Cephaeline dihydrochloride

Name: Cephaeline dihydrochloride
Brand: TargetMol
SKU: TQ0109
Price: 638 USD
Availability: InStock
Rating: 4.5 (1 reviews)

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产品编号 TQ0109Cas号 5853-29-2

别名 盐酸吐根酚碱, NSC 32944, (-)-Cephaeline dihydrochloride

(-)-Cephaeline (dihydrochloride) is an enantiomer of Cephaeline. Cephaeline is a selective CYP2D6 inhibitor (IC50: 121 μM).

还可以

产品编号 TQ0109 别名 盐酸吐根酚碱, NSC 32944, (-)-Cephaeline dihydrochlorideCas号 5853-29-2

(-)-Cephaeline (dihydrochloride) is an enantiomer of Cephaeline. Cephaeline is a selective CYP2D6 inhibitor (IC50: 121 μM).

规格	价格	库存	数量
2 mg	¥ 594	5日内发货
100 mg	¥ 7,410	1-2周

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产品介绍

生物活性

产品描述	(-)-Cephaeline (dihydrochloride) is an enantiomer of Cephaeline. Cephaeline is a selective CYP2D6 inhibitor (IC50: 121 μM).
靶点活性	CYP2D6:121 μM
体外活性	IC50 of Cephaeline against CYP2C9, CYP2D6, and CYP3A4 is over 1000, 121 and 1000 μM, respectively. Further experiments are performed to determine inhibition constants (Ki) for Cephaeline on the CYP2D6 and CYP3A4 activities Graphic analysis of Dixon plots at various Cephaeline concentrations for each of the two CYP enzyme assays yield Kis of 54 and 355 μM for CYP2D6 and CYP3A4, respectively.
别名	盐酸吐根酚碱, NSC 32944, (-)-Cephaeline dihydrochloride

化学信息

储存&溶解度

存储	keep away from direct sunlight \| Powder: -20°C for 3 years \| In solvent: -80°C for 1 year \| Shipping with blue ice.
溶解度信息	DMSO: 80 mg/mL H2O: 60 mg/mL