immunology/Inflammation; Neuroscience
Teriflunomide impurity 3 (4-Amino-N-(4-trifluoromethylphenyl)benzamide) 是一种选择性COX-1抑制剂,IC50为 30 µM。
T40974 Amino-PEG4-C1-Boc

Amino-PEG4-C1-Boc

Others Others
Amino-PEG4-C1-Boc is a PEG-based linker for PROTACs which joins two essential ligands, crucial for forming PROTAC molecules. This linker enables selective protein degradation by leveraging the ubiquitin-proteasome system within cells.
T67967 EOB-DTPA

N-((2s)-2-(bis(carboxymethyl)amino)-3-(4-ethoxyphenyl)propyl)-n-(2-(bis(carboxymethyl)amino)ethyl)glycine

Others Others
EOB-DTPA 是一种生化试剂,可由其他化合物合成,常用于核磁共振成像。
T32039 HADA Hydrochloride

HCC-Amino-D-alanine hydrochloride,HADA HCl

Autophagy Autophagy
HADA Hydrochloride (HCC-Amino-D-alanine hydrochloride) 是一种具有蓝色荧光的D 氨基酸 (λem~450 nm)。FDAAs 在肽聚糖 (PG) 合成位点有效地与多种细菌的 PGs 结合。HADA Hydrochloride 而用于在最小干扰下特异性和共价探测细菌的生长。
T40084 Pomalidomide-amino-PEG5-NH2

Pomalidomide-amino-PEG5-NH2

Others Others
Pomalidomide-amino-PEG5-NH2 is a synthesized conjugate combining the Pomalidomide-based cereblon ligand and a linker utilized in PROTAC technology. It acts as an E3 ligase ligand-linker conjugate.
T39866 Pomalidomide-amino-PEG4-NH2

Pomalidomide-amino-PEG4-NH2

Others Others
Pomalidomide-amino-PEG4-NH2 is a conjugate compound that combines the Pomalidomide-based cereblon ligand and a linker, effectively functioning as a synthesized E3 ligase ligand-linker conjugate utilized in PROTAC technology.
T39952 Pomalidomide-amino-PEG3-NH2

Pomalidomide-amino-PEG3-NH2

Others Others
Pomalidomide-amino-PEG3-NH2 is a compound obtained through synthesis, consisting of a conjugation between the E3 ligase ligand linker and Pomalidomide, a cereblon ligand. This compound is specifically designed for application in PROTAC technology, incorporating a linker that enables effective binding with the targeted proteins.
T9146 ms48107

Benzenemethanol, 2-[4-amino-6-[[(4-phenoxyphenyl)methyl]amino]-1,3,5-triazin-2-yl]-3-fluoro-

Others Others
MS48107 是 G 蛋白偶联受体 68 (GPR68) 的选择性正变构调节剂,对GPR68的选择性高于密切相关的神经递质转运蛋白,质子 GPCR 和 hERG 离子通道。它可以穿越过小鼠的血脑屏障。
T18983 DNP-X acid

6-((2,4-Dinitrophenyl)amino)hexanoic acid

Others Others
DNP-X acid (6-((2,4-Dinitrophenyl)amino)hexanoic acid) 是一种与 Trp 或 Tyr 配对的极好的胺反应性 FRET 淬灭剂,能够用于开发可被 anti-DNP 抗体识别的探针的胺反应性构建块。

化合物

Biotin-C5-amino-C5-amino
Cat.No: T17548
Synonym:
Target: Others, PROTAC Linker
5'-Amino-5'-deoxyadenosine
Cat.No: T21017
Synonym: 5' Amino 5' deoxyadenosine,5'Amino5'deoxyadenosine,Nsc 238990,NH2dAdo
Target: Apoptosis, Adenosine Receptor
Amino-PEG12-acid
Cat.No: T17405
Synonym:
Target: Others, PROTAC Linker
Amino-PEG10-acid
Cat.No: T17402
Synonym:
Target: Others, PROTAC Linker
Amino-PEG12-Boc
Cat.No: T17408
Synonym:
Target: Others, PROTAC Linker
Amino-PEG12-alcohol
Cat.No: T17406
Synonym:
Target: Others, PROTAC Linker
Amino-PEG13-amine
Cat.No: T17411
Synonym: H2N-PEG13-CH2CH2NH2
Target: Others, PROTAC Linker
Amino-PEG8-amine
Cat.No: T14250
Synonym:
Target: Others
4-Amino-6-(trifluoromethyl)benzene-1,3-disulfonamide
Cat.No: T9323
Synonym: 4-氨基-6-(三氟甲基)苯-1,3-二磺酰胺,4-Amino-6-(trifluoromethyl)benzene-1,3-d,2,4-Disulfamyl-5-trifluoromethylaniline,2-amino-4-trifluoromethyl-1,5-benzendisulfonamide
Target: Carbonic Anhydrase
Amino-PEG9-alcohol
Cat.No: T17441
Synonym: 胺基-九聚乙二醇
Target: Others, PROTAC Linker
Amino Tadalafil
Cat.No: T7542
Synonym: 氨基他达那非,氨基他达拉非
Target: PDE
Amino-PEG7-acid
Cat.No: T17440
Synonym: 氨基-七聚乙二醇-羧酸
Target: Others, PROTAC Linker
2-Amino-5-Fluorophenol
Cat.No: T1370
Synonym:
Target: Others
3-Amino-2-oxazolidinone
Cat.No: T9344
Synonym:
Target: Others, Endogenous Metabolite
Amino-PEG11-amine
Cat.No: T14226
Synonym: 氨基-十二聚乙二醇-氨基
Target: Others, PROTAC Linker
3-Amino-5-methylisoxazole
Cat.No: T0644
Synonym:
Target: Others
5-Amino-4-imidazolecarboxamide
Cat.No: T1722
Synonym:
Target: Others
2-Amino-5-chlorobenzophenone
Cat.No: T1685
Synonym:
Target: Others
2-Amino-p-cresol
Cat.No: T9441
Synonym:
Target: Others
5-Amino-2-chloropyridine
Cat.No: T7234
Synonym:
Target: Others
2-Amino-5-nitrobenzophenone
Cat.No: T0526
Synonym:
Target: Others
3-AMINO-1,2,4-TRIAZINE
Cat.No: T8826
Synonym:
Target: Others
Amino-PEG4-Boc
Cat.No: T14238
Synonym: 15-氨基-4,7,10,13-四氧杂十五烷酸叔丁酯
Target: PROTAC Linker
Amino-PEG14-alcohol
Cat.No: T17413
Synonym: 氨基十四聚乙二醇羟基,H2N-PEG14-OH
Target: Others, PROTAC Linker
6-Amino-5-azacytidine
Cat.No: TQ0018
Synonym:
Target: Antibacterial
4-amino-1,8-Naphthalimide
Cat.No: T21524
Synonym:
Target: PARP
Amino-PEG12-amine
Cat.No: T17407
Synonym: H2N-PEG12-CH2CH2NH2,PEODA13,氨基十三聚乙二醇氨基
Target: Others, PROTAC Linker
Tocainide hydrochloride
Cat.No: T9234
Synonym: 2-amino-n-(2,6-dimethylphenyl)propanamide hydrochloride
Target: Sodium Channel
2-Amino-5-chlorobenzoic acid
Cat.No: T0567
Synonym:
Target: Others, Amino Acids and Derivatives
2-Amino-5-methyl-3-thiophenecarbonitrile
Cat.No: T1376
Synonym:
Target: COX
2-amino-4-methyl-1,3-thiazole-5-carbohydrazide
Cat.No: T50016
Synonym:
Target: Others
2-Amino-6-cyclopropylamino-9H-purine
Cat.No: T9462
Synonym:
Target: Others
JFD01307SC
Cat.No: T9085
Synonym: [(1,1-DIOXIDOTETRAHYDROTHIEN-3-YL)AMINO]
Target: Antibacterial
(S)-3'-amino Blebbistatin
Cat.No: T85257
Synonym: meta-amino Blebbistatin,(−)-3'-amino Blebbistatin,m-amino Blebbistatin
Target: Others
(S)-3-AMino-2-Methylpropanoic acid-HCl
Cat.No: T7401
Synonym:
Target: Others
NNMTi
Cat.No: T8760
Synonym: 5-Amino-1-methylquinolinium
Target: Others
2-AMINO-5-PHENYL-THIOPHENE-3-CARBOXYLIC
Cat.No: T8910
Synonym:
Target: IκB/IKK
2-Amino-4-hydroxypyrrolo[2,3- d]pyrimidi
Cat.No: T5445
Synonym:
Target: Others
N-[1-(Aminocarbonyl)-4-[(2-chloro-1-iminoethyl)amino]butyl]benzamide
Cat.No: T9828
Synonym:
Target: PAD
2-Amino-3-(2-chlorophenyl)propanoic acid
Cat.No: T9838
Synonym: 2-Chloro-DL-Phenylalanine
Target: Amino Acids and Derivatives
Hydroxychloroquine
Cat.No: T9287
Synonym: 2-[[4-[(7-Chloroquinolin-4-yl)amino]pentyl](ethyl)amino]ethanol,羟氯喹
Target: SARS-CoV, TLR, Parasite, Autophagy
Teriflunomide impurity 3
Cat.No: T9042
Synonym: 4-Amino-N-(4-trifluoromethylphenyl)benzamide
Target: COX
Amino-PEG4-C1-Boc
Cat.No: T40974
Synonym: Amino-PEG4-C1-Boc
Target: Others
EOB-DTPA
Cat.No: T67967
Synonym: N-((2s)-2-(bis(carboxymethyl)amino)-3-(4-ethoxyphenyl)propyl)-n-(2-(bis(carboxymethyl)amino)ethyl)glycine
Target: Others
HADA Hydrochloride
Cat.No: T32039
Synonym: HCC-Amino-D-alanine hydrochloride,HADA HCl
Target: Autophagy
Pomalidomide-amino-PEG5-NH2
Cat.No: T40084
Synonym: Pomalidomide-amino-PEG5-NH2
Target: Others
Pomalidomide-amino-PEG4-NH2
Cat.No: T39866
Synonym: Pomalidomide-amino-PEG4-NH2
Target: Others
Pomalidomide-amino-PEG3-NH2
Cat.No: T39952
Synonym: Pomalidomide-amino-PEG3-NH2
Target: Others
ms48107
Cat.No: T9146
Synonym: Benzenemethanol, 2-[4-amino-6-[[(4-phenoxyphenyl)methyl]amino]-1,3,5-triazin-2-yl]-3-fluoro-
Target: Others
DNP-X acid
Cat.No: T18983
Synonym: 6-((2,4-Dinitrophenyl)amino)hexanoic acid
Target: Others
Cat. No. Product Name Target Signaling Pathways
TN7178 3-Amino-5-Hydroxybenzoic Acid

3-amino-5-hydroxy-benzoic acid,3-Amino-5-hydroxybenzoicAcid,3-氨基-5-羟基苯甲酸

Others Others
3-Amino-5-Hydroxybenzoic Acid (3-amino-5-hydroxy-benzoic acid) 是一种海洋来源的天然产物,存在于Salinispora arenicola。
T3S1957 9-amino-CPT

9-氨基喜树碱,Aminocamptothecin,9-amino-2(S)-camptothecin,9-Aminocamptothecin

Topoisomerase DNA Damage/DNA Repair
9-amino-CPT (Aminocamptothecin) 是一种拓扑异构酶I 的抑制剂,具有抗肿瘤活性。
T4770 3-Amino-4-hydroxybenzoic acid

3-氨基-4-羟基苯甲酸,3-amino-4-hydroxybenzenecarboxylic acid

Others; Endogenous Metabolite Metabolism; Others
3-Amino-4-hydroxybenzoic acid (3-amino-4-hydroxybenzenecarboxylic acid) 是内源性代谢产物的一种。
T1705 5-Amino-3H-imidazole-4-Carboxamide

4-Amino-5-imidazolecarboxamide,AICA,4-氨基-5-咪唑甲酰胺,5-Aminoimidazole-4-carboxamide

Endogenous Metabolite Metabolism
5-Amino-3H-imidazole-4-Carboxamide (AICA) 是一种合成嘌呤(尤其是核碱基腺嘌呤和鸟嘌呤)的重要前体。
TN1328 7-Amino-4-methylcoumarin-3-acetic acid

7-氨基-4-甲基-3-香豆素醋酸,7-Amino-4-methylcoumarin

Others Others
7-Amino-4-methylcoumarin-3-acetic acid (7-Amino-4-methylcoumarin) 是荧光蛋白质标记剂,能够被紫外光(350 nm) 激活,可在蓝色区域 (440-460 nm) 发光。
T7923 2-Amino-3-hydroxypyridine

Others Others
2-Amino-3-hydroxypyridine 作为显色试剂用于分光光度法测定锇。
T7937 2-Amino-4'-fluorobenzophenone

Others Others
2-Amino-4'-fluorobenzophenone 是一种苯甲酮的衍生物。它可用于合成对氟苯甲酰氯,还被用作生物化学研究的荧光探针,如 DNA 和 RNA 的检测。
T7918 2-Amino-2-dichlorobenzophenone

Others Others
2-Amino-2-dichlorobenzophenone 是一种芳香族天然化合物,已被用于研究各种化合物对细胞代谢、蛋白质合成和酶活性的影响,还被用于药物的合成,如抗肿瘤药物和抗炎药。
T4873 2-Amino-1-phenylethanol

Endogenous Metabolite Metabolism
2-Amino-1-phenylethanol 是去甲肾上腺素类似物。它已在人体睾丸组织中发现,并且主要在血液中检测到。
T13495 3-Amino-2-piperidinone

Cyclo-ornithine

Endogenous Metabolite Metabolism
3-Amino-2-piperidinone 是来自生物体的代谢物,可用作环状鸟氨酸类似物。
T7971 8-Amino-1-Naphthalenesulfonic Acid

Others Others
8-Amino-1-Naphthalenesulfonic Acid 是萘的衍生物,用作荧光染料和有机合成中的试剂。它是一种具有高Stokes 位移的高荧光化合物,使其成为广泛生物系统的理想荧光标记。
T2931 2-Amino-5-ureidopentanoic acid

DL-Citrulline,Citrulline,瓜氨酸

Others; Endogenous Metabolite Metabolism; Others
2-Amino-5-ureidopentanoic acid (Citrulline) 存在于肝脏中,不是蛋白质的构成成分,为人体脲循环的一个重要中间物,可与鸟氨酸、精氨酸合用治疗高氨血症。
TJS0341 7-Amino-4-(trifluoromethyl)coumarin

香豆素151,Coumarin 151,AFC,7-氨基-4-(三氟甲基)香豆素

5-HT Receptor GPCR/G Protein; Neuroscience
7-Amino-4-(trifluoromethyl)coumarin (Coumarin 151) 是一种荧光标记物,其激发和发射波长分别为400和500 nm,可用来灵敏的检测蛋白酶。
T4887 3-Amino-2-methylpropanoic acid

DL-3-AMINOISOBUTYRIC ACID,3-氨基异丁酸,α-Methyl-β-alanine

Endogenous Metabolite Metabolism
3-Amino-2-methylpropanoic acid (α-Methyl-β-alanine) 是 N-carbamyl-beta-aminoisobutyric acid 经 enzyme Beta-ureidopropionase (EC 3.5.1.6)转化后的产物,是嘧啶降解的最后一步。-尿嘧啶丙酸酶缺乏症是一种与神经异常相关的嘧啶降解的先天性错误。
T5569 3-Amino-4-methylpentanoic acid

DL-Homovaline,3-氨基-4-甲基戊酸,DL-beta-leucine,beta-Aminoisocaproic acid,beta-Leucine

Endogenous Metabolite Metabolism
3-Amino-4-methylpentanoic acid (DL-Homovaline) 是 L-亮氨酸的异构体,是 β 氨基酸,通过亮氨酸 2,3-氨基变位酶在人体中由 L-亮氨酸代谢天然产生。
T14065 9-Ethyladenine

6-Amino-9-ethylpurine,9-乙基腺嘌呤

AChR Neuroscience
9-Ethyladenine (6-Amino-9-ethylpurine) 是一种腺嘌呤磷酸核糖基转移酶的部分有效抑制剂。
TN1243 3-Aminocoumarin

3-Amino-2-benzopyrone,3-aminochromen-2-one,Coumarin amine

Others Others
3-Aminocoumarin (3-aminochromen-2-one) 是金属配合物的关键中间体。
T4905 (Z)-4-Amino-4-oxobut-2-enoic acid

Maleamic acid,Acrylic acid,马来酰胺酸

Others; Endogenous Metabolite Metabolism; Others
(Z)-4-Amino-4-oxobut-2-enoic acid (Maleamic acid) 是内源性代谢产物的一种。
T4863 DL-Homocysteine

DL-高半胱氨酸,2-Amino-4-mercaptobutyric acid

Endogenous Metabolite Metabolism
DL-Homocysteine (2-Amino-4-mercaptobutyric acid) 是弱神经毒素,能够影响犬尿酸的产生。
T3011 2-Amino-4-(2-aminophenyl)-4-oxobutanoic acid

Kynurenine,Dl-Kynurenine,Kynurenin,3-Anthraniloylalanine,犬尿氨酸

Others; Endogenous Metabolite Metabolism; Others
2-Amino-4-(2-aminophenyl)-4-oxobutanoic acid 是一种酮类和氨基酸衍生物,具有多种生物功能,包括血管舒张、免疫调节和神经调节活性。2-Amino-4-(2-aminophenyl)-4-oxobutanoic acid 是烟酸的前体。2-Amino-4-(2-aminophenyl)-4-oxobutanoic acid 的异常产生与神经系统疾病相关的认知缺陷和抑郁症状有关。2-Amino-4-(2-aminophenyl)-4-oxobutanoic acid 在某些类型的癌细胞中过度表达,可能被用作评估癌症风险的生物标志物。
T19165 8-Hydroxyguanine

8 Hydroxyguanine,7,8-dihydro-8-oxoguanine,2-Amino-6,8-dihydroxypurine

Endogenous Metabolite Metabolism
8-Hydroxyguanine (8 Hydroxyguanine)是由活性氧物质产生的主要诱变前损伤。 它导致G-T和A-C置换。8-Hydroxyguanine 是一种 RNA 氧化和 DNA 氧化损伤的生物标记物。8-Hydroxyguanine 具有致突变性和致癌性,常用于癌症实验中。
T4709 (2S,3R,4S,5R)-2-Amino-3,4,5,6-tetrahydroxyhexanal hydrochloride

盐酸 D-甘露糖胺,D-Mannosamine hydrochloride

Others; Endogenous Metabolite Metabolism; Others
(2S,3R,4S,5R)-2-Amino-3,4,5,6-tetrahydroxyhexanal hydrochloride (D-Mannosamine hydrochloride) 是内源性代谢产物的一种。
T4757 L-Homoserine

(S)-2-氨基-4-羟基丁酸,(S)-(-)-2-AMINO-4-HYDROXYBUTYRIC ACID

Others; Endogenous Metabolite Metabolism; Others
L-Homoserine ((S)-(-)-2-AMINO-4-HYDROXYBUTYRIC ACID) 是天然存在的非蛋白丝氨酸,是合成苏氨酸、蛋氨酸和赖氨酸的共有中间体。它是氨基酸丝氨酸的更具反应性的变体。
T4933 (S)-2-acetamido-4-amino-4-oxobutanoic acid

Nα-Acetyl-L-asparagine,N-乙酰-L-天门冬酰胺

Endogenous Metabolite Metabolism
(S)-2-acetamido-4-amino-4-oxobutanoic acid (Nα-Acetyl-L-asparagine),也称为acasn,属于一种内源性代谢产物。
T0883 Tramiprosate

Homotaurine,3-Amino-1-propanesulfonic acid,Alzhemed,高牛黄酸

Beta Amyloid; GABA Receptor Membrane transporter/Ion channel; Neuroscience
Tramiprosate (Alzhemed) 是一种具有口服活性的、可透过血脑屏障的天然氨基酸,存在于各种红色海藻中,能够可溶性 Aβ 结合并以非原纤维形式维持 Aβ。它是一种 GABA 类似物,具有神经保护,抗惊厥和抗高血压的活性。
T4832 Cytosine

6-Aminopyrimidin-2(1H)-one,4-Amino-2-hydroxypyrimidine,Cytosinimine,胞嘧啶

Endogenous Metabolite Metabolism
Cytosine (6-Aminopyrimidin-2(1H)-one) 是 DNA 和 RNA 中发现的四个主要碱基之一。它修饰表现出与表观遗传多样性和衰老有关的昼夜节律振荡。
T4752 1-Aminocyclopropane-1-carboxylic acid

1-Aminocyclopropanecarboxylic acid,1-氨基环丙烷羧酸,1-Amino-1-carboxycyclopropane,ACC

Endogenous Metabolite; NMDAR Metabolism; Neuroscience
1-Aminocyclopropane-1-carboxylic acid (ACC) 是内源性代谢产物的一种。
T9143 D-Isoleucine

(2R,3R)-2-Amino-3-methylpentanoic acid,D-异亮氨酸,(R)-Isoleucine

Others Others
D-Isoleucine ((2R,3R)-2-Amino-3-methylpentanoic acid) 是一种异亮氨酸立体异构体,是 Asc-1 反转运蛋白的选择性激活剂。它能够释放内源性 D-丝氨酸,提高海马 CA1-CA3 的长期增效作用。
T5306 H-Abu-OH

L-2-氨基丁酸,L-Aminobutyric Acid,L-α-amino-n-Butyric acid,L(+)-2-Aminobutyric acid

Others; Endogenous Metabolite Metabolism; Others
H-Abu-OH (L-α-amino-n-Butyric acid) 是氨基丁酸的三个同分异构体之一,它在患有雷氏综合征,同型血尿症,酪氨酸血症,非酮糖症以及鸟氨酸转氨酶症等代谢病儿童的血浆中的含量会明显升高。
T10938 D-Kynurenine

D-尿嘧啶,(R)-2-Amino-4-(2-aminophenyl)-4-oxobutanoic acid,ZINC901103

GPR; AhR; Endogenous Metabolite Endocrinology/Hormones; GPCR/G Protein; Immunology/Inflammation; Metabolism
D-Kynurenine (ZINC901103) 是 D-色氨酸的代谢物和 GPR109B 的激动剂。 D-Kynurenine 激活 AhR 并促进上皮细胞向间充质的转化。 D-Kynurenine 在 D-氨基酸氧化酶的荧光分析中用作底物。
T0326 DL-Glutamine

Glutamin,DL-Gl,(±)-Glutamine,DL-谷氨酰胺,2-amino-4-carbamoylbutanoic acid

Ferroptosis; Amino Acids and Derivatives; Endogenous Metabolite Apoptosis; Metabolism
DL-Glutamine (2-amino-4-carbamoylbutanoic acid) 是一种非必需氨基酸,大量存在于全身并参与许多代谢过程。 它由谷氨酸和氨合成,是体内氮的主要载体,是许多细胞的重要能量来源,用于制药和供生物化学研究。
T4514 N-Acetyl-D-Glucosamine

N-乙酰-D-氨基葡萄糖,NAG,N-Acetyl-2-amino-2-deoxyglucose,Marine Sweet,N-Acetyl-2-amino-2-deoxy-D-glucose,N-乙酰氨基葡萄糖,GlcNAc

Endogenous Metabolite Metabolism
N-Acetyl-D-Glucosamine (NAG) 是葡萄糖的单糖衍生物。
T9294 DL-Valine

DL-缬氨酸,Valine, DL-,H-DL-Val-OH,2-Amino-3-methylbutanoic acid

Others Others
DL-Valine (H-DL-Val-OH) 是 2-氨基-3-甲基丁酸。它是在植物中从丙酮酸开始通过几个步骤合成的。
T2O2730 L-Serine

(S)-Serine,L-丝氨酸,丝氨酸,serine,(-)-Serine,(S)-2-Amino-3-hydroxypropanoic acid

Endogenous Metabolite Metabolism
L-Serine (serine) 是一种人体非必需氨基酸,它存在于许多蛋白质中,并且在功能上很重要。L-Serine 也存在于丝氨酸蛋白酶类的活性位点,包括胰蛋白酶和凝乳胰蛋白酶。
T4755 2,3-Diaminopropanoic acid hydrochloride

DL-2,3-Diaminopropionic acid monohydroch,3-Amino-DL-alanine monohydrochloride,DL-2,3-二胺基丙酸盐酸盐

Others; Endogenous Metabolite Metabolism; Others
2,3-Diaminopropanoic acid hydrochloride (3-Amino-DL-alanine monohydrochloride) 是内源性代谢产物的一种。
TQ0273 Neopterin

D-(+)-Neopterin,2-Amino-6-((1S,2R)-1,2,3-trihydroxypropyl)pteridin-4(3H)-one,新蝶呤

Endogenous Metabolite Metabolism
Neopterin (D-(+)-Neopterin) 是三磷酸腺苷的一种分解产物,是细胞免疫系统激活的标志物。
T4772 (±)-Leucine

DL-Leucine,(+/-)-Amino-4-methylpentanoic acid,DL-亮氨酸,DL-2-Aminmo-4-methylvalerianic acid

Others; Endogenous Metabolite; Antibacterial Metabolism; Microbiology/Virology; Others
(±)-Leucine (DL-2-Aminmo-4-methylvalerianic acid) 是亮氨酸的异构体,是一种化学杀菌剂和膳食添加剂,存在于青椒、青西葫芦、意大利甜红辣椒和红甜椒中。
T4871 D-​Glucosamic acid

D-氨基葡萄糖酸,2-Amino-2-deoxy-D-gluconic acid,D-Glucosaminic acid

Others; Endogenous Metabolite Metabolism; Others
D-​Glucosamic acid (2-Amino-2-deoxy-D-gluconic acid) 是内源性代谢产物的一种。
T0710 L-Cycloserine

Levcycloserine,Levcicloserina,(-)-Cycloserine,(S)-Cycloserine,Levcycloserinum,环丝氨酸,(S)-4-Amino-3-isoxazolidone

HIV Protease; GABA Receptor Membrane transporter/Ion channel; Microbiology/Virology; Neuroscience; Proteases/Proteasome
L-Cycloserine ((-)-Cycloserine) 不可逆地抑制大肠杆菌以及各种动物大脑中的 GABA 吡哆醛 5'-磷酸依赖性转氨酶,导致体内抑制性神经递质 γ-氨基丁酸水平升高。
TN7191 4-Amino-5-Bromopyrrolo[2,3-D]Pyrimidine

4-氨基-5-溴吡咯并[2,3-D]嘧啶,5-bromo-1H-pyrrolo[2,3-d]pyrimidin-4-amine,5-bromo-7H-pyrrolo[2,3-d]pyrimidin-4-amine

Others Others
4-Amino-5-Bromopyrrolo[2,3-D]Pyrimidine (5-bromo-1H-pyrrolo[2,3-d]pyrimidin-4-amine) 是一种海洋来源的天然产物,存在于Echinodictyum sp.。
T5057 DL-O-Phosphoserine

DL-O-磷酸丝氨酸,DL-2-Amino-3-hydroxypropanoic acid 3-phosphate,O-PHOSPHO-L-SERINE,DL-SOP

Others; Endogenous Metabolite Metabolism; Others
O-PHOSPHO-L-SERINE 是丝氨酸和磷酸的酯,是人类生物流体中的正常代谢物。O-phospho-L-serine 是一种吞噬抑制剂,抑制光损伤后的神经胶质细胞增殖和锥体细胞再生。
T0043 Octodrine

二甲己胺,2-Amino-6-methylheptane,6-Methyl-2-heptylamine,1,5-Dimethylhexylamine

Dopamine Receptor GPCR/G Protein; Neuroscience
Octodrine (2-Amino-6-methylheptane) 是一种中枢神经刺激剂,可增加痛阈、心率 (正变时效应) 和心肌收缩力 (正变力效应),可增加多巴胺和去甲肾上腺素 (noradrenaline) 的摄取。
T3377 L-Phenylalanine

L-苯丙氨酸,(S)-2-Amino-3-phenylpropionic acid,phenylalanine,3-Phenyl-L-alanine

Calcium Channel; Endogenous Metabolite; iGluR Membrane transporter/Ion channel; Metabolism; Neuroscience
L-Phenylalanine (3-Phenyl-L-alanine) 是分离自大肠杆菌的必需氨基酸,是 NMDARs(KB573 μM) 和非 NMDARs 的甘氨酸和谷氨酸结合位点的竞争性拮抗剂,用于食品香料和药品的生产中。它是一种电压依赖性 α2δ 亚基 Ca2+通道拮抗剂,Ki 为 980 nM。
T19096 2-Amino-5-phenylpyridine

Others Others
2-Amino-5-phenylpyridine is a heterocyclic aromatic amine that is formed by pyrolysis of phenylalanine in proteins. It is in broiled sardines and is considered as potentially carcinogenic.
T0881 6-Aminocaproic acid

氨基己酸,EACA,6-氨基己酸,6-Aminohexanoic acid,Epsilon-Amino-n-caproic Acid,(6-)ε-​Aminocaproic acid

Others Others
6-Aminocaproic acid (EACA) 是一种单氨基羧酸,是一种有效的、具有口服活性的纤溶酶和纤溶酶原的抑制剂。它是一种有效的抗纤维蛋白溶解剂,能够竞争性结合纤溶酶原上的赖氨酸残基,防止血块溶解,并抑制纤溶酶的形成,减少纤维蛋白溶解。它可用于出血性疾病的研究。
T2941 Glucosamine hydrochloride

Chitosamine hydrochloride,盐酸氨基葡萄糖,2-Amino-2-deoxy-glucose HCl,Chitosamine HCl,D-(+)-Glucosamine hydrochloride

Reactive Oxygen Species; HIF/HIF Prolyl-Hydroxylase; Endogenous Metabolite; Autophagy Autophagy; Chromatin/Epigenetic; Immunology/Inflammation; Metabolism; NF-κB
Glucosamine hydrochloride (Chitosamine hydrochloride) 是软骨基质和滑液中糖胺聚糖的天然成分,常用作骨关节炎的治疗方法。它也是一种氨基糖,是糖基化蛋白和脂质生化合成的突出前体,用作膳食补充剂。
T2760 (S)-2-Amino-3-(4-hydroxy-3,5-diiodophenyl)propanoic acid dihydrate

Iodogorgoic acid,apothyrin,jodgorgon,3,5-Diiodotyrosine Dihydrate,双碘酪氨酸

Others; Endogenous Metabolite Metabolism; Others
(S)-2-Amino-3-(4-hydroxy-3,5-diiodophenyl)propanoic acid dihydrate (jodgorgon) 是内源性代谢产物的一种。
T4866 H-Trp-NH2.HCl

L-Tryptophanamide hydrochloride,L-色氨酰胺盐酸盐,(2S)-2-amino-3-(1H-indol-3-yl)propanamide hydrochloride

Others; Endogenous Metabolite Metabolism; Others
H-Trp-NH2.HCl ((2S)-2-amino-3-(1H-indol-3-yl)propanamide hydrochloride) 是一种内源性代谢产物,已在多种生物体液中检测到,如尿液和血液。
TN1208 2-Amino-3-carboxy-1,4-naphthoquinone

NADPH-oxidase Immunology/Inflammation
2-Amino-3-carboxy-1,4-naphthoquinone 是电子转移介质,可改变同型发酵乳酸菌的葡萄糖代谢,可作为双歧杆菌生长刺激剂,它通过NAD(P)H 介导的氧化作用影响双歧杆菌的终产物形态。
TMA2536 4-Amino-4-methyl-2-pentanone

Others Others
4-Amino-4-methyl-2-pentanone 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TMA2536,CAS号为 625-04-7。
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天然产物

3-Amino-5-Hydroxybenzoic Acid
Cat.No: TN7178
Synonym: 3-amino-5-hydroxy-benzoic acid,3-Amino-5-hydroxybenzoicAcid,3-氨基-5-羟基苯甲酸
Target: Others
9-amino-CPT
Cat.No: T3S1957
Synonym: 9-氨基喜树碱,Aminocamptothecin,9-amino-2(S)-camptothecin,9-Aminocamptothecin
Target: Topoisomerase
3-Amino-4-hydroxybenzoic acid
Cat.No: T4770
Synonym: 3-氨基-4-羟基苯甲酸,3-amino-4-hydroxybenzenecarboxylic acid
Target: Others, Endogenous Metabolite
5-Amino-3H-imidazole-4-Carboxamide
Cat.No: T1705
Synonym: 4-Amino-5-imidazolecarboxamide,AICA,4-氨基-5-咪唑甲酰胺,5-Aminoimidazole-4-carboxamide
Target: Endogenous Metabolite
7-Amino-4-methylcoumarin-3-acetic acid
Cat.No: TN1328
Synonym: 7-氨基-4-甲基-3-香豆素醋酸,7-Amino-4-methylcoumarin
Target: Others
2-Amino-3-hydroxypyridine
Cat.No: T7923
Synonym:
Target: Others
2-Amino-4'-fluorobenzophenone
Cat.No: T7937
Synonym:
Target: Others
2-Amino-2-dichlorobenzophenone
Cat.No: T7918
Synonym:
Target: Others
2-Amino-1-phenylethanol
Cat.No: T4873
Synonym:
Target: Endogenous Metabolite
3-Amino-2-piperidinone
Cat.No: T13495
Synonym: Cyclo-ornithine
Target: Endogenous Metabolite
8-Amino-1-Naphthalenesulfonic Acid
Cat.No: T7971
Synonym:
Target: Others
2-Amino-5-ureidopentanoic acid
Cat.No: T2931
Synonym: DL-Citrulline,Citrulline,瓜氨酸
Target: Others, Endogenous Metabolite
7-Amino-4-(trifluoromethyl)coumarin
Cat.No: TJS0341
Synonym: 香豆素151,Coumarin 151,AFC,7-氨基-4-(三氟甲基)香豆素
Target: 5-HT Receptor
3-Amino-2-methylpropanoic acid
Cat.No: T4887
Synonym: DL-3-AMINOISOBUTYRIC ACID,3-氨基异丁酸,α-Methyl-β-alanine
Target: Endogenous Metabolite
3-Amino-4-methylpentanoic acid
Cat.No: T5569
Synonym: DL-Homovaline,3-氨基-4-甲基戊酸,DL-beta-leucine,beta-Aminoisocaproic acid,beta-Leucine
Target: Endogenous Metabolite
9-Ethyladenine
Cat.No: T14065
Synonym: 6-Amino-9-ethylpurine,9-乙基腺嘌呤
Target: AChR
3-Aminocoumarin
Cat.No: TN1243
Synonym: 3-Amino-2-benzopyrone,3-aminochromen-2-one,Coumarin amine
Target: Others
(Z)-4-Amino-4-oxobut-2-enoic acid
Cat.No: T4905
Synonym: Maleamic acid,Acrylic acid,马来酰胺酸
Target: Others, Endogenous Metabolite
DL-Homocysteine
Cat.No: T4863
Synonym: DL-高半胱氨酸,2-Amino-4-mercaptobutyric acid
Target: Endogenous Metabolite
2-Amino-4-(2-aminophenyl)-4-oxobutanoic acid
Cat.No: T3011
Synonym: Kynurenine,Dl-Kynurenine,Kynurenin,3-Anthraniloylalanine,犬尿氨酸
Target: Others, Endogenous Metabolite
8-Hydroxyguanine
Cat.No: T19165
Synonym: 8 Hydroxyguanine,7,8-dihydro-8-oxoguanine,2-Amino-6,8-dihydroxypurine
Target: Endogenous Metabolite
(2S,3R,4S,5R)-2-Amino-3,4,5,6-tetrahydroxyhexanal hydrochloride
Cat.No: T4709
Synonym: 盐酸 D-甘露糖胺,D-Mannosamine hydrochloride
Target: Others, Endogenous Metabolite
L-Homoserine
Cat.No: T4757
Synonym: (S)-2-氨基-4-羟基丁酸,(S)-(-)-2-AMINO-4-HYDROXYBUTYRIC ACID
Target: Others, Endogenous Metabolite
(S)-2-acetamido-4-amino-4-oxobutanoic acid
Cat.No: T4933
Synonym: Nα-Acetyl-L-asparagine,N-乙酰-L-天门冬酰胺
Target: Endogenous Metabolite
Tramiprosate
Cat.No: T0883
Synonym: Homotaurine,3-Amino-1-propanesulfonic acid,Alzhemed,高牛黄酸
Target: Beta Amyloid, GABA Receptor
Cytosine
Cat.No: T4832
Synonym: 6-Aminopyrimidin-2(1H)-one,4-Amino-2-hydroxypyrimidine,Cytosinimine,胞嘧啶
Target: Endogenous Metabolite
1-Aminocyclopropane-1-carboxylic acid
Cat.No: T4752
Synonym: 1-Aminocyclopropanecarboxylic acid,1-氨基环丙烷羧酸,1-Amino-1-carboxycyclopropane,ACC
Target: Endogenous Metabolite, NMDAR
D-Isoleucine
Cat.No: T9143
Synonym: (2R,3R)-2-Amino-3-methylpentanoic acid,D-异亮氨酸,(R)-Isoleucine
Target: Others
H-Abu-OH
Cat.No: T5306
Synonym: L-2-氨基丁酸,L-Aminobutyric Acid,L-α-amino-n-Butyric acid,L(+)-2-Aminobutyric acid
Target: Others, Endogenous Metabolite
D-Kynurenine
Cat.No: T10938
Synonym: D-尿嘧啶,(R)-2-Amino-4-(2-aminophenyl)-4-oxobutanoic acid,ZINC901103
Target: GPR, AhR, Endogenous Metabolite
DL-Glutamine
Cat.No: T0326
Synonym: Glutamin,DL-Gl,(±)-Glutamine,DL-谷氨酰胺,2-amino-4-carbamoylbutanoic acid
Target: Ferroptosis, Amino Acids and Derivatives, Endogenous Metabolite
N-Acetyl-D-Glucosamine
Cat.No: T4514
Synonym: N-乙酰-D-氨基葡萄糖,NAG,N-Acetyl-2-amino-2-deoxyglucose,Marine Sweet,N-Acetyl-2-amino-2-deoxy-D-glucose,N-乙酰氨基葡萄糖,GlcNAc
Target: Endogenous Metabolite
DL-Valine
Cat.No: T9294
Synonym: DL-缬氨酸,Valine, DL-,H-DL-Val-OH,2-Amino-3-methylbutanoic acid
Target: Others
L-Serine
Cat.No: T2O2730
Synonym: (S)-Serine,L-丝氨酸,丝氨酸,serine,(-)-Serine,(S)-2-Amino-3-hydroxypropanoic acid
Target: Endogenous Metabolite
2,3-Diaminopropanoic acid hydrochloride
Cat.No: T4755
Synonym: DL-2,3-Diaminopropionic acid monohydroch,3-Amino-DL-alanine monohydrochloride,DL-2,3-二胺基丙酸盐酸盐
Target: Others, Endogenous Metabolite
Neopterin
Cat.No: TQ0273
Synonym: D-(+)-Neopterin,2-Amino-6-((1S,2R)-1,2,3-trihydroxypropyl)pteridin-4(3H)-one,新蝶呤
Target: Endogenous Metabolite
(±)-Leucine
Cat.No: T4772
Synonym: DL-Leucine,(+/-)-Amino-4-methylpentanoic acid,DL-亮氨酸,DL-2-Aminmo-4-methylvalerianic acid
Target: Others, Endogenous Metabolite, Antibacterial
D-​Glucosamic acid
Cat.No: T4871
Synonym: D-氨基葡萄糖酸,2-Amino-2-deoxy-D-gluconic acid,D-Glucosaminic acid
Target: Others, Endogenous Metabolite
L-Cycloserine
Cat.No: T0710
Synonym: Levcycloserine,Levcicloserina,(-)-Cycloserine,(S)-Cycloserine,Levcycloserinum,环丝氨酸,(S)-4-Amino-3-isoxazolidone
Target: HIV Protease, GABA Receptor
4-Amino-5-Bromopyrrolo[2,3-D]Pyrimidine
Cat.No: TN7191
Synonym: 4-氨基-5-溴吡咯并[2,3-D]嘧啶,5-bromo-1H-pyrrolo[2,3-d]pyrimidin-4-amine,5-bromo-7H-pyrrolo[2,3-d]pyrimidin-4-amine
Target: Others
DL-O-Phosphoserine
Cat.No: T5057
Synonym: DL-O-磷酸丝氨酸,DL-2-Amino-3-hydroxypropanoic acid 3-phosphate,O-PHOSPHO-L-SERINE,DL-SOP
Target: Others, Endogenous Metabolite
Octodrine
Cat.No: T0043
Synonym: 二甲己胺,2-Amino-6-methylheptane,6-Methyl-2-heptylamine,1,5-Dimethylhexylamine
Target: Dopamine Receptor
L-Phenylalanine
Cat.No: T3377
Synonym: L-苯丙氨酸,(S)-2-Amino-3-phenylpropionic acid,phenylalanine,3-Phenyl-L-alanine
Target: Calcium Channel, Endogenous Metabolite, iGluR
2-Amino-5-phenylpyridine
Cat.No: T19096
Synonym:
Target: Others
6-Aminocaproic acid
Cat.No: T0881
Synonym: 氨基己酸,EACA,6-氨基己酸,6-Aminohexanoic acid,Epsilon-Amino-n-caproic Acid,(6-)ε-​Aminocaproic acid
Target: Others
Glucosamine hydrochloride
Cat.No: T2941
Synonym: Chitosamine hydrochloride,盐酸氨基葡萄糖,2-Amino-2-deoxy-glucose HCl,Chitosamine HCl,D-(+)-Glucosamine hydrochloride
Target: Reactive Oxygen Species, HIF/HIF Prolyl-Hydroxylase, Endogenous Metabolite, Autophagy
(S)-2-Amino-3-(4-hydroxy-3,5-diiodophenyl)propanoic acid dihydrate
Cat.No: T2760
Synonym: Iodogorgoic acid,apothyrin,jodgorgon,3,5-Diiodotyrosine Dihydrate,双碘酪氨酸
Target: Others, Endogenous Metabolite
H-Trp-NH2.HCl
Cat.No: T4866
Synonym: L-Tryptophanamide hydrochloride,L-色氨酰胺盐酸盐,(2S)-2-amino-3-(1H-indol-3-yl)propanamide hydrochloride
Target: Others, Endogenous Metabolite
2-Amino-3-carboxy-1,4-naphthoquinone
Cat.No: TN1208
Synonym:
Target: NADPH-oxidase
4-Amino-4-methyl-2-pentanone
Cat.No: TMA2536
Synonym:
Target: Others
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Cat. No. Product Name Species Expression System
TMPH-00857 ABAT Protein, Human, Recombinant (His & Myc & SUMO)

L-AIBAT,GABA aminotransferase,GABA transaminase,GAB...

Human E. coli
Catalyzes the conversion of gamma-aminobutyrate and L-beta-aminoisobutyrate to succinate semialdehyde and methylmalonate semialdehyde, respectively. Can also convert delta-aminovalerate and beta-alanine. ABAT Protein, Human, Recombinant (His & Myc & SUMO) is expressed in E. coli expression system with N-10xHis-SUMO and C-Myc tag. The predicted molecular weight is 73.3 kDa and the accession number is P80404.
TMPY-01938 CD98 Protein, Human, Recombinant (His)

4T2HC,4F2,CD98HC,NACAE,MDU1,4F2HC,CD98,solute carrier family...

Human HEK293 Cells
CD98 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 49.2 kDa and the accession number is P08195-1.
TMPY-02358 CD98 Protein, Mouse, Recombinant (His)

NACAE,AI314110,Ly-m10,Cd98,Mgp-2hc,4F2HC,Ly10,4F2,solute car...

Mouse HEK293 Cells
CD98 Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 49.2 kDa and the accession number is P10852-2.
TMPH-03181 LaaA Protein, Pseudomonas azotoformans, Recombinant (His & Myc & SUMO)

L-amino acid amidase,laaA

Pseudomonas azotoformans E. coli
Hydrolyzes L-prolinamide, L-proline-p-nitroanilide, L-alaninamide, L-methioninamide, piperidine-2-carboxamide and piperazine-2-carboxamide. Has a much lower activity towards piperazine-2-tert-butylcarboxamide. Does not hydrolyze dipeptides and D-prolinamide. LaaA Protein, Pseudomonas azotoformans, Recombinant (His & Myc & SUMO) is expressed in E. coli expression system with N-10xHis-SUMO and C-Myc tag. The predicted molecular weight is 54.5 kDa and the accession number is Q76KX0.
TMPY-02472 DOPA Decarboxylase/DDC Protein, Mouse, Recombinant (His)

Aadc,dopa decarboxylase (aromatic L-amino acid deca...

Mouse Baculovirus Insect Cells
DOPA Decarboxylase/DDC Protein, Mouse, Recombinant (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 55.2 kDa and the accession number is O88533.
TMPJ-00853 DAO Protein, Human, Recombinant (His)

D-Amino-Acid Oxidase,DAMOX,DAAO,DAO

Human E. coli
D-Amino-Acid Oxidase (DAO) belongs to the DAMOX/DASOX family. DAO is a peroxisomal enzyme which founctions as a homodimer to oxidizes D-amino acids to the corresponding imino acids, producing ammonia and hydrogen peroxide. D-amino-acid oxidase regulates the level of the neuromodulator D-serine in the brain, has a high activity towards D-DOPA and contributes to dopamine synthesis. D-amino-acid oxidase could act as a detoxifying agent which removes D-amino acids accumulated during aging. It also a...
TMPY-01060 DOPA Decarboxylase/DDC Protein, Human, Recombinant (His)

dopa decarboxylase (aromatic L-amino acid decarboxy...

Human Baculovirus Insect Cells
DOPA Decarboxylase/DDC Protein, Human, Recombinant (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 55 kDa and the accession number is Q53Y41.
TMPH-03276 DAO Protein, Rat, Recombinant (His & Myc)

D-amino-acid oxidase,Dao1,DAMOX,DAO,DAAO

Rat E. coli
Regulates the level of the neuromodulator D-serine in the brain. Has high activity towards D-DOPA and contributes to dopamine synthesis. Could act as a detoxifying agent which removes D-amino acids accumulated during aging. Acts on a variety of D-amino acids with a preference for those having small hydrophobic side chains followed by those bearing polar, aromatic, and basic groups. Does not act on acidic amino acids. DAO Protein, Rat, Recombinant (His & Myc) is expressed in E. coli expression sy...
TMPH-02621 DAO Protein, Mouse, Recombinant (His)

DAMOX,Dao1,DAO,DAAO,D-amino-acid oxidase

Mouse E. coli
Regulates the level of the neuromodulator D-serine in the brain. Has high activity towards D-DOPA and contributes to dopamine synthesis. Could act as a detoxifying agent which removes D-amino acids accumulated during aging. Acts on a variety of D-amino acids with a preference for those having small hydrophobic side chains followed by those bearing polar, aromatic, and basic groups. Does not act on acidic amino acids. DAO Protein, Mouse, Recombinant (His) is expressed in E. coli expression system...
TMPH-02379 arnT Protein, Klebsiella pneumoniae, Recombinant (His)

Lipid IV(A) 4-amino-4-deoxy-L-arabinosyltransferase...

Klebsiella pneumoniae E. coli
Catalyzes the transfer of the L-Ara4N moiety of the glycolipid undecaprenyl phosphate-alpha-L-Ara4N to lipid A. The modified arabinose is attached to lipid A and is required for resistance to polymyxin and cationic antimicrobial peptides.
TMPH-01604 SLC7A5 Protein, Human, Recombinant (His & Myc & SUMO)

SLC7A5,y+ system cationic amino acid transporter,La...

Human E. coli
SLC7A5 Protein, Human, Recombinant (His & Myc & SUMO) is expressed in E. coli expression system with N-10xHis-SUMO and C-Myc tag. The predicted molecular weight is 19.7 kDa and the accession number is Q01650.
TMPY-04631 CD98 Protein, Rat, Recombinant (hFc)

solute carrier family 3 (amino acid transporter hea...

Rat HEK293 Cells
CD98 Protein, Rat, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 75.8 kDa and the accession number is Q794F9.
TMPY-03307 CD98 Protein, Rat, Recombinant (His)

solute carrier family 3 (amino acid transporter hea...

Rat HEK293 Cells
CD98 Protein, Rat, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 49.7 kDa and the accession number is Q794F9.
TMPH-02554 BCAT2 Protein, Mouse, Recombinant (His & Myc)

Bcat2,BCAT(m),Eca40,Branched-chain-amino-acid a...

Mouse E. coli
Catalyzes the first reaction in the catabolism of the essential branched chain amino acids leucine, isoleucine, and valine. May also function as a transporter of branched chain alpha-keto acids. BCAT2 Protein, Mouse, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 48.2 kDa and the accession number is O35855.
TMPH-00188 BioAB Protein, Bacteroides fragilis, Recombinant (His & Myc)

Adenosylmethionine-8-amino-7-oxononanoate amino...

Bacteroides fragilis E. coli
Catalyzes two activities which are involved in the biotine biosynthesis: the conversion of dethiobiotin (DTB) to biotin by the insertion of a sulfur atom into dethiobiotin via a radical-based mechanism, and the transfer of the alpha-amino group from S-adenosyl-L-methionine (SAM) to 7-keto-8-aminopelargonic acid (KAPA) to form 7,8-diaminopelargonic acid (DAPA). BioAB Protein, Bacteroides fragilis, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The p...
TMPH-02528 SLC7A10 Protein, Mouse, Recombinant (His & SUMOstar)

Slc7a10,Solute carrier family 7 member 10,Asc-type amino...

Mouse P. pastoris (Yeast)
Sodium-independent, high affinity transport of small neutral D- and L-amino acids and amino acid-related compounds. May play a role in the modulation of glutamatergic transmission through mobilization of D-serine at the glutamatergic synapse. SLC7A10 Protein, Mouse, Recombinant (His & SUMOstar) is expressed in yeast with N-His tag. The predicted molecular weight is 22.5 kDa and the accession number is P63115.
TMPH-01314 SLC1A3 Protein, Human, Recombinant (His & KSI)

Excitatory amino acid transporter 1,Solute carrier ...

Human E. coli
SLC1A3 Protein, Human, Recombinant (His & KSI) is expressed in E. coli expression system with N-6xHis-KSI tag. The predicted molecular weight is 25.5 kDa and the accession number is P43003.
TMPH-03434 BIO3 Protein, S. cerevisiae, Recombinant (His & Myc)

Diaminopelargonic acid synthase,BIO3,7,8-diamin...

Saccharomyces cerevisiae E. coli
Catalyzes the transfer of the alpha-amino group from S-adenosyl-L-methionine (SAM) to 7-keto-8-aminopelargonic acid (KAPA) to form 7,8-diaminopelargonic acid (DAPA). It is the only aminotransferase known to utilize SAM as an amino donor. BIO3 Protein, S. cerevisiae, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 58.7 kDa and the accession number is P50277.
TMPY-06611 CD98 Protein, Human, Recombinant (His), Biotinylated

4F2,4F2HC,MDU1,4T2HC,solute carrier family 3 (amino...

Human HEK293 Cells
CD98 Protein, Human, Recombinant (His), Biotinylated is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 49.19 kDa and the accession number is P08195-1.
TMPH-00573 DAPA aminotransferase Protein, E. coli, Recombinant (His & Myc)

DAPA AT,bioA,7,8-diaminononanoate synthase,DAPA

E. coli E. coli
Catalyzes the transfer of the alpha-amino group from S-adenosyl-L-methionine (SAM) to 7-keto-8-aminopelargonic acid (KAPA) to form 7,8-diaminopelargonic acid (DAPA). It is the only animotransferase known to utilize SAM as an amino donor. Complements a bioU deletion in Synechocystis PCC 6803.
TMPH-03750 SLC7A11 Protein, Human, Recombinant (His)

SLC7A11,Calcium channel blocker resistance protein CCBR1,Sol...

Human E. coli
Sodium-independent, high-affinity exchange of anionic amino acids with high specificity for anionic form of cystine and glutamate.
TMPJ-01273 ACY3 Protein, Human, Recombinant (His)

Acylase III,Aminoacylase-3,ACY3,Hepatitis C virus c...

Human E. coli
Aspartoacylase 3, also known as ACY3, N-acyl-aromatic-L-amino acid amidohydrolase (carboxylate-forming), Acylase III, Aminoacylase-3, Aspartoacylase-2, Aspartoacylase-2, HCV core-binding protein 1 and ASPA2, is a member of the Aspartoacylase subfamily. ACY3 plays an important role in deacetylating mercapturic acids in kidney proximal tubules and acts on N-acetyl-aromatic amino acids.ACY3 is located in the cytoplasm of S2 and S3 proximal tubules and the apical domain of S1 proximal tubules. ACY3 ...
TMPY-00665 Aminopeptidase N/CD13 Protein, Human, Recombinant (I603M, His)

alanyl (membrane) aminopeptidase,LAP1,APN,CD13,P150...

Human HEK293 Cells
Aminopeptidase N/CD13 Protein, Human, Recombinant (I603M, His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 104.2 kDa and the accession number is A0A024RC61.
TMPH-03032 Leucyl aminopeptidase Protein, Mycoplasma pneumoniae, Recombinant (His & SUMO)

Probable cytosol aminopeptidase,Leucine amino

Mycoplasma pneumoniae E. coli
Presumably involved in the processing and regular turnover of intracellular proteins. Catalyzes the removal of unsubstituted N-terminal amino acids from various peptides. Leucyl aminopeptidase Protein, Mycoplasma pneumoniae, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 64.8 kDa and the accession number is P75206.
TMPY-03445 Aspartate Aminotransferase Protein, Human, Recombinant (His)

ASTQTL1,glutamic-oxaloacetic transaminase 1, soluble,cCAT,cA...

Human E. coli
GOT1 (Glutamic-Oxaloacetic Transaminase 1) is a Protein Coding gene. GOT1 belongs to the class-I pyridoxal-phosphate-dependent aminotransferase family. Glutamic-oxaloacetic transaminase is a pyridoxal phosphate-dependent enzyme that exists in cytoplasmic and mitochondrial forms, GOT1 and GOT2, respectively. GOT plays a role in amino acid metabolism and the urea and tricarboxylic acid cycles. The two enzymes are homodimeric and show close homology. GOT1 is an important regulator of levels of glut...
TMPH-03099 Aminopeptidase N/CD13 Protein, Pig, Recombinant (His & Myc)

gp130,pAPN,AP-M,Aminopeptidase M,CD13,AP-N,Alanyl <...

Sus scrofa (Pig) E. coli
Aminopeptidase N/CD13 Protein, Pig, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 47.1 kDa and the accession number is P15145.
TMPH-00654 Methionine aminopeptidase Protein, E. coli, Recombinant (His & SUMO)

Methionine aminopeptidase,map,Peptidase M

E. coli E. coli
Removes the N-terminal methionine from nascent proteins. The N-terminal methionine is often cleaved when the second residue in the primary sequence is small and uncharged (Met-Ala-, Cys, Gly, Pro, Ser, Thr, or Val). Requires deformylation of the N(alpha)-formylated initiator methionine before it can be hydrolyzed.
TMPY-00644 Aminopeptidase A Protein, Human, Recombinant (His)

APA,glutamyl aminopeptidase,ENPEP,gp160,CD249

Human Baculovirus Insect Cells
Aminopeptidase A Protein, Human, Recombinant (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 107.2 kDa and the accession number is Q07075.
TMPY-01058 Aminoacylase 1 Protein, Human, Recombinant (His)

ACY-1,ACY1D,aminoacylase 1,HEL-S-5

Human Baculovirus Insect Cells
Aminoacylase 1 Protein, Human, Recombinant (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 47.3 kDa and the accession number is Q03154-1.
TMPY-02896 Aminopeptidase A Protein, Mouse, Recombinant (His)

Ly-51,6030431M22Rik,ENPEP,APA,Bp-1/6C3,glutamyl amino

Mouse Baculovirus Insect Cells
Aminopeptidase A Protein, Mouse, Recombinant (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 106 kDa and the accession number is P16406.
TMPY-00660 Aminoacylase 1 Protein, Mouse, Recombinant (His)

1110014J22Rik,aminoacylase 1,Acy-1

Mouse HEK293 Cells
Aminoacylase 1 Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 45 kDa and the accession number is Q99JW2.
TMPY-03041 Aminopeptidase A Protein, Rat, Recombinant (aa 41-945, His)

ENPEP,glutamyl aminopeptidase

Rat Baculovirus Insect Cells
Aminopeptidase A Protein, Rat, Recombinant (aa 41-945, His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 106 kDa and the accession number is P50123-1.
TMPY-00758 Aminopeptidase N/CD13 Protein, Mouse, Recombinant (His)

Cd13,AP-N,Apn,AP-M,P150,alanyl (membrane) aminopept...

Mouse HEK293 Cells
Aminopeptidase N/CD13 Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 104 kDa and the accession number is P97449.
TMPJ-00745 IFN-alpha 2a/IFNA2 Protein, Human, Recombinant

Interferon α-2,IFNA2,干扰素,IFN α2a,IFN-α-2,IFN-Alpha-2,Interfe...

Human E. coli
At least 23 different variants of IFN-α are known. The individual proteins have molecular masses between 19-26 kDa and consist of proteins with lengths of 156-166 and 172 amino acids. All IFN-α subtypes possess a common conserved sequence region between amino acid positions 115-151 while the amino-terminal ends are variable. Many IFN-α subtypes only differ in their sequences by one or two positions. Naturally occurring variants also include proteins truncated by 10 amino acids at the carboxy-ter...
TMPJ-00746 IFN-alpha 2b/IFNA2 Protein, Human, Recombinant

干扰素,IFNA2,Interferon α-2,Interferon α-A,Interferon Alpha-2,I...

Human E. coli
At least 23 different variants of IFN-α are known. The individual proteins have molecular masses between 19-26 kDa and consist of proteins with lengths of 156-166 and 172 amino acids. All IFN-α subtypes possess a common conserved sequence region between amino acid positions 115-151 while the amino-terminal ends are variable. Many IFN-α subtypes differ in their sequences by only one or two positions. Naturally occurring variants also include proteins that are truncated by 10 amino acids at the ca...
TMPJ-00059 IL-7 Protein, Human, Recombinant (His)

Interleukin-7,IL7,白细胞介素,IL-7,白介素

Human HEK293 Cells
Human Interleukin 7 (IL-7) is a potent lymphoid cell growth factor stimulating the proliferation of lymphoid progenitors. IL7 can associate with the hepatocyte growth factor (HGF) to form a hybrid cytokine that functions as a pre-pro-B cell growth-stimulating factor. Human IL7 cDNA encodes a 177 amino acid precursor protein containing a 25 amino acid signal peptide and a 152 amino acid mature protein. Human and mouse IL7 share 65% sequence identity in the mature region and both exhibit cross-spe...
TMPJ-01469 NGF Protein, Human, Recombinant (E. colli)

NGFB,神经生长因子,β-NGF,NGF,Beta-Nerve Growth Factor,β-Nerve Growt...

Mouse E. coli
NGF is the first member discovered in the Neurotrophin family, which includes brain-derived neurotrophic factor (BDNF), neurotrophin-3 (NT-3), and neurotrophin-4 (NT-4). These proteins belong to the cysteine-knot family of growth factors that assume stable dimeric structures. Mouse beta -NGF is a homodimer of two 120 amino acid polypeptides. It shares approximately 90% homology at the amino acid level with human beta -NGF and 95.8% with rat beta -NGF. NGF signaling has been shown to play an impo...
TMPY-02707 PAH Protein, Human, Recombinant (415 Asn/Asp, His)

phenylalanine hydroxylase,PH,PKU1,PKU

Human Baculovirus Insect Cells
PAH (phenylalanine hydroxylase), also known as PH, belongs to the biopterin-dependent aromatic amino acid hydroxylase family. It contains 1 ACT domain, N-terminal region of PAH is thought to contain allosteric binding sites for phenylalanine and to constitute an "inhibitory" domain that regulates the activity of a catalytic domain in the C-terminal portion of the molecule. In humans, PAH is expressed both in the liver and the kidney, and there is some indication that it may be differentially reg...
TMPY-00105 Recombinant Protein G

E. coli
Protein G is a bacterial cell wall protein expressed at the cell surface of certain group C and group G Streptococcal strains. It has affinity for both Fab- and Fc-fragments of human IgG by independent and separate binding sites. Binding to the Fc region of immunoglobulins from several species by a non-immune mechanism exhibits great affinity for almost all mammalian immunoglobulin G (IgG) classes, including all human IgG subclasses (IgG1, IgG2, IgG3 and IgG4) and also rabbit, mouse, and goat Ig...
TMPJ-00864 VEGF165 Protein, Human, Recombinant

Vascular Endothelial Growth Factor Isoform 165,血管内皮生长因子,VEGF...

Human HEK293 Cells
Human Vascular endothelial growth factor (VEGF), also known as VEGF-A and vascular permeability factor (VPF), belongs to the platelet-derived growth factor family of cysteine-knot growth factors. It is a potent activator in vasculogenesis and angiogenesis both physiologically and pathologically. VEGF-A has 8 differently spliced isoforms, of which VEGF165 is the most abundant one. VEGF165 is a disulfide-linked homodimer consisting of two glycosylated 165 amino acid polypeptide chains. VEGF stimul...
TMPJ-00154 IL-15RA Protein, Mouse, Recombinant (hFc, Human Cells)

sIL-15 receptor subunit α,Il15ra,Interleukin-15 receptor sub...

Mouse HEK293 Cells
Mouse interleukin-15 receptor subunit alpha, also known as Il15ra, is a high-affinity receptor for interleukin-15. Il15ra associates as a heterotrimer with the IL-2 receptor beta and gamma subunits (Common gamma chain, or gamma c) to initiate signal transduction. It can signal both in cis and trans where IL15R from one subset of cells presents IL15 to neighboring IL2RG-expressing cells. Il15ra is expressed in special cells including a wide variety of Tand B cells and non-lymphoid cells. Human Il...
TMPJ-01172 IL-17 Protein, Mouse, Recombinant (His)

CTLA8,IL-17,IL-17A,Interleukin-17A,CTLA-8,Cytotoxic T-Lympho...

Mouse HEK293 Cells
Interleukin-17 is a potent pro-inflammatory cytokine produced by activated memory T cells. There are at least six members of the IL-17 family in humans and in mice. Mature mouse IL-17A shares 61% and 89% amino acid sequence identity with human and rat IL-17A, respectively. As IL-17 shares properties with IL-1 and TNF-alpha, it may induce joint inflammation and bone and cartilage destruction. This cytokine is found in synovial fluids of patients with rheumatoid arthritis, and produced by rheumato...
TMPY-02481 ACOX1 Protein, Human, Recombinant (His)

PALMCOX,ACOX,SCOX,acyl-CoA oxidase 1, palmitoyl

Human Baculovirus Insect Cells
Peroxisomal acyl-coenzyme A oxidase 1(ACOX1 or AOX) is the first enzyme of the fatty acid beta-oxidation pathway and belongs to the Acyl-CoA oxidase family. Human liver peroxisomes contain two acyl-CoA oxidases, namely, palmitoyl-CoA oxidase (ACOX1/AOX) and a branched chain acyl-CoA oxidase. The palmitoyl-CoA oxidase (ACOX1/AOX) oxidizes the CoA esters of straight chain fatty acids and prostaglandins and donates electrons directly to molecular oxygen, thereby producing H2O2. Human ACOX1/AOX is a...
TMPJ-00037 FGF-2 Protein, Mouse, Recombinant

Fibroblast Growth Factor 2,bFGF,HBGF-2,Basic Fibroblast Grow...

Mouse E. coli
FGF basic is one of 22 mitogenic proteins of the FGF family, which show 35-60% amino acid conservation. Unlike other FGFs, FGF acidic and basic lack signal peptides and are secreted by an alternate pathway. The 17 kDa mouse sequence has 98% aa identity with rat, and 95% identity with human, bovine, and sheep FGF basic. Binding of FGF to heparin or cell surface HSPG is necessary for binding, dimerization and activation of tyrosine kinase FGF receptors. FGF basic binds other proteins, polysacchari...
TMPY-02585 Acid sphingomyelinase/SMPD1 Protein, Mouse, Recombinant (His)

aSMase,ASM,Zn-SMase,A-SMase,sphingomyelin phosphodiesterase ...

Mouse Baculovirus Insect Cells
Sphingomyelin phosphodiesterase 1 (SMPD1) , also known as ASM ( acid sphingomyelinase ), is a member of the acid sphingomyelinase family of enzymes. Three isoforms have been identified, isoform 1 is 631 amino acids (aa) in length as the pro form, while Isoform 2 and isoform 3 have lost catalytic activity. The active SMPD1 isoform 1 contains one saposin B-type domain that likely interacts with sphingomyelin, and a catalytic region. Human SMPD1 is 86% aa identical to mouse SMPD1. SMPD1 is a monome...
TMPJ-01065 Noggin/NOG Protein, Mouse, Recombinant (His)

Nog,Noggin

Mouse HEK293 Cells
Noggin is a secreted homodimeric glycoprotein that is an antagonist of bone morphogenetic proteins (BMPs). Mouse Noggin cDNA encodes a 232 amino acid (aa) residue precursor protein with 19 aa residue putative signal peptide that is cleaved to generate the 213 aa residue mature protein which is secreted as a homodimeric glycoprotein. Secreted Noggin probably remains close to the cell surface due to its binding of heparin-containing proteoglycans. Noggin binds some BMPs such as BMP4 with high affi...
TMPJ-00137 APRIL/TNFSF13 Protein, Human, Recombinant (Flag & His)

TRDL-1,TNF- and APOL-related leukocyte expressed ligand 2,Tu...

Human HEK293 Cells
APRIL (a proliferation-inducing ligand), also known as TNFSF13, TALL2, TRDL1, and CD256, is a member of the TNF ligand superfamily. It is synthesized as a 32 kDa proprotein which is cleaved by furin in the Golgi to release the active 17 kDa soluble molecule. Secreted human APRIL, which consists almost entirely of a single TNF homology domain, shares 85% amino acid sequence identity with mouse and rat APRIL. Both APRIL and its close relative BAFF bind and signal through the TNF superfamily recept...
TMPJ-00375 HGF Protein, Human, Recombinant (His)

Scatter factor,Hepatocyte growth factor,HGF,SF,Hepatopoietin...

Human HEK293 Cells
HGF, is a pleiotropic protein in the Plasminogen subfamily of S1 peptidases and contains 4 kringle domains, 1 PAN domain and 1 peptidase S1 domain. HGF is secreted as an inactive 728 amino acid (aa) single chain propeptide. It is cleaved after the fourth Kringle domain by a serine protease to form bioactive disulfide-linked HGF with a 60 kDa alpha and 30 kDa beta chain. HGF binds heparan-sulfate proteoglycans and the widely expressed receptor tyrosine kinase, HGF R/c-MET. HGF regulates epithelia...
TMPJ-00042 TSLP Protein, Human, Recombinant

TSLP,Thymic stromal lymphopoietin

Human E. coli
Thymic stromal lymphopoietin (TSLP) is a novel member of the hemopoietic cytokine family that promotes the development of B cells and shares overlapping activity with IL-7. The human TSLP protein comprises a 28 amino acids (aa) signal sequence and 131 aa mature region. Human TSLP has two isoforms lfTSLP and sfTSLP produced by alternative splicing . lfTSLP is expressed in a number of tissues including heart, liver and prostate, and sfTSLP (63aa) is predominantly expressed in keratinocytes of oral...
TMPY-02550 Eotaxin/CCL11 Protein, Human, Recombinant (His)

SCYA11,chemokine (C-C motif) ligand 11

Human E. coli
CCL11 or chemokine (C-C motif) ligand 11 is a member of the chemokine (C-C motif) ligand family. Chemokin (C-C motif) ligand 11 is a member of the chemokine family. There are four members of the chemokine family: C-C kemokines, C kemokines, CXC kemokines and CX3C kemokines. The C-C kemokines have two cysteines nearby the amino terminus. There have been at least 27 distinct members of this subgroup reported for mammals, called C-C chemokine ligands (CCL)-1 to 28. Chemokines are a family of small ...
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重组蛋白

ABAT Protein, Human, Recombinant (His & Myc & SUMO)
Cat.No: TMPH-00857
Species: Human
Expression System: E. coli
CD98 Protein, Human, Recombinant (His)
Cat.No: TMPY-01938
Species: Human
Expression System: HEK293 Cells
CD98 Protein, Mouse, Recombinant (His)
Cat.No: TMPY-02358
Species: Mouse
Expression System: HEK293 Cells
LaaA Protein, Pseudomonas azotoformans, Recombinant (His & Myc & SUMO)
Cat.No: TMPH-03181
Species: Pseudomonas azotoformans
Expression System: E. coli
DOPA Decarboxylase/DDC Protein, Mouse, Recombinant (His)
Cat.No: TMPY-02472
Species: Mouse
Expression System: Baculovirus Insect Cells
DAO Protein, Human, Recombinant (His)
Cat.No: TMPJ-00853
Species: Human
Expression System: E. coli
DOPA Decarboxylase/DDC Protein, Human, Recombinant (His)
Cat.No: TMPY-01060
Species: Human
Expression System: Baculovirus Insect Cells
DAO Protein, Rat, Recombinant (His & Myc)
Cat.No: TMPH-03276
Species: Rat
Expression System: E. coli
DAO Protein, Mouse, Recombinant (His)
Cat.No: TMPH-02621
Species: Mouse
Expression System: E. coli
arnT Protein, Klebsiella pneumoniae, Recombinant (His)
Cat.No: TMPH-02379
Species: Klebsiella pneumoniae
Expression System: E. coli
SLC7A5 Protein, Human, Recombinant (His & Myc & SUMO)
Cat.No: TMPH-01604
Species: Human
Expression System: E. coli
CD98 Protein, Rat, Recombinant (hFc)
Cat.No: TMPY-04631
Species: Rat
Expression System: HEK293 Cells
CD98 Protein, Rat, Recombinant (His)
Cat.No: TMPY-03307
Species: Rat
Expression System: HEK293 Cells
BCAT2 Protein, Mouse, Recombinant (His & Myc)
Cat.No: TMPH-02554
Species: Mouse
Expression System: E. coli
BioAB Protein, Bacteroides fragilis, Recombinant (His & Myc)
Cat.No: TMPH-00188
Species: Bacteroides fragilis
Expression System: E. coli
SLC7A10 Protein, Mouse, Recombinant (His & SUMOstar)
Cat.No: TMPH-02528
Species: Mouse
Expression System: P. pastoris (Yeast)
SLC1A3 Protein, Human, Recombinant (His & KSI)
Cat.No: TMPH-01314
Species: Human
Expression System: E. coli
BIO3 Protein, S. cerevisiae, Recombinant (His & Myc)
Cat.No: TMPH-03434
Species: Saccharomyces cerevisiae
Expression System: E. coli
CD98 Protein, Human, Recombinant (His), Biotinylated
Cat.No: TMPY-06611
Species: Human
Expression System: HEK293 Cells
DAPA aminotransferase Protein, E. coli, Recombinant (His & Myc)
Cat.No: TMPH-00573
Species: E. coli
Expression System: E. coli
SLC7A11 Protein, Human, Recombinant (His)
Cat.No: TMPH-03750
Species: Human
Expression System: E. coli
ACY3 Protein, Human, Recombinant (His)
Cat.No: TMPJ-01273
Species: Human
Expression System: E. coli
Aminopeptidase N/CD13 Protein, Human, Recombinant (I603M, His)
Cat.No: TMPY-00665
Species: Human
Expression System: HEK293 Cells
Leucyl aminopeptidase Protein, Mycoplasma pneumoniae, Recombinant (His & SUMO)
Cat.No: TMPH-03032
Species: Mycoplasma pneumoniae
Expression System: E. coli
Aspartate Aminotransferase Protein, Human, Recombinant (His)
Cat.No: TMPY-03445
Species: Human
Expression System: E. coli
Aminopeptidase N/CD13 Protein, Pig, Recombinant (His & Myc)
Cat.No: TMPH-03099
Species: Sus scrofa (Pig)
Expression System: E. coli
Methionine aminopeptidase Protein, E. coli, Recombinant (His & SUMO)
Cat.No: TMPH-00654
Species: E. coli
Expression System: E. coli
Aminopeptidase A Protein, Human, Recombinant (His)
Cat.No: TMPY-00644
Species: Human
Expression System: Baculovirus Insect Cells
Aminoacylase 1 Protein, Human, Recombinant (His)
Cat.No: TMPY-01058
Species: Human
Expression System: Baculovirus Insect Cells
Aminopeptidase A Protein, Mouse, Recombinant (His)
Cat.No: TMPY-02896
Species: Mouse
Expression System: Baculovirus Insect Cells
Aminoacylase 1 Protein, Mouse, Recombinant (His)
Cat.No: TMPY-00660
Species: Mouse
Expression System: HEK293 Cells
Aminopeptidase A Protein, Rat, Recombinant (aa 41-945, His)
Cat.No: TMPY-03041
Species: Rat
Expression System: Baculovirus Insect Cells
Aminopeptidase N/CD13 Protein, Mouse, Recombinant (His)
Cat.No: TMPY-00758
Species: Mouse
Expression System: HEK293 Cells
IFN-alpha 2a/IFNA2 Protein, Human, Recombinant
Cat.No: TMPJ-00745
Species: Human
Expression System: E. coli
IFN-alpha 2b/IFNA2 Protein, Human, Recombinant
Cat.No: TMPJ-00746
Species: Human
Expression System: E. coli
IL-7 Protein, Human, Recombinant (His)
Cat.No: TMPJ-00059
Species: Human
Expression System: HEK293 Cells
NGF Protein, Human, Recombinant (E. colli)
Cat.No: TMPJ-01469
Species: Mouse
Expression System: E. coli
PAH Protein, Human, Recombinant (415 Asn/Asp, His)
Cat.No: TMPY-02707
Species: Human
Expression System: Baculovirus Insect Cells
Recombinant Protein G
Cat.No: TMPY-00105
Species:
Expression System: E. coli
VEGF165 Protein, Human, Recombinant
Cat.No: TMPJ-00864
Species: Human
Expression System: HEK293 Cells
IL-15RA Protein, Mouse, Recombinant (hFc, Human Cells)
Cat.No: TMPJ-00154
Species: Mouse
Expression System: HEK293 Cells
IL-17 Protein, Mouse, Recombinant (His)
Cat.No: TMPJ-01172
Species: Mouse
Expression System: HEK293 Cells
ACOX1 Protein, Human, Recombinant (His)
Cat.No: TMPY-02481
Species: Human
Expression System: Baculovirus Insect Cells
FGF-2 Protein, Mouse, Recombinant
Cat.No: TMPJ-00037
Species: Mouse
Expression System: E. coli
Acid sphingomyelinase/SMPD1 Protein, Mouse, Recombinant (His)
Cat.No: TMPY-02585
Species: Mouse
Expression System: Baculovirus Insect Cells
Noggin/NOG Protein, Mouse, Recombinant (His)
Cat.No: TMPJ-01065
Species: Mouse
Expression System: HEK293 Cells
APRIL/TNFSF13 Protein, Human, Recombinant (Flag & His)
Cat.No: TMPJ-00137
Species: Human
Expression System: HEK293 Cells
HGF Protein, Human, Recombinant (His)
Cat.No: TMPJ-00375
Species: Human
Expression System: HEK293 Cells
TSLP Protein, Human, Recombinant
Cat.No: TMPJ-00042
Species: Human
Expression System: E. coli
Eotaxin/CCL11 Protein, Human, Recombinant (His)
Cat.No: TMPY-02550
Species: Human
Expression System: E. coli
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Cat. No. Product Name Target Signaling Pathways
T40376 L-Phenylalanine-15N

L-苯丙氨酸 15N,(S)-2-Amino-3-phenylpropionic acid-15N,L-Phenylalanine-15N

Calcium Channel Membrane transporter/Ion channel; Metabolism
L-Phenylalanine-15N ((S)-2-Amino-3-phenylpropionic acid-15N) 是 15N 标记的 L-Phenylalanine。L-Phenylalanine 是从大肠杆菌中分离出来的一种必需氨基酸。 L-Phenylalanine 广泛用于食品香精和药物的生产。
TMID-0031 WXG02403-d9

(S)-benzyl 2-((tert-butoxycarbonyl)amino)-3,3-dimethylbutanoate-d9

WXG02403-d9 是 WXG02403 的氘代化合物。WXG02403 的 CAS 号为 154092-61-2。
TMIJ-0009 1-Amino Hydantoin-13C3

1-Amino Hydantoin-13C3 是 1-Amino Hydantoin 的 13C 的标记化合物。1-Amino Hydantoin 的 CAS 号为 6301-02-6。1-Aminohydantoin 是一种呋喃妥因在动物组织中的主要代谢物。1-Aminohydantoin 与组织蛋白共价结合,在微酸性条件下从组织中释放出来,与 2-硝基苯甲醛衍生形成 AHD 的硝基苯基衍生物可被检测。1-Aminohydantoin 可作为测定肉、奶等兽药残留的测定指标。
TMIH-0053 4-amino-N-(4-nitrophenyl)benzenesulfonamide-d4

4-amino-N-(4-nitrophenyl)benzenesulfonamide-d4 是 4-amino-N-(4-nitrophenyl)benzenesulfonamide 的氘代化合物。
TMIJ-0008 3-Amino-2-Oxazolidinone-d4

Aoz-d4

3-Amino-2-Oxazolidinone-d4 是 3-Amino-2-Oxazolidinone 的氘代化合物。3-Amino-2-Oxazolidinone 的 CAS 号为 80-65-9。3-Amino-2-oxazolidinone 是一种呋喃唑烷酮的代谢物 (metabolite),可用作检测呋喃唑烷酮残留的一个指标。
TMIJ-0468 Atrazine-desisopropyl-d5 (ethylamino-d5)

Atrazine-desisopropyl-d5 (ethylamino-d5) 是 Atrazine-desisopropyl 的氘代化合物。Atrazine-desisopropyl 的 CAS 号为 1007-28-9。
TMID-0176 4-Aminobutyric acid-2,2,3,3,4,4-d6

4-Aminobutyric acid-2,2,3,3,4,4-d6 是 4-Aminobutyric acid 的氘代化合物。4-Aminobutyric acid 的 CAS 号为 56-12-2。γ-Aminobutyric acid 是成年哺乳动物大脑中主要的抑制性神经递质,能够与离子移变 GABA 受体 (GABAA) 受体和促代谢受体 (GABAB) 受体结合发挥作用。
TMID-0117 Aminophylline-d6

Aminophylline-d6 是 Aminophylline 的氘代化合物。Aminophylline 的 CAS 号为 317-34-0。Aminophylline 是一种竞争性非选择性磷酸二酯酶抑制剂,具有支气管扩张作用。它是竞争性的腺苷受体拮抗剂,有用于哮喘研究的潜力。
TMIJ-0457 Daminozide-d6 (dimethyl-d6)

Daminozide-d6 (dimethyl-d6) 是 Daminozide 的氘代化合物。Daminozide 的 CAS 号为 1596-84-5。Daminozide 是一种植物生长调节剂,选择性地抑制 KDM2/7 JmjC 亚家族,对PHF8、KDM2A和KIAA1718的IC50值分别为 0.55、1.5 和 2.1 μM。
TMIJ-0030 1-Aminoadamantane-d15

1-Aminoadamantane-d15 是 1-Aminoadamantane 的氘代化合物。1-Aminoadamantane 的 CAS 号为 768-94-5。Amantadine (1-Aminoadamantane) 是抗病毒药物,也是是 NMDA 型谷氨酸受体的弱拮抗剂,能促进高多巴胺的释放,并阻断多巴胺的再摄取。
TMID-0278 4-AMinoantipyrine-d3

4-AMinoantipyrine-d3 是 4-AMinoantipyrine 的氘代化合物。4-AMinoantipyrine 的 CAS 号为 83-07-8。4-Aminoantipyrine是一种检测试剂,在过氧化物酶与苯酚存在时,用于葡萄糖测定。
TMID-0103 N-Nitroso-N-(methyl-d3)-4-aminobutyric Acid

NMBA-d3

N-Nitroso-N-(methyl-d3)-4-aminobutyric Acid 是 N-Nitroso-N-(methyl)-4-aminobutyric Acid 的氘代化合物。N-Nitroso-N-(methyl)-4-aminobutyric Acid 的 CAS 号为 61445-55-4。
T32902 L-Serine-1-13C

L-(1-13C)Serine,L-(l-13C)Serine

L-Serine-1-13C is an amino acid.
T40915 L-Aspartic acid 13C

L-Aspartic acid 13C is a 13C labeled L-Aspartic acid. L-Aspartic acid is is an amino acid, shown to be a suitable prodrug for colon-specific drug deliverly.
TMIJ-0055 DL-Norepinephrine-d6 HCl

DL-Norepinephrine-d6 HCl 是 DL-NorepinephrineHCl 的氘代化合物。DL-NorepinephrineHCl 的 CAS 号为 55-27-6。DL-Norepinephrine hydrochloride 是一种靶向α1 adrenoceptor和β1 adrenoceptor的神经递质,可降低心内膜下氧分压。它是一种模拟内源性去甲肾上腺素的拟交感神经作用的合成苯乙胺。
TMIJ-0372 L-Threonine-d2

L-Threonine-d2 是 L-Threonine 的氘代化合物。L-Threonine 的 CAS 号为 72-19-5。L-Threonine 是人体必需氨基酸,是神经系统的重要氨基酸。L-Threonine 在卟啉和脂肪代谢中也起着重要作用,防止肝脏脂肪堆积。L-Threonine 可用于治疗肠道疾病和消化不良,也可用于缓解焦虑和轻度抑郁。
TMIJ-0089 L-Valine-d8

L-Valine-d8 是 L-Valine 的氘代化合物。L-Valine 的 CAS 号为 72-18-4。L-Valine 是蛋白二十种氨基酸中的其中一种。它是必需氨基酸。
TMIJ-0381 L-Valine-13C5-15N

L-Valine-13C5-15N 是 L-Valine 的 13C 和 15 N 的标记化合物。L-Valine 的 CAS 号为 72-18-4。L-Valine 是蛋白二十种氨基酸中的其中一种。它是必需氨基酸。
TMID-0171 Kynurenic Acid-d5

Kynurenic Acid-d5 是 Kynurenic Acid 的氘代化合物。Kynurenic Acid 的 CAS 号为 492-27-3。Kynurenic acid 是一种内源性色氨酸代谢物,是针对靶点NMDA、谷氨酸、α7烟碱型乙酰胆碱受体的广谱拮抗剂。它也是GPR35/CXCR8激动剂。
TMIJ-0082 Benserazide-d3 HCl

Benserazide-d3 HCl 是 Benserazide HCl 的氘代化合物。Benserazide HCl 的 CAS 号为 14919-77-8。Benserazide hydrochloride 是一种芳香族 L-氨基酸脱羧酶(AADC)的抑制剂,常用于帕金森病。
TMIJ-0363 DL-Valine-d8

DL-Valine-d8 是 DL-Valine 的氘代化合物。DL-Valine 的 CAS 号为 516-06-3。DL-Valine 是 2-氨基-3-甲基丁酸。它是在植物中从丙酮酸开始通过几个步骤合成的。
TMID-0152 Pyridoxine-d2 HCl

Pyridoxine-d2 HCl 是 Pyridoxine HCl 的氘代化合物。Pyridoxine HCl 的 CAS 号为 58-56-0。Pyridoxine hydrochloride 是一种吡啶衍生物。在于阿尔茨海默病细胞模型中,通过Nrf-2/HO-1 途径发挥抗氧化作用。
TMID-0185 (±)-Ropivacaine-d7

(±)-Ropivacaine-d7 是 (±)-Ropivacaine 的氘代化合物。(±)-Ropivacaine 的 CAS 号为 84057-95-4。Ropivacaine 是有效的钠通道阻断剂,通过可逆地抑制钠离子内流从而引起神经纤维脉冲传导阻滞。Ropivacaine 也是一种 K2P(双孔钾通道)TREK-1的抑制剂,在 COS-7 细胞膜上的 IC50值为 402.7 μM。Ropivacaine 可以用于神经性疼痛的缓解的相关研究。
TMIJ-0373 Biotin-d2

Biotin-d2 是 Biotin 的氘代化合物。Biotin 的 CAS 号为 58-85-5。Biotin 是一种水溶性B族维生素,是细胞生长、脂肪酸产生以及脂肪和氨基酸代谢所必需的。
TMIJ-0078 Glycine-d2

Glycine-d2 是 Glycine 的氘代化合物。Glycine 的 CAS 号为 56-40-6。Glycine 是中枢神经系统的抑制性神经递质,也是谷氨酸的联合激动剂,有促进谷氨酸能NMDA受体兴奋的潜力。它主要存在于明胶和丝素蛋白中,并在治疗上用作营养物质。
TMIJ-0265 Homovanillic Acid-13C-d3

Homovanillic Acid-13C-d3 是 Homovanillic Acid 的 13C 和氘代化合物。Homovanillic Acid 的 CAS 号为 306-08-1。Homovanillic acid 是一种多巴胺代谢物,它与乳糜泻、生长激素缺乏、芳香族氨基酸脱羧酶缺乏症以及脂联素还原酶缺乏症相关。
TMIJ-0521 L-Lysine-4,4,5,5-d4 Hydrochloride

L-Lysine-4,4,5,5-d4 Hydrochloride 是 L-Lysine Hydrochloride 的氘代化合物。L-Lysine Hydrochloride 的 CAS 号为 657-27-2。L-lysine hydrochloride 是一种人类必需氨基酸,能增加钙吸收,减少糖尿病相关疾病和改善肠道健康,可用于疱疹的研究。
TMIJ-0102 Ropivacaine-d7

Ropivacaine-d7 是 Ropivacaine 的氘代化合物。Ropivacaine 的 CAS 号为 84057-95-4。Ropivacaine 是有效的钠通道阻断剂,通过可逆地抑制钠离子内流从而引起神经纤维脉冲传导阻滞。Ropivacaine 也是一种 K2P(双孔钾通道)TREK-1的抑制剂,在 COS-7 细胞膜上的 IC50值为 402.7 μM。Ropivacaine 可以用于神经性疼痛的缓解的相关研究。
TMIJ-0384 L-Cysteine-d3

L-Cysteine-d3 是 L-Cysteine 的氘代化合物。L-Cysteine 的 CAS 号为 52-90-4。L-Cysteine 是人体非必需的含硫氨基酸。L-Cysteine 对蛋白质合成、解毒和多种代谢功能很重要。L-Cysteine 存在于指甲、皮肤和头发的主要蛋白质-角蛋白中,对胶原蛋白的生成、皮肤弹性和质地都很重要。L-Cysteine 是抗氧化剂谷胱甘肽的一种成分,在辅酶A、肝素和生物素等基本生化物质的代谢中起着重要作用,也是氨基酸牛磺酸的制造所必需的。
T36384 DL-Tyrosine-13C9,15N

L-Tyrosine-13C9,15N

L-Tyrosine-13C9,15N is intended for use as an internal standard for the quantification of L-tyrosine by GC- or LC-MS. L-Tyrosine is a non-essential amino acid.1It is produced by hydroxylation of phenylalanine by phenylalanine hydroxylase but can also be obtained from dietary sources or degradation of endogenous proteins, resulting in L-tyrosine release.1,2L-Tyrosine is a precursor in the biosynthesis of catecholamine neurotransmitters, melanins, and thyroid hormones.3Plasma, skeletal muscle, and...
TMIJ-0380 L-Lysine-13C6-15N2 Hydrochloride

L-Lysine-13C6-15N2 Hydrochloride 是 L-Lysine Hydrochloride 的 13C 和 15 N 的标记化合物。L-Lysine Hydrochloride 的 CAS 号为 657-27-2。L-lysine hydrochloride 是一种人类必需氨基酸,能增加钙吸收,减少糖尿病相关疾病和改善肠道健康,可用于疱疹的研究。
TMIJ-0090 L-Carnitine-d9

L-Carnitine-d9 是 L-Carnitine 的氘代化合物。L-Carnitine 的 CAS 号为 541-15-1。L-carnitine 是一种人内源性分子,在人体内以蛋氨酸和赖氨酸为底物进行生物合成,并参与脂肪酸代谢。L-Carnitine 将长链脂肪酰辅酶A转运到线粒体。L-Carnitine 能够改善许多先天性代谢错误的代谢失衡。
TMID-0057 (4-Hydroxy-3-methoxyphenyl)acetic-2,2-d2 Acid

(4-Hydroxy-3-methoxyphenyl)acetic-2,2-d2 Acid 是 (4-Hydroxy-3-methoxyphenyl)acetic Acid 的氘代化合物。(4-Hydroxy-3-methoxyphenyl)acetic Acid 的 CAS 号为 306-08-1。Homovanillic acid 是一种多巴胺代谢物,它与乳糜泻、生长激素缺乏、芳香族氨基酸脱羧酶缺乏症以及脂联素还原酶缺乏症相关。
TMIJ-0081 L-Leucine-d10

L-Leucine-d10 是 L-Leucine 的氘代化合物。L-Leucine 的 CAS 号为 61-90-5。L-Leucine 是必需的支链氨基酸,能够激活mTOR信号通路。
TMIJ-0377 Thiamine Hydrochloride-13C4

Thiamine Hydrochloride-13C4 是 Thiamine Hydrochloride 的 13C 的标记化合物。Thiamine Hydrochloride 的 CAS 号为 67-03-8。Thiamine hydrochloride 是一种必需的微量营养素,是许多中枢代谢酶的辅因子。
TMIJ-0374 L-Leucine-d3

L-Leucine-d3 是 L-Leucine 的氘代化合物。L-Leucine 的 CAS 号为 61-90-5。L-Leucine 是必需的支链氨基酸,能够激活mTOR信号通路。
TMIJ-0240 Lacosamide-d3 (Acetyl-d3)

Lacosamide-d3 (Acetyl-d3) 是 Lacosamide 的氘代化合物。Lacosamide 的 CAS 号为 175481-36-4。Lacosamide是一种功能化氨基酸。Lacosamide以一种新的方式调节钠通道:它选择性地增强钠通道缓慢失活,而对快速失活没有影响Lacosamine在不同的啮齿类动物癫痫发作模型中显示出抗癫痫作用,在反映神经性疼痛和慢性炎性疼痛的不同类型和症状的实验动物模型中显示了抗伤害潜力。
TMID-0247 LacosaMide-d3

LacosaMide-d3 是 LacosaMide 的氘代化合物。LacosaMide 的 CAS 号为 175481-36-4。Lacosamide是一种功能化氨基酸。Lacosamide以一种新的方式调节钠通道:它选择性地增强钠通道缓慢失活,而对快速失活没有影响Lacosamine在不同的啮齿类动物癫痫发作模型中显示出抗癫痫作用,在反映神经性疼痛和慢性炎性疼痛的不同类型和症状的实验动物模型中显示了抗伤害潜力。
TMIH-0257 Glycoursodeoxycholic Acid-d4

Glycoursodeoxycholic Acid-d4 是 Glycoursodeoxycholic Acid 的氘代化合物。Glycoursodeoxycholic Acid 的 CAS 号为 64480-66-6。Glycoursodeoxycholic acid 是一种酰基甘氨酸和胆汁酸-甘氨酸缀合物,是熊去氧胆酸的代谢物。
TMIJ-0312 L-Dopa-2,5,6-d3

L-Dopa-2,5,6-d3 是 L-Dopa 的氘代化合物。L-Dopa 的 CAS 号为 59-92-7。Levodopa 是的神经递质多巴胺的代谢前体,具有口服活性。Levodopa 能够透过血脑屏障,并在大脑中转化为多巴胺。Levodopa具有抗痛觉过敏作用。Levodopa还具有帕金森氏病的研究潜力。
TMIJ-0101 DL-Alanine-2,3,3,3-d4

DL-Alanine-2,3,3,3-d4 是 DL-Alanine 的氘代化合物。DL-Alanine 的 CAS 号为 302-72-7。DL-Alanine 是一种氨基酸,是L-和D-丙氨酸的外消旋化合物。DL-Alanine 与硝酸银水溶液一起用于纳米颗粒生成时常作为还原剂和封端剂。DL-Alanine 是一种甜味剂,可把它位与甘氨酸和糖精钠归为一类。DL-Alanine 在组织和肝脏之间的葡萄糖-丙氨酸循环中起重要作用。DL-Alanine 可用于研究 Cu、Zn、Cd 等过渡金属螯合。
TMID-0096 P-CRESOL-d3 (METHYL-d3)

P-CRESOL-d3 (METHYL-d3) 是 P-CRESOL 的氘代化合物。P-CRESOL 的 CAS 号为 106-44-5。p-Cresol 是一种部分亲脂性部分,在正常条件下与血浆蛋白(接近 100%)强烈结合。对甲酚通过结合代谢,主要是硫酸化和葡萄糖醛酸化,但未结合的对甲酚至少部分通过尿液去除。
T38356 1,2-Dipalmitoyl-13C-sn-glycero-3-PC

1,2-Dipalmitoyl-13C-sn-glycero-3-PC is intended for use as an internal standard for the quantification of 1,2-dipalmitoyl-sn-glycero-3-PC by GC- or LC-MS. 1,2-Dipalmitoyl-sn-glycero-3-PC (DPPC) is a zwitterionic glycerophospholipid commonly used in the formation of lipid monolayers, bilayers, and liposomes for use in a variety of applications.1,2,3,4 It has been used in the formation of proteoliposomes for implantation of γ-glutamyl transpeptidase into human erythrocyte membranes.3 Incorporation...

同位素标记化合物

L-Phenylalanine-15N
Cat.No: T40376
Synonym: L-苯丙氨酸 15N,(S)-2-Amino-3-phenylpropionic acid-15N,L-Phenylalanine-15N
Target: Calcium Channel
WXG02403-d9
Cat.No: TMID-0031
Synonym: (S)-benzyl 2-((tert-butoxycarbonyl)amino)-3,3-dimethylbutanoate-d9
Target:
1-Amino Hydantoin-13C3
Cat.No: TMIJ-0009
Synonym:
Target:
4-amino-N-(4-nitrophenyl)benzenesulfonamide-d4
Cat.No: TMIH-0053
Synonym:
Target:
3-Amino-2-Oxazolidinone-d4
Cat.No: TMIJ-0008
Synonym: Aoz-d4
Target:
Atrazine-desisopropyl-d5 (ethylamino-d5)
Cat.No: TMIJ-0468
Synonym:
Target:
4-Aminobutyric acid-2,2,3,3,4,4-d6
Cat.No: TMID-0176
Synonym:
Target:
Aminophylline-d6
Cat.No: TMID-0117
Synonym:
Target:
Daminozide-d6 (dimethyl-d6)
Cat.No: TMIJ-0457
Synonym:
Target:
1-Aminoadamantane-d15
Cat.No: TMIJ-0030
Synonym:
Target:
4-AMinoantipyrine-d3
Cat.No: TMID-0278
Synonym:
Target:
N-Nitroso-N-(methyl-d3)-4-aminobutyric Acid
Cat.No: TMID-0103
Synonym: NMBA-d3
Target:
L-Serine-1-13C
Cat.No: T32902
Synonym: L-(1-13C)Serine,L-(l-13C)Serine
Target:
L-Aspartic acid 13C
Cat.No: T40915
Synonym:
Target:
DL-Norepinephrine-d6 HCl
Cat.No: TMIJ-0055
Synonym:
Target:
L-Threonine-d2
Cat.No: TMIJ-0372
Synonym:
Target:
L-Valine-d8
Cat.No: TMIJ-0089
Synonym:
Target:
L-Valine-13C5-15N
Cat.No: TMIJ-0381
Synonym:
Target:
Kynurenic Acid-d5
Cat.No: TMID-0171
Synonym:
Target:
Benserazide-d3 HCl
Cat.No: TMIJ-0082
Synonym:
Target:
DL-Valine-d8
Cat.No: TMIJ-0363
Synonym:
Target:
Pyridoxine-d2 HCl
Cat.No: TMID-0152
Synonym:
Target:
(±)-Ropivacaine-d7
Cat.No: TMID-0185
Synonym:
Target:
Biotin-d2
Cat.No: TMIJ-0373
Synonym:
Target:
Glycine-d2
Cat.No: TMIJ-0078
Synonym:
Target:
Homovanillic Acid-13C-d3
Cat.No: TMIJ-0265
Synonym:
Target:
L-Lysine-4,4,5,5-d4 Hydrochloride
Cat.No: TMIJ-0521
Synonym:
Target:
Ropivacaine-d7
Cat.No: TMIJ-0102
Synonym:
Target:
L-Cysteine-d3
Cat.No: TMIJ-0384
Synonym:
Target:
DL-Tyrosine-13C9,15N
Cat.No: T36384
Synonym: L-Tyrosine-13C9,15N
Target:
L-Lysine-13C6-15N2 Hydrochloride
Cat.No: TMIJ-0380
Synonym:
Target:
L-Carnitine-d9
Cat.No: TMIJ-0090
Synonym:
Target:
(4-Hydroxy-3-methoxyphenyl)acetic-2,2-d2 Acid
Cat.No: TMID-0057
Synonym:
Target:
L-Leucine-d10
Cat.No: TMIJ-0081
Synonym:
Target:
Thiamine Hydrochloride-13C4
Cat.No: TMIJ-0377
Synonym:
Target:
L-Leucine-d3
Cat.No: TMIJ-0374
Synonym:
Target:
Lacosamide-d3 (Acetyl-d3)
Cat.No: TMIJ-0240
Synonym:
Target:
LacosaMide-d3
Cat.No: TMID-0247
Synonym:
Target:
Glycoursodeoxycholic Acid-d4
Cat.No: TMIH-0257
Synonym:
Target:
L-Dopa-2,5,6-d3
Cat.No: TMIJ-0312
Synonym:
Target:
DL-Alanine-2,3,3,3-d4
Cat.No: TMIJ-0101
Synonym:
Target:
P-CRESOL-d3 (METHYL-d3)
Cat.No: TMID-0096
Synonym:
Target:
1,2-Dipalmitoyl-13C-sn-glycero-3-PC
Cat.No: T38356
Synonym:
Target:
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