918
345
1
101
40
Cat. No. | Product Name | ||
---|---|---|---|
L1100 | 蛋白酶抑制剂库 | 343 compounds | |
343 种已知的小分子蛋白酶抑制剂的特有集合,可用于高通量筛选和高内涵筛选; |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T21588 |
Olomoucine
|
ERK; CDK | Cell Cycle/Checkpoint; MAPK |
Olomoucine 是 Cdk2/cyclin A、Cdc2/CyclinB、CDK2/CyclinE、CDK5/p35 和 ERK1/p44 MAP 激酶的 ATP 竞争性抑制剂,IC50 分别为 7、7、7、3 和 25 µM。 Olomoucine 调节细胞周期并表现出抗黑色素肿瘤活性。 | |||
T6798 |
Tretazicar
5-Aziridino-2,4-dinitrobenzamide,CB1954,NSC 115829 |
DNA Alkylator/Crosslinker; DNA Alkylation | DNA Damage/DNA Repair |
Tretazicar (NSC-115829) 是一种抗肿瘤前药,由 NAD(P)H 醌氧化还原酶 2 激活。它在酶促活化后生成细胞毒性双功能烷基剂,可以形成 DNA-DNA 链间交联。 | |||
T4297 |
Flibanserin
BIMT-17BS,氟立班丝氨,Girosa,BIMT-17 |
Dopamine Receptor; 5-HT Receptor | GPCR/G Protein; Neuroscience |
Flibanserin (Girosa) 一种具有口服活性的 5-HT1A 受体激动剂和 5-HT2A 受体拮抗剂,Ki 值分别为 1 和 49 nM。它与多巴胺 D4 受体结合,Ki 值在 4 到 24 nM 之间。它是一种血清素能抗抑郁药,用于治疗性欲减退症。 | |||
T8810 |
Terbutaline
|
Adrenergic Receptor | GPCR/G Protein; Neuroscience |
Terbutaline 是 bambuterol 的活性代谢物,也是β2肾上腺素能受体的短效激动剂,可预防早产及用作支气管扩张剂。 | |||
T9835 |
4-QUinolinecarboxamide, N-[3-[[[2-[4-(aminosulfonyl)phenyl]ethyl]amino]carbonyl]phenyl]-1,2-dihydro-2-oxo-
|
Others | Others |
4-QUinolinecarboxamide, N-[3-[[[2-[4-(aminosulfonyl)phenyl]ethyl]amino]carbonyl]phenyl]-1,2-dihydro-2-oxo-是胺。 | |||
TP1253 |
Argireline
六胜肽,Acetyl hexapeptide-3,阿基瑞林 |
Others | Others |
Argireline (Acetyl hexapeptide-3) 是可渗透皮肤的、无毒的抗皱肽。它对神经肌肉接头处依赖 Ca2+的神经递质释放具有显著的抑制作用。它具有抗皱和抗衰老的活性。 | |||
T3526 |
Dasotraline hydrochloride
SEP-225289 hydrochloride,达索曲林盐酸盐 |
Dopamine Receptor; 5-HT Receptor; Serotonin Transporter; Norepinephrine | GPCR/G Protein; Neuroscience |
Dasotraline hydrochloride (SEP-225289 hydrochloride) 是具有阻断多巴胺 (IC50=4 nM),去甲肾上腺素 (IC50=6 nM) 和三羟色胺转运蛋白 (IC50=11 nM)的三重再摄取抑制剂。 | |||
T1888 |
Tacedinaline
Acetyldinaline,N-acetyldinaline,PD-123654,CI994,Goe-5549 |
Apoptosis; HDAC | Apoptosis; Chromatin/Epigenetic; DNA Damage/DNA Repair |
Tacedinaline (CI994) 是一种组蛋白脱乙酰酶抑制剂,抑制重组 HDAC 1, 2 和 3 的IC50值分别为 0.9,0.9,1.2 μM。 | |||
T4635 |
Ralinepag
APD811 |
Others; Prostaglandin Receptor | GPCR/G Protein; Immunology/Inflammation; Others |
Ralinepag (APD811) 是一种可口服的非前列腺素前列环素 (IP) 受体激动剂,对人和大鼠 IP 受体以及人 DP1 受体的 EC50 分别为 8.5、530 和 850 nM。 | |||
T9816 |
Arofylline
阿罗茶碱,LAS 31025 |
PDE | Metabolism |
Arofylline (LAS 31025) 是一种 PDE4 抑制剂,可用于哮喘的研究。 | |||
T0327 |
Fendiline hydrochloride
Fendiline HCl,盐酸芬他林 |
Calcium Channel | Membrane transporter/Ion channel; Metabolism |
Fendiline hydrochloride (Fendiline HCl) 是一种非选择性钙通道抑制剂。 | |||
T67965 |
Torbafylline
|
cAMP; PI3K; PDE | GPCR/G Protein; Metabolism; PI3K/Akt/mTOR signaling |
Torbafylline 是黄嘌呤衍生物,是 磷酸二酯酶 (PDE) 抑制剂,通过 激活 PDE4/cAMP/EPAC/PI3K/Akt 途径减弱烧伤诱导的大鼠骨骼肌蛋白水解,抑制癌症和败血症大鼠增强的骨骼肌泛素 - 蛋白酶体依赖性蛋白水解。 | |||
T7477 |
Antazoline
|
Others | Others |
Antazoline 具有抗组胺和抗胆碱能作用。它用于治疗各种心律失常。 | |||
T13353 |
Xanomeline oxalate
LY246708 oxalate |
AChR | Neuroscience |
Xanomeline oxalate (LY246708 oxalate)作为一种高效且选择性的胆碱能受体激动剂(SMRA),在体内有效促进磷脂酰肌醇水解。Xanomeline oxalate 对于阿尔茨海默病的研究具有重要价值。 | |||
T8104 |
Glycyl-L-valine
|
Others; Endogenous Metabolite | Metabolism; Others |
Glycyl-L-valine 是含有甘氨酸和缬氨酸的二肽。 | |||
T5983 |
o-Phenanthroline
1,10-菲罗啉,1,10-Phenanthroline |
MMP; Others | Others; Proteases/Proteasome |
o-Phenanthroline (1,10-Phenanthroline) 是一种金属螯合剂,能够与 Fe2+形成红色螯合物,在 510 nm 处最大吸收,可防止链脲佐菌素诱导染色体畸变。它也是一种MMP 的抑制剂。 | |||
T9793 |
Methyl Ergoline Acid
|
Others | Others |
Methyl Ergoline Acid 是一种麦角碱衍生物,可用作趋化因子受体配体。 | |||
T0248 |
Clorprenaline hydrochloride
盐酸氯丙那林,Clorprenaline HCl,NSC 334693 |
Adrenergic Receptor | GPCR/G Protein; Neuroscience |
Clorprenaline hydrochloride (Clorprenaline HCl) 是 β2-肾上腺素受体激动剂,与支气管扩张有关,可用于研究哮喘。 | |||
T1140 |
Doxycycline hydrochloride
Doxylin,盐酸多西环素,Vibramycin,Hyclate |
MMP; Antibacterial; Antibiotic | Microbiology/Virology; Proteases/Proteasome |
Doxycycline hydrochloride (Hyclate) 是一种四环素抗生素,是口服有效的广谱金属蛋白酶抑制剂,具有抗菌活性。 | |||
T3941 |
Choline Fenofibrate
Trilipix,ABT-335,非诺贝特胆碱 |
P450; COX; PPAR | DNA Damage/DNA Repair; Immunology/Inflammation; Metabolism; Neuroscience |
Choline Fenofibrate (Trilipix) 是 Fenofibric acid 的胆碱盐,在胃肠道中释放游离的 Fenofibric acid。Fenofibric acid 是一种合成的苯氧基异丁酸衍生物和具有抗高血脂活性的前药。 | |||
T0059 |
Diphenylpyraline hydrochloride
盐酸双苯比拉林,4-Diphenylmethoxy-1-methylpiperidine hydrochloride |
Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Diphenylpyraline hydrochloride (4-Diphenylmethoxy-1-methylpiperidine hydrochloride) 是一种组胺 H1 受体的拮抗剂,抑制多巴胺的吸收。它是可口服的抗组胺试剂,具有抗胆碱和抗过敏作用,可用于缓解过敏性疾病,如鼻炎、花粉热和瘙痒性皮肤疾病等。 | |||
T1083L |
Theophylline monohydrate
Quibron,茶碱一水合物 |
HDAC; PDE; Adenosine Receptor | Chromatin/Epigenetic; DNA Damage/DNA Repair; GPCR/G Protein; Metabolism; Neuroscience |
Theophylline monohydrate (Quibron) 似乎抑制磷酸二酯酶和前列腺素的产生,调节钙通量和细胞内钙分布,并拮抗腺苷。茶碱是黄嘌呤的天然生物碱衍生物,从植物山茶花和小粒咖啡中分离出来。在生理上,该药剂可放松支气管平滑肌,产生血管舒张(脑血管除外),刺激中枢神经系统,刺激心肌,利尿,增加胃酸分泌;它还可以抑制炎症并改善横膈膜的收缩性。 | |||
T20344 |
Acetylcholine bromide
|
Others | Others |
Acetylcholine bromide 是乙酰胆碱的溴化物盐。它是一种神经递质,存在于神经肌肉接头、自主神经节、副交感神经效应器接头、交感神经效应器接头的一个子集以及中枢神经系统的许多部位。 | |||
T38173 |
Propargylcholine
Propargylcholine (bromide) |
Antibacterial | Microbiology/Virology |
Propargylcholine (Propargylcholine (bromide)) 是一种炔烃修饰的胆碱类似物,在铜绿假单胞菌中 Dgc 酶催化的二甲基甘氨酸去甲基化水平上抑制胆碱分解代谢。 | |||
T21447 |
Tolazoline
Priscol,妥拉苏林,Priscoline,Pridazole,Divascol,Vasimid,Benzalolin |
Adrenergic Receptor | GPCR/G Protein; Neuroscience |
Tolazoline (Benzalolin) 是一种竞争性的α-肾上腺素受体拮抗剂。 | |||
T1578 |
Pargyline hydrochloride
优降宁盐酸盐,Pargylamine hydrochloride |
MAO; Monoamine Oxidase | Metabolism; Neuroscience |
Pargyline hydrochloride (Pargylamine hydrochloride) 是不可逆的单胺氧化酶抑制剂,可作用于 MAO-A (Ki=13 μM) 和 MAO-B (Ki=0.5 μM) ,具有降压和抗癌作用。 | |||
T21694 |
(R)-Lisofylline
(R)-Lisophylline |
STAT | JAK/STAT signaling; Stem Cells |
(R)-Lisofylline ((R)-Lisophylline) 是溶血磷脂酸酰基转移酶的抑制剂 (IC50 = 0.6 µM)。 (R)-Lisofylline 可中断 IL-12 信号介导的 STAT4 激活,可用于治疗 1 型糖尿病和自身免疫性疾病的研究。 | |||
T35048 |
Verofylline
CK 0383,Verofilina,CK-0383,Verofyllinum,CK0383 |
PDE | Metabolism |
Verofylline (Verofyllinum) 是一种可口服的长效多效取代甲基黄嘌呤支气管扩张剂,对 PDE4 具有抑制作用,可用于治疗哮喘疾病研究肥胖症。 | |||
T10861 |
Collagen proline hydroxylase inhibitor-1
|
Others | Others |
Collagen proline hydroxylase inhibitor-1 具有抗纤维增生活性。 | |||
T1177 |
Sulfaquinoxaline
磺胺喹恶啉,Avicocid,磺胺喹噁啉,Sulphaquinoxaline,Sulfabenzpyrazine |
Others; Antibacterial; Antibiotic; Parasite | Microbiology/Virology; Others |
Sulfaquinoxaline (Sulfabenzpyrazine) 是一种兽用抗菌剂,对革兰氏阴性菌和革兰氏阳性菌均有活性。它能用于预防球虫病和细菌感染。 | |||
T72079 |
Biotin-aniline
|
||
Biotin-aniline 是一种会对 RNA 和 DNA做出强烈反应的探针。Biotin-aniline具有高效性,用于捕获具有高空间特异性的活细胞中的亚细胞转录组。 | |||
T0400 |
Nitroxoline
5-Nitro-8-quinolinol,8-Hydroxy-5-nitroquinoline,5-Nitro-8-hydroxyquinoline,5-nitroquinolin-8-ol,硝羟喹啉 |
Antibacterial; Antibiotic; Autophagy | Autophagy; Microbiology/Virology |
Nitroxoline (5-nitroquinolin-8-ol) 是一种抗生素,防治生物膜感染。它通过从生物膜基质螯合Fe2+和Zn2+离子而发挥作用。 | |||
T22604 |
(-)-Bicuculline methiodide
|
Others | Others |
(-)-Bicuculline methiodide is a GABAA receptor antagonist. | |||
T9817 |
Isbufylline
|
Others | Others |
Isbufylline 具有显着的抗炎作用和支气管扩张剂活性。 | |||
T22576 |
Anpirtoline hydrochloride
D-16949 hydrochloride |
5-HT Receptor | GPCR/G Protein; Neuroscience |
Anpirtoline hydrochloride (D-16949 hydrochloride) 是一种新型高效的 5-HT1B 受体激动剂和 5-HT3 受体拮抗剂,具有抗伤害、镇痛和抗抑郁活性,可用于研究运动障碍。 | |||
T25742 |
Linzagolix choline
|
GNRH Receptor | GPCR/G Protein |
Linzagolix choline 是一种可口服的非肽类的促性腺激素释放激素(GnRH)拮抗剂。可用于研究子宫肌瘤和子宫内膜异位症相关疼痛。 | |||
T60536 |
Terodiline
|
Calcium Channel; HER; AChR | Angiogenesis; JAK/STAT signaling; Membrane transporter/Ion channel; Metabolism; Neuroscience; Tyrosine Kinase/Adaptors |
Terodiline 是一种具有抗胆碱能和钙拮抗特性的仲胺,可阻断 hERG 电流(IC50:375 nM)。Terodiline 具有心脏毒性,可用于研究逼尿肌不稳定引起的疾病。 | |||
T68080 |
Gevotroline
|
5-HT Receptor | GPCR/G Protein; Neuroscience |
Gevotroline 是棕榈酒中的一种可用来治疗精神病的化学物,是5-HT2 receptor 拮抗剂,可用于研究行为障碍。 | |||
T64331 |
Fmoc-L-Proline
Fmoc-Pro-OH |
Amino Acids and Derivatives | Metabolism |
Fmoc-L-Proline (Fmoc-Pro-OH) 是一种脯氨酸衍生物。 | |||
T11097 |
Drobuline hydrochloride
|
Others | Others |
Drobuline hydrochloride 是一种抗心律失常剂。 | |||
T72072 |
2-benzylsulfanyl-6-methoxy-4-methylquinazoline
|
ROS | Immunology/Inflammation |
2-benzylsulfanyl-6-methoxy-4-methylquinazoline 可作为TRPML 调节剂,可用于治疗与TRPML 活性相关的疾病,如溶酶体储存病、肌肉萎缩症、氧化应激或活性氧(ROS)相关疾病和衰老。 | |||
T9342 |
4-(6,7-dimethoxyquinolin-4-yl)oxyaniline
4-(6,7-Dimethoxy-quinolin-4-yloxy)-phenylamine,BenzenaMine, 4-[(6,7-diMethoxy-4-quinolinyl)oxy]- |
Others | Others |
4-(6,7-dimethoxyquinolin-4-yl)oxyaniline (4-(6,7-Dimethoxy-quinolin-4-yloxy)-phenylamine) 是一种喹啉的衍生物,已用于合成一系列化合物,包括药物、农药和其他有机分子。 | |||
T16782 |
Rolofylline
KW-3902,MK-7418,KF-15372 |
Adenosine Receptor | GPCR/G Protein; Neuroscience |
Rolofylline (KW-3902) 是一种具有选择性腺苷 A1 受体拮抗剂,可用于研究急性充血性心力衰竭和肾功能障碍,可用与研究神经退行性疾病。 | |||
T3052 |
Sancycline
Bonomycin,Norcycline,Sancyclinum,山环素,6-Demethyl-6-deoxytetracycline |
Antibacterial | Microbiology/Virology |
Sancycline (Bonomycin) 是半合成四环素,通过可逆地结合 30S 核糖体亚基并通过阻断氨酰-tRNA 进入核糖体 A 位点来抑制蛋白质翻译。 | |||
T36013 |
Lysophosphatidylcholines
Lyso-Lecithins (egg) |
Apoptosis | Apoptosis |
Lysophosphatidylcholines (Lyso-Lecithins (egg)) 是一种具有口服活性的脂质,可诱导细胞损伤和凋亡 (apoptosis),诱导脱髓鞘。Lysophosphatidylcholines 在炎症、纤维化和癌症的介导中发挥作用,可用于研究动脉粥样硬化。 | |||
T1117 |
Clorgyline hydrochloride
盐酸氯吉林,Clorgiline hydrochloride,N-[3-(2,4-二氯苯氧基)丙基]-N-甲基-2-丙炔胺盐酸盐 |
MAO; Monoamine Oxidase | Metabolism; Neuroscience |
Clorgyline hydrochloride (Clorgiline hydrochloride) 是一种选择性、不可逆的单胺氧化酶A 抑制剂,结构上与Pargyline 相关。 | |||
T7042 |
1,5-Isoquinolinediol
|
PARP | Chromatin/Epigenetic; DNA Damage/DNA Repair |
1,5-Isoquinolinediol 是一种多聚(ADP-核糖)合成酶抑制剂,对PARP1的IC50值为 0.39 µM。它用于研究 PARP1 在 DNA 修复和氧化应激诱导的细胞死亡中的作用。 | |||
T8415 |
4-Benzyl-2-carboxymorpholine hydrochloride
|
Others | Others |
4-Benzyl-2-carboxymorpholine hydrochloride 是一种用于蛋白质组学研究应用的专业产品,来自 Santa Cruz。 | |||
T1006 |
Propantheline bromide
Neopepulsan,溴丙胺太林,Pro-Banthine,Neometantyl |
AChR | Neuroscience |
Propantheline bromide (Pro-Banthine) 是一种抗毒蕈碱剂,用于研究多汗症,遗尿,胃肠和膀胱痉挛。 | |||
T21023 |
Bedaquiline fumarate
TMC 207,R403323,TMC-207,TMC207,R-403323,贝达喹啉富马酸盐,R 403323 |
Antibacterial; Antibiotic | Microbiology/Virology |
Bedaquiline fumarate (TMC207) 是二芳基喹啉抗生素,作用于 ATP 合成酶,常用于结核杆菌感染的研究。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T1680 |
Tolazoline hydrochloride
Imidaline hydrochloride,苯甲唑啉盐酸盐,Imidaline (hydrochloride),Benzidazol hydrochloride,Tolazoline HCl,NSC35110 (hydrochloride) |
Adrenergic Receptor | GPCR/G Protein; Neuroscience |
Tolazoline hydrochloride (NSC35110(hydrochloride)) 是一种 α 肾上腺素受体抑制剂。 | |||
T2773 |
Vindoline
文朵灵,文多灵 |
Microtubule Associated | Cytoskeletal Signaling |
Vindoline 是从长春花叶片中提取的一种生物碱,通过抑制微管组装而表现出抗有丝分裂活性。 | |||
T3S0631 |
Fuziline
|
Anti-infection | Microbiology/Virology |
Fuziline 是一种在附子侧根中发现的二萜生物碱。它在功能上与乌头有关。 | |||
T9294 |
DL-Valine
DL-缬氨酸,Valine, DL-,H-DL-Val-OH,2-Amino-3-methylbutanoic acid |
Others | Others |
DL-Valine (H-DL-Val-OH) 是 2-氨基-3-甲基丁酸。它是在植物中从丙酮酸开始通过几个步骤合成的。 | |||
TN1480 |
Cephaeline
吐根鹼,吐根酚碱 |
Virus Protease; Influenza Virus; HIF | Angiogenesis; Chromatin/Epigenetic; Microbiology/Virology |
Cephaeline 对受保护的原代 CLL 细胞具有高度活性(相对 IC50 为 35nM),并通过抑制 HIF-1α± 和扰乱细胞内氧化还原稳态发挥作用。 | |||
T8287 |
Edpetiline
Sipeimine-3β-D-glucoside,西贝母碱苷 |
Others | Others |
Sipeimine-3β-D-glucoside 是一种来自 P.eduardi 的主要生物碱。它具有显著的抗炎活性。 | |||
T0895 |
Oxytetracycline
土霉素,Terramycin |
ribosome; Endogenous Metabolite; Antibacterial; Antibiotic; HSV | Metabolism; Microbiology/Virology |
Oxytetracycline (Terramycin) 是一种四环素类抗生素。它强力抑制革兰氏阴性和革兰氏阳性细菌。它是一种蛋白质合成抑制剂,可阻止 aminoacil-tRNA 与复杂的核糖体 RNA 结合,具有抗 HSV-1的活性。 | |||
T0268 |
Lobeline hydrochloride
盐酸洛贝林,α-Lobeline hydrochloride,L-Lobeline hydrochloride |
AChR | Neuroscience |
Lobeline hydrochloride (α-Lobeline hydrochloride) 是一种烟碱样受体激动剂,是神经元烟碱受体α3β2和α4β2拮抗剂。 | |||
T0480 |
Doxofylline
Doxophylline,多索茶碱 |
PDE; Adenosine Receptor | GPCR/G Protein; Metabolism; Neuroscience |
Doxofylline (Doxophylline) 是腺苷 A1 受体拮抗剂,且能抑制磷酸二酯酶 IV,用于治疗哮喘。 | |||
T25664 |
Lepidiline A
Macaline A |
Others | Others |
Lepidiline A (Macaline A) 是一种具有抗炎症活性的黄酮木质素。Lepidiline A 对HL-60细胞具有细胞毒活性,IC50值为 32.3 μM。它是从芸苔科植物Lepidium meyenii Walpers 的活性成分,可改善小鼠内源性性激素的平衡,提高果蝇的繁殖力。Lepidiline A 靶向HSD17B1基因的机制来增强酶的活性,提高性激素的生物转化效率,提高生殖能力。Lepidiline A 具有抗癌活性。 | |||
T6805 |
Choline bitartrate
2,3,4-trihydroxy-4-oxobutanoate,2-hydroxyethyl(trimethyl)azanium,酒石酸氢胆碱 |
Others; AChR | Neuroscience; Others |
Choline bitartrate (2-hydroxyethyl(trimethyl)azanium) 是一种存在于食物中的营养胆碱,可影响肝脏疾病、动脉粥样硬化和神经系统疾病等疾病。它是神经递质乙酰胆碱的前体,作为甲基供体参与各种代谢过程和脂质代谢。 | |||
T1681 |
Aminophylline
氨茶碱,Phyllocontin |
PDE; Adenosine Receptor | GPCR/G Protein; Metabolism; Neuroscience |
Aminophylline (Phyllocontin) 是一种竞争性非选择性磷酸二酯酶抑制剂,具有支气管扩张作用。它是竞争性的腺苷受体拮抗剂,有用于哮喘研究的潜力。 | |||
T5693 |
Pyrroloquinoline quinone disodium salt
吡咯喹啉醌二钠盐,Methoxatin disodium salt |
Others; Endogenous Metabolite | Metabolism; Others |
Pyrroloquinoline quinone disodium salt (Methoxatin disodium salt) 一种阴离子型氧化还原循环原醌,作为氧化还原辅助因子。它是从嗜甲基细菌的培养物中分离的,也存在于哺乳动物的组织。它是哺乳动物的必需营养素,对免疫功能很重要。 | |||
T6751 |
Acetylcholine iodide
Acetylcolina |
Others | Others |
Acetylcholine iodide (Acetylcolina) 是一种在中枢和外周神经系统中常见的神经递质。 | |||
T3054 |
Daurisoline
蝙蝠葛苏林碱,(R,R)-Daurisoline |
Others; Potassium Channel; Autophagy | Autophagy; Membrane transporter/Ion channel; Others |
Daurisoline ((R,R)-Daurisoline) 是一种 hERG 抑制剂,也是一种自噬阻滞剂。 | |||
T3S0629 |
Delsoline
Belsoline,硬飞燕草碱 |
Others | Others |
Delsoline (Belsoline) 是一种还亮草的主要生物碱,具有类似箭毒的效果和神经节阻滞作用,可用于肌肉紧张或运动过度的缓解。其中还亮草具有祛风除湿,止痛,活络的功效,可用于风湿,偏瘫,消化不良和咳嗽的研究。 | |||
TN1078 |
Seneciphylline
千里光菲灵碱,千里光非灵 |
P450; GST | Metabolism; oxidation-reduction |
Seneciphylline 是一种有毒的吡咯烷核生物碱,存在于千里光植物中。它显著增加了环氧水合酶和谷胱甘肽-S-转移酶的特性,但导致细胞色素 P-450 和相关单加氧酶特性的抑制。 | |||
TN7193 |
2,4,6-Triphenylaniline
2,4,6-Triphenyl-anilin,2,4,6-三苯基苯胺,5'-Phenyl-[1,1':3',1''-terphenyl]-2'-amine |
Others | Others |
2,4,6-Triphenylaniline (5'-Phenyl-[1,1':3',1''-terphenyl]-2'-amine) 是一种海洋来源的天然产物,存在于Alternaria longipes。 | |||
T4S0537 |
Neoline
Bullatine B,雪上一枝蒿乙素 |
Others; Sodium Channel | Membrane transporter/Ion channel; Others |
Neoline 是一种乌头根 (PA) 的活性成分,可改善奥沙利铂引起的小鼠周围神经病变。Neoline 通对Nav1.7 电压门控钠通道电流 (VGSC)有抑制作用。它可用作标记化合物,从而测定用于研究神经性疼痛的 PA 产品的质量。 | |||
T38095 |
Acetylvaline
Ac-Val-OH |
Others | Others |
Acetylvaline (Ac-Val-OH) 可作为 2 型糖尿病、肥胖和视网膜病变等疾病的一个指标。 | |||
T2809 |
(R)-Fangchinoline
防己醇灵,Thaligine,(+)-Thalrugosine,Demethyl tetrandrine |
FAK; Antibacterial; Antibiotic | Angiogenesis; Cytoskeletal Signaling; Microbiology/Virology; Tyrosine Kinase/Adaptors |
(R)-Fangchinoline ((+)-Thalrugosine) 是一种来自Stephania 属的生物碱,具有抗菌和降血压活性。它可用作中药,可用于发烧,腹泻,消化不良和泌尿疾病的研究。 | |||
T5S2358 |
Dehydrocorydaline
Dehydrocorydalin,脱氢紫堇碱,13-Methylpalmatine |
BCL; PARP; p38 MAPK; Caspase; Parasite; Autophagy | Apoptosis; Autophagy; Chromatin/Epigenetic; DNA Damage/DNA Repair; MAPK; Microbiology/Virology; Proteases/Proteasome |
Dehydrocorydaline (13-Methylpalmatine) 是一种生物碱。它调节Bax,Bcl-2蛋白表达,激活caspase-7,caspase-8,并使PARP 失活。它能增强p38 MAPK 活化,具有抗炎、抗癌等功效。它具有强大的抗疟疾作用,并具低细胞毒性。 | |||
TN7150 |
Pygmaniline B
1,3-Bis-(2,4-dimethoxy-phenyl)-urea,1,3-bis(2,4-dimethoxyphenyl)urea,N,N'-bis(2,4-dimethoxyphenyl)urea |
Others | Others |
Pygmaniline B (1,3-bis(2,4-dimethoxyphenyl)urea) 是一种海洋来源的天然产物,存在于Lichina pygmaea。 | |||
TN2213 |
Imperialine 3-β-D-glucoside
Sipeimine-3-beta-D-glucoside,西贝母碱苷 |
Others | Others |
Imperialine 3-β-D-glucoside (Sipeimine-3-beta-D-glucoside) 是 Imperialine 的糖苷。它对多重耐药肿瘤细胞表现出抗肿瘤特性。 | |||
T4780 |
Quinoline-2-carboxylic acid
喹哪啶酸,Quinaldic acid,RARECHEM AL BO 1348 |
Others; Endogenous Metabolite | Metabolism; Others |
Quinaldic acid 是内源性代谢产物的一种。Quinaldic acid 是一种金属螯合剂。 | |||
T5257 |
L-Homocitrulline
高瓜氨酸,Homo-L-citrulline,Homocitrulline |
Others; Endogenous Metabolite | Metabolism; Others |
L-Homocitrulline (Homocitrulline) 是一种代谢物,可在尿素循环障碍患者的尿液中大量检测到。在某些情况下,由于尿素循环的鸟氨酸供应耗尽而导致的氨甲酰磷酸酯的积累可能是 L-Homocitrulline 和高精氨酸合成增强的原因。 | |||
T4813 |
L-Citrulline
|
Endogenous Metabolite | Metabolism |
L-Citrulline 是一种氨基酸,源自于精氨酸-瓜氨酸途径获得的 l-精氨酸,或脯氨酸、谷氨酰胺和谷氨酸盐的分解代谢过程中产生的鸟氨酸。 | |||
T2803 |
Monocrotaline
野百合碱,Crotaline |
TGF-beta/Smad | Stem Cells |
Monocrotaline (Crotaline) 是一种吡咯里西啶生物碱,从猪屎豆植物的种子中提取得到,可诱导啮齿动物产生肺动脉高血压。 | |||
T1039 |
Choline chloride
Biocolina,Biocoline,Hepacholine,氯化胆碱 |
AChR | Neuroscience |
Choline chloride (Biocoline) 是一种必需营养素,可激活 α7 烟碱受体,具有抗炎、镇痛的活性。对动脉粥样硬化、神经系统疾病和肝脏疾病等具有影响。 | |||
T37784 |
2,6-Dimethylquinoline
|
P450 | Metabolism |
2,6-Dimethylquinoline 是一种从前胡根中提取的天然产物。2,6-Dimethylquinoline 是 CYP1A2 和 CYP2B6 的抑制剂,IC50 分别为 3.3 和 480 µM。 | |||
T10990 |
Dehydrocorydaline chloride
盐酸脱氢紫堇碱,13-Methylpalmatine chloride |
BCL; PARP; p38 MAPK; Caspase; Parasite; Autophagy | Apoptosis; Autophagy; Chromatin/Epigenetic; DNA Damage/DNA Repair; MAPK; Microbiology/Virology; Proteases/Proteasome |
Dehydrocorydaline chloride (13-Methylpalmatine chloride) 是生物碱。Dehydrocorydaline 调节 Bax,Bcl-2蛋白表达;激活 caspase-7,caspase-8,并使 PARP 失活。它能增强 p38 MAPK 活化,具有抗炎、抗癌等功效。它具有强大的抗疟疾作用,并具低细胞毒性。 | |||
T1221 |
Acetylcholine chloride
ACh chloride,Pilofrin,氯化乙酰胆碱 |
Calcium Channel; Endogenous Metabolite; AChR | Membrane transporter/Ion channel; Metabolism; Neuroscience |
Acetylcholine chloride (Pilofrin) 是一种神经递质,是胆碱能激动剂,通过刺激烟碱乙酰胆碱受体调节多巴胺能神经元活性,在体外抑制 p53 突变肽的聚集。 | |||
T5S2360 |
Corydaline
Corydalin,紫堇碱,延胡索甲素,(+)-Corydaline |
P450; Virus Protease; Opioid Receptor; AChE | Endocrinology/Hormones; GPCR/G Protein; Metabolism; Microbiology/Virology; Neuroscience |
Corydaline (Corydalin) 是从 Corydalis yanhusuo 提取的一种异喹啉生物碱,是一种新型促动力植物药的主要活性成分之一。它促进胃排空和小肠转运,促进胃的调节,具有抗乙酰胆碱酯酶、抗过敏和镇痛活性。 | |||
T5692 |
Pyrroloquinoline quinone
|
Others; Endogenous Metabolite | Metabolism; Others |
Pyrroloquinoline quinone 是氧化还原辅助因子,一种阴离子型氧化还原循环原醌。它是哺乳动物的必需营养素,对免疫功能很重要。它是从嗜甲基细菌的培养物中分离的,也存在于哺乳动物的组织。 | |||
T0136 |
Citicoline
CDP-Choline,Citicholine,尼古林,cytidine 5'-diphosphocholine,cytidine diphosphate-choline |
Apoptosis; Dopamine Receptor; Endogenous Metabolite | Apoptosis; GPCR/G Protein; Metabolism; Neuroscience |
Citicoline (CDP-Choline) 是一种合成细胞膜组分磷脂酰胆碱的中间体,有神经保护作用。 | |||
T6624 |
Oxytetracycline Dihydrate
土霉素二水合物,地霉素,Terramycin Dihydrate |
Others; Endogenous Metabolite; Antibacterial; Antibiotic; HSV | Metabolism; Microbiology/Virology; Others |
Oxytetracycline Dihydrate (Terramycin Dihydrate) 是一种四环素类抗生素,可抑制革兰氏阴性和革兰氏阳性细菌。它是一种蛋白质合成抑制剂,可阻止 aminoacil-tRNA 与复杂的核糖体 RNA 结合,还具有抗 HSV-1的活性。 | |||
T37512 |
cis-4-Hydroxy-L-proline
|
Endogenous Metabolite | Metabolism |
cis-4-Hydroxy-L-proline 是脯氨酸的一种类似物,抑制胶原蛋白的产生。它通过阻止三层螺旋胶原在细胞层上的沉积从而抑制成纤维细胞的生长。它还可抑制原发性N-亚硝基甲基脲诱导的大鼠乳腺肿瘤的生长。 | |||
T2O2776 |
L-Valine
|
Others; Endogenous Metabolite | Metabolism; Others |
L-Valine 是蛋白二十种氨基酸中的其中一种。它是必需氨基酸。 | |||
T6S0657 |
Isorhynchophylline
IsoRhy,异钩藤碱,Isorhyncophylline,Isorhychophylline,7-Isorhyncophylline |
Others | Others |
Isorhynchophylline (7-Isorhyncophylline) 是一种分离自钩藤中的生物碱类化合物,具有舒张血管、降血压、保护神经免于局部缺血造成损伤的作用。 | |||
T8713 |
1-Oleoyl-sn-glycero-3-phosphocholine
|
Others | Others |
1-Oleoyl-sn-glycero-3-phosphocholine 是分析溶血卵磷脂的参考。 | |||
T68953 |
Arecoline
|
Reactive Oxygen Species; AChR | Immunology/Inflammation; Metabolism; Neuroscience; NF-κB |
Arecoline 是一种来自棕榈科植物槟榔的天然生物碱,是有效的烟碱和毒蕈碱乙酰胆碱受体的部分激动剂。Arecoline 具有抗焦虑和抗寄生虫活性,可诱导氧化应激,可用于研究阿尔茨海默病和老年性痴呆。 | |||
T2797 |
Harmaline
|
Others | Others |
Harmaline 是一种来自harmala 生物碱和β-咔啉的荧光精神活性吲哚生物碱。它是harmine 的还原氢化形式。 | |||
T1687L |
Doxycycline (hyclate)
Doxycycline hydrochloride hemiethanolate hemihydrate,盐酸强力霉素,WC2031,Doxycycline hyclate |
MMP; ribosome; Antibacterial; Antibiotic | Microbiology/Virology; Proteases/Proteasome |
Doxycycline hyclate (WC2031) 属于四环素类抗生素,是一种广谱的金属蛋白酶 (MMP) 抑制剂,具有口服活性。Doxycycline hyclate 具有抗菌活性和抗肿瘤活性。 | |||
TN2549 |
1-Methoxycarbonyl-β-carboline
1-Methoxycarbonyl-beta-carboline |
Others | Others |
1-Methoxycarbonyl-β-carboline (1-Methoxycarbonyl-beta-carboline) 是一种来自 Ailanthus altissima 的生物碱。 | |||
TN6739 |
Angoline
6-Methoxyldihydrochelerythrine |
IL Receptor; STAT | Immunology/Inflammation; JAK/STAT signaling; Stem Cells |
Angoline (6-Methoxyldihydrochelerythrine) 是选择性 IL6/STAT3信号通路的抑制剂,IC50为 11.56 μM。它抑制 STAT3 磷酸化及其靶基因表达,并抑制癌细胞增殖。 | |||
T0912 |
Tetracycline hydrochloride
NCI-c55561,盐酸四环素,Tetracycline HCl |
ribosome; Antibacterial; Antibiotic | Microbiology/Virology |
Tetracycline hydrochloride (NCI-c55561) 是一种广谱抗生素,抑制多种革兰氏阳性和革兰氏阴性细菌。 | |||
T9525 |
1,2-Dimyristoyl-sn-glycero-3-phosphocholine
DMPC,1,2-DIMYRISTOYL-SN-GLYCERO-3-PHOSPHOCHOL,二肉豆蔻酰磷脂酰胆碱(DMPC) |
Others | Others |
1,2-Dimyristoyl-sn-glycero-3-phosphocholine (DMPC) 是一种用于脂质体和脂质双层的合成磷脂。它可用于脂质单层和双层的研究。 | |||
T73602 |
Phosphorylcholine
Phosphocholine |
Endogenous Metabolite | Metabolism |
Phosphorylcholine 广泛存在于生物界,是存在于真核生物膜中的磷脂,也存在于与真核生物相关联的共生菌或致病菌中。Phosphorylcholine 具有免疫调节特性,可用于研究动脉粥样硬化。 | |||
T0281 |
Meclocycline sulfosalicylate salt
磺基水杨酸甲氯环素,Meclutin,Mecloderm,甲环素磺基水杨酸盐,Meclan Cream |
Antibacterial; Antibiotic | Microbiology/Virology |
Meclocycline sulfosalicylate salt (Mecloderm) 是一种具有广谱抗菌活性的四环素抗生素,可预防皮肤细菌感染。 | |||
T4550 |
Ajmaline
Cardiorythmine,Raugalline,阿义吗啉,阿义马林,Tachmalin,(+)-Ajmaline |
Sodium Channel | Membrane transporter/Ion channel |
Ajmaline (Cardiorythmine) 是一种钠通道阻断剂,属于1A 类抗心律失常剂。Ajmaline 阻断 HERG 电流,在 HEK 细胞的 IC50为 1 μM,爪蟾卵母细胞的IC50为 42.3 μM。Ajmaline 在室性心动过速方面具有研究价值。 | |||
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Cat. No. | Product Name | Species | Expression System |
---|---|---|---|
TMPH-02759 |
LIRE1 Protein, Mouse, Recombinant (His & Myc)
Transposase element L1Md-A101/L1Md-A102/L1Md-A2,LINE |
Mouse | E. coli |
LIRE1 Protein, Mouse, Recombinant (His & Myc) is expressed in E. coli. | |||
TMPH-01381 |
GDNF Protein, Human, Recombinant (His & SUMO)
Astrocyte-derived trophic factor,GDNF,Glial cell line |
Human | E. coli |
Neurotrophic factor that enhances survival and morphological differentiation of dopaminergic neurons and increases their high-affinity dopamine uptake. GDNF Protein, Human, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 31.1 kDa and the accession number is P39905. | |||
TMPY-00663 |
Alkaline Phosphatase/ALPL Protein, Human, Recombinant (His)
alkaline phosphatase, liver/bone/kidney,TNSALP,AP-T... |
Human | HEK293 Cells |
Alkaline Phosphatase/ALPL Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 55 kDa and the accession number is A0A024RAB4. | |||
TMPK-00639 |
Alkaline Phosphatase (Germ type) /ALPG Protein, Rat, Recombinant (His)
GCAP,ALP-1,Alkaline Phosphatase,ALPPL2,PLAP-like,AL... |
Rat | HEK293 Cells |
Alkaline phosphatase can be considered "our favorite enzyme" for reasons apparent to those who diagnose and treat metabolic bone diseases or who study skeletal biology. Few might know, however, that alkaline phosphatase likely represents the most frequently assayed enzyme in all of medicine. Elevated activity in the circulation is universally recognized as a marker for skeletal or hepatobiliary disease. Alkaline Phosphatase (Germ type) /ALPG Protein, Rat, Recombinant (His) is expressed in HEK293... | |||
TMPY-00570 |
Alkaline Phosphatase/PLAP Protein, Human, Recombinant (His)
ALPI,PALP,PLAP,PLAP-1,alkaline phosphatase, placent... |
Human | P. pastoris (Yeast) |
Most importantly, placental alkaline phosphatase (ALPP), an ectoenzyme that locates on cell surface with catalytic domains outside the plasma membrane and is overexpressed on many cancer cells, dephosphorylate the d-tyrosine phosphates on the surface of the magnetic nanoparticle and enable the magnetic nanoparticles to adhere selectively to the cancer cells, such as HeLa cells. Placental alkaline phosphatase (PLAP), encoded by the ALPP gene, is produced by the fetal side of the placenta. | |||
TMPY-02650 |
Alkaline phosphatase Protein, Human, Recombinant (His)
IAP,alkaline phosphatase, intestinal |
Human | HEK293 Cells |
Alkaline phosphatase Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 54 kDa and the accession number is P09923. | |||
TMPY-01693 |
Butyrylcholinesterase Protein, Human, Recombinant (His)
CHE1,E1,butyrylcholinesterase,CHE2 |
Human | HEK293 Cells |
Butyrylcholinesterase Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 66.5 kDa and the accession number is P06276. | |||
TMPY-00446 |
Alkaline Phosphatase/ALPL Protein, Mouse, Recombinant (His)
TNSALP,Akp2,alkaline phosphatase, liver/bone/kidney... |
Mouse | HEK293 Cells |
Alkaline Phosphatase/ALPL Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 55 kDa and the accession number is B7XGA6. | |||
TMPY-04299 |
West Nile Virus (WNV) (lineage 1, strain NY99) E/Envelope Protein (His)
WNV-E Protein |
WNV | P. pastoris (Yeast) |
West Nile Virus (WNV) (lineage 1, strain NY99) E/Envelope Protein (His) is expressed in yeast with His tag. The predicted molecular weight is 12.9 kDa and the accession number is ABA62343.1. | |||
TMPY-06524 |
EGFR Protein, Feline, Recombinant (His)
epidermal growth factor receptor |
Feline | Baculovirus Insect Cells |
EGFR Protein, Feline, Recombinant (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 70.18 kDa and the accession number is A0A337S424. | |||
TMPY-02397 |
IL-1 beta/IL-1F2 Protein, Feline, Recombinant
interleukin 1, beta,白细胞介素,白介素,interleukin 1, β,IL-1 β |
Feline | E. coli |
IL-1 beta/IL-1F2 Protein, Feline, Recombinant is expressed in E. coli expression system. The predicted molecular weight is 17.5 kDa and the accession number is P41687. | |||
TMPK-00684 |
Alkaline phosphatase (Intestinal type) /ALPI Protein, Mouse, Recombinant (His)
IAP,TNSALP,APTNAP,FLJ40094,AP-TNAP,MGC161443,TNAP,Akp2,HOPS,... |
Mouse | HEK293 Cells |
Alkaline phosphatase can be considered "our favorite enzyme" for reasons apparent to those who diagnose and treat metabolic bone diseases or who study skeletal biology. Few might know, however, that alkaline phosphatase likely represents the most frequently assayed enzyme in all of medicine. Elevated activity in the circulation is universally recognized as a marker for skeletal or hepatobiliary disease. Alkaline phosphatase (Intestinal type) /ALPI Protein, Mouse, Recombinant (His) is expressed i... | |||
TMPK-00855 |
Alkaline Phosphatase (Germ type) /ALPG Protein, Mouse, Recombinant (His)
Alkaline Phosphatase,Alppl2,Akp5,Alpg,Alkaline<... |
Mouse | HEK293 Cells |
Alkaline phosphatase can be considered "our favorite enzyme" for reasons apparent to those who diagnose and treat metabolic bone diseases or who study skeletal biology. Few might know, however, that alkaline phosphatase likely represents the most frequently assayed enzyme in all of medicine. Elevated activity in the circulation is universally recognized as a marker for skeletal or hepatobiliary disease. Alkaline Phosphatase (Germ type) /ALPG Protein, Mouse, Recombinant (His) is expressed in HEK2... | |||
TMPH-03234 |
Acetylcholinesterase Protein, Rat, Recombinant (His)
AChE,EC:3.1.1.7 |
Rat | E. coli |
Terminates signal transduction at the neuromuscular junction by rapid hydrolysis of the acetylcholine released into the synaptic cleft. Acetylcholinesterase Protein, Rat, Recombinant (His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 68.9 kDa and the accession number is P37136. | |||
TMPH-02343 |
Hypodermin-A Protein, Hypoderma lineatum, Recombinant (His)
Hypodermin-A |
Hypoderma lineatum | E. coli |
Specificity, limited to carboxyl side of arginine residue in B-chain of insulin. | |||
TMPY-00525 |
IL-10 Protein, Feline, Recombinant
interleukin 10 |
Feline | E. coli |
IL-10 Protein, Feline, Recombinant is expressed in E. coli expression system. The predicted molecular weight is 18.9 kDa and the accession number is P55029.2. | |||
TMPY-01596 |
Butyrylcholinesterase Protein, Mouse, Recombinant (His)
C730038G20Rik,butyrylcholinesterase |
Mouse | HEK293 Cells |
Butyrylcholinesterase Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 66.7 kDa and the accession number is Q03311. | |||
TMPH-00352 |
CKM Protein, Feline, Recombinant
M-CK,Creatine kinase M-type,Creatine phosphokinase M-type,CK... |
Feline | E. coli |
CKM Protein, Feline, Recombinant is expressed in E. coli expression system. The predicted molecular weight is 27.9 kDa and the accession number is M3VYX8. | |||
TMPH-00355 |
Major allergen I polypeptide chain 1 Protein, Feline, Recombinant (His & Myc)
Allergen Cat-1,Allergen Fel d I-A,AG4,Major allergen I polyp... |
Feline | E. coli |
Major allergen I polypeptide chain 1 Protein, Feline, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 15.3 kDa and the accession number is P30438. | |||
TMPH-00757 |
Reticuline oxidase Protein, Eschscholzia californica, Recombinant (His)
BBE1,Tetrahydroprotoberberine synthase,Berberine bridge-form... |
Eschscholzia californica | E. coli |
Essential to the formation of benzophenanthridine alkaloids in the response of plants to pathogenic attack. Catalyzes the stereospecific conversion of the N-methyl moiety of (S)-reticuline into the berberine bridge carbon of (S)-scoulerine. | |||
TMPY-06335 |
SARS-CoV-2 B.1.1.529 sublineage BA.2 (Omicron) Spike RBD Protein (His)
|
SARS-CoV-2 | HEK293 Cells |
SARS-CoV-2 B.1.1.529 sublineage BA.2 (Omicron) Spike RBD Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 26.71 kDa and the accession number is YP_009724390.1. | |||
TMPY-04735 |
West Nile Virus (WNV) (lineage 1, strain NY99) NS1 Protein (His)
interferon regulatory factor 3 |
WNV | HEK293 Cells |
West Nile Virus (WNV) (lineage 1, strain NY99) NS1 Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 42.1 kDa and the accession number is YP_001527881.1. | |||
TMPH-00354 |
CSF1R Protein, Feline, Recombinant (His & SUMO)
FMS,M-CSF-R,CSF-1-R,CSF1R,Proto-oncogene c-Fms,CSF-1R,CD115,... |
Feline | E. coli |
CSF1R Protein, Feline, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 70.8 kDa and the accession number is P13369. | |||
TMPH-03236 |
Alkaline phosphatase/ALPL Protein, Rat, Recombinant (His & SUMO)
ALPase,PiALP |
Rat | E. coli |
Alkaline phosphatase/ALPL Protein, Rat, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 69.5 kDa and the accession number is P08289. | |||
TMPH-03161 |
Alkaline Phosphatase Protein, Prevotella intermedia, Recombinant (GST & His & Myc)
PiALP,ALPase |
Prevotella intermedia | E. coli |
Acts against tyrosine-phosphatases. Alkaline Phosphatase Protein, Prevotella intermedia, Recombinant (GST & His & Myc) is expressed in E. coli expression system with N-10xHis-GST and C-Myc tag. The predicted molecular weight is 32.1 kDa and the accession number is P81800. | |||
TMPY-00594 |
Alkaline Phosphatase/ALPL Protein, Mouse, Recombinant (hFc)
Akp-2,TNSALP,TNAP,alkaline phosphatase, liver/bone/... |
Mouse | HEK293 Cells |
Alkaline Phosphatase/ALPL Protein, Mouse, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 80.3 kDa and the accession number is B7XGA6. | |||
TMPY-06467 |
SARS-CoV-2 (B.1.1.529 sublineage BA.2) Spike S1 Protein (His)
|
SARS-CoV-2 | HEK293 Cells |
SARS-CoV-2 (B.1.1.529 sublineage BA.2) Spike S1 Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 76.39 kDa and the accession number is YP_009724390.1. | |||
TMPY-01742 |
Acetylcholinesterase Protein, Mouse, Recombinant (His)
Acre,Chrne,acetylcholinesterase (Yt blood group) |
Mouse | HEK293 Cells |
Acetylcholinesterase, also known as ACHE, is an enzyme that degrades (through its hydrolytic activity) the neurotransmitter acetylcholine, producing choline and an acetate group. Acetylcholinesterase plays a crucial role in nerve impulse transmission at cholinergic synapses by rapid hydrolysis of the neurotransmitter acetylcholine (ACh). ACHE appears to be a potential therapeutic target at muscle injuries including organophosphate myopathy. It is an externally oriented membrane-bound enzyme and ... | |||
TMPK-00803 |
Alkaline Phosphatase (Germ type) /ALPG Protein, Human, Recombinant (His)
ALPG,ALPPL,Alkaline phosphatase, placental-like,Alk... |
Human | HEK293 Cells |
Alkaline phosphatase can be considered "our favorite enzyme" for reasons apparent to those who diagnose and treat metabolic bone diseases or who study skeletal biology. Few might know, however, that alkaline phosphatase likely represents the most frequently assayed enzyme in all of medicine. Elevated activity in the circulation is universally recognized as a marker for skeletal or hepatobiliary disease. Alkaline Phosphatase (Germ type) /ALPG Protein, Human, Recombinant (His) is expressed in HEK2... | |||
TMPK-00796 |
Alkaline phosphatase (Intestinal type) /ALPI Protein, Human, Recombinant (His & Flag)
FLJ40094,ALPI,APTNAP,EC 3.1.3.1,AP-TNAP,IAP,TNAP,HOPS,FLJ930... |
Human | HEK293 Cells |
Alkaline phosphatase can be considered "our favorite enzyme" for reasons apparent to those who diagnose and treat metabolic bone diseases or who study skeletal biology. Few might know, however, that alkaline phosphatase likely represents the most frequently assayed enzyme in all of medicine. Elevated activity in the circulation is universally recognized as a marker for skeletal or hepatobiliary disease. Alkaline phosphatase (Intestinal type) /ALPI Protein, Human, Recombinant (His & Flag) is expr... | |||
TMPK-01326 |
Alkaline Phosphatase (Placental type) /ALPP Protein, Cynomolgus, Recombinant (His)
Alkaline phosphatase,PLAP,PLAP-1,ALPP |
Cynomolgus | HEK293 Cells |
Alkaline phosphatase can be considered "our favorite enzyme" for reasons apparent to those who diagnose and treat metabolic bone diseases or who study skeletal biology. Few might know, however, that alkaline phosphatase likely represents the most frequently assayed enzyme in all of medicine. Elevated activity in the circulation is universally recognized as a marker for skeletal or hepatobiliary disease. Alkaline Phosphatase (Placental type) /ALPP Protein, Cynomolgus, Recombinant (His) is express... | |||
TMPK-00801 |
Alkaline Phosphatase (Germ type) /ALPG Protein, Human, Recombinant (His & Avi), Biotinylated
ALPPL2,PLAP-like,GCAP,ALPG,Alkaline phosphatase, pl... |
Human | HEK293 Cells |
Alkaline phosphatase can be considered "our favorite enzyme" for reasons apparent to those who diagnose and treat metabolic bone diseases or who study skeletal biology. Few might know, however, that alkaline phosphatase likely represents the most frequently assayed enzyme in all of medicine. Elevated activity in the circulation is universally recognized as a marker for skeletal or hepatobiliary disease. Alkaline Phosphatase (Germ type) /ALPG Protein, Human, Recombinant (His & Avi), Biotinylated ... | |||
TMPK-00802 |
Alkaline Phosphatase (Germ type) /ALPG Protein, Human, Recombinant (hFc)
GCAP,ALPPL,Alkaline phosphatase, placental-like,Alk... |
Human | HEK293 Cells |
Alkaline phosphatase can be considered "our favorite enzyme" for reasons apparent to those who diagnose and treat metabolic bone diseases or who study skeletal biology. Few might know, however, that alkaline phosphatase likely represents the most frequently assayed enzyme in all of medicine. Elevated activity in the circulation is universally recognized as a marker for skeletal or hepatobiliary disease. Alkaline Phosphatase (Germ type) /ALPG Protein, Human, Recombinant (hFc) is expressed in HEK2... | |||
TMPH-02342 |
Collagenase Protein, Hypoderma lineatum, Recombinant (His & Myc)
Collagenase,HC,Hypodermin C |
Hypoderma lineatum | E. coli |
This enzyme is a serine protease capable of degrading the native triple helix of collagen. Also cleaves the B chain of insulin at the 15-Leu-|-Try-16 and 22-Arg-|-Gly-23 bonds. Hydrolyzes casein, but not Px-Pro-Leu-Gly-Pro-DArg, BzArgNHPh, AcTyrNHPh, 2-naphthyl phosphate, 2-naphthyl butyrate, 2-naphthyl caprylate, 2-naphthyl myristate, L-leucine 2-2-naphthylamide, L-valine 2-naphthylamide, L-cysteine 2-naphthylamide or L-glutarylphenylalanine 2-naphthylamide. | |||
TMPH-00358 |
SAA1 Protein, Feline, Recombinant (B2M & His)
Serum amyloid A protein,SAA1 |
Feline | E. coli |
Major acute phase reactant. Apolipoprotein of the HDL complex. SAA1 Protein, Feline, Recombinant (B2M & His) is expressed in E. coli expression system with N-6xHis-B2M tag. The predicted molecular weight is 24.1 kDa and the accession number is P19707. | |||
TMPH-00351 |
Fel d 4 Protein, Feline, Recombinant (His & SUMO)
Allergen Fel d 4 |
Feline | E. coli |
May be a pheromone carrier. Acts as a kairomone, detected by the prey vomeronasal organ and inducing fear reactions in mice. Fel d 4 Protein, Feline, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 35.7 kDa and the accession number is Q5VFH6. | |||
TMPH-02344 |
Hypodermin-B Protein, Hypoderma lineatum, Recombinant (His & Myc)
Hypodermin-B |
Hypoderma lineatum | E. coli |
Protease that shows preferential cleavage after Arg and Lys residues. | |||
TMPH-00356 |
PAI-1 Protein, Feline, Recombinant
PAI-1,Endothelial plasminogen activator inhibitor,Serpin E1,... |
Feline | E. coli |
PAI-1 Protein, Feline, Recombinant is expressed in E. coli expression system. The predicted molecular weight is 29.7 kDa and the accession number is A9NJ78. | |||
TMPH-00353 |
GDF8 Protein, Feline, Recombinant
Myostatin,MSTN,Growth/differentiation factor 8 |
Feline | E. coli |
GDF-8 Protein, Feline, Recombinant is expressed in E. coli expression system. The predicted molecular weight is 40.7 kDa and the accession number is M3WPT7. | |||
TMPY-02713 |
Alkaline phosphatase Protein, Human, Recombinant (hFc)
alkaline phosphatase, intestinal,IAP |
Human | HEK293 Cells |
Alkaline phosphatase Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 79.5 kDa and the accession number is P09923. | |||
TMPY-06493 |
EGF Protein, Feline, Recombinant (hFc)
表皮生长因子,epidermal growth factor |
Feline | HEK293 Cells |
EGF Protein, Feline, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 34.63 kDa and the accession number is NP_001009381.1. | |||
TMPY-04787 |
West Nile Virus (WNV) (lineage 2, strain Nea Santa-Greece-2010) E/Envelope Protein (His)
WNV-E Protein |
WNV | P. pastoris (Yeast) |
West Nile Virus (WNV) (lineage 2, strain Nea Santa-Greece-2010) E/Envelope Protein (His) is expressed in yeast with His tag. The predicted molecular weight is 12.9 kDa and the accession number is AED99787.1. | |||
TMPY-06473 |
SARS-CoV-2 (B.1.1.529 sublineage BA.2) Nucleocapsid Protein (His)
|
SARS-CoV-2 | E. coli |
SARS-CoV-2 (B.1.1.529 sublineage BA.2) Nucleocapsid Protein (His) is expressed in E. coli expression system with His tag. The predicted molecular weight is 46.38 kDa and the accession number is YP_009724397.2. | |||
TMPK-00804 |
Alkaline Phosphatase (Germ type) /ALPG Protein, Human, Recombinant (mFc)
GCAP,Alkaline Phosphatase,PLAP-like,Alkaline |
Human | HEK293 Cells |
Alkaline phosphatase can be considered "our favorite enzyme" for reasons apparent to those who diagnose and treat metabolic bone diseases or who study skeletal biology. Few might know, however, that alkaline phosphatase likely represents the most frequently assayed enzyme in all of medicine. Elevated activity in the circulation is universally recognized as a marker for skeletal or hepatobiliary disease. Alkaline Phosphatase (Germ type) /ALPG Protein, Human, Recombinant (mFc) is expressed in HEK2... | |||
TMPJ-00784 |
Alkaline Phosphatase Protein, Human, Recombinant (aa 23-506, His)
Alkaline phosphatase Regan isozyme,placental type,P... |
Human | HEK293 Cells |
ALPP is a membrane protein and exits as a homodimer. ALPP is expressed only in normal term placenta, endocervix and fallopian tube and also in ovarian and proximal gastrointestinal tumors. It has been shown to play a role in a number of processes including cell signaling, long-term potentiation, and cell adhesion, however, the best known and most commonly studied role is implicated in Alzheimer's research. | |||
TMPH-00350 |
Adiponectin Protein, Feline, Recombinant
apM-1,30 kDa adipocyte complement-related protein,APM1,ACRP3... |
Feline | E. coli |
Adiponectin Protein, Feline, Recombinant is expressed in E. coli expression system. The predicted molecular weight is 24.9 kDa and the accession number is A4PB30. | |||
TMPH-00513 |
Proline iminopeptidase Protein, Elizabethkingia meningoseptica, Recombinant (His & Myc)
Proline iminopeptidase,Prolyl aminopeptidase,fpaP |
Elizabethkingia meningoseptica | E. coli |
Releases the N-terminal proline from various substrates. Cleaves specifically Pro-betaNA and small peptides containing proline at the amino terminal. No activity against hydroxyproline-betaNA. Proline iminopeptidase Protein, Elizabethkingia meningoseptica, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 41.6 kDa and the accession number is O05420. | |||
TMPH-00357 |
SAA1 Protein, Feline, Recombinant (His)
Serum amyloid A protein,SAA1 |
Feline | P. pastoris (Yeast) |
Major acute phase reactant. Apolipoprotein of the HDL complex. SAA1 Protein, Feline, Recombinant (His) is expressed in yeast with N-6xHis tag. The predicted molecular weight is 12.1 kDa and the accession number is P19707. | |||
TMPK-00925 |
Noggin/NOG Protein, Mouse, Recombinant
NOG,SYM1,SYNS1,Noggin |
Mouse | HEK293 Cells |
Noggin is an antagonist of bone morphogenetic proteins (BMP), being indispensable for certain developmental events.Noggin expression positively correlated with EGFR expression in both GC cell line models and The Cancer Genome Atlas human GC cohort. Targeting EGFR and its downstream pathways diminished cell proliferation which was promoted by Noggin. Noggin promotes the proliferation of GC cells by upregulating EGFR and enhancing a vicious circle formed by β‑catenin, EGFR, ERK and Akt. Noggin/NOG... | |||
TMPJ-00042 |
TSLP Protein, Human, Recombinant
TSLP,Thymic stromal lymphopoietin |
Human | E. coli |
Thymic stromal lymphopoietin (TSLP) is a novel member of the hemopoietic cytokine family that promotes the development of B cells and shares overlapping activity with IL-7. The human TSLP protein comprises a 28 amino acids (aa) signal sequence and 131 aa mature region. Human TSLP has two isoforms lfTSLP and sfTSLP produced by alternative splicing . lfTSLP is expressed in a number of tissues including heart, liver and prostate, and sfTSLP (63aa) is predominantly expressed in keratinocytes of oral... | |||
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Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TMIH-0396 |
N-Nitroso-N-methylaniline-d5
|
||
N-Nitroso-N-methylaniline-d5 是 N-Nitroso-N-methylaniline 的氘代化合物。 | |||
TMIJ-0027 |
3-Methyl-2-quinoxalinecarboxylic Acid-d4
MQCA-d4 |
||
3-Methyl-2-quinoxalinecarboxylic Acid-d4 是 3-Methyl-2-quinoxalinecarboxylic Acid 的氘代化合物。3-Methyl-2-quinoxalinecarboxylic Acid 的 CAS 号为 74003-63-7。3-Methyl-2-quinoxalinecarboxylic acid 在生命科学相关研究中具有广泛的应用。 | |||
TMIH-0564 |
Tetracycline-d6
|
||
Tetracycline-d6 是 Tetracycline 的氘代化合物。 | |||
TMIH-0207 |
E-10-Hydroxynortriptyline-d3
|
||
E-10-Hydroxynortriptyline-d3 是 E-10-Hydroxynortriptyline 的氘代化合物。E-10-Hydroxynortriptyline 的 CAS 号为 47132-16-1。 | |||
TMIH-0149 |
Choline-d4 Chloride
|
||
Choline-d4 Chloride 是 Choline Chloride 的氘代化合物。 | |||
TMIJ-0215 |
Doxofylline-d4
|
||
Doxofylline-d4 是 Doxofylline 的氘代化合物。Doxofylline 的 CAS 号为 69975-86-6。Doxofylline 是腺苷 A1 受体拮抗剂,且能抑制磷酸二酯酶 IV,用于治疗哮喘。 | |||
TMIJ-0247 |
Doxycycline-d3 HCl
|
||
Doxycycline-d3 HCl 是 Doxycycline HCl 的氘代化合物。Doxycycline HCl 的 CAS 号为 100929-47-3。 | |||
TMID-0118 |
Doxofylline-d6
|
||
Doxofylline-d6 是 Doxofylline 的氘代化合物。Doxofylline 的 CAS 号为 69975-86-6。Doxofylline 是腺苷 A1 受体拮抗剂,且能抑制磷酸二酯酶 IV,用于治疗哮喘。 | |||
TMID-0232 |
Choline-d13 Bromide (N,N,N-trimethyl-d9; 1,1,2,2-d4)
|
||
Choline-d13 Bromide (N,N,N-trimethyl-d9; 1,1,2,2-d4) 是 Choline Bromide 的氘代化合物。Choline Bromide 的 CAS 号为 1927-06-6。 | |||
TMID-0117 |
Aminophylline-d6
|
||
Aminophylline-d6 是 Aminophylline 的氘代化合物。Aminophylline 的 CAS 号为 317-34-0。Aminophylline 是一种竞争性非选择性磷酸二酯酶抑制剂,具有支气管扩张作用。它是竞争性的腺苷受体拮抗剂,有用于哮喘研究的潜力。 | |||
T71329 |
Theophylline-d6
|
||
Theophylline-d6 is intended for use as an internal standard for the quantification of theophylline by GC- or LC-MS. Theophylline is an inhibitor of phosphodiesterase. It is also an adenosine A1 and A2 receptor antagonist. Theophylline induces relaxation of isolated cat bronchial smooth muscle segments precontracted with acetylcholine. It inhibits ovalbumin-induced increases in bronchoalveolar lavage fluid (BALF) eosinophil infiltration in an ovalbumin-sensitized mouse model of allergic asthma. F... | |||
TMIH-0165 |
Clorprenaline-d7
|
||
Clorprenaline-d7 是 Clorprenaline 的氘代化合物。Clorprenaline 的 CAS 号为 3811-25-4。 | |||
TMIH-0565 |
Tetracycline EP Impurity A-d6
4-Epitetracycline-d6 |
||
Tetracycline EP Impurity A-d6 是 Tetracycline EP Impurity A 的氘代化合物。Tetracycline EP Impurity A 的 CAS 号为 79-85-6。 | |||
TMIJ-0231 |
Hydroxy Pentoxifylline-d6
rac-Lisofylline-d6 |
||
Hydroxy Pentoxifylline-d6 是 Hydroxy Pentoxifylline 的氘代化合物。Hydroxy Pentoxifylline 的 CAS 号为 6493-06-7。(±)-Lisofylline 是一种对映异构体特异性、烷基取代的甲基黄嘌呤,在下调白细胞活化方面具有特异性和有效的活性。它是一种抗炎剂。 | |||
TMID-0187 |
Amitriptyline-d6 Hydrochloride
|
||
Amitriptyline-d6 Hydrochloride 是 Amitriptyline Hydrochloride 的氘代化合物。Amitriptyline Hydrochloride 的 CAS 号为 549-18-8。Amitriptyline hydrochloride 是血清素再摄取转运体和去甲肾上腺素再摄取转运体抑制剂,还与多巴胺再摄取转运体结合,其Ki为 2.58 μM。它也抑制肾上腺素能受体、毒蕈碱受体、组胺受体、5-羟色胺受体。它是TrkA和TrkA受体的激动剂,具有强神经营养活性和有抗抑郁作用。 | |||
TMIJ-0381 |
L-Valine-13C5-15N
|
||
L-Valine-13C5-15N 是 L-Valine 的 13C 和 15 N 的标记化合物。L-Valine 的 CAS 号为 72-18-4。L-Valine 是蛋白二十种氨基酸中的其中一种。它是必需氨基酸。 | |||
TMIJ-0251 |
Nicergoline-13C-d3
|
||
Nicergoline-13C-d3 是 Nicergoline 的 13C 和氘代化合物。Nicergoline 的 CAS 号为 27848-84-6。Nicergoline 是一种有效的,选择性的、具有口服活性的α1A-肾上腺素能受体拮抗剂,是一种溴烟碱酸的麦角林衍生物。它具有血管舒张作用,可以改善阿尔茨海默症小鼠的认知功能。 | |||
TMIJ-0342 |
Aniline-d5
|
||
Aniline-d5 是 Aniline 的氘代化合物。Aniline 的 CAS 号为 62-53-3。Aniline 通过铁过载和通过血红素加氧酶 1 上调诱导氧化应激对脾脏产生毒性。它会导致 p-IKKα 和 p-IKKβ 显着增加,进而增加 NF-κB 和 AP-1 结合活性。 | |||
T71300 |
Pentoxifylline-d6
|
||
Pentoxifylline-d6 is intended for use as an internal standard for the quantification of pentoxifylline by GC- or LC-MS. Pentoxifylline is a hemorrheologic agent. It increases the deformability of washed isolated human erythrocytes when used at a concentration of 100 µM. Pentoxifylline (1, 2, and 3 mM) inhibits ADP-induced platelet aggregation in isolated human whole blood. It inhibits thrombus formation induced by ADP in a hamster cheek pouch model when administered at doses of 5, 10, and 20 mg/... | |||
T36903 |
Rasagiline-13C3 (mesylate)
Rasagiline-13C3 (mesylate) |
||
Rasagiline-13C3is intended for use as an internal standard for the quantification of rasagiline by GC- or LC-MS. Rasagiline is an inhibitor of monoamine oxidase B (MAO-B; IC50= 4.43 nM for the rat brain enzyme).1It is selective for MAO-B over MAO-A (IC50= 412 nM for the rat brain enzyme). It inhibits serum and NGF withdrawal-induced apoptosis of PC12 cells when used at concentrations ranging from 0.01 to 100 μM.2Rasagiline inhibits rat brain MAO-Bin vivo(ED50= 0.1 mg/kg).1It reduces cerebral ede... | |||
T33348 |
Methyl-d9-choline
J2.078.736H |
||
Methyl -D9- choline is an isotopically labeled choline tracer. | |||
TMID-0054 |
2-Quinoxalinecarboxylic acid-d4
|
||
2-Quinoxalinecarboxylic acid-d4 是 2-Quinoxalinecarboxylic acid 的氘代化合物。2-Quinoxalinecarboxylic acid 的 CAS 号为 879-65-2。 | |||
T70960 |
Maprotiline-d3 hydrochloride
|
||
Maprotiline-d3 is intended for use as an internal standard for the quantification of maprotiline by GC- or LC-MS. Maprotiline is a tricyclic antidepressant. It binds to the norepinephrine transporter (NET) and is selective for NET over the serotonin and dopamine transporters. Maprotiline also binds to the serotonin (5-HT) receptor subtype 5-HT2A, as well as histamine H1, muscarinic acetylcholine, α1-adrenergic, and dopamine D2 receptors. In vivo, maprotiline inhibits norepinephrine reuptake in r... | |||
TMIH-0559 |
Terbutaline-d9
|
||
Terbutaline-d9 是 Terbutaline 的氘代化合物。 | |||
TMIH-0542 |
Sulfaquinoxaline-d4
|
||
Sulfaquinoxaline-d4 是 Sulfaquinoxaline 的氘代化合物。 | |||
TMIJ-0218 |
Nortriptyline-d3 HCl
|
||
Nortriptyline-d3 HCl 是 Nortriptyline HCl 的氘代化合物。Nortriptyline HCl 的 CAS 号为 894-71-3。Nortriptyline hydrochloride 是一种三环类抗抑郁药,用于缓解抑郁症的症状。它是 Amitriptyline 的主要活性代谢产物,是有效自噬抑制剂。 | |||
TMID-0119 |
Diprophylline-d6
|
||
Diprophylline-d6 是 Diprophylline 的氘代化合物。Diprophylline 的 CAS 号为 479-18-5。Diphylline 是一种A1/A2腺苷受体拮抗剂,也是环状核苷酸磷酸二酯酶抑制剂。它是一种黄嘌呤衍生物,具有支气管扩张和血管扩张作用,有用于治疗慢性支气管炎和肺气肿的潜力。 | |||
TMID-0307 |
Sertraline-d3 Hydrochloride
|
||
Sertraline-d3 Hydrochloride 是 Sertraline Hydrochloride 的氘代化合物。Sertraline Hydrochloride 的 CAS 号为 79559-97-0。Sertraline hydrochloride 是选择性 5- 羟色胺再吸收抑制剂类的抗抑郁剂,可用于多种疾病的研究,如重度抑郁症和强迫症。 | |||
T12693 |
Rasagiline 13C3 mesylate racemic
TVP1012 13C3 racemic,AGN1135 13C3 racemic |
Others | Others |
Rasagiline 13C3 mesylate racemic is the deuterium labeled Rasagiline, which is an irreversible monoamine oxidase inhibitor. | |||
TMIH-0210 |
Eluxadoline-13C-d3
|
||
Eluxadoline-13C-d3 是 Eluxadoline 的 13C 和氘代化合物。Eluxadoline 的 CAS 号为 864825-13-8。 | |||
TMIH-0460 |
Protriptyline-d3 Hydrochloride
|
||
Protriptyline-d3 Hydrochloride 是 Protriptyline Hydrochloride 的氘代化合物。 | |||
TMIH-0424 |
Pentoxyfylline-d6
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Pentoxyfylline-d6 是 Pentoxyfylline 的氘代化合物。Pentoxyfylline 的 CAS 号为 。Questiomycin A derivatives 20 是一种Questiomycin A衍生物。 | |||
TMIH-0064 |
8-Chlorotheophylline-d6
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8-Chlorotheophylline-d6 是 8-Chlorotheophylline 的氘代化合物。8-Chlorotheophylline 的 CAS 号为 85-18-7。 | |||
TMIJ-0363 |
DL-Valine-d8
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DL-Valine-d8 是 DL-Valine 的氘代化合物。DL-Valine 的 CAS 号为 516-06-3。DL-Valine 是 2-氨基-3-甲基丁酸。它是在植物中从丙酮酸开始通过几个步骤合成的。 | |||
TMID-0257 |
Quinoline-d7
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Quinoline-d7 是 Quinoline 的氘代化合物。Quinoline 的 CAS 号为 91-22-5。Quinoline 存在于酒精饮料中。 它是一种来自包括薄荷在内的多种植物的生物碱。 也存在于可可、红茶和苏格兰威士忌中。 老化的样品,如果暴露在光线下,会变成黄色,然后变成棕色。 | |||
T11853 |
Linezolid-d3
Linezolid D3,PNU-100766 D3 |
Others | Others |
Linezolid D3, a deuterium-labeled version of Linezolid, is a synthetic antibiotic designed to halt the initiation of bacterial protein synthesis. | |||
TMIH-0608 |
Z-10-Hydroxynortriptyline-d3
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Z-10-Hydroxynortriptyline-d3 是 Z-10-Hydroxynortriptyline 的氘代化合物。Z-10-Hydroxynortriptyline 的 CAS 号为 47132-19-4。 | |||
TMIJ-0089 |
L-Valine-d8
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L-Valine-d8 是 L-Valine 的氘代化合物。L-Valine 的 CAS 号为 72-18-4。L-Valine 是蛋白二十种氨基酸中的其中一种。它是必需氨基酸。 | |||
TMID-0207 |
Maprotiline-d5 Hydrochloride
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Maprotiline-d5 Hydrochloride 是 Maprotiline Hydrochloride 的氘代化合物。Maprotiline Hydrochloride 的 CAS 号为 10347-81-6。Maprotiline hydrochloride 是一种桥环四环类抗抑郁药,是去甲肾上腺素重吸收抑制剂。 | |||
TMID-0084 |
Tigecycline-d9
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Tigecycline-d9 是 Tigecycline 的氘代化合物。Tigecycline 的 CAS 号为 220620-09-7。Tigecycline是甘氨酰环素抗生素,对Acinetobacter baumannii(A. baumannii) 的 MIC50和 MIC90分别为 1 和 2 mg/L。它对E. coli(MG1655 菌株) 的平均抑制浓度 (MIC) 约 125 ng/ mL。 |